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1Academic Journal
المؤلفون: Schimunek, Johannes, Seidl, Philipp, Elez, Katarina, Hempel, Tim, Le, Tuan, Noé, Frank, Olsson, Simon, Raich, Lluís, Winter, Robin, Gokcan, Hatice, Gusev, Filipp, Gutkin, Evgeny, Isayev, Olexandr, Kurnikova, Maria, Narangoda, Chamali, Zubatyuk, Roman, Bosko, Ivan, Furs, Konstantin, Karpenko, Anna, Kornoushenko, Yury, Shuldau, Mikita, Yushkevich, Artsemi, Benabderrahmane, Mohammed, Bousquet-Melou, Patrick, Bureau, Ronan, Charton, Beatrice, Cirou, Bertrand, Gil, Gérard, Allen, William, Sirimulla, Suman, Watowich, Stanley, Antonopoulos, Nick, Epitropakis, Nikolaos, Krasoulis, Agamemnon, Pitsikalis, Vassilis, Theodorakis, Stavros, Kozlovskii, Igor, Maliutin, Anton, Medvedev, Alexander, Popov, Petr, Zaretckii, Mark, Eghbal-Zadeh, Hamid, Halmich, Christina, Hochreiter, Sepp, Mayr, Andreas, Ruch, Peter, Widrich, Michael, Berenger, Francois, Kumar, Ashutosh, Yamanishi, Yoshihiro, Zhang, Kam, Bengio, Emmanuel, Bengio, Yoshua, Jain, Moksh, Korablyov, Maksym, Liu, Cheng-Hao, Gilles, Marcous, Glaab, Enrico, Barnsley, Kelly, Iyengar, Suhasini, Ondrechen, Mary Jo, Haupt, V. Joachim, Kaiser, Florian, Schroeder, Michael, Pugliese, Luisa, Albani, Simone, Athanasiou, Christina, Beccari, Andrea, Carloni, Paolo, d'Arrigo, Giulia, Gianquinto, Eleonora, Goßen, Jonas, Hanke, Anton, Joseph, Benjamin, Kokh, Daria, Kovachka, Sandra, Manelfi, Candida, Mukherjee, Goutam, Muñiz-Chicharro, Abraham, Musiani, Francesco, Nunes-Alves, Ariane, Paiardi, Giulia, Rossetti, Giulia, Sadiq, S. Kashif, Spyrakis, Francesca, Talarico, Carmine, Tsengenes, Alexandros, Wade, Rebecca, Copeland, Conner, Gaiser, Jeremiah, Olson, Daniel, Roy, Amitava, Venkatraman, Vishwesh, Wheeler, Travis, Arthanari, Haribabu, Blaschitz, Klara, Cespugli, Marco, Durmaz, Vedat, Fackeldey, Konstantin, Fischer, Patrick, Gorgulla, Christoph, Gruber, Christian, Gruber, Karl, Hetmann, Michael, Kinney, Jamie, Das, Krishna, Pandita, Shreya, Singh, Amit, Steinkellner, Georg, Tesseyre, Guilhem, Wagner, Gerhard, Wang, Zi-Fu, Yust, Ryan, Druzhilovskiy, Dmitry, Filimonov, Dmitry, Pogodin, Pavel, Poroikov, Vladimir, Rudik, Anastassia, Stolbov, Leonid, Veselovsky, Alexander, de Rosa, Maria, Simone, Giada De, Gulotta, Maria, Lombino, Jessica, Mekni, Nedra, Perricone, Ugo, Casini, Arturo, Embree, Amanda, Gordon, D. Benjamin, Lei, David, Pratt, Katelin, Voigt, Christopher, Chen, Kuang-Yu, Jacob, Yves, Krischuns, Tim, Lafaye, Pierre, Zettor, Agnès, Rodríguez, M. Luis, White, Kris, Fearon, Daren, von Delft, Frank, Walsh, Martin, Horvath, Dragos, Brooks, Charles, Falsafi, Babak, Ford, Bryan, García-Sastre, Adolfo, Lee, Sang Yup, Naffakh, Nadia, Varnek, Alexandre, Klambauer, Guenter, Hermans, Thomas
المساهمون: Johannes Kepler Universität (JKU), Laboratoire de Photophysique et Photochimie Supramoléculaires et Macromoléculaires (PPSM), École normale supérieure - Cachan (ENS Cachan)-Institut de Chimie - CNRS Chimie (INC-CNRS)-Centre National de la Recherche Scientifique (CNRS), Freie Universität Berlin, Departament de Quimica Fisica and Institut de Quimica Teorica i Computacional (IQTCUB), Universitat de Barcelona (UB), Carnegie Mellon University Pittsburgh (CMU), Institute for Scintillation Materials of NASU, National Academy of Sciences of Ukraine = Національна академія наук України = Académie nationale des sciences d'Ukraine (NASU / НАН України), Centre d'Etudes et de Recherche sur le Médicament de Normandie (CERMN), Université de Caen Normandie (UNICAEN), Normandie Université (NU)-Normandie Université (NU), CRIANN, Centre de Ressources Informatiques de Haute-Normandie, France (CRIHAN), Biologie des ARN et virus influenza - RNA Biology of Influenza Virus (CNRS-UMR3569), Institut Pasteur Paris (IP)-Centre National de la Recherche Scientifique (CNRS)-Université Paris Cité (UPCité), Génétique moléculaire des virus à ARN, Institut Pasteur Paris (IP)-Centre National de la Recherche Scientifique (CNRS), Ingénierie des Anticorps (plate-forme) - Antibody Engineering (Platform), Criblage chémogénomique et biologique (Plateforme) - Chemogenomic and Biological Screening Platform (PF-CCB), Institut Pasteur Paris (IP)-Institut de Chimie - CNRS Chimie (INC-CNRS)-Centre National de la Recherche Scientifique (CNRS)-Université Paris Cité (UPCité)
المصدر: ISSN: 1868-1743.
