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1Academic Journal
المؤلفون: J Matthew Hutzler, Larissa M Balogh, Michael Zientek, Vikas Kumar, Timothy S Tracy, St Louis Development, J M H Labs, V K, La Jolla Labs, M Z, L M B, Dr J Matthew Hutzler
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.1046.7819; http://dmd.aspetjournals.org/content/dmd/early/2008/10/06/dmd.108.023358.full.pdf
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2
المؤلفون: Taysir Chamem, Xiaochun Zhu, Todd Hieronymus, Richard D. Burton, J. Matthew Hutzler, Shelby Anderson, David Heim
المصدر: Drug Metabolism and Disposition. 46:1617-1625
مصطلحات موضوعية: Pharmacology, Taurine, biology, Metabolite, Pharmaceutical Science, Cytochrome P450, Metabolism, 030226 pharmacology & pharmacy, 03 medical and health sciences, chemistry.chemical_compound, Metabolic pathway, 0302 clinical medicine, medicine.anatomical_structure, Biochemistry, chemistry, In vivo, 030220 oncology & carcinogenesis, Hepatocyte, biology.protein, medicine, Aldehyde oxidase
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3
المؤلفون: John D. Huber, J. Matthew Hutzler, Doris Riether, Tom Simpson, Alan Olague, Asitha Abeywardane, Renee Zindell, John Broadwater, Peter Allen Nemoto, Hidenori Takahashi, Todd Bosanac, Yunlong Zhang, Alessandra Bartolozzi, Zhidong Chen, Lifen Wu
المصدر: Bioorganic & Medicinal Chemistry Letters. 27:4652-4659
مصطلحات موضوعية: Male, 0301 basic medicine, ERG1 Potassium Channel, 5-Lipoxygenase-Activating Proteins, Clinical Biochemistry, hERG, Drug Evaluation, Preclinical, Pharmaceutical Science, Oxadiazole, macromolecular substances, 01 natural sciences, Biochemistry, Rats, Sprague-Dawley, Inhibitory Concentration 50, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, In vivo, Drug Discovery, Animals, Humans, Structure–activity relationship, Rats, Wistar, Molecular Biology, Oxadiazoles, biology, Chemistry, Organic Chemistry, Combinatorial chemistry, Rats, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 030104 developmental biology, Solubility, 5-Lipoxygenase-Activating Protein Inhibitors, Microsomes, Liver, biology.protein, Molecular Medicine, Functional activity, Half-Life
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4
المؤلفون: J. Matthew Hutzler, Rachel D. Crouch, J. Scott Daniels
المصدر: Xenobiotica. 48:219-231
مصطلحات موضوعية: Male, Guanine, Swine, Health, Toxicology and Mutagenesis, Guinea Pigs, Biology, Toxicology, Guanidines, 030226 pharmacology & pharmacy, Biochemistry, Article, Rats, Sprague-Dawley, Guinea pig, Mice, 03 medical and health sciences, 0302 clinical medicine, Species Specificity, Pharmacokinetics, In vivo, Acetamides, Animals, Humans, Aldehyde oxidase, Pharmacology, General Medicine, Triazoles, Macaca mulatta, In vitro, Aldehyde Oxidase, Pyridazines, SSS, Macaca fascicularis, Pyrimidines, Liver, 030220 oncology & carcinogenesis, Pyrazoles, Swine, Miniature, Female, Allometry, Drug metabolism
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5Academic Journal
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.1036.7675; http://dmd.aspetjournals.org/content/dmd/31/7/878.full.pdf
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6
المصدر: The AAPS Journal. 18:1391-1405
مصطلحات موضوعية: Glucuronosyltransferase, Metabolic Clearance Rate, Pharmaceutical Science, Pharmacology, 030226 pharmacology & pharmacy, Article, Carboxylesterase, 03 medical and health sciences, 0302 clinical medicine, In vivo, Animals, Humans, Aldehyde oxidase, chemistry.chemical_classification, biology, Metabolism, Aldehyde Oxidase, Metabolic pathway, Phenotype, Enzyme, Pharmaceutical Preparations, chemistry, Biochemistry, 030220 oncology & carcinogenesis, biology.protein, Microsome, Forecasting
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7
المؤلفون: Michael Huskin, Jennifer Wood, Nicholas Ingram, J. Matthew Hutzler, Sherri Smith, Christopher Dishinger
المصدر: The AAPS journal. 21(1)
