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1
المؤلفون: Jean-François Fournier
المصدر: The Medicinal Chemist's Guide to Solving ADMET Challenges ISBN: 9781788012270
مصطلحات موضوعية: chemistry.chemical_compound, Photosensitivity, Chemistry, Aryl, Drug administration, Drug-induced photosensitivity, Combinatorial chemistry, Scavenger (chemistry)
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2
المؤلفون: Jean-François Fournier
المصدر: French Forum. 44:345-360
مصطلحات موضوعية: Literature and Literary Theory, Visual Arts and Performing Arts
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3
المؤلفون: Corinne Millois, Loïc Tomas, Catherine Comino, Laurence Dumais, Sandrine Talano, Kevin Reverse, Céline Mathieu, Craig S. Harris, Nicolas Vanthuyne, Grégoire Mouis, Anne-Laurence Ghilini, Laurent F. Hennequin, Claire Bouix-Peter, Vincent Rodeschini, Ghizlane El-Bazbouz, Laurence Clary, Sandrine Chambon, Romain Pierre, Jean-François Fournier, Anne Brethon
المساهمون: Nestle Skin Health GALDERMA R&D, Institut des Sciences Moléculaires de Marseille (ISM2), Aix Marseille Université (AMU)-École Centrale de Marseille (ECM)-Institut de Chimie du CNRS (INC)-Centre National de la Recherche Scientifique (CNRS), edelris
المصدر: Tetrahedron
Tetrahedron, Elsevier, 2018, 74 (37), pp.4805-4822. ⟨10.1016/j.tet.2018.07.029⟩
Tetrahedron, 2018, 74 (37), pp.4805-4822. ⟨10.1016/j.tet.2018.07.029⟩مصطلحات موضوعية: 0301 basic medicine, Drug, Peptidomimetic, media_common.quotation_subject, Caspase 1, 01 natural sciences, Biochemistry, 03 medical and health sciences, chemistry.chemical_compound, Drug Discovery, [CHIM]Chemical Sciences, media_common, 010405 organic chemistry, Drug discovery, Organic Chemistry, Acetal, Uracil, Combinatorial chemistry, 0104 chemical sciences, 3. Good health, 030104 developmental biology, chemistry, Caspase-1 inhibitors 1, Hemiacetal, 5-Trisubstitued uracil Peptidomimetics Topical application Excipient stability Chiral stability
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4
المؤلفون: Catherine Soulet, Laurent F. Hennequin, Nicolas Fleury-Brégeot, Craig S. Harris, Blanche Gauthier, Gwenaëlle Duvert, Etienne Thoreau, Laurent Chantalat, Karine Grisendi, Jean-François Fournier, Jerome Aubert, Michèle Aurelly, Rémy Morgentin, Claire Bouix-Peter, Bénédicte Drean, Guillaume Lafitte, Yushma Bhurruth-Alcor, Florence Joly, Jonathan Pascau, Branislav Musicki, Yves Rival, David Piwnica, Karinne Bouquet, Marion Delorme, T. Isabet, Corinne Millois, Loïc Tomas
المصدر: Bioorganic & Medicinal Chemistry Letters. 28:2985-2992
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Skin Neoplasms, Clinical Biochemistry, Histone Deacetylase 2, Pharmaceutical Science, Antineoplastic Agents, Apoptosis, Histone Deacetylase 1, Pharmacology, Crystallography, X-Ray, Biochemistry, Structure-Activity Relationship, 03 medical and health sciences, 0302 clinical medicine, Cell Line, Tumor, Drug Discovery, Hydrolase, medicine, Humans, Solubility, Molecular Biology, Cell Proliferation, chemistry.chemical_classification, Mycosis fungoides, Dose-Response Relationship, Drug, Molecular Structure, Quinine, Organic Chemistry, Cutaneous T-cell lymphoma, Squaramide, medicine.disease, Lymphoma, T-Cell, Cutaneous, Histone Deacetylase Inhibitors, 030104 developmental biology, Enzyme, chemistry, Cell culture, 030220 oncology & carcinogenesis, Molecular Medicine, Histone deacetylase, Drug Screening Assays, Antitumor
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5
المؤلفون: Didier M. Roche, Danielle Orfila, Ghizlane El-Bazbouz, Laurence Dumais, Laurent F. Hennequin, Céline Mathieu, Michèle Aurelly, Jerome Aubert, Claude Lardy, Etienne Thoreau, Anne-Pascale Luzy, Claire Bouix-Peter, Kenny Mebrouk, T. Isabet, Jean-François Fournier, Kevin Reverse, Catherine Comino, Corinne Millois, Anne-Laurence Ghilini, Jonathan Pascau, Sandrine Talano, Anne Brethon, Craig S. Harris, Romain Pierre, Sandrine Chambon, Laurence Clary, Olivier Christin, Laurent Chantalat, Vincent Rodeschini