مصطلحات موضوعية: SARS-Cov2, computational drug discovery, covid-19, [SDV]Life Sciences [q-bio], [CHIM]Chemical Sciences, [INFO]Computer Science [cs]
Relation: info:eu-repo/semantics/altIdentifier/pmid/37833243; pasteur-04269641; https://pasteur.hal.science/pasteur-04269641; https://pasteur.hal.science/pasteur-04269641/document; https://pasteur.hal.science/pasteur-04269641/file/Molecular%20Informatics%20-%202023%20-%20Schimunek%20-%20A%20community%20effort%20in%20SARS%E2%80%90CoV%E2%80%902%20drug%20discovery.pdf; PUBMED: 37833243
الاتاحة: https://pasteur.hal.science/pasteur-04269641
https://pasteur.hal.science/pasteur-04269641/document
https://pasteur.hal.science/pasteur-04269641/file/Molecular%20Informatics%20-%202023%20-%20Schimunek%20-%20A%20community%20effort%20in%20SARS%E2%80%90CoV%E2%80%902%20drug%20discovery.pdf
https://doi.org/10.1002/minf.202300262 -
2Academic Journal
المؤلفون: Lombino, Jessica, Vallone, Rosario, Cimino, Maura, Gulotta, Maria Rita, De Simone, Giada, Morando, Maria Agnese, Sabbatella, Raffaele, Di Martino, Simona, Fogazza, Mario, Sarno, Federica, Coronnello, Claudia, De Rosa, Maria, Cipollina, Chiara, Altucci, Lucia, Perricone, Ugo, Alfano, Caterina
المصدر: Lombino , J , Vallone , R , Cimino , M , Gulotta , M R , De Simone , G , Morando , M A , Sabbatella , R , Di Martino , S , Fogazza , M , Sarno , F , Coronnello , C , De Rosa , M , Cipollina , C , Altucci , L , Perricone , U & Alfano , C 2023 , ' In-silico guided chemical exploration of KDM4A fragments hits ' , Clinical Epigenetics , vol. 15 , no. 1 , 197 . https://doi.org/10.1186/s13148-023-01613-7
مصطلحات موضوعية: Epigenetic regulation, Fragment-based drug discovery (FBDD), KDM4 inhibitors, KDM4A, Lysine demethylases, Rational drug design
وصف الملف: application/pdf
الاتاحة: https://hdl.handle.net/11370/1f72f9e4-e237-4c3f-a220-787265437197
https://research.rug.nl/en/publications/1f72f9e4-e237-4c3f-a220-787265437197
https://doi.org/10.1186/s13148-023-01613-7
https://pure.rug.nl/ws/files/909181922/s13148-023-01613-7.pdf
http://www.scopus.com/inward/record.url?scp=85180244483&partnerID=8YFLogxK -
3Academic Journal
المؤلفون: Costanzo, Giuliana, Patamia, Vincenzo, Turnaturi, Rita, Parenti, Carmela, Zagni, Chiara, Lombino, Jessica, Amata, Emanuele, Marrazzo, Agostino, Pasquinucci, Lorella, Rescifina, Antonio
المساهمون: Università di Catania
المصدر: Chemical Biology & Drug Design ; volume 101, issue 6, page 1382-1392 ; ISSN 1747-0277 1747-0285
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4Academic Journal
المؤلفون: Dichiara, Maria, Ambrosio, Francesca Alessandra, Lee, Sang Min, Ruiz-Cantero, M. Carmen, Lombino, Jessica, Coricello, Adriana, Costa, Giosuè, Shah, Dhara, Costanzo, Giuliana, Pasquinucci, Lorella, Son, Kyung No, Cosentino, Giuseppe, González-Cano, Rafael, Marrazzo, Agostino, Aakalu, Vinay Kumar, Cobos, Enrique J., Alcaro, Stefano, Amata, Emanuele
المساهمون: National Institute of Neurological Disorders and Stroke, National Eye Institute, Research to Prevent Blindness, Junta de Andalucía, Agencia Estatal de Investigación, Ministero dell’Istruzione, dell’Università e della Ricerca
المصدر: Journal of Medicinal Chemistry ; volume 66, issue 16, page 11447-11463 ; ISSN 0022-2623 1520-4804
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5Academic JournalA new family of Jumonji C domain-containing KDM inhibitors inspired by natural product Purpurogallin
المؤلفون: Souto Salgado, Jose Antonio, Sarno, Federica, Nebbioso, Ángela, Papulino, Chiara, Álvarez Rodríguez, Maria Rosana, Lombino, Jessica, Perricone, Ugo, Padova, Alessandro, Altucci, Lucia, Rodríguez de Lera, Ángel
