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1
المؤلفون: Joseph T. Repine, Lorraine Kathleen Fay, Favor David, Hyacinth Akunne, Kim Nicholls, Bradley Snyder, Liming Zhang, Kevin A. Serpa, Douglas S. Johnson, Lawrence W. Fitzgerald, Andrew D. White, Chung Choi, Steven Z. Whetzel
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:2621-2625
مصطلحات موضوعية: Male, Bipolar Disorder, Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Catalepsy, Biochemistry, Partial agonist, Chemical synthesis, Piperazines, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Drug Discovery, medicine, Animals, Naphthyridines, Antipsychotic, Receptor, Piperazine, Molecular Biology, Molecular Structure, Receptors, Dopamine D2, Chemistry, Aryl, Organic Chemistry, Haplorhini, medicine.disease, Rats, Schizophrenia, Molecular Medicine, Antipsychotic Agents
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2
المؤلفون: Kay Ahn, Benjamin F. Cravatt, Cory Michael Stiff, Yuntao Song, Sarah E. Smith, Mark Morris, Douglas S. Johnson, Tyzoon K. Nomanbhoy, James B. Dunbar, David Beidler, Lorraine Kathleen Fay, Marya Liimatta, Lazerwith Scott E, Tracy Fay Gregory, Suzanne Ross Kesten
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:2865-2869
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Thiophenes, Biochemistry, Article, Piperazines, Amidohydrolases, Amidase, Serine, Structure-Activity Relationship, chemistry.chemical_compound, Piperidines, Fatty acid amide hydrolase, Drug Discovery, Animals, Humans, Urea, Computer Simulation, Enzyme Inhibitors, Molecular Biology, biology, Organic Chemistry, Activity-based proteomics, Benzothiophene, Biological activity, Rats, Piperazine, Models, Chemical, nervous system, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, lipids (amino acids, peptides, and proteins), psychological phenomena and processes
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3
المؤلفون: Dong Liming, Xinjun Hou, Elizabeth A. Lunney, Corinne E. Augelli-Szafran, Deal Judith G, Christopher F. Bigge, Darin Vanderpool, Raymond Andrew Hudack, Nancy Sue Barta, Bradley William Caprathe, Chuangxing Guo, Steve Bender, Richard E. Showalter, Lorraine Kathleen Fay, Arindam Chatterjee
المصدر: Journal of Medicinal Chemistry. 49:1202-1206
مصطلحات موضوعية: Peptidylprolyl isomerase, Aza Compounds, Binding Sites, Neurite, Chemistry, Hydrogen Bonding, Biological activity, Tacrolimus Binding Protein 1A, Isoquinolines, Ligands, Amides, Heterocyclic Compounds, 4 or More Rings, Tacrolimus, Structure-Activity Relationship, Neuroprotective Agents, FKBP, Biochemistry, Cis-trans-Isomerases, Drug Discovery, Molecular Medicine, Structure–activity relationship, Binding site, Cognitive decline
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4
المؤلفون: David T. Dudley, Tyzoon K. Nomanbhoy, Benjamin F. Cravatt, Nalini Sadagopan, Stephen J. Kesten, Shobha N. Bhattachar, David Beidler, Lorraine Kathleen Fay, Cory Michael Stiff, Marya Liimatta, Mark Morris, Lazerwith Scott E, Douglas S. Johnson, Kay Ahn, Suzanne Ross Kesten, Sarah E. Smith
المصدر: ACS medicinal chemistry letters. 2(2)
مصطلحات موضوعية: Fatty acid amide, Organic Chemistry, Serine hydrolase, Cannabinoid Receptor Agonists, Anandamide, Biology, Pharmacology, Biochemistry, Endocannabinoid system, Serine, chemistry.chemical_compound, nervous system, chemistry, Fatty acid amide hydrolase, Drug Discovery, lipids (amino acids, peptides, and proteins), PF-04457845, psychological phenomena and processes