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1Academic Journal
المؤلفون: Xie, Stanley C., Wang, Yinuo, Morton, Craig J., Metcalfe, Riley D., Dogovski, Con, Pasaje, Charisse Flerida A., Dunn, Elyse, Luth, Madeline R., Kumpornsin, Krittikorn, Istvan, Eva S., Park, Joon Sung, Fairhurst, Kate J., Ketprasit, Nutpakal, Yeo, Tomas, Yildirim, Okan, Bhebhe, Mathamsanqa N., Klug, Dana M., Rutledge, Peter J., Godoy, Luiz C., Dey, Sumanta, De Souza, Mariana Laureano, Siqueira-Neto, Jair L., Du, Yawei, Puhalovich, Tanya, Amini, Mona, Shami, Gerry, Loesbanluechai, Duangkamon, Nie, Shuai, Williamson, Nicholas, Jana, Gouranga P., Maity, Bikash C., Thomson, Patrick, Foley, Thomas, Tan, Derek S., Niles, Jacquin C., Han, Byung Woo, Goldberg, Daniel E., Burrows, Jeremy, Fidock, David A., Lee, Marcus C.S., Winzeler, Elizabeth A., Griffin, Michael D.W., Todd, Matthew H., Tilley, Leann
مصطلحات موضوعية: Pharmaceutical chemistry
وصف الملف: text
Relation: https://strathprints.strath.ac.uk/88229/1/Xie-etal-NC-2024-Reaction-hijacking-inhibition-of-Plasmodium-falciparum.pdf; Xie, Stanley C. and Wang, Yinuo and Morton, Craig J. and Metcalfe, Riley D. and Dogovski, Con and Pasaje, Charisse Flerida A. and Dunn, Elyse and Luth, Madeline R. and Kumpornsin, Krittikorn and Istvan, Eva S. and Park, Joon Sung and Fairhurst, Kate J. and Ketprasit, Nutpakal and Yeo, Tomas and Yildirim, Okan and Bhebhe, Mathamsanqa N. and Klug, Dana M. and Rutledge, Peter J. and Godoy, Luiz C. and Dey, Sumanta and De Souza, Mariana Laureano and Siqueira-Neto, Jair L. and Du, Yawei and Puhalovich, Tanya and Amini, Mona and Shami, Gerry and Loesbanluechai, Duangkamon and Nie, Shuai and Williamson, Nicholas and Jana, Gouranga P. and Maity, Bikash C. and Thomson, Patrick and Foley, Thomas and Tan, Derek S. and Niles, Jacquin C. and Han, Byung Woo and Goldberg, Daniel E. and Burrows, Jeremy and Fidock, David A. and Lee, Marcus C.S. and Winzeler, Elizabeth A. and Griffin, Michael D.W. and Todd, Matthew H. and Tilley, Leann (2024 ) Reaction hijacking inhibition of Plasmodium falciparum asparagine tRNA synthetase. Nature Communications , 15 (1). 937. ISSN 2041-1723
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2Academic Journal
المؤلفون: Xie, Stanley, Wang, Yinuo, Morton, Craig, Metcalfe, Riley, Dogovski, Con, Flerida Pasaje, Charisse, Dunn, Elyse, Luth, Madeline R., Kumpornsin, Krittikorn, Istvan, Eva, Sung Park, Joon, Fairhurst, Kate J., Ketprasit, Nutpakal, Yeo, Tomas, Yildirim, Okan, Bhebhe, Mathamsanqa, Klug, Dana M., Rutledge, Peter, Godoy, Luiz C., Laureano de Souza, Mariana, Siqueira-Neto, Jair L., Du, Yawei, Puhalovich, Tanya, Amini, Mona, Shami, Gerald, Loesbanluechai, Duangkamon, Nie, Shuai, Williamson, Nicholas, Jana, Gouranga P., Maity, Bikash C., Thomson, Patrick, Foley, Thomas, Tan, Derek, Niles, Jacquin, Woo Han, Byung, Goldberg, Daniel, Burrows, Jeremy, Fidock, David, Lee, Marcus C.S., Winzeler, Elizabeth A., Griffin, M.D.W., Todd, Matthew, Tilley, Leann
وصف الملف: text
