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1
المؤلفون: Nick Hartley, Jonathan Coates, Katy Woodward, Ian Briedis, Millie Dias
المصدر: Clinical Psychology Forum. 1:72-81
مصطلحات موضوعية: Clinical Psychology
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2
المؤلفون: Renate Griffith, Neal Dalton, Stephen G. Pyne, John B. Bremner, Nicholas Vandegraaff, Christopher P. Gordon, David Ian Rhodes, John Deadman, Paul A. Keller, Jonathan Coates
المصدر: Tetrahedron. 74:1253-1268
مصطلحات موضوعية: 0301 basic medicine, biology, Chemistry, Stereochemistry, Organic Chemistry, Human immunodeficiency virus (HIV), Active site, Tripeptide, medicine.disease_cause, Biochemistry, Integrase, Core domain, 03 medical and health sciences, 030104 developmental biology, Docking (molecular), Drug Discovery, biology.protein, medicine, HIV Integrase Inhibitors, Structure based
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3Academic Journal
المؤلفون: Jonathan Coates, Kate Smith
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.564.8378; http://journal.nzma.org.nz/journal/117-1201/1050/content.pdf
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4
المؤلفون: Fraser Gething, Jonathan Coates, Mark I. Johnson
المصدر: Pain Management. 7:223-227
مصطلحات موضوعية: Physician-Patient Relations, medicine.medical_specialty, Primary Health Care, business.industry, General Medicine, Primary care, 03 medical and health sciences, 0302 clinical medicine, Ambulatory care, General Practitioners, Managing pain, 030220 oncology & carcinogenesis, Family medicine, Outcome Assessment, Health Care, Humans, Pain Management, Medicine, 030212 general & internal medicine, business
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5
المؤلفون: Jonathan Coates, Jan Stolarek, Frank Emrich, James Cheney, Sam Lindley
المصدر: Proceedings of the 41st ACM SIGPLAN Conference on Programming Language Design and Implementation
Emrich, F, Lindley, S, Stolarek, J, Cheney, J & Coates, J 2020, FreezeML : Complete and Easy Type Inference for First-Class Polymorphism . in Proceedings of the 41st ACM SIGPLAN Conference on Programming Language Design and Implementation . Association for Computing Machinery (ACM), pp. 423-437, 41st ACM SIGPLAN Conference on Programming Language Design and Implementation, London, United Kingdom, 15/06/20 . https://doi.org/10.1145/3385412.3386003
PLDIمصطلحات موضوعية: FOS: Computer and information sciences, type inference, Computer Science - Programming Languages, Computer science, Programming language, System F, Inference, Type inference, 020207 software engineering, 0102 computer and information sciences, 02 engineering and technology, computer.software_genre, 01 natural sciences, First class, Undecidable problem, 010201 computation theory & mathematics, Conservative extension, Polymorphism (computer science), first-class polymorphism, impredicative types, 0202 electrical engineering, electronic engineering, information engineering, Programmer, computer, Programming Languages (cs.PL)
وصف الملف: application/pdf
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6
المؤلفون: Christopher P. Gordon, Timothy P. Boyle, Stephen G. Pyne, Nicholas Vandegraaf, Neal Dalton, David Ian Rhodes, John B. Bremner, John Deadman, Paul A. Keller, Jonathan Coates
المصدر: Organic & Biomolecular Chemistry. 14:6010-6023
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Protein Conformation, Stereochemistry, Antimicrobial peptides, HIV Integrase, Tripeptide, 01 natural sciences, Biochemistry, Inhibitory Concentration 50, Structure-Activity Relationship, 03 medical and health sciences, Protein structure, Structure–activity relationship, HIV Integrase Inhibitors, Physical and Theoretical Chemistry, IC50, chemistry.chemical_classification, Oligopeptide, biology, 010405 organic chemistry, Organic Chemistry, Combinatorial chemistry, 0104 chemical sciences, Amino acid, Integrase, 030104 developmental biology, chemistry, Drug Design, biology.protein, Tyrosine, Oligopeptides
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7
المؤلفون: Philip Rea, Nicholas J. Ede, John Deadman, Thomas S. Peat, Jonathan Coates, Janet Newman, Dharshini Jeevarajah, David Ian Rhodes, Nick Vandegraaff, John Martyn
المصدر: ChemBioChem. 12:2311-2315
