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1Academic Journal
المؤلفون: Magda Horejsi, Juraj Sedlacek, Graham A. Bentley
المساهمون: The Pennsylvania State University CiteSeerX Archives
مصطلحات موضوعية: cross-reactivity, crystal structure, drug design
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.570.7706; http://www.pasteur.fr/recherche/unites/ImmStr/publis-pdf/1999_ProtSci_8_2686.pdf
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2
المؤلفون: Tomáš Etrych, Michal Pechar, Juraj Sedlacek, Milan Fábry, Irena Sieglová, Leonid I. Kaberov, Sergey K. Filippov, Vlastimil Král, Robert Pola
المصدر: Biomacromolecules. 20(1)
مصطلحات موضوعية: Polymers and Plastics, medicine.drug_class, Bioengineering, Peptide, Antineoplastic Agents, 02 engineering and technology, Nanoconjugates, 010402 general chemistry, Monoclonal antibody, 01 natural sciences, law.invention, Biomaterials, chemistry.chemical_compound, Mice, Antigen, Polymethacrylic Acids, law, Cell Line, Tumor, Gangliosides, Materials Chemistry, medicine, Methacrylamide, Animals, Cytotoxicity, Cell Proliferation, chemistry.chemical_classification, Chemistry, 3T3 Cells, 021001 nanoscience & nanotechnology, Bungarotoxins, 0104 chemical sciences, Biochemistry, Covalent bond, Doxorubicin, Recombinant DNA, 0210 nano-technology, Conjugate, Protein Binding, Single-Chain Antibodies
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3
المؤلفون: Juraj Sedlacek, Vaclav Veverka, Pavlína Řezáčová, Milan Fábry, Jana Škerlová, Vlastimil Král
المصدر: Acta Crystallographica Section F Structural Biology Communications. 70:1701-1706
مصطلحات موضوعية: biology, Chemistry, Laboratory Communications, Molecular Sequence Data, Biophysics, Single chain, Condensed Matter Physics, Biochemistry, Molecular biology, Antibody fragments, Structural Biology, Chromatography, Gel, Genetics, biology.protein, Humans, Amino Acid Sequence, Antibody, Crystallization, Single-Chain Antibodies
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4
المؤلفون: Leo Kronrád, Pavlína Řezáčová, Juraj Sedlacek, Vlastimil Král, Milan Fábry, Bronislava Uhnáková, Irena Sieglová, Agnieszka Sawicka, Renata Mikolajczak, Marcela Múdra
المصدر: Journal of Labelled Compounds and Radiopharmaceuticals. 55:52-56
مصطلحات موضوعية: biology, Chemistry, Fragment (computer graphics), Organic Chemistry, Biochemistry, Fusion protein, Analytical Chemistry, law.invention, law, Drug Discovery, Recombinant DNA, biology.protein, Single-chain variable fragment, Radiology, Nuclear Medicine and imaging, Antibody, Spectroscopy
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5
المؤلفون: Jan Konvalinka, Jana Pokorná, Bohumír Grüner, Jaromír Plešek, Pavlina Rezacova, Heike Oberwinkler, Klára Grantz Šašková, Václav Šícha, Petr Cigler, Vladimír Král, Pavel Hobza, Hans-Georg Kräusslich, Martin Lepšík, Jindrich Fanfrlík, Juraj Sedlacek, Irena Sieglová, Milan Kozisek, Jan Rezac, Jiri Brynda
المصدر: Journal of Medicinal Chemistry. 52:7132-7141
مصطلحات موضوعية: Boron Compounds, Models, Molecular, Molecular model, Stereochemistry, medicine.medical_treatment, Molecular Conformation, Electrons, Crystal structure, Crystallography, X-Ray, HIV Protease, Drug Discovery, medicine, HIV Protease Inhibitor, Protease inhibitor (pharmacology), chemistry.chemical_classification, Protease, biology, Chemistry, Cobalt, HIV Protease Inhibitors, Carbon, Enzyme, Enzyme inhibitor, Drug Design, HIV-1, biology.protein, Molecular Medicine, Linker
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6
المؤلفون: Jarmila Dušková, Milan Fábry, Eva Vondráčková, Tereza Skálová, Jan Dohnálek, Jiří Brynda, Jan Konvalinka, Juraj Sedlacek, Milan Souček, Hana Petroková, Jindřich Hašek, Martin Hradilek
المصدر: Acta Crystallographica Section D Biological Crystallography. 62:489-497
