نتائج البحث - "Kalinin, Stanislav"

Relation: This research was supported by the Ministry of Education of the Russian Federation [government contract 073-00077-21-02 `Development of an innovative glaucoma drug based on selective inhibition of carbonic anhydrase II', registry number 730000 Phi.99.1.(sic)B10AA00006] and by Megagrant of the Government of Russian Federation [075-15-2021-637] and Academy of Finland.; Kalinin , S , Kovalenko , A , Valtari , A , Nocentini , A , Gureev , M , Urtti , A , Korsakov , M , Supuran , C T & Krasavin , M 2022 , ' 5-(Sulfamoyl)thien-2-yl 1,3-oxazole inhibitors of carbonic anhydrase II with hydrophilic periphery ' , Journal of Enzyme Inhibition and Medicinal Chemistry , vol. 37 , no. 1 , pp. 1005-1011 . https://doi.org/10.1080/14756366.2022.2056733; http://hdl.handle.net/10138/343075; 7178c164-23dd-4799-bd59-de4bbf85273e; 000776808200001

الاتاحة: http://hdl.handle.net/10138/343075

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7

Academic Journal

Diversely substituted sulfamides for fragment-based drug discovery of carbonic anhydrase inhibitors: synthesis and inhibitory profile

المؤلفون: Sharonova, Tatiana, Zhmurov, Petr, Kalinin, Stanislav, Nocentini, Alessio, Angeli, Andrea, Ferraroni, Marta, Korsakov, Mikhail, Supuran, Claudiu T., Krasavin, Mikhail

المساهمون: Ministry of Education of the Russian Federation

المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry ; volume 37, issue 1, page 857-865 ; ISSN 1475-6366 1475-6374

الاتاحة: http://dx.doi.org/10.1080/14756366.2022.2051023
https://www.tandfonline.com/doi/pdf/10.1080/14756366.2022.2051023

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8

Academic Journal

Novel melanin‐binding carbonic anhydrase II inhibitor for long‐acting topical glaucoma treatment

المؤلفون: Valtari, Annika, Kalinin, Stanislav, Jäntti, Janika, Stenberg, Katja, Vellonen, Kati‐Sisko, Toropainen, Elisa, Ruponen, Marika, Urtti, Arto

المصدر: Acta Ophthalmologica ; volume 102, issue S279 ; ISSN 1755-375X 1755-3768

الاتاحة: http://dx.doi.org/10.1111/aos.15829

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9

Academic Journal

Discovery and characterization of potent spiro-isoxazole-based cereblon ligands with a novel binding mode

المؤلفون: Shevalev, Robert, Bischof, Luca, Sapegin, Alexander, Bunev, Alexander, Olga, Grigor'eva, Kantin, Grigory, Kalinin, Stanislav, Hartmann, Marcus D.

المساهمون: Max-Planck-Gesellschaft, Russian Science Foundation

المصدر: European Journal of Medicinal Chemistry ; volume 270, page 116328 ; ISSN 0223-5234

الاتاحة: http://dx.doi.org/10.1016/j.ejmech.2024.116328
https://api.elsevier.com/content/article/PII:S0223523424002083?httpAccept=text/xml
https://api.elsevier.com/content/article/PII:S0223523424002083?httpAccept=text/plain

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10

Academic Journal

Direct assembly of N-sulfamoyl lactam scaffolds bearing a zinc-binding group for inhibiting metalloenzymes based on desymmetrization of sulfamide and the Castagnoli-Cushman reaction

المؤلفون: Karchuganova, Elizaveta, Martynova, Sofiia, Kalinin, Stanislav, Angeli, Andrea, Dar'in, Dmitry, Vullo, Daniella, Supuran, Claudiu T., Bakulina, Olga

المساهمون: Russian Science Foundation, Saint Petersburg State University

المصدر: Tetrahedron ; volume 154, page 133890 ; ISSN 0040-4020

الاتاحة: http://dx.doi.org/10.1016/j.tet.2024.133890
https://api.elsevier.com/content/article/PII:S004040202400070X?httpAccept=text/xml
https://api.elsevier.com/content/article/PII:S004040202400070X?httpAccept=text/plain

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11

Academic Journal

Biochemical profiling of anti-HIV prodrug Elsulfavirine (Elpida ® ) and its active form VM1500A against a panel of twelve human carbonic anhydrase isoforms

المؤلفون: Supuran, Claudiu T., Nocentini, Alessio, Yakubova, Elena, Savchuk, Nikolay, Kalinin, Stanislav, Krasavin, Mikhail

المساهمون: Russian Federation Government Megagrant, Italian Ministry for Research and University, PRIN prot.

المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry ; volume 36, issue 1, page 1056-1060 ; ISSN 1475-6366 1475-6374

الاتاحة: http://dx.doi.org/10.1080/14756366.2021.1927007
https://www.tandfonline.com/doi/pdf/10.1080/14756366.2021.1927007

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12

Academic Journal

Corrigendum to “Investigation of 3-sulfamoyl coumarins against cancer-related IX and XII isoforms of human carbonic anhydrase as well as cancer cells leads to the discovery of 2-oxo-2H-benzo[h]chromene-3-sulfonamide – A new caspase-activating proapoptotic agent” [J. Med. Chem. 222 (2021) 113589]

المؤلفون: Dar'in, Dmitry, Kantin, Grigory, Kalinin, Stanislav, Sharonova, Tatiana, Bunev, Alexander, Ostapenko, Gennady I., Nocentini, Alessio, Sharoyko, Vladimir, Supuran, Claudiu T., Krasavin, Mikhail

المساهمون: Russian Foundation for Basic Research, Russian Science Foundation

المصدر: European Journal of Medicinal Chemistry ; volume 225, page 113788 ; ISSN 0223-5234

الاتاحة: https://doi.org/10.1016/j.ejmech.2021.113788
https://api.elsevier.com/content/article/PII:S0223523421006371?httpAccept=text/xml
https://api.elsevier.com/content/article/PII:S0223523421006371?httpAccept=text/plain

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13

Academic Journal

Unraveling multi-state molecular dynamics in single-molecule FRET experiments. II. Quantitative analysis of multi-state kinetic networks.

المؤلفون: Opanasyuk, Oleg, Barth, Anders, Peulen, Thomas-Otavio, Felekyan, Suren, Kalinin, Stanislav, Sanabria, Hugo, Seidel, Claus A. M.

المصدر: Journal of Chemical Physics; 7/21/2022, Vol. 157 Issue 3, p1-24, 24p

مصطلحات موضوعية: FLUORESCENCE resonance energy transfer, QUANTITATIVE research, MOLECULAR dynamics, BREMSSTRAHLUNG, STRUCTURAL dynamics, FLUORESCENCE spectroscopy

14

Academic Journal

Unraveling multi-state molecular dynamics in single-molecule FRET experiments. I. Theory of FRET-lines.

المؤلفون: Barth, Anders, Opanasyuk, Oleg, Peulen, Thomas-Otavio, Felekyan, Suren, Kalinin, Stanislav, Sanabria, Hugo, Seidel, Claus A. M.

المصدر: Journal of Chemical Physics; 4/14/2022, Vol. 156 Issue 14, p1-29, 29p

مصطلحات موضوعية: MOLECULAR dynamics, FLUORESCENCE resonance energy transfer, BIOMOLECULES

15

Academic Journal

New Biocides Based on N 4 -Alkylcytidines: Effects on Microorganisms and Application for the Protection of Cultural Heritage Objects of Painting.

المؤلفون: Alexandrova, Liudmila A., Oskolsky, Ivan A., Makarov, Dmitry A., Jasko, Maxim V., Karpenko, Inna L., Efremenkova, Olga V., Vasilyeva, Byazilya F., Avdanina, Darya A., Ermolyuk, Anna A., Benko, Elizaveta E., Kalinin, Stanislav G., Kolganova, Tat'yana V., Berzina, Maria Ya., Konstantinova, Irina D., Chizhov, Alexander O., Kochetkov, Sergey N., Zhgun, Alexander A.

المصدر: International Journal of Molecular Sciences; Mar2024, Vol. 25 Issue 5, p3053, 20p

مصطلحات موضوعية: CULTURAL property, BIOCIDES, NUCLEOSIDE derivatives, DRUG resistance in microorganisms, PROTECTION of cultural property, BENZALKONIUM chloride, MYCOBACTERIUM smegmatis, MOLDS (Fungi), GRAM-positive bacteria

مصطلحات جغرافية: MOSCOW (Russia), RUSSIA

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16

Academic Journal

Continued exploration of 1,2,4-oxadiazole periphery for carbonic anhydrase-targeting primary arene sulfonamides: Discovery of subnanomolar inhibitors of membrane-bound hCA IX isoform that selectively kill cancer cells in hypoxic environment

المؤلفون: Krasavin, Mikhail, Shetnev, Anton, Sharonova, Tatyana, Baykov, Sergey, Kalinin, Stanislav, Nocentini, Alessio, Sharoyko, Vladimir, Poli, Giulio, Tuccinardi, Tiziano, Presnukhina, Sofia, Tennikova, Tatiana B., Supuran, Claudiu T.

المساهمون: Krasavin, Mikhail, Shetnev, Anton, Sharonova, Tatyana, Baykov, Sergey, Kalinin, Stanislav, Nocentini, Alessio, Sharoyko, Vladimir, Poli, Giulio, Tuccinardi, Tiziano, Presnukhina, Sofia, Tennikova, Tatiana B., Supuran, Claudiu T.

مصطلحات موضوعية: 1,2,4-Oxadiazole, Cancer cell, Carbonic anhydrase, Hypoxic environment, Isoform-selective inhibitor, Isosteric replacement, Periphery group, Primary sulfonamide, Subnanomolar inhibition, Pharmacology

وصف الملف: ELETTRONICO

Relation: info:eu-repo/semantics/altIdentifier/pmid/30594030; info:eu-repo/semantics/altIdentifier/wos/WOS:000458221400007; volume:164; firstpage:92; lastpage:105; numberofpages:14; journal:EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY; http://hdl.handle.net/11568/963886; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85058993622; https://www.sciencedirect.com/science/article/pii/S0223523418310870

الاتاحة: http://hdl.handle.net/11568/963886
https://doi.org/10.1016/j.ejmech.2018.12.049
https://www.sciencedirect.com/science/article/pii/S0223523418310870

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