نتائج البحث - "Lavoi, Travis M."

1

Academic Journal

N-Branched Tricyclic Guanidines as Novel Melanocortin-3 Receptor Agonists and Melanocortin-4 Receptor Antagonists

المؤلفون: Weirath, Nicholas A., Zajac, Jonathan W. P., Donow, Haley M., Lavoi, Travis M., Pinilla, Clemencia, Santos, Radleigh G., Prajapati, Ritu, Speth, Robert, Ericson, Mark D., Sarupria, Sapna, Giulianotti, Marcello A., Haskell-Luevano, Carrie

المساهمون: National Institute of Diabetes and Digestive and Kidney Diseases

المصدر: Journal of Medicinal Chemistry ; ISSN 0022-2623 1520-4804

الاتاحة: https://doi.org/10.1021/acs.jmedchem.4c01556
https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.4c01556

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2

Academic Journal

Correction to “Discovery of Nanomolar Melanocortin-3 Receptor (MC3R)-Selective Small Molecule Pyrrolidine Bis-Cyclic Guanidine Agonist Compounds Via a High Throughput ‘Unbiased’ Screening Campaign”

المؤلفون: Doering, Skye R., Freeman, Katie, Debevec, Ginamarie, Geer, Phaedra, Santos, Radleigh G., Lavoi, Travis M., Giulianotti, Marc A., Pinilla, Clemencia, Appel, Jon R., Houghten, Richard A., Ericson, Mark D., Haskell-Luevano, Carrie

المساهمون: National Institute of Diabetes and Digestive and Kidney Diseases, National Institute on Drug Abuse, Executive Office of the Governor?s Office of Tourism, Trade, and Economic Development, State of Florida

المصدر: Journal of Medicinal Chemistry ; volume 66, issue 10, page 7063-7065 ; ISSN 0022-2623 1520-4804

الاتاحة: http://dx.doi.org/10.1021/acs.jmedchem.3c00588
https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.3c00588

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3

Academic Journal

The Parallel Structure–Activity Relationship Screening of Three Compounds Identifies the Common Agonist Pharmacophore of Pyrrolidine Bis-Cyclic Guanidine Melanocortin-3 Receptor (MC3R) Small-Molecule Ligands.

المؤلفون: Ericson, Mark D., Freeman, Katie T., LaVoi, Travis M., Donow, Haley M., Santos, Radleigh G., Giulianotti, Marc A., Pinilla, Clemencia, Houghten, Richard A., Haskell-Luevano, Carrie

المصدر: International Journal of Molecular Sciences; Jun2023, Vol. 24 Issue 12, p10145, 29p

مصطلحات موضوعية: STRUCTURE-activity relationships, MELANOCORTIN receptors, LIGANDS (Biochemistry), PYRROLIDINE, GUANIDINE, MOLECULAR weights, GUANIDINES

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4

Academic Journal

Functional Mixture-Based Positional Scan Identifies a Library of Antagonist Tetrapeptide Sequences (LAtTeS) with Nanomolar Potency for the Melanocortin-4 Receptor and Equipotent with the Endogenous AGRP(86-132) Antagonist

المؤلفون: Ericson, Mark D., Doering, Skye R., Larson, Courtney M., Freeman, Katie T., LaVoi, Travis M., Donow, Haley M., Santos, Radleigh G, Cho, Rachel H., Koerperich, Zoe M., Giulianotti, Marc A., Pinilla, Clemencia, Houghten, Richard A., Haskell-Luevano, Carrie

المصدر: Mathematics Faculty Articles

مصطلحات موضوعية: Antagonists, Peptides and proteins, Agonists, Monomers, Mixtures, Mathematics

Relation: https://nsuworks.nova.edu/math_facarticles/323

الاتاحة: https://nsuworks.nova.edu/math_facarticles/323

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5

Periodical

Discovery of Nanomolar Melanocortin-3 Receptor (MC3R)-Selective Small Molecule Pyrrolidine Bis-Cyclic Guanidine Agonist Compounds Via a High-Throughput “Unbiased” Screening Campaign

المؤلفون: Doering, Skye R., Freeman, Katie, Debevec, Ginamarie, Geer, Phaedra, Santos, Radleigh G., Lavoi, Travis M., Giulianotti, Marc A., Pinilla, Clemencia, Appel, Jon R., Houghten, Richard A., Ericson, Mark D., Haskell-Luevano, Carrie

المصدر: Journal of Medicinal Chemistry; May 2021, Vol. 64 Issue: 9 p5577-5592, 16p