المصدر: Journal of Medicinal Chemistry. 61:4030-4051
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Protein Conformation, Administration, Topical, medicine.medical_treatment, Caspase 1, Drug design, Pharmacology, 01 natural sciences, Cell Line, Mice, 03 medical and health sciences, chemistry.chemical_compound, Acne Vulgaris, Drug Discovery, medicine, Animals, Humans, Tissue Distribution, Caspase, Acne, Protease, biology, 010405 organic chemistry, Uracil, medicine.disease, Caspase Inhibitors, 0104 chemical sciences, 030104 developmental biology, chemistry, Drug Design, Solvents, biology.protein, Molecular Medicine, Pharmacophore, Phototoxicity
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6
المصدر: Journal of Medicinal Chemistry. 61:3231-3236
مصطلحات موضوعية: Keratinocytes, 0301 basic medicine, Ultraviolet Rays, Chemistry, Pharmaceutical, Electrons, Mice, Structure-Activity Relationship, 03 medical and health sciences, 0302 clinical medicine, Drug Discovery, Animals, Heuristics, Humans, Photosensitizing Agents, Chemistry, Liability, 3T3 Cells, Rule of thumb, 030104 developmental biology, Skin irritation, 030220 oncology & carcinogenesis, Molecular Medicine, Biochemical engineering, Phototoxicity, Algorithms, Dermatitis, Phototoxic, Forecasting
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7
المؤلفون: Marcus Gastreich, Laurence Clary, Jonathan Pascau, Anne Brethon, Laurent Chantalat, Olivier Christin, Etienne Thoreau, Jean-François Fournier, Craig S. Harris, Didier Roche, T. Isabet, Vincent Rodeschini
المصدر: Bioorganic & Medicinal Chemistry Letters. 27:5373-5377
مصطلحات موضوعية: 0301 basic medicine, Scaffold, Stereochemistry, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, CASPASE 1 INHIBITOR, Crystallography, X-Ray, Scaffold hopping, 01 natural sciences, Biochemistry, Inhibitory Concentration 50, 03 medical and health sciences, chemistry.chemical_compound, 4-Butyrolactone, Drug Discovery, Molecular Biology, Biological Products, Binding Sites, Natural product, 010405 organic chemistry, Caspase 1, Organic Chemistry, Hydrogen Bonding, Dipeptides, Caspase Inhibitors, Combinatorial chemistry, Protein Structure, Tertiary, 0104 chemical sciences, Molecular Docking Simulation, 030104 developmental biology, chemistry, Docking (molecular), Molecular Medicine, Azabicyclo Compounds
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8
المؤلفون: Jean-François Fournier, Didier Roche, Craig S. Harris, Sandrine Talano, Anne Brethon, Claude Lardy, Laurence Clary, Claire Bouix-Peter, Vincent Rodeschini
المصدر: Tetrahedron Letters. 57:5924-5927
مصطلحات موضوعية: 010405 organic chemistry, Chemistry, Peptidomimetic, Organic Chemistry, Drug Discovery, Alkylation, 010402 general chemistry, 01 natural sciences, Biochemistry, Combinatorial chemistry, 0104 chemical sciences, Stereocenter
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9
المؤلفون: Nicolas Rodeville, Jean-Guy Boiteau, Sebastien Daver, Corinne Millois, Jean-François Fournier, Laurence Dumais, Loïc Tomas, Laurence Clary, Kenny Mebrouk, Sandrine Talano, Romain Pierre, Craig S. Harris, Claire Bouix-Peter, Sandrine Chambon
المصدر: Tetrahedron Letters. 57:2367-2371
مصطلحات موضوعية: chemistry.chemical_classification, 5-nitrouracil, 010405 organic chemistry, Component (thermodynamics), Stereochemistry, Organic Chemistry, Uracil, Alkylation, 010402 general chemistry, 01 natural sciences, Biochemistry, 0104 chemical sciences, Amino acid, chemistry.chemical_compound, chemistry, Drug Discovery, Protecting group
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10
