-
1
المؤلفون: Jeffrey H. Hager, Nicholas D. Smith, Tadimeti S. Rao, Stewart A. Noble, Andrew K. Shiau, Jerry Muhammad, Robert L. Davis, James W. Malecha, Alan Saven, Brandon M. Wiley, Sara J. Dozier, Timothy Z. Hoffman, Elena L. Milkova, John V. Anzola, Yan Wang, Carol Trotter, Céline Bonnefous, David A. Jenkins, Joseph E. Payne, Paul L. Wash, Tami Annable, Phan-Manh Nguyen, Xin Guo, Kent T. Symons, Christian A. Hassig
-
2
المؤلفون: Jeffrey H. Hager, Nicholas D. Smith, Tadimeti S. Rao, Stewart A. Noble, Andrew K. Shiau, Jerry Muhammad, Robert L. Davis, James W. Malecha, Alan Saven, Brandon M. Wiley, Sara J. Dozier, Timothy Z. Hoffman, Elena L. Milkova, John V. Anzola, Yan Wang, Carol Trotter, Céline Bonnefous, David A. Jenkins, Joseph E. Payne, Paul L. Wash, Tami Annable, Phan-Manh Nguyen, Xin Guo, Kent T. Symons, Christian A. Hassig
-
3
المؤلفون: Jeffrey H. Hager, Nicholas D. Smith, Tadimeti S. Rao, Stewart A. Noble, Andrew K. Shiau, Jerry Muhammad, Robert L. Davis, James W. Malecha, Alan Saven, Brandon M. Wiley, Sara J. Dozier, Timothy Z. Hoffman, Elena L. Milkova, John V. Anzola, Yan Wang, Carol Trotter, Céline Bonnefous, David A. Jenkins, Joseph E. Payne, Paul L. Wash, Tami Annable, Phan-Manh Nguyen, Xin Guo, Kent T. Symons, Christian A. Hassig
-
4
المؤلفون: Jeffrey H. Hager, Nicholas D. Smith, Tadimeti S. Rao, Stewart A. Noble, Andrew K. Shiau, Jerry Muhammad, Robert L. Davis, James W. Malecha, Alan Saven, Brandon M. Wiley, Sara J. Dozier, Timothy Z. Hoffman, Elena L. Milkova, John V. Anzola, Yan Wang, Carol Trotter, Céline Bonnefous, David A. Jenkins, Joseph E. Payne, Paul L. Wash, Tami Annable, Phan-Manh Nguyen, Xin Guo, Kent T. Symons, Christian A. Hassig
-
5
المؤلفون: James W. Malecha, Christina N. Steininger, Melanie L. Williams, Kristen E. Shannon, Thomas Rogers, Bryan H. Landis, Tiffany Duffin, Srinivasan Nagarajan, Pegg Jodi Ann, Hwang-Fun Lu, Rico Joseph G, Maureen A. Nickols, Jun Zhu, Sandra K. Freeman, V. Wayne Engleman, David W. Griggs, G. Alan Nickols, Jeffery L. Keene, Devadas Balekudru, Debra M. Meyer, Marisa M. Westlin, Larry Miller, Laura D. Marrufo, Nawasa F. Green, Melissa K. Lantz, Mark A. Russell, Peter G. Ruminski, Mary Beth Finn, H. Peter Kleine, Joe T. Collins
المصدر: Bioorganic & Medicinal Chemistry. 15:3783-3800
مصطلحات موضوعية: chemistry.chemical_classification, Dipeptide, biology, Chemistry, Cell adhesion molecule, Stereochemistry, Angiogenesis, Organic Chemistry, Clinical Biochemistry, Integrin, Pharmaceutical Science, Peptide, Tripeptide, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Drug Discovery, biology.protein, Molecular Medicine, Vitronectin, Molecular Biology
-
6
المؤلفون: Walter G. Smith, Suzanne H Kim, Doreen Villani-Price, Matthew W Mahoney, Nayereh S Ghoreishi-Haack, Helen Y. Chen, Thomas D. Penning, Stella Siu-Tzyy Yu, James W. Malecha, Leslie J Askonas, Chi-Dean Liang, Elizabeth I Harding, E.Yvonne Pyla, Maureen K Highkin, James K. Gierse, Julie M Miyashiro, Mark A Russell, James F Kachur, Chen Barbara B
المصدر: Journal of Medicinal Chemistry. 45:3482-3490
مصطلحات موضوعية: Epoxide Hydrolases, chemistry.chemical_classification, biology, Stereochemistry, Administration, Oral, Leukotriene A4, Chemical synthesis, Proinflammatory cytokine, Leukotriene-A4 hydrolase, Mice, Structure-Activity Relationship, Enzyme, chemistry, Enzyme inhibitor, In vivo, Drug Discovery, Hydrolase, beta-Alanine, biology.protein, Animals, Humans, Molecular Medicine, Structure–activity relationship, Enzyme Inhibitors
