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1A class of 5-benzylidene-2-phenylthiazolinones with high potency as direct 5-lipoxygenase inhibitors
المؤلفون: Carmen B. Rödl, Gisbert Schneider, Andreas Kiehl, Sebastian Barzen, Holger Stark, Julia Borig, Dieter Steinhilber, Aleksandra Zivkovic, Bettina Hofmann
المصدر: Journal of medicinal chemistry. 54(6)
مصطلحات موضوعية: Virtual screening, Arachidonate 5-Lipoxygenase, biology, Stereochemistry, Cancer, Stereoisomerism, medicine.disease, Benzylidene Compounds, chemistry.chemical_compound, Structure-Activity Relationship, Thiazoles, chemistry, Benzylidene compounds, Drug Discovery, Arachidonate 5-lipoxygenase, biology.protein, medicine, Molecular Medicine, Potency, Moiety, Structure–activity relationship, Lipoxygenase Inhibitors
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2
المؤلفون: Andreas Pfützner, Johannes Pfützner, Julia Borig, Anna M. Pfützner, Alexander Weise, PB Musholt, Michael Safinowski, Heike Hänel
المصدر: Journal of diabetes science and technology. 3(1)
مصطلحات موضوعية: Type 1 diabetes, medicine.medical_specialty, business.industry, Endocrinology, Diabetes and Metabolism, Insulin, medicine.medical_treatment, Injections, Subcutaneous, Biomedical Engineering, Dose accuracy, Bioengineering, Type 2 diabetes, Original Articles, medicine.disease, Specific density, Surgery, Animal science, Drug Delivery Systems, Diabetes mellitus, Instructions for use, Internal Medicine, medicine, Dosing, business
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3Academic Journal
المؤلفون: Bettina Hofmann, Sebastian Barzen, Carmen B. Rödl, Andreas Kiehl, Julia Borig, Aleksandra Živković, Holger Stark, Gisbert Schneider, Dieter Steinhilber
المصدر: Journal of Medicinal Chemistry; Mar2011, Vol. 54 Issue 6, p1943-1947, 5p