مصطلحات موضوعية: Stereochemistry, Allosteric regulation, HIV Infections, Peptide, HIV Integrase, Crystallography, X-Ray, Peptides, Cyclic, Biochemistry, Molecular Docking Simulation, Humans, Amino Acid Sequence, HIV Integrase Inhibitors, Binding site, Molecular Biology, Peptide sequence, chemistry.chemical_classification, Binding Sites, biology, Chemistry, Hydrogen bond, Organic Chemistry, Hydrogen Bonding, Cyclic peptide, Integrase, HIV-1, biology.protein, Molecular Medicine
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8
المؤلفون: John Deadman, G. Paul Savage, Craig L. Francis, John H. Ryan, Thomas S. Peat, Jessica A. Smith, Dharshini Jeevarajah, Jonathan Coates, Janet Newman, Lisa Jane Winfield, Del Lucent, Giang Thanh Le, Neeranat Thienthong, Eric Dale Jones, David Ian Rhodes, Nick Vandegraaff
المصدر: Antiviral Chemistry and Chemotherapy. 21:155-168
مصطلحات موضوعية: Isatin, Crystallography, Indoles, Magnetic Resonance Spectroscopy, Alkylation, biology, Mechanism (biology), HIV Infections, Dioxoles, General Medicine, Computational biology, Surface Plasmon Resonance, Ligands, Integrase, Structure-Activity Relationship, Biochemistry, Catalytic Domain, Drug Design, HIV-1, biology.protein, Hiv 1 integrase, Structure based, HIV Integrase Inhibitors, Protein Binding
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9
المؤلفون: Xiao Feng, Changjiang Yu, Katherine Macfarlane, Giang Thanh Le, Eric Dale Jones, John Deadman, David Ian Rhodes, Neeranat Thienthong, Nick Vandegraaff, Long Lu, Xinming Li, Lisa Jane Winfield, Jonathan Coates, Neil Choi, William Issa
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:5913-5917
مصطلحات موضوعية: Scaffold, Pyridines, Stereochemistry, T-Lymphocytes, Clinical Biochemistry, Pharmaceutical Science, Integrase inhibitor, HIV Integrase, Biochemistry, Bridged Bicyclo Compounds, Structure-Activity Relationship, Drug Discovery, Humans, HIV Integrase Inhibitors, Molecular Biology, chemistry.chemical_classification, biology, Bicyclic molecule, Chemistry, Organic Chemistry, Wild type, biology.organism_classification, Nucleotidyltransferase, Integrase, Pyrimidines, Enzyme, Drug Design, Lentivirus, HIV-1, biology.protein, Molecular Medicine
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10Design of a series of bicyclic HIV-1 integrase inhibitors. Part 2: Azoles: Effective metal chelators
المؤلفون: John Deadman, Eric Dale Jones, David Ian Rhodes, Changjiang Yu, Nick Vandegraaff, Jonathan Coates, Xinming Li, Xiao Feng, Giang Thanh Le, Lisa Jane Winfield, Long Lu, Neeranat Thienthong
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:5909-5912
مصطلحات موضوعية: Azoles, Stereochemistry, Isostere, Clinical Biochemistry, Pharmaceutical Science, Integrase inhibitor, HIV Integrase, Biochemistry, Chemical synthesis, Bridged Bicyclo Compounds, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Humans, Structure–activity relationship, HIV Integrase Inhibitors, Thiazole, Molecular Biology, Chelating Agents, Oxazole, biology, Bicyclic molecule, Organic Chemistry, Integrase, chemistry, Metals, Drug Design, HIV-1, biology.protein, Molecular Medicine
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11
المؤلفون: John Deadman, Xiao Feng, Changjiang Yu, Jonathan Coates, Xinming Li, Eric Dale Jones, David Ian Rhodes, Nick Vandegraaff, Long Lu, Giang Thanh Le
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:5013-5018
مصطلحات موضوعية: Clinical Biochemistry, Pharmaceutical Science, Integrase inhibitor, medicine.disease_cause, Biochemistry, Virus, Structure-Activity Relationship, Raltegravir Potassium, Drug Resistance, Viral, Drug Discovery, medicine, HIV Integrase Inhibitors, Molecular Biology, chemistry.chemical_classification, Mutation, biology, Chemistry, Organic Chemistry, HIV, Nucleotidyltransferase, Raltegravir, biology.organism_classification, Virology, Pyrrolidinones, Integrase, Enzyme, Lentivirus, biology.protein, Molecular Medicine, medicine.drug
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12
المؤلفون: Jonathan Coates, Eric Dale Jones, Susan Cox, Nick Vandegraaff, Paula J De Bruyn, David Rhodes, David Gerard Bourke, Alan D. Robertson, Ian Travers Crosby
المصدر: Bioorganic & Medicinal Chemistry. 18:6442-6450
مصطلحات موضوعية: Anti-HIV Agents, Stereochemistry, Dihydropyran, Clinical Biochemistry, Pharmaceutical Science, HIV Integrase, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Drug Discovery, Animals, Humans, HIV Integrase Inhibitors, Molecular Biology, Maleimide, biology, Bicyclic molecule, Chemistry, Organic Chemistry, Naphthoquinone, Rats, Quinone, Integrase, Pyran, HIV-1, biology.protein, Molecular Medicine, Naphthoquinones
