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1
المؤلفون: Cindy Q. Xia, Bei-Ching Chuang, Johnny J. Yang, Yuexian Li, Shaoxia Yu, Shimoga Prakash, Mingxiang Liao, Emily Guan, Qing Zhu
المصدر: Xenobiotica. 48:467-477
مصطلحات موضوعية: Male, Cell Membrane Permeability, Time Factors, Abcg2, Health, Toxicology and Mutagenesis, Breast Neoplasms, Diketopiperazines, Pharmacology, Toxicology, 030226 pharmacology & pharmacy, Biochemistry, 03 medical and health sciences, Dogs, 0302 clinical medicine, Pharmacokinetics, ATP Binding Cassette Transporter, Subfamily G, Member 2, Animals, Humans, Distribution (pharmacology), ADME, Mice, Knockout, biology, Chemistry, Transporter, General Medicine, Metabolism, In vitro, Absorption, Physiological, Neoplasm Proteins, Rats, Sulfasalazine, Macaca fascicularis, 030220 oncology & carcinogenesis, Hepatocytes, Microsomes, Liver, biology.protein, Female, Efflux, Caco-2 Cells
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2
المؤلفون: Yuexian Li, Mingxiang Liao, Miao Y. Guan, Jiyeon Woo, Johnny J. Yang, Shimoga Prakash, Jessica M. Chmielecki, Bei-Ching Chuang, Cindy Q. Xia, Mihaela Plesescu
المصدر: Bioorganic & Medicinal Chemistry Letters. 26:551-555
مصطلحات موضوعية: Compound a, Abcg2, Estrone, Clinical Biochemistry, Pharmaceutical Science, Diketopiperazines, Pharmacology, 010402 general chemistry, Heterocyclic Compounds, 4 or More Rings, 01 natural sciences, Biochemistry, Structure-Activity Relationship, Pharmacokinetics, In vivo, Drug Discovery, ATP Binding Cassette Transporter, Subfamily G, Member 2, Animals, Humans, Potency, ATP Binding Cassette Transporter, Subfamily B, Member 1, Molecular Biology, biology, 010405 organic chemistry, Chemistry, Organic Chemistry, Stereoisomerism, In vitro, Rats, 0104 chemical sciences, Bioavailability, Inhibitory potency, biology.protein, Molecular Medicine, Caco-2 Cells
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3
المؤلفون: Tim Wyant, Melissa Gallery, Daniel Bradley, Adnan O. Abu-Yousif, Mark Williamson, Jose Estevam, Qing Zhu, Ping Li, Johnny J. Yang, Mark Manfredi, Claudia Rabino, Huay-Keng Loke, Edward A. Greenfield, O. Petter Veiby, Julie Zhang, Brad Stringer, Hadi Danaee, Donna Cvet, Pamela Brauer
المصدر: PLoS ONE, Vol 13, Iss 1, p e0191046 (2018)
PLoS ONEمصطلحات موضوعية: 0301 basic medicine, Immunoconjugates, Physiology, Cancer Treatment, Receptors, Enterotoxin, lcsh:Medicine, Mice, SCID, Biochemistry, Mice, chemistry.chemical_compound, Spectrum Analysis Techniques, 0302 clinical medicine, Immune Physiology, Medicine and Health Sciences, Cytotoxic T cell, Intestinal Mucosa, lcsh:Science, Immune System Proteins, Multidisciplinary, biology, Reverse Transcriptase Polymerase Chain Reaction, Antibodies, Monoclonal, Guanylate cyclase 2C, Flow Cytometry, Oncology, Monomethyl auristatin E, Spectrophotometry, 030220 oncology & carcinogenesis, Monoclonal, Female, Cytophotometry, Anatomy, Antibody, Colorectal Neoplasms, Oligopeptides, Research Article, Colon, medicine.drug_class, Immunology, Blotting, Western, Research and Analysis Methods, Antibodies, Monoclonal, Humanized, Monoclonal antibody, Antibodies, 03 medical and health sciences, Antigen, In vivo, medicine, Animals, Humans, Immunohistochemistry Techniques, Colorectal Cancer, lcsh:R, Biology and Life Sciences, Proteins, Cancers and Neoplasms, Xenograft Model Antitumor Assays, Monoclonal Antibodies, Gastrointestinal Tract, Histochemistry and Cytochemistry Techniques, HEK293 Cells, 030104 developmental biology, Metastatic Tumors, chemistry, Immunologic Techniques, Cancer research, biology.protein, lcsh:Q, Digestive System