Relation: https://eprints.gla.ac.uk/319051/1/319051.pdf; Xie, S. et al. (2024) Reaction hijacking inhibition of Plasmodium falciparum asparagine tRNA synthetase. Nature Communications , 15, 937. (doi:10.1038/s41467-024-45224-z ) (PMID:38297033) (PMCID:PMC10831071)
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3Academic Journal
المؤلفون: Xie, Stanley C, Wang, Yinuo, Morton, Craig J, Metcalfe, Riley D, Dogovski, Con, Pasaje, Charisse Flerida A, Dunn, Elyse, Luth, Madeline R, Kumpornsin, Krittikorn, Istvan, Eva S, Park, Joon Sung, Fairhurst, Kate J, Ketprasit, Nutpakal, Yeo, Tomas, Yildirim, Okan, Bhebhe, Mathamsanqa N, Klug, Dana M, Rutledge, Peter J, Godoy, Luiz C, Dey, Sumanta, De Souza, Mariana Laureano, Siqueira-Neto, Jair L, Du, Yawei, Puhalovich, Tanya, Amini, Mona, Shami, Gerry, Loesbanluechai, Duangkamon, Nie, Shuai, Williamson, Nicholas, Jana, Gouranga P, Maity, Bikash C, Thomson, Patrick, Foley, Thomas, Tan, Derek S, Niles, Jacquin C, Han, Byung Woo, Goldberg, Daniel E, Burrows, Jeremy, Fidock, David A, Lee, Marcus CS, Winzeler, Elizabeth A, Griffin, Michael DW, Todd, Matthew H, Tilley, Leann
المصدر: Nature Communications , 15 , Article 937. (2024)
مصطلحات موضوعية: Animals, Humans, Plasmodium falciparum, Asparagine, Aspartate-tRNA Ligase, RNA, Transfer, Amino Acyl, Antimalarials, Mammals
وصف الملف: application/pdf
Relation: https://discovery.ucl.ac.uk/id/eprint/10186744/1/Todd_Reaction%20hijacking%20inhibition%20of%20Plasmodium%20falciparum%20asparagine%20tRNA%20synthetase_VoR.pdf; https://discovery.ucl.ac.uk/id/eprint/10186744/
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4Academic Journal
المؤلفون: Bachovchin, Kelly A, Sharma, Amrita, Bag, Seema, Klug, Dana M, Schneider, Katherine M, Singh, Baljinder, Jalani, Hitesh B, Buskes, Melissa J, Mehta, Naimee, Tanghe, Scott, Momper, Jeremiah D, Sciotti, Richard J, Rodriguez, Ana, Mensa-Wilmot, Kojo, Pollastri, Michael P, Ferrins, Lori
المصدر: Journal of Medicinal Chemistry. 62(2)
مصطلحات موضوعية: Rare Diseases, Orphan Drug, Vector-Borne Diseases, Infectious Diseases, Development of treatments and therapeutic interventions, 5.1 Pharmaceuticals, Good Health and Well Being, Animals, Blood Proteins, Disease Models, Animal, Drug Design, Drug Evaluation, Preclinical, Half-Life, Hepatocytes, Humans, Lapatinib, Mice, Microsomes, Liver, Quinazolines, Rats, Solubility, Structure-Activity Relationship, Thermodynamics, Trypanocidal Agents, Trypanosoma brucei brucei, Trypanosomiasis, African, Water, Medicinal and Biomolecular Chemistry, Organic Chemistry, Pharmacology and Pharmaceutical Sciences, Medicinal & Biomolecular Chemistry
وصف الملف: application/pdf
URL الوصول: https://escholarship.org/uc/item/0qv0q4v1
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5Academic Journal
المؤلفون: Dichiara, Maria, Simpson, Quillon J., Quotadamo, Antonio, Jalani, Hitesh B., Huang, Anson X., Millard, Caroline C., Klug, Dana M., Tse, Edwin G., Todd, Matthew H., Silva, Daniel Gedder, Emery, Flavio da Silva, Carlson, J. Eric, Zheng, Shao-Liang, Vleminckx, Margot, Matheeussen, An, Caljon, Guy, Pollastri, Michael P., Sjo, Peter, Perry, Benjamin, Ferrins, Lori
