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1
المؤلفون: Zenichi Ikeda, Keiko Kakegawa, Fumiaki Kikuchi, Sachiko Itono, Hideyuki Oki, Hiroaki Yashiro, Hideyuki Hiyoshi, Kazue Tsuchimori, Kenichi Hamagami, Masanori Watanabe, Masako Sasaki, Youko Ishihara, Kimio Tohyama, Tomoyuki Kitazaki, Tsuyoshi Maekawa, Minoru Sasaki
المصدر: Journal of medicinal chemistry. 65(12)
مصطلحات موضوعية: Enteropeptidase, Mice, Drug Discovery, Molecular Medicine, Animals, Mice, Obese, Obesity, Benzoates, Guanidines, Rats
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2
المؤلفون: Tsuyoshi Maekawa, Minoru Sasaki, Kazue Tsuchimori, Yusuke Moritoh, Hideyuki Hiyoshi, Hiroaki Yashiro, Kenichi Hamagami, Fuminari Yamaguchi, Yukio Yamada, Masanori Watanabe, Jun Sugama
المصدر: Diabetes, Obesity & Metabolism
مصطلحات موضوعية: Blood Glucose, Male, Enteropeptidase, FGF21, Endocrinology, Diabetes and Metabolism, Mice, Obese, 030204 cardiovascular system & hematology, Mice, chemistry.chemical_compound, 0302 clinical medicine, Endocrinology, Insulin, animal pharmacology, diabetes, biology, Trypsin, Protein catabolism, Original Article, medicine.drug, medicine.medical_specialty, Serine Proteinase Inhibitors, Trypsinogen, mouse model, 030209 endocrinology & metabolism, Diabetes Mellitus, Experimental, Small Molecule Libraries, 03 medical and health sciences, In vivo, Internal medicine, Diabetes mellitus, Internal Medicine, medicine, Animals, Obesity, Benzofurans, Aspartic Acid, business.industry, Body Weight, Original Articles, medicine.disease, drug development, Mice, Inbred C57BL, Disease Models, Animal, chemistry, Alanine transaminase, obesity therapy, biology.protein, business
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3
المؤلفون: Shoki Okuda, Yasuyoshi Arikawa, Tomohiro Okawa, Junichi Sakamoto, Nobuyuki Amano, Shinobu Sasaki, Masanori Nakakariya, Yugo Habata, Shizuo Kasai, Natsu Hotta, Kenichi Hamagami, Masaaki Funata, Yasutaka Nagisa, Minoru Maruyama, Toshimi Nagi, Yasunori Nio
المصدر: Endocrinology. 158:1298-1313
مصطلحات موضوعية: Male, 0301 basic medicine, Agonist, Hypothalamo-Hypophyseal System, endocrine system, Sympathetic nervous system, medicine.medical_specialty, medicine.drug_class, Pituitary-Adrenal System, Diet, High-Fat, Rats, Sprague-Dawley, 03 medical and health sciences, 0302 clinical medicine, Endocrinology, Internal medicine, Weight Loss, medicine, Animals, Obesity, Circadian rhythm, business.industry, Suprachiasmatic nucleus, Body Weight, Lipid Metabolism, Rats, Inbred F344, Circadian Rhythm, Rats, Receptors, Bombesin, 030104 developmental biology, medicine.anatomical_structure, Hypothalamus, Anorectic, Bombesin Receptor Subtype-3, Anti-Obesity Agents, Corticosterone, Energy Metabolism, business, Diet-induced obese, hormones, hormone substitutes, and hormone antagonists, 030217 neurology & neurosurgery
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4
المؤلفون: Kazue Tsuchimori, Masanori Watanabe, Tomohiro Kawamoto, Ikuo Miyahisa, Minoru Sasaki, Hideyuki Hiyoshi, Hiroaki Yashiro, Masako Sasaki, Junichi Sakamoto, Yusuke Moritoh, Kenichi Hamagami, Kimio Tohyama, Sachiko Itono
المصدر: Pharmacology Research & Perspectives
Pharmacology Research & Perspectives, Vol 7, Iss 5, Pp n/a-n/a (2019)مصطلحات موضوعية: Enteropeptidase, Brush border, Trypsinogen, Protein digestion, Drug Evaluation, Preclinical, Administration, Oral, RM1-950, 030226 pharmacology & pharmacy, Small Molecule Libraries, Inhibitory Concentration 50, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, In vivo, Fluorescence Resonance Energy Transfer, medicine, Animals, Humans, Enzyme Inhibitors, General Pharmacology, Toxicology and Pharmaceutics, chemistry.chemical_classification, covalent, enteropeptidase, Original Articles, Trypsin, In vitro, SCO‐792, Rats, Enzyme, Neurology, chemistry, Biochemistry, 030220 oncology & carcinogenesis, FRET, Original Article, Therapeutics. Pharmacology, medicine.drug
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5
المؤلفون: Mayumi Nishida, Natsu Hotta, Kenichi Hamagami, Masaaki Mori, Nobuyuki Amano, Masaaki Funata, Tomohiro Okawa, Shinobu Sasaki, Yasunori Nio, Junichi Sakamoto, Yasutaka Nagisa, Masanori Nakakariya, Yasuyoshi Arikawa, Minoru Maruyama, Toshimi Nagi, Shizuo Kasai, Yugo Habata
المصدر: Brain and Behavior
مصطلحات موضوعية: 0301 basic medicine, Agonist, Male, medicine.medical_specialty, obesity, medicine.drug_class, Hypothalamus, Nerve Tissue Proteins, CHO Cells, Biology, Energy homeostasis, Rats, Sprague-Dawley, 03 medical and health sciences, Behavioral Neuroscience, bombesin receptor subtype‐3, Eating, Cricetulus, Internal medicine, medicine, Animals, Homeostasis, Receptors, Somatostatin, Dorsomedial hypothalamic nucleus, energy homeostasis, Original Research, Mice, Knockout, Neurons, fungi, Feeding Behavior, Thermoregulation, Bombesin receptor, Rats, Receptors, Bombesin, 030104 developmental biology, Endocrinology, nervous system, neuronal pathway, Bombesin Receptor Subtype-3, Energy Metabolism, Immunostaining