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4
المؤلفون: Emily F. Calderwood, Kathleen Aertgeerts, Michael D. Smith, Dylan Bradley England, Roushan Afroze, Ryan Chau, Stepan Vyskocil, Nancy E. Forsyth, Dong Mei Zhang, Ruth Adams, Stephen G. Stroud, O. P. Veiby, Christelle C. Renou, R. Scott Rowland, Erin Paske, Jane X. Liu, Ming Tregay, Michael D. Sintchak, Juliet A Williams, Shih-Chung Huang, Xu Tianlin, Bheemashankar Kulkarni, Sharmila Adhikari, Yuan Tian, Jason Yano, Christopher Blackburn, Paul D. Greenspan, Cheryl A. Farrer, Matthew O. Duffey, Liting Ma, Mi-Sook Kim, Qin Zhang, Sean Harrison, Hirotake Mizutani, Katherine M. Galvin, Alexandra E. Gould, Johnny J. Yang, Steven P. Langston, Dave Janowick, Natalia Iartchouk, Mansoureh Rezaei, Jeffery Gaulin, Khristofer Garcia, Hongbo Zeng, Ribo Guo, Tricia J. Vos, Jouhara Chouitar, Saurabh Menon
المصدر: Journal of Medicinal Chemistry. 54:1836-1846
مصطلحات موضوعية: Models, Molecular, Proto-Oncogene Proteins B-raf, Tetrahydronaphthalenes, Mutant, Melanoma, Experimental, Administration, Oral, Biological Availability, Mice, Nude, Antineoplastic Agents, Pharmacology, Crystallography, X-Ray, Mice, Structure-Activity Relationship, Pharmacokinetics, Mouse xenograft, In vivo, Drug Discovery, medicine, Animals, chemistry.chemical_classification, Chemistry, Melanoma, Stereoisomerism, medicine.disease, Xenograft Model Antitumor Assays, In vitro, Bioavailability, Enzyme, Drug Design, Mutation, Molecular Medicine
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5
المؤلفون: Frank W. Lee, Suresh K. Balani, Mingxiang Liao, Johnny J. Yang, Ning Liu, Liang-Shang Gan, Shaoxia Yu, Shimoga R. Prakash, Cindy Q. Xia, Jing-Tao Wu, Mark N. Milton
المصدر: Drug Metabolism Letters. 4:202-212
مصطلحات موضوعية: Male, medicine.medical_specialty, ATP Binding Cassette Transporter, Subfamily B, Abcg2, medicine.drug_class, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Pharmacology, Piperazines, Tyrosine-kinase inhibitor, Rats, Sprague-Dawley, Mice, Oral administration, Tetrahydroisoquinolines, Internal medicine, medicine, ATP Binding Cassette Transporter, Subfamily G, Member 2, Animals, Humans, Pharmacology (medical), ATP Binding Cassette Transporter, Subfamily B, Member 1, Intestinal Mucosa, Protein Kinase Inhibitors, P-glycoprotein, Mice, Knockout, biology, Biochemistry (medical), Wild type, Brain, Biological Transport, Transporter, Neoplasm Proteins, Rats, Endocrinology, Caco-2, Injections, Intravenous, Quinazolines, biology.protein, Acridines, ATP-Binding Cassette Transporters, Efflux, Caco-2 Cells
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6
المؤلفون: Johnny J. Yang, Weirong Wang, Nagendra Chemuturi, Ramaswamy A. Iyer, Eugenia Kraynov, Markus Walles, Priya Sriraman, David J Moore, Amita Datta-Mannan, Edit Tarcsa, Guangqing Xiao, Amrita V. Kamath, Enrique Escandón, Matthew Barfield, Michaela Bairlein, Antoine Deslandes, Dan A. Rock
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 44(5)
مصطلحات موضوعية: 0301 basic medicine, Drug, Immunoconjugates, Drug Industry, media_common.quotation_subject, Pharmaceutical Science, Computational biology, Pharmacology, Drug molecule, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, White paper, Antibodies monoclonal, Distribution (pharmacology), Animals, Humans, Hardware_ARITHMETICANDLOGICSTRUCTURES, Drug industry, ADME, media_common, Chemistry, Antibodies, Monoclonal, body regions, 030104 developmental biology, Pharmaceutical Preparations