المصدر: 2373-8227 ; ACS Infectious Diseases
مصطلحات موضوعية: Pharmacology. Therapy, Human medicine
Relation: info:eu-repo/semantics/altIdentifier/isi/001024841700001
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6Academic Journal
المؤلفون: Klug, Dana M, Tse, Edwin G, Silva, Daniel G, Cao, Yafeng, Charman, Susan A, Chauhan, Jyoti, Crighton, Elly, Dichiara, Maria, Drake, Chris, Drewry, David, da Silva Emery, Flavio, Ferrins, Lori, Graves, Lee, Hopkins, Emily, Kresina, Thomas AC, Lorente-Macías, Álvaro, Perry, Benjamin, Phipps, Richard, Quiroga, Bruno, Quotadamo, Antonio, Sabatino, Giada N, Sama, Anthony, Schätzlein, Andreas, Simpson, Quillon J, Steele, Jonathan, Shanu-Wilson, Julia, Sjö, Peter, Stapleton, Paul, Swain, Christopher J, Vaideanu, Alexandra, Xie, Huanxu, Zuercher, William, Todd, Matthew H
المصدر: ACS Infectious Diseases (2023) (In press).
مصطلحات موضوعية: Drug discovery, antibacterials, antibiotics, bioactive molecules, open science, organic synthesis
وصف الملف: application/pdf
Relation: https://discovery.ucl.ac.uk/id/eprint/10182369/1/klug-et-al-2023-open-source-antibiotics-simple-diarylimidazoles-are-potent-against-methicillin-resistant-staphylococcus.pdf; https://discovery.ucl.ac.uk/id/eprint/10182369/
الاتاحة: https://discovery.ucl.ac.uk/id/eprint/10182369/1/klug-et-al-2023-open-source-antibiotics-simple-diarylimidazoles-are-potent-against-methicillin-resistant-staphylococcus.pdf
https://discovery.ucl.ac.uk/id/eprint/10182369/ -
7Academic Journal
المؤلفون: Ferrins, Lori, Buskes, Melissa J., Kapteyn, Madison M., Engels, Hannah N., Enos, Suzanne E., Lu, Chenyang, Klug, Dana M., Singh, Baljinder, Quotadamo, Antonio, Bachovchin, Kelly, Tear, Westley F., Spaulding, Andrew E., Forbes, Katherine C., Bag, Seema, Rivers, Mitch, LeBlanc, Catherine, Burchfield, Erin, Armand, Jeremy R., Diaz-Gonzalez, Rosario, Ceballos-Perez, Gloria, García-Hernández, Raquel, Pérez-Moreno, Guiomar, Bosch-Navarrete, Cristina, Gómez-Liñ�n, Claudia, Ruiz-Pérez, Luis Miguel, Gamarro, Francisco, González-Pacanowska, Dolores, Navarro, Miguel, Mensa-Wilmot, Kojo, Pollastri, Michael P., Kyle, Dennis E., Rice, Christopher A.
المصدر: Frontiers in Microbiology ; volume 14 ; ISSN 1664-302X
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8Academic Journal
المؤلفون: Ferrins, Lori, Buskes, Melissa J., Kapteyn, Madison M., Engels, Hannah N., Enos, Suzanne E., Lu, Chenyang, Klug, Dana M., Singh, Baljinder, Quotadamo, Antonio, Bachovchin, Kelly, Tear, Westley F., Spaulding, Andrew E., Forbes, Katherine C., Bag, Seema, Rivers, Mitch, LeBlanc, Catherine, Burchfield, Erin, Armand, Jeremy R., Diaz-Gonzalez, Rosario, Ceballos-Perez, Gloria, García-Hernández, Raquel, Pérez-Moreno, Guiomar, Bosch-Navarrete, Cristina, Gómez-Liñ�n, Claudia, Ruiz-Pérez, Luis Miguel, Gamarro, Francisco, González-Pacanowska, Dolores, Navarro, Miguel, Mensa-Wilmot, Kojo, Pollastri, Michael P., Kyle, Dennis E., Rice, Christopher A.