مصطلحات موضوعية: Models, Molecular, Isostere, Stereochemistry, Peptidomimetic, medicine.medical_treatment, Protein Data Bank (RCSB PDB), Stereoisomerism, Crystallography, X-Ray, HIV Protease, HIV-1 protease, Structural Biology, medicine, Peptide bond, HIV Protease Inhibitor, Binding Sites, Protease, biology, Chemistry, Hydrogen Bonding, HIV Protease Inhibitors, General Medicine, Ethanolamines, HIV-1, biology.protein, Oligopeptides, Protein Binding
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7
المؤلفون: Juraj Sedlacek, Jaromír Plešek, Vladimír Král, Jan Konvalinka, Jiří Brynda, Jochen Bodem, Martin Máša, Hans-Georg Kräusslich, Jana Pokorná, Zbyszek Otwinowski, Pavlína Řezáčová, Bohumír Grüner, Lucie Dolečková-Marešová, Petr Cigler, Milan Kožíšek
المصدر: Proceedings of the National Academy of Sciences. 102:15394-15399
مصطلحات موضوعية: Multidisciplinary, Protease, Chemistry, Stereochemistry, medicine.medical_treatment, Cathepsin D, Drug design, HIV Protease Inhibitors, Biological Sciences, Crystallography, X-Ray, Structure-Activity Relationship, Papain, chemistry.chemical_compound, Non-competitive inhibition, HIV Protease, Drug Design, medicine, Aspartic Acid Endopeptidases, HIV Protease Inhibitor, Structure–activity relationship, Pharmacophore, Boranes
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8
المؤلفون: Martin Hradilek, Jan Konvalinka, Jiri Brynda, Milan Fábry, M. Horejsi, R. Stouracova, Milan Souček, Juraj Sedlacek, Pavlina Rezacova
المصدر: Acta Crystallographica Section D Biological Crystallography. 60:1943-1948
مصطلحات موضوعية: Models, Molecular, Binding Sites, biology, Protein Conformation, Ligand, Stereochemistry, Chemistry, Active site, HIV Protease Inhibitors, General Medicine, Crystallography, X-Ray, Ligands, Sensitivity and Specificity, Crystallography, Protein structure, HIV Protease, HIV-1 protease, Structural Biology, biology.protein, Molecule, HIV Protease Inhibitor, Orthorhombic crystal system, Binding site
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9
المؤلفون: Martin Hradilek, Juraj Sedlacek, Jiri Brynda, Pavlina Rezacova, Milan Souček, Martin Lepšík, R. Stouracova, M. Horejsi, Milan Fábry, Jan Konvalinka
المصدر: Journal of Medicinal Chemistry. 47:2030-2036
مصطلحات موضوعية: Models, Molecular, Molecular model, Stereochemistry, medicine.medical_treatment, Protonation, Crystallography, X-Ray, Phenylbutyrate, HIV Protease, HIV-1 protease, Drug Resistance, Viral, Drug Discovery, medicine, HIV Protease Inhibitor, Moiety, Binding Sites, Protease, biology, Chemistry, Hydrogen bond, Stereoisomerism, HIV Protease Inhibitors, Phenylbutyrates, Crystallography, Mutation, biology.protein, Thermodynamics, Molecular Medicine, Protein Binding
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10
المؤلفون: Jindrich Hasek, Jan Dohnálek, Milan Fábry, Jiri Brynda, Jarmila Dušková, Juraj Sedlacek, Martin Hradilek, Hana Petroková, Jan Konvalinka, Milan Souček
المصدر: Journal of Medicinal Chemistry. 45:1432-1438
مصطلحات موضوعية: Glycerol, Models, Molecular, Protein Conformation, Stereochemistry, Isostere, medicine.medical_treatment, Dimer, Tripeptide, Catalysis, chemistry.chemical_compound, HIV Protease, X-Ray Diffraction, HIV-1 protease, Endopeptidases, Drug Discovery, medicine, Amines, Amino Acids, Aspartic Acid, Binding Sites, Protease, biology, Chemistry, Hydrogen bond, Active site, Hydrogen Bonding, HIV Protease Inhibitors, Peptide Fragments, Protease inhibitor (biology), Oxygen, Kinetics, Models, Chemical, Ethanolamines, biology.protein, Molecular Medicine, Dimerization, Synchrotrons, Protein Binding, medicine.drug
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11
المؤلفون: Milan Fábry, Klára Grantz Šašková, Jan Konvalinka, Vlastimil Král, Juraj Sedlacek, Irena Sieglová, Pavlína Řezáčová, Magdalena Hořejší, Milan Kožíšek, Jiří Brynda, Vanda Bartoňová
المصدر: Antiviral Research. 78:275-277