-
7
المؤلفون: James A. Hendrix, Shun ichiro Hachiya, Kiyoshi Horita, Anthony G. M. Barrett, James W. Malecha, Andrew Vansickle, Oren P. Anderson, Christopher J. Parkinson, Jeremy J. Edmunds
المصدر: Canadian Journal of Chemistry. 79:1562-1592
مصطلحات موضوعية: chemistry.chemical_compound, Aldol reaction, Chemistry, Stereochemistry, Metabolite, Organic Chemistry, Total synthesis, Organic chemistry, Phosphatase inhibitor, General Chemistry, Calyculin A, Catalysis, Calyculin
-
8
المؤلفون: Doreen Villani-Price, Suzanne H Kim, Walter G. Smith, Leslie J Askonas, Elizabeth I Harding, Maureen K Highkin, Thomas D. Penning, Alan F. Gasiecki, Nayereh S Ghoreishi-Haack, Nizal S Chandrakumar, E.Yvonne Pyla, Bipin N Desai, James F Kachur, Mark A Russell, Stevan W Djuric, James W. Malecha, James K. Gierse, Julie M Miyashiro
المصدر: Bioorganic & Medicinal Chemistry Letters. 13:1137-1139
مصطلحات موضوعية: Imidazopyridine, Pyridines, Clinical Biochemistry, Pharmaceutical Science, Purine analogue, In Vitro Techniques, Biochemistry, Chemical synthesis, Leukotriene-A4 hydrolase, Mice, Structure-Activity Relationship, Heterocyclic Compounds, Drug Discovery, Animals, Humans, Structure–activity relationship, Enzyme Inhibitors, Purine metabolism, Molecular Biology, Epoxide Hydrolases, biology, Chemistry, Organic Chemistry, Recombinant Proteins, stomatognathic diseases, Purines, Enzyme inhibitor, biology.protein, Molecular Medicine, Indicators and Reagents, Ex vivo
-
9
المؤلفون: Jeremy J. Edmunds, Anthony G. M. Barrett, James A. Hendrix, Christopher J. Parkinson, James W. Malecha
المصدر: ChemInform. 23
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Stereochemistry, Amide, Diisopinocampheylborane, General Medicine, Alkylation, Calyculin A, Unit (ring theory), Calyculin, Oxazole
-
10
المؤلفون: James W. Malecha, Anthony G. M. Barrett
المصدر: ChemInform. 23
مصطلحات موضوعية: chemistry.chemical_compound, Chemistry, Reagent, Diisopinocampheylborane, Organic chemistry, Stereoselectivity, General Medicine, Vicinal
-
11
المؤلفون: Kiyoshi Horita, Anthony G. M. Barrett, Andrew Vansickle, James A. Hendrix, Jeremy J. Edmunds, Christopher J. Parkinson, Oren P. Anderson, James W. Malecha, Shun ichiro Hachiya
المصدر: ChemInform. 33
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Stereochemistry, Metabolite, Total synthesis, General Medicine, Calyculin A
-
12
المؤلفون: Avery R. Coyle, Mark R. Hellberg, James W. Malecha, Daniel A. Gamache, Andrew K. Shiau, Guy Oshiro, John V. Anzola, John C. Liao, Lena M. Staszewski, C. Beauregard, Jennifer N. Hsien, Jasmine Chen, John M. Yanni, Stewart A. Noble, Julia M. Lerch, Steven P. Govek, David J. Thomas
المصدر: Bioorganicmedicinal chemistry letters. 20(9)
مصطلحات موضوعية: Clinical Biochemistry, Anti-Inflammatory Agents, Pharmaceutical Science, Inflammation, Pharmacology, Biochemistry, chemistry.chemical_compound, Coumarins, Drug Discovery, medicine, Animals, Tear secretion, Computer Simulation, PDE4 Inhibitors, 4-Aminopyridine, Molecular Biology, Binding Sites, Organic Chemistry, Water, Coumarin, Cyclic nucleotide phosphodiesterases, eye diseases, Cyclic Nucleotide Phosphodiesterases, Type 4, Rats, Disease Models, Animal, Water soluble, chemistry, Rabbit model, Molecular Medicine, Water chemistry, Dry Eye Syndromes, sense organs, Phosphodiesterase 4 Inhibitors, Rabbits, medicine.symptom