مصطلحات موضوعية: Drug, endocrine system, media_common.quotation_subject, Pharmaceutical Science, Orosomucoid, Plasma protein binding, 030226 pharmacology & pharmacy, Vial, 03 medical and health sciences, chemistry.chemical_compound, Plasma, 0302 clinical medicine, Plasticizers, Diethylhexyl Phthalate, Humans, Tissue Distribution, media_common, Blood Specimen Collection, Chromatography, biology, Chemistry, Phthalate, Plasticizer, Blood collection, In vitro, Pharmaceutical Preparations, 030220 oncology & carcinogenesis, biology.protein, Protein Binding
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8
المؤلفون: Richard D, Burton, Todd, Hieronymus, Taysir, Chamem, David, Heim, Shelby, Anderson, Xiaochun, Zhu, J Matthew, Hutzler
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 46(11)
مصطلحات موضوعية: Cytochrome P-450 Enzyme System, Pharmaceutical Preparations, Metabolic Clearance Rate, Taurine, Glycine, Hepatocytes, Humans, Oxidation-Reduction, Biotransformation, Cells, Cultured, Metabolic Networks and Pathways
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9
المؤلفون: Adam Flegg, Tina Morwick, Ho Yin Lo, Todd Bosanac, Weimin Liu, Valentina Berger, Steven Kerr, Stéphane De Lombaert, Paige Erin Mahaney, Ralph Binetti, John Broadwater, Spencer Napier, Alessandra Bartolozzi, Lifen Wu, Hidenori Takahashi, Asitha Abeywardane, Heather Tye, Tazmeen Fadra-Khan, John D. Huber, Adrian Kotey, Ming-Hong Hao, Dines Jonathon Alan, Anil Kumar Padyana, Alan Olague, Michael Garrigou, David S. Thomson, J. Matthew Hutzler, Pui Leng Loke, Renee Zindell, Edward Pack, Zhidong Chen, Rebecca Crux, Thomas Simpson, Rajvee Dave, Doris Riether
المصدر: Journal of Medicinal Chemistry. 58:1669-1690
مصطلحات موضوعية: Models, Molecular, Oxadiazoles, Arachidonate 5-Lipoxygenase, Dose-Response Relationship, Drug, CYP3A4, Stereochemistry, Chemistry, Molecular Conformation, Oxadiazole, 5-Lipoxygenase-Activating Protein Inhibitors, Crystallography, X-Ray, Structure-Activity Relationship, chemistry.chemical_compound, Pharmacokinetics, Acetamides, Drug Discovery, Humans, Molecular Medicine, Lipoxygenase Inhibitors, IC50, Ex vivo, Drug metabolism, Whole blood
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10
المؤلفون: Constance Asher, Diane Wong, J. Matthew Hutzler, Young-Sun Yang, Matthew A. Cerny, Kyle E. Gilpin, Kosea Frederick
المصدر: Drug Metabolism and Disposition. 42:1751-1760
مصطلحات موضوعية: medicine.medical_specialty, Metabolite, Biological Availability, Pharmaceutical Science, Pharmacology, Biology, Excretion, chemistry.chemical_compound, Cytosol, Dogs, Pharmacokinetics, Oral administration, Internal medicine, medicine, Animals, Humans, Toxicokinetics, Organic Chemicals, Aldehyde oxidase, Metabolism, Macaca mulatta, Rats, Bioavailability, Aldehyde Oxidase, ErbB Receptors, Macaca fascicularis, Endocrinology, Liver, chemistry, Raloxifene Hydrochloride, Hepatocytes
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11
المؤلفون: Jeffrey M. Weber, Lori Bunkowfst, Brian Staton, J. Matthew Hutzler
المصدر: Drug Metabolism and Pharmacokinetics. 33:S68-S69
مصطلحات موضوعية: Pharmacology, Chromatography, Human liver, Chemistry, Lc ms ms, Microsome, Pharmaceutical Science, Pharmacology (medical), Selectivity
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12
المصدر: Drug Metabolism and Disposition. 40:1336-1344
مصطلحات موضوعية: CYP3A, Cell, Pharmaceutical Science, Biology, Pharmacology, Troleandomycin, Clarithromycin, medicine, Cytochrome P-450 CYP3A, Humans, Drug Interactions, Cells, Cultured, Cryopreservation, Mibefradil, In vitro, Kinetics, medicine.anatomical_structure, Verapamil, Hepatocytes, Microsomes, Liver, Microsome, Cytochrome P-450 CYP3A Inhibitors, medicine.drug
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13
المصدر: Drug Metabolism and Disposition. 38:1113-1121
مصطلحات موضوعية: Male, Metabolite, Drug Evaluation, Preclinical, Pharmaceutical Science, In Vitro Techniques, Sulfides, Pharmacology, Models, Biological, Rats, Sprague-Dawley, chemistry.chemical_compound, Dogs, Pharmacokinetics, In vivo, Animals, Cytochrome P-450 Enzyme Inhibitors, Humans, Drug Interactions, Lipoxygenase Inhibitors, Enzyme Inhibitors, biology, CYP3A4, Imidazoles, Cytochrome P450, In vitro, Genetic translation, Rats, Kinetics, chemistry, Microsomes, Liver, biology.protein, Microsome
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14
المصدر: Drug Metabolism and Disposition. 37:59-65
