-
1Academic Journal
المصدر: 0365-6233 ; Archiv der Pharmazie
مصطلحات موضوعية: Chemistry, Pharmacology. Therapy
Relation: info:eu-repo/semantics/altIdentifier/isi/001268339800001
-
2Academic Journal
المؤلفون: Hartman, Carla B., Dube, Phelelisiwe S., Legoabe, Lesetja J., Van Pelt, Natascha, Matheeussen, An, Caljon, Guy, Beteck, Richard M.
المصدر: 0365-6233 ; Archiv der Pharmazie
مصطلحات موضوعية: Chemistry, Pharmacology. Therapy
Relation: info:eu-repo/semantics/altIdentifier/isi/001169705500001
-
3Academic Journal
المصدر: 1747-0277 ; Chemical biology and drug design
مصطلحات موضوعية: Chemistry, Biology, Pharmacology. Therapy
Relation: info:eu-repo/semantics/altIdentifier/isi/001108369100001
-
4Academic Journal
المؤلفون: Chirwa, Kgothatso A., Francisco, Karol R., Dube, Phelelisiwe S., Park, Hayoung, Legoabe, Lesetja J., Teixeira, Thaiz Rodrigues, Caffrey, Conor R., Beteck, Richard M.
المصدر: ChemMedChem ; volume 19, issue 9 ; ISSN 1860-7179 1860-7187
-
5Academic JournalSynthesis and in vitro biological activity of chalcone derivatives as potential antiparasitic agents
المؤلفون: Setshedi, Koketso J., Beteck, Richard M., Ilbeigi, Kayhan, Mabille, Dorien, Caljon, Guy, Legoabe, Lesetja J.
المصدر: Medicinal Chemistry Research ; ISSN 1054-2523 1554-8120
-
6Academic Journal
المؤلفون: Plaatjie, Moitshepi T. A., Onyiche, ThankGod E., Ramatla, Tsepo, Bezuidenhout, Johannes J., Legoabe, Lesetja, Nyembe, Nthatisi I., Thekisoe, Oriel
المساهمون: North-West University
المصدر: Tropical Medicine and Health ; volume 52, issue 1 ; ISSN 1349-4147
-
7Academic Journal
المؤلفون: Dube, Phelelisiwe S., Legoabe, Lesetja J., Joordan, Audrey, Sigauke, Lester, Warner, Digby F., Beteck, Richard M.
المساهمون: Legoabe, Lesetja- 12902608, Beteck, Richard- 25159194
مصطلحات موضوعية: DprE1, Quinolone, Nitro compounds, Mycobacterium tuberculosis, Benzothiazinone
وصف الملف: application/pdf
Relation: Dube, P.S. et al. 2023. Quinolone analogues of benzothiazinone: Synthesis, antitubercular structure-activity relationship and ADME profiling. European Journal of Medicinal Chemistry 258 (2023) 115539 [https://doi.org/10.1016/j.ejmech.2023.115539]; https://doi.org/10.1016/j.ejmech.2023.115539; http://hdl.handle.net/10394/42560
-
8Academic Journal
المؤلفون: Setshedi, Koketso J.J., Beteck, Richard M.M., Jesumoroti, Omobolanle J.J., Ilbeigi, Kayhan, Mabille, Dorien, Caljon, Guy, Van der Kooy, Frank, Legoabe, Lesetja J.J.
المصدر: 1747-0277 ; Chemical biology and drug design
مصطلحات موضوعية: Chemistry, Biology, Pharmacology. Therapy
Relation: info:eu-repo/semantics/altIdentifier/isi/001019416500001
-
9Academic Journal
المؤلفون: Setshedi, Koketso J., Beteck, Richard M., Jesumoroti, Omobolanle J., Ilbeigi, Kayhan, Mabille, Dorien, Caljon, Guy, Van der Kooy, Frank, Legoabe, Lesetja J.
المساهمون: National Research Foundation
المصدر: Chemical Biology & Drug Design ; volume 102, issue 4, page 763-772 ; ISSN 1747-0277 1747-0285
-
10Academic Journal
المصدر: Chemical Biology & Drug Design ; volume 103, issue 1 ; ISSN 1747-0277 1747-0285
-
11Academic Journal
المساهمون: North-West University
المصدر: Steroids ; volume 197, page 109258 ; ISSN 0039-128X
-
12Academic Journal
المؤلفون: Dube, Phelelisiwe S., Angula, Klaudia T., Legoabe, Lesetja J., Jordaan, Audrey, Boitz Zarella, Jan M., Warner, Digby F., Doggett, J. Stone, Beteck, Richard M.
المساهمون: Schlumberger Foundation, North-West University, National Research Foundation, South African Medical Research Council
المصدر: ACS Omega ; volume 8, issue 19, page 17086-17102 ; ISSN 2470-1343 2470-1343
-
13
-
14
-
15Academic Journal
المؤلفون: Beteck, Richard M., Isaacs, Michelle, Legoabe, Lesetja J., Hoppe, Heinrich C., Tam, Christina C., Kim, Jong H., Petzer, Jacobus P., Cheng, Luisa W., Quiambao, Quincel, Land, Kirkwood M., Khanye, Setshaba D.
المصدر: Archiv der Pharmazie ; volume 356, issue 3 ; ISSN 0365-6233 1521-4184
-
16Academic Journal
المؤلفون: du Preez, Charné, Legoabe, Lesetja J., Jordaan, Audrey, Jesumoroti, Omobolanle J., Warner, Digby F., Beteck, Richard M.
