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1
المؤلفون: Sean P. Henry, Maria-Elena Liosi, Joseph A. Ippolito, Kara J. Cutrona, Stefan G. Krimmer, Ana S. Newton, Joseph Schlessinger, William L. Jorgensen
المصدر: ACS Med Chem Lett
مصطلحات موضوعية: Organic Chemistry, Drug Discovery, Biochemistry
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2
المؤلفون: Maria-Elena Liosi, Joseph A. Ippolito, Sean P. Henry, Stefan G. Krimmer, Ana S. Newton, Kara J. Cutrona, Rene A. Olivarez, Jyotidarsini Mohanty, Joseph Schlessinger, William L. Jorgensen
المصدر: J Med Chem
مصطلحات موضوعية: STAT Transcription Factors, Myeloproliferative Disorders, Drug Discovery, Mutation, Molecular Medicine, Humans, Janus Kinase 2, Ligands, Article, Janus Kinases, Signal Transduction
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3
المؤلفون: Shengyan Jin, José A. Cisneros, Karen S. Anderson, Krasimir A. Spasov, Kara J. Cutrona, M. Valhondo, Haichan Niu, Nicole Bertoletti, Zachary J Carter, William L. Jorgensen, Joseph A. Ippolito
المصدر: ACS Med Chem Lett
مصطلحات موضوعية: chemistry.chemical_classification, Catechol, 010405 organic chemistry, Stereochemistry, Organic Chemistry, Wild type, Crystal structure, 01 natural sciences, Biochemistry, In vitro, Reverse transcriptase, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, chemistry.chemical_compound, Enzyme, chemistry, Covalent bond, Drug Discovery, Mass spectrum
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4
المؤلفون: Elizabeth A Stone, Kara J. Cutrona, Scott J. Miller
المصدر: J Am Chem Soc
مصطلحات موضوعية: Stereochemistry, Histamine Antagonists, Molecular Conformation, Peptide, Loratadine, 010402 general chemistry, 01 natural sciences, Biochemistry, Article, Catalysis, Colloid and Surface Chemistry, Aspartic acid, medicine, Humans, chemistry.chemical_classification, Aspartic Acid, Desloratadine, Enantioselective synthesis, Stereoisomerism, General Chemistry, 0104 chemical sciences, Molecular Docking Simulation, chemistry, Docking (molecular), Receptors, Histamine, Enantiomer, Peptides, medicine.drug
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5
المصدر: J Chem Inf Model
مصطلحات موضوعية: Virtual screening, Binding Sites, Computer science, Extramural, General Chemical Engineering, Scoring methods, Metadynamics, General Chemistry, Computational biology, Library and Information Sciences, Ligand (biochemistry), Ligands, Article, Computer Science Applications, Docking (molecular), Research Design, False positive paradox, Potential of mean force, Protein Binding
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6
المؤلفون: Thomas K. Dawson, S.G. Krimmer, Maria-Elena Liosi, Kara J. Cutrona, Ana S. Newton, David E. Puleo, Joseph Schlessinger, Yoshihisa Suzuki, William L. Jorgensen
المصدر: J Med Chem
مصطلحات موضوعية: Enzyme Activators, Ligands, 01 natural sciences, Article, 03 medical and health sciences, Myeloproliferative Disorders, X-Ray Diffraction, hemic and lymphatic diseases, Drug Discovery, Sf9 Cells, Animals, Humans, Binding site, 030304 developmental biology, Amitrole, 0303 health sciences, Janus kinase 2, biology, Chemistry, Autophosphorylation, biochemical phenomena, metabolism, and nutrition, Janus Kinase 2, 0104 chemical sciences, Cell biology, 010404 medicinal & biomolecular chemistry, HEK293 Cells, Protein kinase domain, biology.protein, Molecular Medicine, Signal transduction, Janus kinase, Tyrosine kinase, Protein Binding
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7