المساهمون: Georgia Research Alliance, National Institute of Allergy and Infectious Diseases, National Science Foundation
المصدر: Frontiers in Microbiology ; volume 14 ; ISSN 1664-302X
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9Academic Journal
المؤلفون: Klug, Dana M., Tse, Edwin G., Silva, Daniel G., Cao, Yafeng, Charman, Susan A., Chauhan, Jyoti, Crighton, Elly, Dichiara, Maria, Drake, Chris, Drewry, David, da Silva Emery, Flavio, Ferrins, Lori, Graves, Lee, Hopkins, Emily, Kresina, Thomas A. C., Lorente-Macías, Álvaro, Perry, Benjamin, Phipps, Richard, Quiroga, Bruno, Quotadamo, Antonio, Sabatino, Giada N., Sama, Anthony, Schätzlein, Andreas, Simpson, Quillon J., Steele, Jonathan, Shanu-Wilson, Julia, Sjö, Peter, Stapleton, Paul, Swain, Christopher J., Vaideanu, Alexandra, Xie, Huanxu, Zuercher, William, Todd, Matthew H.
المساهمون: Monash University, University of North Carolina at Chapel Hill, National Institute of Allergy and Infectious Diseases, Direktion f?r Entwicklung und Zusammenarbeit, Agence Fran?aise de D?veloppement, M?decins Sans Fronti?res, Foreign, Commonwealth and Development Office, Ministerio de Educaci?n, Cultura y Deporte, Funda??o de Amparo ? Pesquisa do Estado de S?o Paulo, University College London
المصدر: ACS Infectious Diseases ; volume 9, issue 12, page 2423-2435 ; ISSN 2373-8227 2373-8227
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10Academic Journal
المؤلفون: Klug, Dana M., Idiris, Fahima I.M., Blaskovich, Mark A.T., von Delft, Frank, Dowson, Christopher G., Kirchhelle, Claas, Roberts, Adam P., Singer, Andrew C., Todd, Matthew H.
مصطلحات موضوعية: Medicine
وصف الملف: text
Relation: https://nora.nerc.ac.uk/id/eprint/530675/1/N530675JA.pdf; Klug, Dana M.; Idiris, Fahima I.M.; Blaskovich, Mark A.T.; von Delft, Frank; Dowson, Christopher G.; Kirchhelle, Claas; Roberts, Adam P.; Singer, Andrew C. orcid:0000-0003-4705-6063; Todd, Matthew H. 2021 There is no market for new antibiotics: this allows an open approach to research and development. Wellcome Open Research, 6, 146. 14, pp. https://doi.org/10.12688/wellcomeopenres.16847.1
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11Academic Journal
المؤلفون: Klug, Dana M., Díaz-González, Rosario, Pérez-Moreno, Guiomar, Ceballos-Pérez, Gloria, García-Hernández, Raquel, Gómez-Pérez, Veronica, Ruiz-Pérez, Luis Miguel, Rojas-Barros, Domingo I., Gamarro, Francisco, González-Pacanowska, D., Martínez-Martínez, María S., Manzano, Pilar, Ferrins, Lori, Caffrey, Conor R., Navarro, M., Pollastri, M.P.
المساهمون: National Institute of Allergy and Infectious Diseases (US), Ministerio de Economía, Industria y Competitividad (España), Junta de Andalucía, Instituto de Salud Carlos III, Klug, Dana M., Gamarro, Francisco, González-Pacanowska, D., Navarro, M., Pollastri, M.P.