المصدر: Chemical Biology & Drug Design ; volume 101, issue 3, page 717-726 ; ISSN 1747-0277 1747-0285
-
17Academic Journal
المؤلفون: Mahomoodally, Mohamad Fawzi, Aumeeruddy, Muhammad Zakariyyah, Legoabe, Lesetja Jan, Dall’Acqua, Stefano, Zengin, Gokhan
المصدر: Frontiers in Pharmacology ; volume 13 ; ISSN 1663-9812
-
18Academic Journal
المؤلفون: Marais, Lereze, Petzer, Anél, Petzer, Jacobus P., Legoabe, Lesetja J.
المساهمون: 10727388 - Petzer, Jacobus Petrus, 12264954 - Petzer, Anél, 12902608 - Legoabe, Lesetja Jan, 22161333 - Marais, Lereze
مصطلحات موضوعية: Monoamine oxidase, MAO, Inhibition, Reversible, Quinazolinone, Neurodegenerative disorders
Relation: Marais, L. et al. 2020. The monoamine oxidase inhibition properties of C6- and N1-substituted 3-methyl-3,4-dihydroquinazolin-2(1H)-one derivatives. Molecular diversity, 24:391-406. [https://doi.org/10.1007/s11030-019-09960-5]; 1573-501X (Online); http://hdl.handle.net/10394/32503; https://link.springer.com/article/10.1007/s11030-019-09960-5; https://doi.org/10.1007/s11030-019-09960-5
-
19Academic Journal
المؤلفون: Ahmadu, Augustine A., Delehouze, Claire, Haruna, Anas, Mustapha, Lukman, Lawal, Bilqis A., Udobre, Aniefiok, Baratte, Blandine, Triscornia, Camilla, Autret, Axelle, Robert, Thomas, Bulinski, Jeannette Chloe, Rousselot, Morgane, Eugenio, Melanie Simoes, Dimanche-Boitrel, Marie-Thérèse, Petzer, Jacobus P., Legoabe, Lesetja J., Bach, Stéphane
المساهمون: University of Calabar (UNICAL), Kaduna State University, Laboratoire de Biologie Intégrative des Modèles Marins (LBI2M), Sorbonne Université (SU)-Centre National de la Recherche Scientifique (CNRS)-Station biologique de Roscoff = Roscoff Marine Station (SBR), Sorbonne Université (SU)-Centre National de la Recherche Scientifique (CNRS)-Centre National de la Recherche Scientifique (CNRS), Station biologique de Roscoff = Roscoff Marine Station (SBR), Sorbonne Université (SU)-Centre National de la Recherche Scientifique (CNRS), SeaBeLife Biotech, University of Ilorin Ilorin, Nigeria, University of Uyo, Plate-forme de criblage d'inhibiteurs de protéines kinases=Kinase Inhibitor Specialized Screening facility (KISSf), Fédération de recherche de Roscoff (FR2424), Sorbonne Université (SU)-Centre National de la Recherche Scientifique (CNRS)-Sorbonne Université (SU)-Centre National de la Recherche Scientifique (CNRS)-Station biologique de Roscoff = Roscoff Marine Station (SBR), Sorbonne Université (SU)-Centre National de la Recherche Scientifique (CNRS)-Sorbonne Université (SU)-Centre National de la Recherche Scientifique (CNRS), Columbia University New York, Institut de recherche en santé, environnement et travail (Irset), Université d'Angers (UA)-Université de Rennes (UR)-École des Hautes Études en Santé Publique EHESP (EHESP)-Institut National de la Santé et de la Recherche Médicale (INSERM)-Structure Fédérative de Recherche en Biologie et Santé de Rennes ( Biosit : Biologie - Santé - Innovation Technologique ), Biosit : biologie, santé, innovation technologique (SFR UMS CNRS 3480 - INSERM 018), Université de Rennes (UR)-Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS)-Structure Fédérative de Recherche en Biologie et Santé de Rennes ( Biosit : Biologie - Santé - Innovation Technologique ), North-West University South Aftrica (NWU), Nigeria Institution Based Research grant, Tertiary Education Trust Fund (TETFund), French National Agency for Research and Technology (ANRT), Cifre PhD fellowship French National Research Agency (ANR) 2019/0686, Fondation d'Entreprise Grand Ouest, French ANR/Investissements d'Avenir program via the OCEANOMICs project French National Research Agency (ANR) ANR-11-BTBR-0008, ANR-11-BTBR-0008,OCEANOMICS,Biotechnologies et bioressources pour la valorisation des écosystèmes marins planctoniques(2011)
المصدر: ISSN: 1420-3049 ; Molecules ; https://hal.science/hal-03331756 ; Molecules, 2021, 26 (15), pp.4599. ⟨10.3390/molecules26154599⟩.
مصطلحات موضوعية: protein kinase inhibitors, polypharmacology, triterpenoids, Acacia stem bark, [SDV]Life Sciences [q-bio]
Relation: info:eu-repo/semantics/altIdentifier/pmid/34361750; hal-03331756; https://hal.science/hal-03331756; https://hal.science/hal-03331756/document; https://hal.science/hal-03331756/file/molecules-26-04599-v2.pdf; PUBMED: 34361750; PUBMEDCENTRAL: PMC8347092
-
20Academic Journal
المؤلفون: Dube, Phelelisiwe S., Hart, Dylan, Legoabe, Lesetja J., Jordaan, Audrey, Warner, Digby F., Beteck, Richard M.
المصدر: Molbank; Mar2024, Vol. 2024 Issue 1, pM1793, 8p
مصطلحات موضوعية: MANNICH bases, MYCOBACTERIUM tuberculosis, ERYTHROCYTES, CYTOTOXINS, THIAZOLES