المؤلفون: José A. Cisneros, Joseph Schlessinger, Kara J. Cutrona, Luca Deiana, William L. Jorgensen, David E. Puleo, Ana S. Newton
المصدر: ACS Medicinal Chemistry Letters. 8:614-617
مصطلحات موضوعية: 0301 basic medicine, Filgotinib, Chemistry, Stereochemistry, Organic Chemistry, Allosteric regulation, Crystal structure, biochemical phenomena, metabolism, and nutrition, Biochemistry, Small molecule, Fluorescence, 03 medical and health sciences, Crystallography, chemistry.chemical_compound, 030104 developmental biology, Diaminopyrimidine, Drug Discovery, Molecule, Fluorescence anisotropy
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8Role of arginine and lysine in the antimicrobial mechanism of histone-derived antimicrobial peptides
المصدر: FEBS Letters. 589:3915-3920
مصطلحات موضوعية: Arginine, Molecular Sequence Data, Lysine, Antimicrobial peptides, Biophysics, Biology, Biochemistry, Article, Microbiology, Histones, Structure-Activity Relationship, Structural Biology, Genetics, Structure–activity relationship, Amino Acid Sequence, Molecular Biology, Peptide sequence, Cell Membrane, Cell Biology, Antimicrobial, Protein Transport, Mutation, Cell-penetrating peptide, Antibacterial activity, Antimicrobial Cationic Peptides
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b1a07dc7809c84157b41d485e93954a1
https://doi.org/10.1016/j .febslet.2015.11.002 -
9
المؤلفون: Sukin Sim, Mala L. Radhakrishnan, Penny Wang, Kara J. Cutrona, Brittany Beyer, Donald E. Elmore
المصدر: FEBS letters. 591(5)
مصطلحات موضوعية: 0301 basic medicine, DNA, Bacterial, Antimicrobial peptides, Biophysics, Plasma protein binding, Molecular Dynamics Simulation, 010402 general chemistry, Arginine, 01 natural sciences, Biochemistry, Protein Structure, Secondary, Article, Histones, 03 medical and health sciences, chemistry.chemical_compound, Structure-Activity Relationship, Structural Biology, Genetics, Animals, Amino Acid Sequence, Molecular Biology, Peptide sequence, Binding selectivity, biology, Lysine, Molecular Mimicry, Proteins, Cell Biology, biology.organism_classification, 0104 chemical sciences, Anti-Bacterial Agents, Kinetics, 030104 developmental biology, Histone, chemistry, Amino Acid Substitution, Nucleic acid, biology.protein, Thermodynamics, Anura, Bacteria, DNA, Protein Binding
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10
المصدر: Journal of chemical theory and computation. 11(9)
مصطلحات موضوعية: Models, Molecular, Aqueous medium, Chemistry, Thermodynamics, Force field (chemistry), Article, Computer Science Applications, Vaporization, Physical chemistry, Molecule, Quantum Theory, Free energies, Atomic charge, Organic liquids, Physical and Theoretical Chemistry, Quantum
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11
المؤلفون: Penny Wang, Brittany Beyer, Sukin Sim, Mala L. Radhakrishnan, Donald E. Elmore, Kara J. Cutrona
المصدر: Biophysical Journal. 110(3):560a-561a
مصطلحات موضوعية: chemistry.chemical_classification, 0303 health sciences, biology, Antimicrobial peptides, Lysine, Biophysics, Peptide, biology.organism_classification, Bacterial cell structure, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Histone, Biochemistry, chemistry, biology.protein, Nucleic acid, 030217 neurology & neurosurgery, DNA, Bacteria, 030304 developmental biology
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12
المؤلفون: Donald E. Elmore, Kara J. Cutrona
المصدر: The FASEB Journal. 27
مصطلحات موضوعية: Histone, Arginine, biology, Biochemistry, Chemistry, Mechanism (biology), Lysine, Genetics, biology.protein, Antimicrobial, Molecular Biology, Biotechnology