المؤلفون: Loïc Tomas, Rodolphe Vatinel, Craig S. Harris, Veronique Parnet, Gilles Ouvry, Catherine Raffin, Bénédicte Drean, Claire Bouix-Peter, Kana Kunihiro, Guillaume Lafitte, Branislav Musicki, Jean-François Fournier, Frédéric Gaigne, Romain Pierre, Céline Bonneaud
المصدر: Tetrahedron Letters. 58:3757-3759
مصطلحات موضوعية: Scope (project management), 010405 organic chemistry, Chemistry, Organic Chemistry, Drug Discovery, One-pot synthesis, Substrate (chemistry), Organic chemistry, 010402 general chemistry, 01 natural sciences, Biochemistry, 0104 chemical sciences, Butyl lithium
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11
المؤلفون: Coralie Pascau, Nicolas Atrux-Tallau, Laurent F. Hennequin, Christophe Feret, Gilles Ouvry, Feriel Hacini-Rachinel, Craig S. Harris, Claire Defoin-Platel, Nathalie Taquet, Sophie Deret, Mathieu Forissier, Hélène Huguet, Etienne Thoreau, Benjamin Ozello, Olivier Christin, Emmanuel Vial, Guillaume Lafitte, Danielle Orfila, Isabelle Carlavan, Franck Bihl, David Froude, Jean-François Fournier, Denis Duvert, Anne-Pascale Luzy, Delphine Spiesse, Patricia Rossio, Marie-Josée Cuadrado, Jonathan Pascau, Catherine Raffin, Aline Bondu, Claire Bouix-Peter, Catherine Hervouet, Guillaume Peluchon, Veronique Parnet, David Piwnica, Branislav Musicki, Rodolphe Vatinel, Romain Pierre
المساهمون: Laboratoire de synthèse organique (DCSO), École polytechnique (X)-Institut de Chimie du CNRS (INC)-Centre National de la Recherche Scientifique (CNRS), Institut de pharmacologie moléculaire et cellulaire (IPMC), Université Nice Sophia Antipolis (1965 - 2019) (UNS), COMUE Université Côte d'Azur (2015-2019) (COMUE UCA)-COMUE Université Côte d'Azur (2015-2019) (COMUE UCA)-Centre National de la Recherche Scientifique (CNRS), Nestle Skin Health GALDERMA R&D, Religions et croyances (LARHRA REC ), LAboratoire de Recherche Historique Rhône-Alpes - UMR5190 (LARHRA), École normale supérieure de Lyon (ENS de Lyon)-Université Lumière - Lyon 2 (UL2)-Université Jean Moulin - Lyon 3 (UJML), Université de Lyon-Université de Lyon-Centre National de la Recherche Scientifique (CNRS)-Université Grenoble Alpes [2016-2019] (UGA [2016-2019])-École normale supérieure de Lyon (ENS de Lyon)-Université Lumière - Lyon 2 (UL2)-Université Jean Moulin - Lyon 3 (UJML), Université de Lyon-Université de Lyon-Centre National de la Recherche Scientifique (CNRS)-Université Grenoble Alpes [2016-2019] (UGA [2016-2019]), Laboratoire d'Immunologie et Immunopathologie [CHU Poitiers] (CNRS URA 1172), Centre hospitalier universitaire de Poitiers (CHU Poitiers)-Centre National de la Recherche Scientifique (CNRS), Mucosal Immunity, Vaccination, and Biometrics -- Immunité des muqueuses, vaccinations et biothérapies, Centre International de Recherche en Infectiologie (CIRI), École normale supérieure de Lyon (ENS de Lyon)-Université Claude Bernard Lyon 1 (UCBL), Université de Lyon-Université de Lyon-Université Jean Monnet - Saint-Étienne (UJM)-Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS)-École normale supérieure de Lyon (ENS de Lyon)-Université Claude Bernard Lyon 1 (UCBL), Université de Lyon-Université de Lyon-Université Jean Monnet - Saint-Étienne (UJM)-Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS), Transporteurs et Imagerie, Radiothérapie en Oncologie et Mécanismes biologiques des Altérations du Tissu Osseux (TIRO-MATOs - UMR E4320), Service Hospitalier Frédéric Joliot (SHFJ), Université Paris-Saclay-Direction de Recherche Fondamentale (CEA) (DRF (CEA)), Commissariat à l'énergie atomique et aux énergies alternatives (CEA)-Commissariat à l'énergie atomique et aux énergies alternatives (CEA)-Université Paris-Saclay-Direction de Recherche Fondamentale (CEA) (DRF (CEA)), Commissariat à l'énergie atomique et aux énergies alternatives (CEA)-Commissariat à l'énergie atomique et aux énergies