مصطلحات موضوعية: Stereochemistry, Kinetics, Ticrynafen, Suprofen, Pharmaceutical Science, Substrate Specificity, Hydroxylation, chemistry.chemical_compound, Tandem Mass Spectrometry, medicine, Carboxylate, Enzyme Inhibitors, Diuretics, Cytochrome P-450 CYP2C9, Pharmacology, chemistry.chemical_classification, biology, Anti-Inflammatory Agents, Non-Steroidal, Active site, Substrate (chemistry), Articles, Enzyme, chemistry, Tienilic acid, biology.protein, Spectrophotometry, Ultraviolet, Aryl Hydrocarbon Hydroxylases, Chromatography, Liquid, medicine.drug
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15
المؤلفون: Michael Zientek, J. Matthew Hutzler
المصدر: New Horizons in Predictive Drug Metabolism and Pharmacokinetics ISBN: 9781849738286
مصطلحات موضوعية: chemistry.chemical_classification, Metabolic pathway, Enzyme, chemistry, biology, Biochemistry, Oxidative enzyme, biology.protein, Cytochrome P450, Metabolism, Monooxygenase, Aldehyde oxidase, Drug metabolism
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16
المؤلفون: Barbara J. Ring, J. Matthew Hutzler, Shelby Anderson
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 43(12)
مصطلحات موضوعية: Drug, Metabolic Clearance Rate, Metabolite, media_common.quotation_subject, Pharmaceutical Science, Biology, Pharmacology, chemistry.chemical_compound, Animals, Humans, Cells, Cultured, media_common, chemistry.chemical_classification, In vitro toxicology, Metabolism, In vitro, Coculture Techniques, Enzyme, chemistry, Biochemistry, Pharmaceutical Preparations, Inactivation, Metabolic, Microsome, Hepatocytes, Microsomes, Liver, Drug metabolism
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17
المؤلفون: Rick C. Steenwyk, J. Matthew Hutzler, Jim Sams, Gary Siuzdak, Zhouxin Shen
المصدر: Rapid Communications in Mass Spectrometry. 20:3717-3722
مصطلحات موضوعية: Silicon, Spectrometry, Mass, Electrospray Ionization, Metabolic Clearance Rate, Midazolam, Kinetics, Desorption/ionization on silicon, Hydroxylation, Mass spectrometry, Analytical Chemistry, chemistry.chemical_compound, Pharmacokinetics, Desorption, Animals, Humans, Cells, Cultured, Spectroscopy, Detection limit, Chromatography, Organic Chemistry, Rats, Atmospheric Pressure, chemistry, Microsomes, Liver, Microsome
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18
المصدر: Archives of Biochemistry and Biophysics. 438:21-28
مصطلحات موضوعية: Cytochrome, Stereochemistry, Kinetics, Biophysics, Biochemistry, Catalysis, chemistry.chemical_compound, Cytochrome P-450 Enzyme System, Multienzyme Complexes, Cytochrome b5, Cytochrome P-450 CYP3A, Computer Simulation, Molecular Biology, Pyrenes, biology, Chemistry, Active site, Cooperative binding, Substrate (chemistry), Metabolism, Enzyme Activation, Cytochromes b5, Models, Chemical, biology.protein, Pyrene, Oxidation-Reduction
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19
المؤلفون: Stephen C. Strom, Shimin Zhang, Hongbo Cai, Raman Venkataramanan, Catharina Y. W. Ang, Bernard J. Komoroski, J. Matthew Hutzler, Timothy S. Tracy, Yan Yan Cui, Reginald F. Frye, Thomas Lehmann
المصدر: Drug Metabolism and Disposition. 32:512-518
مصطلحات موضوعية: Pharmaceutical Science, Phloroglucinol, Pharmacology, Bridged Bicyclo Compounds, chemistry.chemical_compound, Cytochrome P-450 Enzyme System, Cytochrome P-450 Enzyme Inhibitors, Humans, RNA, Messenger, Enzyme Inhibitors, Enzyme inducer, Cells, Cultured, Dose-Response Relationship, Drug, biology, Terpenes, CYP1A2, Cytochrome P450, Hypericum perforatum, biology.organism_classification, Hypericin, Hyperforin, Biochemistry, chemistry, Enzyme Induction, Hepatocytes, biology.protein, Hypericum
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20
المصدر: Archives of Biochemistry and Biophysics. 417:165-175
مصطلحات موضوعية: Anions, Hydrochloride, Inorganic chemistry, Carbonates, Biophysics, Biochemistry, Medicinal chemistry, Substrate Specificity, chemistry.chemical_compound, medicine, Sulfate, Molecular Biology, biology, Cytochrome P450, Dextromethorphan, Metabolism, Hydrogen-Ion Concentration, Phosphate, Enzyme Activation, Oxygen, Cytochrome P-450 CYP2D6, chemistry, Cumene hydroperoxide, biology.protein, Carbonate, Reactive Oxygen Species, Oxidation-Reduction, medicine.drug