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7
المؤلفون: Jasmine Davda, Vinod Labhasetwar, Mohamed G. Qaddoumi, Vincent H.L. Lee, Johnny J. Yang, Hideo Ueda
المصدر: Pharmaceutical Research. 21:641-648
مصطلحات موضوعية: Male, Polymers, Pharmaceutical Science, Nanoparticle, macromolecular substances, Absorption (skin), Pharmacology, Endocytosis, Plga nanoparticles, chemistry.chemical_compound, Polylactic Acid-Polyglycolic Acid Copolymer, Coumarins, Animals, Nanotechnology, Pharmacology (medical), Lactic Acid, Particle Size, Polylactic acid-polyglycolic acid copolymer, Dose-Response Relationship, Drug, Organic Chemistry, technology, industry, and agriculture, Epithelial Cells, Rabbit (nuclear engineering), Conjunctival epithelial cell, PLGA, chemistry, Biophysics, Molecular Medicine, Rabbits, Conjunctiva, Polyglycolic Acid, Biotechnology
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8
المؤلفون: Santhosh Palani, Johnny J. Yang, Mayankbhai Patel, Wen Chyi Shyu, Arijit Chakravarty, Jerome T. Mettetal
المصدر: PLoS ONE
PLoS ONE, Vol 9, Iss 10, p e109892 (2014)مصطلحات موضوعية: Male, Neutropenia, Physiology, Hematopoietic System, Cmax, Predictive Toxicology, lcsh:Medicine, Antineoplastic Agents, Docetaxel, Bioinformatics, Toxicology, Models, Biological, Drug Administration Schedule, Dose schedule, Rats, Sprague-Dawley, Pharmacokinetics, In vivo, hemic and lymphatic diseases, medicine, Medicine and Health Sciences, Animals, Humans, lcsh:Science, Etoposide, Multidisciplinary, Toxicity, business.industry, Systems Biology, lcsh:R, Biology and Life Sciences, Computational Biology, Models, Theoretical, medicine.disease, Toxicokinetics, Oncology, lcsh:Q, Taxoids, Oncology drugs, business, Topotecan, medicine.drug, Research Article
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9
المؤلفون: Kwang-Jin Kim, Hideo Ueda, Johnny J. Yang, Vincent H.L. Lee
المصدر: Journal of Controlled Release. 65:1-11
مصطلحات موضوعية: Passive transport, Chemistry, Stereochemistry, Pharmaceutical Science, Ouabain, Cell culture, Biophysics, medicine, Electrochemical gradient, Ion transporter, Bumetanide, medicine.drug, Transepithelial potential difference, Uridine transport
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10
المؤلفون: Kwang-Jin Kim, Vincent H.L. Lee, Johnny J. Yang
المصدر: Pharmaceutical Research. 17:533-538
مصطلحات موضوعية: Pharmacology, Pathology, medicine.medical_specialty, Lagomorpha, Conjunctiva, biology, medicine.diagnostic_test, Organic Chemistry, Pharmaceutical Science, Apical membrane, biology.organism_classification, Immunofluorescence, Molecular biology, In vitro, Epithelium, medicine.anatomical_structure, Cell culture, medicine, biology.protein, Molecular Medicine, Pharmacology (medical), Biotechnology, P-glycoprotein
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11
المؤلفون: Mayankbhai Patel, Johnny J. Yang, Suresh K. Balani, Santhosh Palani, Arijit Chakravarty, Jerome T. Mettetal, Susan Chen, Mark Manfredi, Jessica Huck, Mengkun Zhang, Jeffrey Ecsedy, Wen Chyi Shyu
المصدر: Cancer chemotherapy and pharmacology. 72(6)