alternatives (CEA)-UMR E4320 (TIRO-MATOs), COMUE Université Côte d'Azur (2015-2019) (COMUE UCA)-COMUE Université Côte d'Azur (2015-2019) (COMUE UCA)-Commissariat à l'énergie atomique et aux énergies alternatives (CEA)-Université Côte d'Azur (UCA)-Université Nice Sophia Antipolis (1965 - 2019) (UNS), COMUE Université Côte d'Azur (2015-2019) (COMUE UCA)-COMUE Université Côte d'Azur (2015-2019) (COMUE UCA)-Commissariat à l'énergie atomique et aux énergies alternatives (CEA)-Université Côte d'Azur (UCA), Nestlé Institute of Health Sciences SA [Lausanne, Switzerland], Institut de Recherches SERVIER (IRS), GALDERMA R&D, Galderma Recherche et Développement [Biot, France] (Galderma R&D), Virologie humaine, École normale supérieure de Lyon (ENS de Lyon)-IFR128-Institut National de la Santé et de la Recherche Médicale (INSERM), Université Nice Sophia Antipolis (... - 2019) (UNS), École normale supérieure - Lyon (ENS Lyon)-Université Lumière - Lyon 2 (UL2)-Université Jean Moulin - Lyon 3 (UJML), Université de Lyon-Université de Lyon-Centre National de la Recherche Scientifique (CNRS)-Université Grenoble Alpes [2016-2019] (UGA [2016-2019])-École normale supérieure - Lyon (ENS Lyon)-Université Lumière - Lyon 2 (UL2)-Université Jean Moulin - Lyon 3 (UJML), Centre International de Recherche en Infectiologie - UMR (CIRI), Institut National de la Santé et de la Recherche Médicale (INSERM)-École normale supérieure - Lyon (ENS Lyon)-Université Claude Bernard Lyon 1 (UCBL), Université de Lyon-Université de Lyon-Centre National de la Recherche Scientifique (CNRS)-Institut National de la Santé et de la Recherche Médicale (INSERM)-École normale supérieure - Lyon (ENS Lyon)-Université Claude Bernard Lyon 1 (UCBL), Université de Lyon-Université de Lyon-Centre National de la Recherche Scientifique (CNRS), UMR E4320 (TIRO-MATOs), COMUE Université Côte d'Azur (2015-2019) (COMUE UCA)-COMUE Université Côte d'Azur (2015-2019) (COMUE UCA)-Commissariat à l'énergie atomique et aux énergies alternatives (CEA)-Université Côte d'Azur (UCA)-Université Nice Sophia Antipolis (... - 2019) (UNS), COMUE Université Côte d'Azur (2015-2019) (COMUE UCA)-COMUE Université Côte d'Azur (2015-2019) (COMUE UCA)-Commissariat à l'énergie atomique et aux énergies alternatives (CEA)-Université Côte d'Azur (UCA)-Service Hospitalier Frédéric Joliot (SHFJ), Direction de Recherche Fondamentale (CEA) (DRF (CEA)), Commissariat à l'énergie atomique et aux énergies alternatives (CEA)-Commissariat à l'énergie atomique et aux énergies alternatives (CEA)-Université Paris-Saclay, École normale supérieure - Lyon (ENS Lyon)-IFR128-Institut National de la Santé et de la Recherche Médicale (INSERM)
المصدر: ChemMedChem
ChemMedChem, 2018, 13 (4), pp.321-337. ⟨10.1002/cmdc.201700758⟩
ChemMedChem, Wiley-VCH Verlag, 2018, 13 (4), pp.321-337. ⟨10.1002/cmdc.201700758⟩مصطلحات موضوعية: 0301 basic medicine, Keratinocytes, Administration, Topical, [SDV]Life Sciences [q-bio], Retinoic acid, Drug Evaluation, Preclinical, Pharmacology, 01 natural sciences, Biochemistry, Interleukin-23, chemistry.chemical_compound, Mice, Drug Discovery, heterocyclic compounds, General Pharmacology, Toxicology and Pharmaceutics, ComputingMilieux_MISCELLANEOUS, Orphan receptor, Mice, Inbred BALB C, Sulfonamides, Interleukin-17, Nuclear Receptor Subfamily 1, Group F, Member 3, 3. Good health, Molecular Medicine, medicine.symptom, Drug Inverse Agonism, Inflammation, Topical treatment, Skin Diseases, 03 medical and health sciences, Inhibitory Concentration 50, Structure-Activity Relationship, In vivo, Psoriasis, medicine, Inverse agonist, Animals, Humans, [CHIM]Chemical Sciences, 010405 organic chemistry, business.industry, Organic Chemistry, medicine.disease, 0104 chemical sciences, Disease Models, Animal, 030104 developmental biology, chemistry, Mouse skin, Th17 Cells, business