مصطلحات موضوعية: Models, Molecular, medicine.drug_class, medicine.medical_treatment, HIV Infections, Monoclonal antibody, Virus, Epitope, HIV Protease, Antiretroviral Therapy, Highly Active, Virology, Drug Resistance, Viral, medicine, Humans, Protease inhibitor (pharmacology), Immunoglobulin Fragments, Pharmacology, chemistry.chemical_classification, Protease, biology, Antibodies, Monoclonal, Genetic Variation, HIV Protease Inhibitors, Molecular biology, Recombinant Proteins, In vitro, Enzyme, chemistry, Mutation, HIV-1, biology.protein, Antibody, Dimerization
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12
المؤلفون: Milan Fábry, Juraj Sedlacek, Pavel Tichý, F. Kaprálek
المصدر: Folia Microbiologica. 43:63-67
مصطلحات موضوعية: Hot Temperature, Gene Dosage, Gene Expression, Biology, medicine.disease_cause, Microbiology, Gene dosage, law.invention, Plasmid, law, Gene expression, Escherichia coli, medicine, Animals, Topoisomerase II Inhibitors, Novobiocin, Enzyme Precursors, Expression vector, DNA, Superhelical, General Medicine, biology.organism_classification, Molecular biology, Enterobacteriaceae, Recombinant Proteins, Recombinant DNA, Cattle, Chymosin, Plasmids, medicine.drug
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13
المؤلفون: Milan Fábry, Anusch Peyman, Rolf Hilgenfeld, Alexander Liesum, Karl-Heinz Budt, Jochen Knolle, Juraj Sedlacek, Harald Berchtold, Gudrun Lange-Savage
المصدر: European Journal of Biochemistry. 248:313-322
مصطلحات موضوعية: Models, Molecular, Polyproteins, Protein Conformation, Stereochemistry, medicine.medical_treatment, Dimer, Molecular Sequence Data, Diol, Crystallography, X-Ray, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Protein structure, HIV Protease, medicine, Structure–activity relationship, chemistry.chemical_classification, Protease, biology, Active site, Valine, HIV Protease Inhibitors, Crystallography, Enzyme, chemistry, biology.protein
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14
المؤلفون: V. Chitarra, J. Lescar, Magda Horejsi, Milan Fábry, Juraj Sedlacek, M.-M. Riottot, Renata Stouracova, Jiri Brynda, Graham A. Bentley
المصدر: Journal of Molecular Biology. 267:1207-1222
مصطلحات موضوعية: Models, Molecular, Structural similarity, Stereochemistry, medicine.medical_treatment, Proteolysis, Molecular Sequence Data, Peptide, Cross Reactions, Crystallography, X-Ray, Antiparallel (biochemistry), Immunoglobulin Fab Fragments, HIV Protease, HIV-1 protease, Structural Biology, medicine, Computer Simulation, Amino Acid Sequence, Cloning, Molecular, Tyrosine, Molecular Biology, chemistry.chemical_classification, Binding Sites, Hybridomas, Protease, Base Sequence, medicine.diagnostic_test, biology, Antibodies, Monoclonal, HIV Protease Inhibitors, Sequence Analysis, DNA, Enzyme, chemistry, biology.protein
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15
المؤلفون: Milan Fábry, Jiří Brynda, Juraj Sedlacek, Magda Hořejšı́
المصدر: Virology. 207:185-190
مصطلحات موضوعية: viruses, Molecular Sequence Data, Peptide, Biology, medicine.disease_cause, Cleavage (embryo), Catalysis, Substrate Specificity, Enzyme catalysis, Frameshift mutation, Retrovirus, Proteinase 3, Virology, Escherichia coli, medicine, Aspartic Acid Endopeptidases, Amino Acid Sequence, Cloning, Molecular, Protein Precursors, chemistry.chemical_classification, Avian Myeloblastosis Virus, Base Sequence, biology.organism_classification, Molecular biology, Fusion Proteins, gag-pol, Amino acid, Kinetics, chemistry, Biochemistry, Protein Biosynthesis, Protein Processing, Post-Translational, Sequence Analysis
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16
المؤلفون: Olga Hrušková-Heidingsfeldová, Petr Štrop, Hans-Georg Kräusslich, Anke-Mareil Heuser, Jan Konvalinka, Volker M. Vogt, Juraj Sedlacek
المصدر: European Journal of Biochemistry. 228:191-198