-
13
المؤلفون: Timothy Z. Hoffman, Tami Annable, Michael Sertic, Paul L. Wash, Celine Bonnefous, Jeffrey H. Hager, Kent T. Symons, Stewart A. Noble, James W. Malecha, Charles Lawrence, Christian A. Hassig, Nicholas D. Smith, Xin Guo, Brandon M. Wiley, Kevin D. Lustig, Phan-Manh Nguyen
المصدر: Bioorganicmedicinal chemistry letters. 18(24)
مصطلحات موضوعية: medicine.drug_class, Chemistry, Pharmaceutical, Clinical Biochemistry, Pharmaceutical Science, Antineoplastic Agents, Biochemistry, Structure-Activity Relationship, In vivo, Neoplasms, Drug Discovery, medicine, Humans, Prodrugs, Enzyme Inhibitors, Molecular Biology, Chelating Agents, chemistry.chemical_classification, Histone deacetylase 5, biology, Chemistry, Histone deacetylase 2, HDAC11, Organic Chemistry, Histone deacetylase inhibitor, Ketones, Histone Deacetylase Inhibitors, Zinc, Enzyme, Models, Chemical, Enzyme inhibitor, Drug Design, biology.protein, Cancer research, Molecular Medicine, Histone deacetylase, Drug Screening Assays, Antitumor, HeLa Cells
-
14
المؤلفون: Tadimeti S. Rao, Christian A. Hassig, Timothy Z. Hoffman, Celine Bonnefous, James W. Malecha, Andrew K. Shiau, Xin Guo, Kent T. Symons, Paul L. Wash, Tami Annable, Jeffrey H. Hager, Nicholas D. Smith, Joseph E. Payne, Phan-Manh Nguyen, Stewart A. Noble
المصدر: Bioorganicmedicinal chemistry letters. 18(23)
مصطلحات موضوعية: medicine.drug_class, Pyridines, Clinical Biochemistry, Pharmaceutical Science, Mice, Nude, Antineoplastic Agents, Biochemistry, Histone H3, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, In vivo, Cell Line, Tumor, Drug Discovery, medicine, Cytotoxic T cell, Animals, Humans, Prodrugs, Enzyme Inhibitors, Cytotoxicity, Molecular Biology, Sulfonamides, biology, Molecular Structure, Chemistry, Organic Chemistry, Histone deacetylase inhibitor, HCT116 Cells, Xenograft Model Antitumor Assays, Histone Deacetylase Inhibitors, Cell culture, Enzyme inhibitor, Cancer research, biology.protein, Molecular Medicine, Histone deacetylase, Drug Screening Assays, Antitumor
-
15
المؤلفون: Timothy Z. Hoffman, Celine Bonnefous, Tadimeti S. Rao, Jerry Muhammad, James W. Malecha, Paul L. Wash, Christian A. Hassig, Nicholas D. Smith, Kent T. Symons, Xin Guo, John V. Anzola, Elena L. Milkova, Alan Saven, Tami Annable, Jeffrey H. Hager, Andrew K. Shiau, Stewart A. Noble, David A. Jenkins, Carol Trotter, Joseph E. Payne, Yan Wang, Phan-Manh Nguyen, Brandon M. Wiley, Sara J. Dozier, Robert L. Davis
المصدر: Molecular cancer therapeutics. 7(5)
مصطلحات موضوعية: Male, Cancer Research, medicine.drug_class, Pyridines, Cell, Mice, Nude, Antineoplastic Agents, Biology, Pharmacology, HeLa, Inhibitory Concentration 50, Mice, In vivo, Cell Line, Tumor, medicine, Animals, Humans, Enzyme Inhibitors, Histone H3 acetylation, Vorinostat, Mice, Inbred BALB C, Sulfonamides, Histone deacetylase inhibitor, Prostatic Neoplasms, biology.organism_classification, Xenograft Model Antitumor Assays, Histone Deacetylase Inhibitors, medicine.anatomical_structure, Oncology, Cell culture, Female, Histone deacetylase, Drug Screening Assays, Antitumor, Colorectal Neoplasms, medicine.drug
-
16