مصطلحات موضوعية: Cancer Research, Mitotic index, Population, Aurora A kinase, Mice, Nude, Antineoplastic Agents, Pharmacology, Biology, Toxicology, Bioinformatics, Models, Biological, chemistry.chemical_compound, Inhibitory Concentration 50, Mice, Pharmacokinetics, In vivo, Animals, Humans, Pharmacology (medical), education, Protein Kinase Inhibitors, Aurora Kinase A, education.field_of_study, Dose-Response Relationship, Drug, Azepines, HCT116 Cells, Xenograft Model Antitumor Assays, Pyrimidines, Oncology, chemistry, Pharmacodynamics, Alisertib, Spindle organization, Female, Colorectal Neoplasms
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12
المؤلفون: Swaminathan Padmanabhan, Johnny J. Yang, Jennifer S. Carew, Claudia M. Espitia, Mengkun Zhang, Steffan T. Nawrocki, Francis J. Giles, Kevin R. Kelly, Jeffrey Ecsedy
مصطلحات موضوعية: Cancer Research, Cell Survival, Aurora A kinase, Apoptosis, HL-60 Cells, Mice, SCID, Pharmacology, Protein Serine-Threonine Kinases, Article, chemistry.chemical_compound, Mice, Aurora Kinases, hemic and lymphatic diseases, Cell Line, Tumor, Proto-Oncogene Proteins, Antineoplastic Combined Chemotherapy Protocols, medicine, Animals, Humans, Viability assay, Molecular Targeted Therapy, Protein Kinase Inhibitors, Aurora Kinase A, Gene knockdown, Bcl-2-Like Protein 11, business.industry, Cell Cycle, Forkhead Box Protein O3, Cytarabine, Myeloid leukemia, Membrane Proteins, Drug Synergism, Forkhead Transcription Factors, Azepines, Cell cycle, Xenograft Model Antitumor Assays, Leukemia, Myeloid, Acute, Pyrimidines, Oncology, chemistry, Alisertib, Female, business, Apoptosis Regulatory Proteins, Cyclin-Dependent Kinase Inhibitor p27, medicine.drug
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13
المؤلفون: Paul D. Greenspan, Susan Chen, Liting Ma, Jane X. Liu, Johnny J. Yang, Qin Zhang, Ruth Adams, Shih-Chung Huang, Bheemashankar Kulkarni, Ryan W. Chau, Masayuki Nagayoshi, Matthew O. Duffey, Shaoxia Yu, Christopher Blackburn, Khristofer Garcia, Katherine M. Galvin, Tricia J. Vos, Sean Harrison, R. Scott Rowland, Xu Tianlin, Steven P. Langston, Mi-Sook Kim, Saurabh Menon, Alexandra E. Gould
المصدر: Bioorganicmedicinal chemistry letters. 20(16)
مصطلحات موضوعية: Proto-Oncogene Proteins B-raf, Stereochemistry, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Pyrazoline, Pyrazoline derivatives, Non-specific serine/threonine protein kinase, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, Computer Simulation, Molecular Biology, Protein Kinase Inhibitors, chemistry.chemical_classification, Binding Sites, biology, Organic Chemistry, Chemical modification, Thiophene derivatives, Recombinant Proteins, Enzyme, chemistry, Amino Acid Substitution, Enzyme inhibitor, biology.protein, Molecular Medicine, Pyrazoles
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14
المؤلفون: Cindy Q. Xia, Johnny J. Yang
المصدر: Enzyme Inhibition in Drug Discovery and Development: The Good and the Bad
مصطلحات موضوعية: Drug, business.industry, media_common.quotation_subject, Medicine, Transporter, Pharmacology, business, media_common
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15
المؤلفون: Suresh K. Balani, Johnny J. Yang, Cindy Q. Xia
المصدر: Drug Metabolism in Drug Design and Development: Basic Concepts and Practice
مصطلحات موضوعية: Drug, Drug disposition, business.industry, media_common.quotation_subject, Medicine, Transporter, Drug resistance, Pharmacology, business, media_common
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16
المؤلفون: Vincent H.L. Lee, Johnny J. Yang, David K. Ann, Ram Kannan