مصطلحات موضوعية: chemistry.chemical_classification, Oligopeptide, Avian Myeloblastosis Virus, Polyproteins, Bovine leukemia virus, biology, viruses, Gene Products, gag, HIV, Peptide, Group-specific antigen, Cleavage (embryo), biology.organism_classification, Molecular biology, Biochemistry, Virus, Alpharetrovirus, law.invention, Fusion Proteins, gag-pol, Retroviridae, chemistry, law, Endopeptidases, Recombinant DNA, Cells, Cultured
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17
المؤلفون: Juraj Sedlacek, J. J. Wendoloski, S. I. Foundling, Douglas H. Ohlendorf, Petr Štrop, F. R. Salemme
المصدر: Proteins: Structure, Function, and Genetics. 14:382-391
مصطلحات موضوعية: Models, Molecular, Macromolecular Substances, Protein Conformation, viruses, Molecular Sequence Data, Avian myeloblastosis virus, Human immunodeficiency virus (HIV), medicine.disease_cause, Biochemistry, Virus, Substrate Specificity, Peptide substrate, Viral Proteins, Structural Biology, Homologous chromosome, medicine, Aspartic Acid Endopeptidases, Amino Acid Sequence, Molecular Biology, chemistry.chemical_classification, Avian Myeloblastosis Virus, Rous sarcoma virus, Sequence Homology, Amino Acid, biology, biology.organism_classification, Virology, Enzyme, Avian Sarcoma Viruses, chemistry, Oncovirinae, Protein Binding
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18
المؤلفون: Vladimír Kostka, F. Kaprálek, Iva Pichová, Juraj Sedlacek, Vladimir Benes, S. Foundling, Petr Štrop, Milan Souček, L. Pavlíčková, M. Trávníček
المصدر: International Journal of Biochemistry. 24:235-242
مصطلحات موضوعية: Cytoplasm, Sequence analysis, Molecular Sequence Data, Gene Products, gag, Biology, Biochemistry, Inclusion bodies, law.invention, law, Escherichia coli, Aspartic Acid Endopeptidases, Amino Acid Sequence, Isoelectric Point, Peptide sequence, Chromatography, High Pressure Liquid, chemistry.chemical_classification, Avian Myeloblastosis Virus, Rous sarcoma virus, Base Sequence, Fast protein liquid chromatography, biology.organism_classification, Molecular biology, Recombinant Proteins, Enzyme, Isoelectric point, chemistry, DNA, Viral, Recombinant DNA, Electrophoresis, Polyacrylamide Gel, Crystallization, Protein Processing, Post-Translational
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19
المؤلفون: Iva Pichová, Rostislav Skrabana, Jan Konvalinka, Frantisek Kapralek, Petr Štrop, Juraj Sedlacek, Vladimír Kostka, Ivo Bláha
المصدر: FEBS Letters. 282:73-76
مصطلحات موضوعية: Stereochemistry, Molecular Sequence Data, Norleucine, Kinetics, Biophysics, Peptide, Cleavage (embryo), Biochemistry, Substrate Specificity, chemistry.chemical_compound, Structural Biology, Genetics, Peptide synthesis, Aspartic Acid Endopeptidases, Amino Acid Sequence, Retroviral proteinase, Enzyme kinetics, Molecular Biology, Peptide sequence, chemistry.chemical_classification, Avian Myeloblastosis Virus, Chemistry, Spectrum Analysis, Cell Biology, Hydrogen-Ion Concentration, Chromogenic substrate, Enzyme, HIV-1 proteinase, Subsite specificity, MAV
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20
المؤلفون: Jiri Velek, Ivo Bláha, Miloslav Trávníček, L. Pavlíčková, Juraj Sedlacek, Petr Štrop, Vladimír Kostka, Jan Konvalinka, Dalibor Stys
المصدر: Biochemistry. 30:3437-3443
مصطلحات موضوعية: Molecular Sequence Data, Retroviridae Proteins, Sodium Chloride, Cleavage (embryo), Biochemistry, Avian sarcoma virus, Substrate Specificity, Endopeptidases, Aspartic Acid Endopeptidases, Amino Acid Sequence, Enzyme kinetics, Binding site, Peptide sequence, chemistry.chemical_classification, Avian Myeloblastosis Virus, Rous sarcoma virus, Binding Sites, Avian Leukosis Virus, biology, Hydrolysis, Serum Albumin, Bovine, Hydrogen-Ion Concentration, biology.organism_classification, Genes, gag, Kinetics, Enzyme, Avian Sarcoma Viruses, chemistry, Ionic strength, Peptide Hydrolases