6

Academic Journal

SAR Studies of Exosite-Binding Substrate-Selective Inhibitors of ADisintegrin And Metalloprotease 17 (ADAM17) and Application as Selective in Vitro Probes

المؤلفون: Knapinska, Anna M., Dreymuller, Daniela, Ludwig, Andreas, Smith, Lyndsay, Golubkov, Vladislav, Sohail, Anjum, Fridman, Rafael, Giulianotti, Marc, LaVoi, Travis M., Houghten, Richard A., Fields, Gregg B., Minond, Dmitriy

المصدر: Chemistry Faculty Publications

Relation: https://digitalcommons.usf.edu/chm_facpub/192; https://doi.org/10.1021/acs.jmedchem.5b00354

الاتاحة: https://digitalcommons.usf.edu/chm_facpub/192
https://doi.org/10.1021/acs.jmedchem.5b00354

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7

Academic Journal

SAR Studies of Exosite-Binding Substrate-Selective Inhibitors of A Disintegrin And Metalloprotease 17 (ADAM17) and Application as Selective in Vitro Probes

المؤلفون: Knapinska, Anna M., Dreymüller, Daniela, Fields, Gregg B., Minond, Dmitriy, Ludwig, Andreas, Smith, Lyndsay, Golubkov, Vladislav, Sohail, Anjum, Fridman, Rafael, Giulianotti, Marc, LaVoi, Travis M., Houghten, Richard A.

المصدر: Journal of medicinal chemistry 58(15), 5808-5824 (2015). doi:10.1021/acs.jmedchem.5b00354

جغرافية الموضوع: DE

Relation: info:eu-repo/semantics/altIdentifier/issn/0022-2623; info:eu-repo/semantics/altIdentifier/issn/0095-9065; info:eu-repo/semantics/altIdentifier/issn/1943-2992; info:eu-repo/semantics/altIdentifier/wos/WOS:000359683700009; info:eu-repo/semantics/altIdentifier/pmid/pmid:26192023; info:eu-repo/semantics/altIdentifier/issn/1520-4804; https://publications.rwth-aachen.de/record/567723; https://publications.rwth-aachen.de/search?p=id:%22RWTH-CONV-092097%22

الاتاحة: https://publications.rwth-aachen.de/record/567723
https://publications.rwth-aachen.de/search?p=id:%22RWTH-CONV-092097%22

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8

Academic Journal

Combinatorial Libraries As a Tool for the Discovery of Novel, Broad-Spectrum Antibacterial Agents Targeting the ESKAPE Pathogens

المؤلفون: Fleeman, Renee, LaVoi, Travis M., Santos, Radleigh G., Morales, Angela, Nefzi, Adel, Welmaker, Gregory S., Medina-Franco, José L., Giulianotti, Marc A., Houghten, Richard A., Shaw, Lindsey N.

المساهمون: Florida Department of Health, National Institute of Allergy and Infectious Diseases

المصدر: Journal of Medicinal Chemistry ; volume 58, issue 8, page 3340-3355 ; ISSN 0022-2623 1520-4804

الاتاحة: http://dx.doi.org/10.1021/jm501628s
https://pubs.acs.org/doi/pdf/10.1021/jm501628s

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9

Academic Journal

Scaffold Ranking and Positional Scanning Utilized in the Discovery of nAChR-Selective Compounds Suitable for Optimization Studies

المؤلفون: Wu, Jinhua, Zhang, Yaohong, Maida, Laura E., Santos, Radleigh G., Welmaker, Gregory S., LaVoi, Travis M., Nefzi, Adel, Yu, Yongping, Houghten, Richard A., Toll, Lawrence, Giulianotti, Marc A.

المصدر: Journal of Medicinal Chemistry ; volume 56, issue 24, page 10103-10117 ; ISSN 0022-2623 1520-4804

الاتاحة: http://dx.doi.org/10.1021/jm401543h
https://pubs.acs.org/doi/pdf/10.1021/jm401543h

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10

Academic Journal

Scaffold Ranking and PositionalScanning Utilized in the Discovery of nAChR-Selective Compounds Suitablefor Optimization Studies.

المؤلفون: Wu, Jinhua, Zhang, Yaohong, Maida, Laura E., Santos, Radleigh G., Welmaker, Gregory S., LaVoi, Travis M., Nefzi, Adel, Yu, Yongping, Houghten, Richard A., Toll, Lawrence, Giulianotti, Marc A.

المصدر: Journal of Medicinal Chemistry; Dec2013, Vol. 56 Issue 24, p10103-10117, 15p

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