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12Academic Journal
المؤلفون: Pierre Matthieu Joubert, Thomas Marie Gabriel Desmazières, Jean-François Fournier de la Pommeraye, René Lecesve
المساهمون: Librairie Administrative P. Dupont
المصدر: Archives parlementaires 24(1):444
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13
المؤلفون: Joel Robichaud, Nicolas Morin, Sébastien Gagné, Michel Belley, Lianhai Li, Genevieve Lavallee, Geoffrey K. Tranmer, Yves Gareau, Erin F. Mulrooney, W. Cameron Black, Stacia Kargman, Jean-François Lévesque, Joseph A. Mancini, Jacques Yves Gauthier, Jean-François Fournier, Denis Deschenes, Jin Wu, Martine Hamel, Zhaoyin Wang, Michel Therien, Martin Henault, Yaël Mamane, Huda Hyjazie
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:2836-2839
مصطلحات موضوعية: Pan troglodytes, Stereochemistry, Carboxylic acid, Clinical Biochemistry, Carboxylic Acids, Glucuronidation, Pharmaceutical Science, Naphthalenes, Binding, Competitive, Biochemistry, Chemical synthesis, Uridine Diphosphate, Mice, Structure-Activity Relationship, Pharmacokinetics, Drug Discovery, Purinergic P2 Receptor Antagonists, Animals, Structure–activity relationship, Molecular Biology, chemistry.chemical_classification, Molecular Structure, Receptors, Purinergic P2, Chemistry, Organic Chemistry, Antagonist, Bioavailability, Competitive antagonist, Receptors, Purinergic P2Y, Molecular Medicine, Protein Binding
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14
المؤلفون: Jean-François Fournier
المصدر: French Forum. 36:79-96
مصطلحات موضوعية: Literature and Literary Theory, Visual Arts and Performing Arts
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15
المؤلفون: Jean-François Fournier
المصدر: Dix-Neuf. 12:25-36
مصطلحات موضوعية: Cultural Studies, Linguistics and Language, Literature and Literary Theory, Music, Language and Linguistics
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16
المؤلفون: Jean-François Fournier, André B. Charette, Simon Mathieu
المصدر: Synlett. :1779-1782
مصطلحات موضوعية: Cyclopropanation, Potassium, Organic Chemistry, chemistry.chemical_element, General Medicine, Zinc, Allylic alcohol, Medicinal chemistry, Cycloaddition, chemistry, Organic chemistry, Boron, Carbenoid, Sequence (medicine)
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17
المؤلفون: Jean-François Fournier
المصدر: Symposium: A Quarterly Journal in Modern Literatures. 65:231-233
مصطلحات موضوعية: Literature and Literary Theory
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18
المؤلفون: Sébastien Gagné, Joseph A. Mancini, W. Cameron Black, Jean-François Lévesque, Martine Hamel, Yongxin Han, Jin Wu, Erin F. Mulrooney, Jacques Yves Gauthier, Joel Robichaud, Martin Henault, Stacia Kargman, Nicolas Morin, Yaël Mamane, Jean-François Fournier
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:4366-4368
مصطلحات موضوعية: Clinical Biochemistry, Serum albumin, Biological Availability, Pharmaceutical Science, Plasma protein binding, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Drug Discovery, Purinergic P2 Receptor Antagonists, medicine, Humans, Prodrugs, Molecular Biology, biology, Receptors, Purinergic P2, Chemistry, Ligand binding assay, Organic Chemistry, Prodrug, Human serum albumin, Combinatorial chemistry, Bioavailability, Microsomes, Liver, biology.protein, Molecular Medicine, Lead compound, Protein Binding, medicine.drug
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19
المصدر: Organic Letters. 7:2703-2705
مصطلحات موضوعية: Lactones, Molecular Structure, Chemistry, Computational chemistry, Simple (abstract algebra), Organic Chemistry, Diastereomer, Stereoisomerism, Physical and Theoretical Chemistry, Biochemistry, Catalysis, Methylomuralide
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20eBook