مصطلحات موضوعية: 3207.03 Carcinogénesis, 2302 Bioquímica, 2306 Química Orgánica
Relation: Frontiers in Chemistry, 8, 00312 (2020); http://hdl.handle.net/11093/2344; https://www.frontiersin.org/article/10.3389/fchem.2020.00312/full
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6Academic Journal
المؤلفون: Gulotta, Maria Rita, Lombino, Jessica, Perricone, Ugo, De Simone, Giada, Mekni, Nedra, De Rosa, Maria, Diana, Patrizia, Padova, Alessandro
المصدر: ChemMedChem ; volume 15, issue 20, page 1921-1931 ; ISSN 1860-7179 1860-7187
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7Academic Journal
المؤلفون: Elkholy, Nada, Abdelwaly, Ahmad, Mohamed, Karim, Amata, Emanuele, Lombino, Jessica, Cosentino, Giuseppe, Intagliata, Sebastiano, Helal, Mohamed A.
المساهمون: Academy of Scientific Research and Technology
المصدر: Chemical Biology & Drug Design ; volume 100, issue 1, page 25-40 ; ISSN 1747-0277 1747-0285
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8
المؤلفون: LOMBINO, Jessica
المساهمون: DIANA, Patrizia
مصطلحات موضوعية: Drug Design, KDM4A, Epigenetic, Carbenoid, PCR2, Dynamic pharmacophore, Settore CHIM/08 - Chimica Farmaceutica
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9Academic Journal
المؤلفون: Lombino, Jessica, Gulotta, Maria Rita, De Simone, Giada, Mekni, Nedra, De Rosa, Maria, Carbone, Daniela, Parrino, Barbara, Cascioferro, Stella Maria, Diana, Patrizia, Padova, Alessandro, Perricone, Ugo
المصدر: Molecular Informatics ; volume 40, issue 2 ; ISSN 1868-1743 1868-1751
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10Academic Journal
المؤلفون: Ielo, Laura, Castoldi, Laura, Touqeer, Saad, Lombino, Jessica, Roller, Alexander, Prandi, Cristina, Holzer, Wolfgang, Pace, Vittorio
المصدر: Angewandte Chemie International Edition ; volume 59, issue 47, page 20852-20857 ; ISSN 1433-7851 1521-3773
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11Academic Journal
المؤلفون: Perricone, Ugo, Gulotta, Maria Rita, Lombino, Jessica, Parrino, Barbara, Cascioferro, Stella, Diana, Patrizia, Cirrincione, Girolamo, Padova, Alessandro
المصدر: MedChemComm ; volume 9, issue 6, page 920-936 ; ISSN 2040-2503 2040-2511
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12Academic Journal
المؤلفون: Lombino, Jessica, Gulotta, Maria Rita, De Simone, Giada, Mekni, Nedra, De Rosa, Maria, Carbone, Daniela, Parrino, Barbara, Cascioferro, Stella Maria, Diana, Patrizia, Padova, Alessandro, Perricone, Ugo
المصدر: Molecular Informatics; Feb2021, Vol. 40 Issue 2, p1-9, 9p
مصطلحات موضوعية: COMPUTER-assisted drug design, RECEIVER operating characteristic curves, PROTEIN structure, GENE silencing, CHROMATIN-remodeling complexes, PROTEIN-ligand interactions
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13Academic Journal
المؤلفون: Ielo, Laura, Castoldi, Laura, Touqeer, Saad, Lombino, Jessica, Roller, Alexander, Prandi, Cristina, Holzer, Wolfgang, Pace, Vittorio
المصدر: Angewandte Chemie; 11/16/2020, Vol. 132 Issue 47, p21038-21043, 6p
مصطلحات موضوعية: CATALYSIS, AZIRIDINES, LIGANDS (Chemistry), METALATION, CHLORIDES
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14Academic Journal
المؤلفون: Mekni, Nedra, De Rosa, Maria, Cipollina, Chiara, Gulotta, Maria Rita, De Simone, Giada, Lombino, Jessica, Padova, Alessandro, Perricone, Ugo
المصدر: International Journal of Molecular Sciences; Oct2019, Vol. 20 Issue 20, p4974, 1p, 5 Color Photographs, 1 Chart, 4 Graphs
مصطلحات موضوعية: PYRIN (Protein), ALZHEIMER'S disease, RHEUMATOID arthritis, ANTIBIOTIC residues