Relation: #PLACEHOLDER_PARENT_METADATA_VALUE#; MINECO/ICT2013-2016/SAF2015-71444-P; MINECO/ICT2013-2016/SAF2016-79957-R; Publisher's version; https://journals.plos.org/plosntds/article?id=10.1371/journal.pntd.0007129; Sí; PLoS Neglected Tropical Diseases; http://hdl.handle.net/10261/178459; http://dx.doi.org/10.13039/501100010198; http://dx.doi.org/10.13039/100000060; http://dx.doi.org/10.13039/501100004587; http://dx.doi.org/10.13039/501100011011; http://dx.doi.org/10.13039/100006492
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12Academic Journal
المؤلفون: Buskes, Melissa J., Clements, Monica, Bachovchin, Kelly A., Jalani, Hitesh B., Leonard, Allison, Bag, Seema, Klug, Dana M., Singh, Baljinder, Campbell, Robert F., Sciotti, Richard J., El-Sakkary, Nelly, Caffrey, Conor R., Pollastri, Michael P., Ferrins, Lori
المساهمون: National Institute of Allergy and Infectious Diseases, Bill and Melinda Gates Foundation, South African Agency for Science and Technology Advancement
المصدر: ACS Medicinal Chemistry Letters ; volume 11, issue 3, page 258-265 ; ISSN 1948-5875 1948-5875
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13Academic Journal
المؤلفون: Ferrins, Lori, Araujo, Erika, Boudreau, Matthew W., Grenier-Davies, Melissa C., Haranahalli, Krupanandan, Journigan, V. Blair, Klug, Dana M., Olson, Margaret E.
المصدر: Journal of Medicinal Chemistry ; volume 65, issue 9, page 6353-6355 ; ISSN 0022-2623 1520-4804
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14Academic Journal
المؤلفون: Klug, Dana M., Mavrogiannaki, Eftychia M., Forbes, Katherine C., Silva, Lisseth, Díaz-González, Rosario, Pérez-Moreno, Guiomar, Ceballos-Pérez, Gloria, García-Hernández, Raquel, Bosch-Navarrete, Cristina, Cordon-Obras, Carlos, Gómez-Liñán, Claudia, Saura, Andreu, Momper, Jeremiah D., Martínez-Martínez, María S., Manzano, Miguel, Syed, Ali Asgher, El-Sakkary, Nelly, Caffrey, Conor R., Gamarro, Francisco, Ruiz-Pérez, Luis Miguel, González Pacanowska, Dolores, Ferrins, L, Navarro, Miquel, Pollastri, M.P.
المساهمون: Instituto Nacional de Alergias y Enfermedades Infecciosas, Ministerio de Economía, Industria y Competitividad (España), National Science Foundation for K.F., Subdireccion General de Redes ́ y Centros de Investigacion Cooperativa (RICET
Relation: Publisher's version; http://dx.doi.org/10.1021/acs.jmedchem.1c00674; Sí; Journal of Medicinal Chemistry 64: 9404- 9430 (2021); http://hdl.handle.net/10261/359703
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15Electronic Resource
المؤلفون: National Institute of Allergy and Infectious Diseases (US), Ministerio de Economía, Industria y Competitividad (España), Junta de Andalucía, Instituto de Salud Carlos III, Klug, Dana M. [0000-0002-8982-0640], Gamarro, Francisco [0000-0003-1347-3440], González-Pacanowska, D. [0000-0002-4303-5209], Navarro, M. [0000-0003-2301-2699], Pollastri, M.P. [0000-0001-9943-7197], Klug, Dana M., Díaz-González, Rosario, Pérez-Moreno, Guiomar, Ceballos-Pérez, Gloria, García-Hernández, Raquel, Gómez-Pérez, Veronica, Ruiz-Pérez, Luis Miguel, Rojas-Barros, Domingo I., Gamarro, Francisco, González-Pacanowska, Dolores, Martínez-Martínez, María S., Manzano, Pilar, Ferrins, Lori, Caffrey, Conor R., Navarro, M., Pollastri, M.P.
مصطلحات الفهرس: artículo
URL:
http://hdl.handle.net/10261/178459 https://journals.plos.org/plosntds/article?id=10.1371/journal.pntd.0007129
Publisher's versionhttps://journals.plos.org/plosntds/article?id=10.1371/journal.pntd.0007129
Sí
MINECO/ICT2013-2016/SAF2015-71444-P
MINECO/ICT2013-2016/SAF2016-79957-R -
16Electronic Resource
المؤلفون: Instituto Nacional de Alergias y Enfermedades Infecciosas, Ministerio de Economía, Industria y Competitividad (España), National Science Foundation for K.F., Subdireccion General de Redes ́ y Centros de Investigacion Cooperativa (RICET, Klug, Dana M., Mavrogiannaki, Eftychia M., Forbes, Katherine C., Silva, Lisseth, Díaz-González, Rosario, Pérez-Moreno, Guiomar, Ceballos-Pérez, Gloria, García-Hernández, Raquel, Bosch-Navarrete, Cristina, Cordon-Obras, Carlos, Gómez-Liñán, Claudia, Saura, Andreu, Momper, Jeremiah D., Martínez-Martínez, María S., Manzano, Miguel, Syed, Ali Asgher, El-Sakkary, Nelly, Caffrey, Conor R., Gamarro, Francisco, Ruiz-Pérez, Luis Miguel, González Pacanowska, Dolores, Ferrins, L, Navarro, Miquel, Pollastri, M.P.