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13
المؤلفون: Allan H. White, John B. Bremner, Brian W. Skelton, Paul A. Keller, Jonathan Coates, Yasmine S. Torkamani, Mohammed K. Abdel-Hamid, Anthony C. Willis, Celia Miländer
المصدر: Tetrahedron Letters. 50:6947-6950
مصطلحات موضوعية: chemistry.chemical_classification, Chemical structure, Organic Chemistry, One-pot synthesis, Biochemistry, Combinatorial chemistry, Indigo, chemistry.chemical_compound, Cascade reaction, chemistry, Indigo carmine, Heterocyclic compound, Microwave heating, Drug Discovery, Microwave irradiation, Organic chemistry
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14
المؤلفون: John Deadman, John B. Bremner, Kittiya Somphol, Paul A. Keller, Jonathan Coates, Timothy P. Boyle, Stephen G. Pyne
المصدر: European Journal of Medicinal Chemistry. 44:1001-1009
مصطلحات موضوعية: Pharmacology, chemistry.chemical_classification, Spectrometry, Mass, Electrospray Ionization, Staphylococcus aureus, Magnetic Resonance Spectroscopy, Tetrapeptide, Stereochemistry, Phenylalanine, Organic Chemistry, Cationic polymerization, Peptoid, Peptide, Microbial Sensitivity Tests, General Medicine, Tripeptide, Chemical synthesis, Anti-Bacterial Agents, chemistry.chemical_compound, chemistry, Drug Discovery, Lipophilicity, Antibacterial agent
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15
المؤلفون: David Ian Rhodes, John B. Bremner, Timothy P. Boyle, Stephen G. Pyne, Paul A. Keller, Jonathan Coates, John Deadman
المصدر: Tetrahedron. 64:11270-11290
مصطلحات موضوعية: chemistry.chemical_classification, Dipeptide, Allylglycine, Organic Chemistry, medicine.disease_cause, Metathesis, Biochemistry, Combinatorial chemistry, Cyclic peptide, chemistry.chemical_compound, Ring-closing metathesis, chemistry, Staphylococcus aureus, Drug Discovery, medicine, Salt metathesis reaction, Tyrosine
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16
المؤلفون: Vicki S. Au, Stephen G. Pyne, Paul A. Keller, Jonathan Coates, John B. Bremner
المصدر: Tetrahedron. 62:9373-9382
مصطلحات موضوعية: Indole test, Ring-closing metathesis, Chemistry, Organic Chemistry, Drug Discovery, Organic chemistry, Metathesis, Antibacterial activity, Biochemistry, Combinatorial chemistry
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17
المصدر: Tetrahedron. 61:7271-7276
مصطلحات موضوعية: Olefin fiber, Arginine, Chain (algebraic topology), Chemistry, Stereochemistry, Organic Chemistry, Drug Discovery, Lysine, Salt metathesis reaction, General Medicine, Metathesis, Biochemistry
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18
المؤلفون: David Ian Rhodes, Susan Cox, Neville G. Walsh, Simon P. B. Ovenden, Jin Yu, R. Murray Tait, Barbara Meurer-Grimes, Gian Sberna, Soo San Wan, Jonathan Coates
المصدر: Phytochemistry. 65:3255-3259
مصطلحات موضوعية: Lignan, Bioassay guided fractionation, biology, Stereochemistry, Plant Science, General Medicine, Horticulture, Eucalyptus globoidea, biology.organism_classification, Biochemistry, Strand transfer, Integrase, chemistry.chemical_compound, chemistry, biology.protein, Globoidnan A, Molecular Biology
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19
المصدر: Synlett. 2002:0219-0222
مصطلحات موضوعية: chemistry.chemical_compound, Ring-closing metathesis, Chemistry, Carbazole, Organic Chemistry, Salt metathesis reaction, Moiety, Peptoid, Tripeptide, Antibacterial activity, Combinatorial chemistry
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20
المؤلفون: Ben Li, Dawei Ma, Xing He, Miao Wang, Jonathan Coates, Eric Dale Jones, Xin Xie, David Ian Rhodes, Enkun Zhou, Li Chen, John Deadman, Shanghai Yu, Gang Pei, Dean Baylis
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:5334-5336
مصطلحات موضوعية: Pyrrolidines, Anti-HIV Agents, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, CHO Cells, CCR5 receptor antagonist, Ring (chemistry), Biochemistry, Chemical synthesis, Pyrrolidine, Structure-Activity Relationship, chemistry.chemical_compound, Cricetulus, Cricetinae, Drug Discovery, Animals, Structure–activity relationship, Molecular Biology, Organic Chemistry, Antagonist, Stereoisomerism, Tropane, chemistry, CCR5 Receptor Antagonists, Molecular Medicine, Piperidine