المصدر: Pharmaceutical research. 24(8)
مصطلحات موضوعية: medicine.medical_treatment, Blotting, Western, Indomethacin, Molecular Sequence Data, Pharmaceutical Science, Biological Transport, Active, Gene Expression, Biology, Adenoviridae, Western blot, Multidrug Resistance Protein 1, Sequence Homology, Nucleic Acid, medicine, Animals, Humans, Pharmacology (medical), Amino Acid Sequence, Buthionine Sulfoximine, Cells, Cultured, Epithelial polarity, Pharmacology, medicine.diagnostic_test, Base Sequence, Sequence Homology, Amino Acid, Reverse Transcriptase Polymerase Chain Reaction, Organic Chemistry, Anti-Inflammatory Agents, Non-Steroidal, Interleukin, Epithelial Cells, Molecular biology, Leukotriene C4, Blot, Cytokine, Pharmaceutical Preparations, Caco-2, Molecular Medicine, Cytokines, Tumor necrosis factor alpha, Fluorescein, Rabbits, Caco-2 Cells, Multidrug Resistance-Associated Proteins, Conjunctiva, Biotechnology
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17
المؤلفون: Johnny J Yang, Liang-Shang Gan, Cindy Q. Xia
المصدر: Expert opinion on drug metabolismtoxicology. 1(4)
مصطلحات موضوعية: Drug, Abcg2, media_common.quotation_subject, ATP-binding cassette transporter, Pharmacology, Toxicology, Absorption, chemistry.chemical_compound, Food-Drug Interactions, Pharmacokinetics, In vivo, ATP Binding Cassette Transporter, Subfamily G, Member 2, Humans, Drug Interactions, media_common, Polymorphism, Genetic, biology, Transporter, General Medicine, In vitro, Neoplasm Proteins, chemistry, Blood-Brain Barrier, Area Under Curve, biology.protein, ATP-Binding Cassette Transporters, Xenobiotic
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18
المؤلفون: Petter Veiby, John W. Hoppin, Mary Carsillo, Shu-Wen Teng, Daniel Bradley, Nicolas Salem, Melissa Saylor, Steven Mather, Donna Cvet, Mary Ruscowski, Jennifer Terkelsen, Robert Robertson, Kelly Davis Orcutt, Marc Berridge, Jeffery Norenberg, Ozlem Yardibi, Maria Borland, Mike Schulz, Tamara Anderson, Johnny J. Yang, Jacob Hesterman, Sells Todd B
المصدر: Cancer Research. 74:4949-4949
مصطلحات موضوعية: Cancer Research, medicine.medical_specialty, business.industry, Guanylate cyclase 2C, Effective dose (pharmacology), In vitro, Malignant transformation, chemistry.chemical_compound, Endocrinology, Oncology, chemistry, In vivo, Internal medicine, Cancer research, Medicine, DOTA, business, Receptor, Ex vivo
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19
المؤلفون: Shu-Wen Teng, Jerome T. Mettetal, Johnny J. Yang, Brad Stringer, Arijit Chakravarty, Wen Chyi Shyu, Julie Zhang, Christopher J. Zopf, Petter Veiby
المصدر: Cancer Research. 74:4649-4649
مصطلحات موضوعية: Drug, Cancer Research, media_common.quotation_subject, Cancer, Biological activity, Guanylate cyclase 2C, Pharmacology, Biology, medicine.disease, Oncology, Pharmacokinetics, Linear regression, medicine, Dosing, media_common, Conjugate
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20
المؤلفون: Johnny J. Yang, Kelly Davis Orcutt, Petter Veiby, Wen Chyi Shyu, Julie Zhang, Ozlem Yardibi, Arijit Chakravarty, Shu-Wen Teng, Donna Cvet, Melissa Gallery, Daniel Bradley, Jerome T. Mettetal
المصدر: Cancer Research. 74:365-365
مصطلحات موضوعية: Cancer Research, Pathology, medicine.medical_specialty, Chemistry, Cancer, Biological activity, medicine.disease, Tumor antigen, In vitro, Oncology, Antigen, In vivo, Cancer research, medicine, Viability assay, Preclinical imaging