مصطلحات الفهرس: artículo
URL:
http://hdl.handle.net/10261/359703
Publisher's versionhttp://dx.doi.org/10.1021/acs.jmedchem.1c00674
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17Academic Journal
المؤلفون: Klug, Dana M., Díaz-González, Rosario, DeLano, Travis J., Mavrogiannaki, Eftychia M., Buske, Melissa J., Dalton, Raeann M., Fisher, John K., Schneider, Katherine M., Hilborne, Vivian, Fritsche, Melanie G., Simpson, Quillon J., Tear, Westley F., Devine, William G., Pérez-Moreno, Guiomar, Ceballos-Pérez, Gloria, García-Hernández, Raquel, Bosch-Navarrete, Cristina, Ruiz-Pérez, Luis Miguel, Gamarro, Francisco, González-Pacanowska, D., Martínez-Martínez, María S., Manzano-Chinchón, Pilar, Navarro, M., Pollastri, M.P., Ferrins, L
Relation: http://dx.doi.org/10.1039/d0md00103a; Sí; RSC Medicinal Chemistry 11: 950- 959 (2020); http://hdl.handle.net/10261/246477
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18Academic Journal
المؤلفون: Singh, Baljinder, Bernatchez, Jean A., McCall, Laura-Isobel, Calvet, Claudia M., Ackermann, Jasmin, Souza, Julia M., Thomas, Diane, Silva, Everton M., Bachovchin, Kelly A., Klug, Dana M., Jalani, Hitesh B., Bag, Seema, Buskes, Melissa J., Leed, Susan E., Roncal, Norma E., Penn, Erica C., Erath, Jessey, Rodriguez, Ana, Sciotti, Richard J., Campbell, Robert F., McKerrow, James, Siqueira-Neto, Jair L., Ferrins, Lori, Pollastri, Michael P.
المساهمون: National Institute of Allergy and Infectious Diseases
المصدر: ACS Medicinal Chemistry Letters ; volume 11, issue 3, page 249-257 ; ISSN 1948-5875 1948-5875
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19Academic Journal
المؤلفون: Klug, Dana M., Tschiegg, Laura, Diaz, Rosario, Rojas-Barros, Domingo, Perez-Moreno, Guiomar, Ceballos, Gloria, García-Hernández, Raquel, Martinez-Martinez, Maria Santos, Manzano, Pilar, Ruiz, Luis Miguel, Caffrey, Conor R., Gamarro, Francisco, Pacanowska, Dolores Gonzalez, Ferrins, Lori, Navarro, Miguel, Pollastri, Michael P.
المساهمون: Ministerio de Econom?a y Competitividad, National Institute of Allergy and Infectious Diseases, American Chemical Society, Instituto de Salud Carlos III
المصدر: Journal of Medicinal Chemistry ; volume 63, issue 5, page 2527-2546 ; ISSN 0022-2623 1520-4804
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20Academic Journal
المؤلفون: Bachovchin, Kelly A., Sharma, Amrita, Bag, Seema, Klug, Dana M., Schneider, Katherine M., Singh, Baljinder, Jalani, Hitesh B., Buskes, Melissa J., Mehta, Naimee, Tanghe, Scott, Momper, Jeremiah D., Sciotti, Richard J., Rodriguez, Ana, Mensa-Wilmot, Kojo, Pollastri, Michael P., Ferrins, Lori
المساهمون: National Institute of Allergy and Infectious Diseases
المصدر: Journal of Medicinal Chemistry ; volume 62, issue 2, page 665-687 ; ISSN 0022-2623 1520-4804