المؤلفون: Srinivasan R, Nagarajan, Balekudru, Devadas, James W, Malecha, Hwang-Fun, Lu, Peter G, Ruminski, Joseph G, Rico, Thomas E, Rogers, Laura D, Marrufo, Joe T, Collins, H Peter, Kleine, Melissa K, Lantz, Jun, Zhu, Nawasa F, Green, Mark A, Russell, Bryan H, Landis, Lawrence M, Miller, Debra M, Meyer, Tiffany D, Duffin, V Wayne, Engleman, Mary B, Finn, Sandra K, Freeman, David W, Griggs, Melanie L, Williams, Maureen A, Nickols, Jodi A, Pegg, Kristen E, Shannon, Christina, Steininger, Marisa M, Westlin, G Alan, Nickols, Jeffery L, Keene
المصدر: Bioorganicmedicinal chemistry. 15(11)
مصطلحات موضوعية: Skin Neoplasms, Molecular Mimicry, Antineoplastic Agents, Mice, Inbred Strains, Integrin alphaVbeta3, Xenograft Model Antitumor Assays, Mice, Isomerism, Colonic Neoplasms, Hypercalcemia, Animals, Amino Acids, Melanoma, Oligopeptides
-
17
المؤلفون: Kristen E. Shannon, Barbara B. Chen, James W. Malecha, Stephen H Docter, G. Allen Nickols, Thomas D. Penning, Marisa M. Westlin, Glen J. Gesicki, Chi-Dean Liang, Helen Y. Chen, David J. Edwards, Melanie L. Hanneke, Bipin N. Desai, Stella S. Yu, Sandra K. Freeman, Mark A. Russell, V. Wayne Engleman
المصدر: Bioorganicmedicinal chemistry letters. 14(6)
مصطلحات موضوعية: chemistry.chemical_classification, Chemistry, Peptidomimetic, Stereochemistry, Carboxylic acid, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Alpha (ethology), Stereoisomerism, Integrin alphaVbeta3, Biochemistry, Chemical synthesis, Cinnamic acid, chemistry.chemical_compound, Cinnamates, Drug Discovery, Molecular Medicine, Humans, Beta (finance), Selectivity, Molecular Biology
-
18
المؤلفون: James W. Malecha, Anthony G. M. Barrett
المصدر: The Journal of Organic Chemistry. 56:5243-5245
مصطلحات موضوعية: chemistry.chemical_classification, chemistry.chemical_compound, chemistry, Reagent, Organic Chemistry, Organic chemistry, Diisopinocampheylborane, Stereoselectivity, Aldehyde, Vicinal
-
19Academic Journal
المؤلفون: Christian A Hassig, Kent T Symons, Xin Guo, Phan-Manh Nguyen, Tami Annable, Paul L Wash, Joseph E Payne, David A Jenkins, Cé Line Bonnefous, Carol Trotter, Yan Wang, John V Anzola, Elena L Milkova, Timothy Z Hoffman, Sara J Dozier, Brandon M Wiley, Alan Saven, James W Malecha, Robert L Davis, Jerry Muhammad, Andrew K Shiau, Stewart A Noble, Tadimeti S Rao, Nicholas D Smith, Jeffrey H Hager
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.1035.1289; http://mct.aacrjournals.org/content/molcanther/7/5/1054.full.pdf
-
20
المؤلفون: Karen Seibert, AndersonGD, John J. Talley, Susan A. Gregory, Matthew J. Graneto, Yan Y. Zhang, James W. Malecha, Len F. Lee, Stella S. Yu, Stephen H. Docter, Bertenshaw, P. C. Isakson, P. W. Collins, E. G. Burton, J. N. Cogburn, Jeffery S. Carter, A. W. Veenhuizen, Carol M. Koboldt, T. D. Penning, Julie M. Miyashiro, D. J. Rogier, W E Perkins, Roland S. Rogers
المصدر: Journal of medicinal chemistry. 40(9)
مصطلحات موضوعية: Male, Magnetic Resonance Spectroscopy, Stereochemistry, Pyrazole, Pharmacology, Carrageenan, Prostaglandin-endoperoxide synthase 2, Arthritis, Rheumatoid, Rats, Sprague-Dawley, chemistry.chemical_compound, Structure-Activity Relationship, Pharmacokinetics, In vivo, Drug Discovery, Osteoarthritis, medicine, Animals, Cyclooxygenase Inhibitors, Sulfonamides, Trifluoromethyl, biology, Cyclooxygenase 2 Inhibitors, Molecular Structure, Membrane Proteins, Arthritis, Experimental, In vitro, Rats, Isoenzymes, chemistry, Celecoxib, Cyclooxygenase 2, Hyperalgesia, Prostaglandin-Endoperoxide Synthases, Rats, Inbred Lew, biology.protein, Cyclooxygenase 1, Molecular Medicine, Pyrazoles, Cyclooxygenase, medicine.drug