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1Academic Journal
المؤلفون: Erdogan, Fettah (University of Toronto), Gunning, Patrick Thomas (University of Toronto), Orlova, Anna (University of Veterinary Medicine Vienna), Moriggl, Richard (University of Veterinary Medicine Vienna), Herling, Marco (University of Leipzig), Mustjoki, Satu M (University of Helsinki), Valent, Peter (Medical University of Vienna), Israelian, Johan (University of Toronto), de Araujo, Elvin Dominic (University of Toronto), Qadree, Abdul Khawazak (University of Toronto), Radu, Tudor Bogdan (University of Toronto)
المصدر: Journal of Cellular and Molecular Medicine 26(7), 2049-2062 (2022)
مصطلحات موضوعية: Cytokinesmetabolism, ErbB Receptorsmetabolism, Humans, Neoplasmsgenetics, STAT Transcription Factorsgeneticsmetabolism
وصف الملف: application/pdf
Relation: isPartOf:https://phaidra.vetmeduni.ac.at/o:605[Open Access Publications]; https://phaidra.vetmeduni.ac.at/o:1791
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2Academic Journal
المؤلفون: Toutah, Krimo, Nawar, Nabanita, Timonen, Sanna, Sorger, Helena, Raouf, Yasir S., Bukhari, Shazreh, von Jan, Jana, Ianevski, Aleksandr, Gawel, Justyna M., Olaoye, Olasunkanmi O., Geletu, Mulu, Abdeldayem, Ayah, Israelian, Johan, Radu, Tudor B., Sedighi, Abootaleb, Bhatti, Muzaffar N., Hassan, Muhammad Murtaza, Manaswiyoungkul, Pimyupa, Shouksmith, Andrew E., Neubauer, Heidi A., de Araujo, Elvin D., Aittokallio, Tero, Kraemer, Oliver H., Moriggl, Richard, Mustjoki, Satu, Herling, Marco, Gunning, Patrick T.
المساهمون: Computational Systems Medicine, TRIMM - Translational Immunology Research Program, Institute for Molecular Medicine Finland, Helsinki Institute for Information Technology, Tero Aittokallio / Principal Investigator, Bioinformatics, HUS Comprehensive Cancer Center, Department of Clinical Chemistry and Hematology, Clinicum
مصطلحات موضوعية: HISTONE DEACETYLASE INHIBITOR, SUBEROYLANILIDE HYDROXAMIC ACID, ACCURATE DOCKING, BCL-2 INHIBITOR, TUBULIN, RICOLINOSTAT, COMBINATION, EXPRESSION, BORTEZOMIB, MODEL, Cancers
وصف الملف: application/pdf
Relation: The authors would like to thank Ruth Villalonga for her contributions with cytotoxicity assays using NHF, pPF and HUVEC. They would also like to thank Andrew Sedmihradsky and family, who have raised funds, awareness for DMD and generated support for Max's Big Fellowship. Funding: This work was supported by the EU consortia ERAPerMed "JAKSTAT-TARGET" (S.M., H.A.N., M.H., P.T.G.) and the "ERANETPLL" (M.H., R.M.). S.M. was funded by European Research Council (M-IMM project), Academy of Finland, Sigrid Juselius Foundation and the Cancer Foundation Finland. T.A. was funded by the Academy of Finland (grants 310507, 313267, 326238), Cancer Society of Finland, Sigrid Juselius Foundation and Helse Sor-Ost. R.M., H.A.N., and H.S. were supported by the Austrian Science Fund (FWF) (SFBF04707, SFB-F06105). R.M. and H.A.N. were also generously supported by a private cancer metabolism grant donation from Liechtenstein. P.T.G is supported by research grants from NSERC (RGPIN-2014-05767), CIHR (MOP-130424, MOP137036), Canada Research Chair (950-232042), Canadian Cancer Society (703963), Canadian Breast Cancer Foundation (705456), Leukemia and Lymphoma Society of Canada and infrastructure grants from CFI (33536) and the Ontario Research Fund (34876). O.O.O. is supported by an OGS Fellowship. Y.S.R and N.N are supported by grants from Jesse's Journey.; Toutah , K , Nawar , N , Timonen , S , Sorger , H , Raouf , Y S , Bukhari , S , von Jan , J , Ianevski , A , Gawel , J M , Olaoye , O O , Geletu , M , Abdeldayem , A , Israelian , J , Radu , T B , Sedighi , A , Bhatti , M N , Hassan , M M , Manaswiyoungkul , P , Shouksmith , A E , Neubauer , H A , de Araujo , E D , Aittokallio , T , Kraemer , O H , Moriggl , R , Mustjoki , S , Herling , M & Gunning , P T 2021 , ' Development of HDAC Inhibitors Exhibiting Therapeutic Potential in T-Cell Prolymphocytic Leukemia ' , Journal of Medicinal Chemistry , vol. 64 , no. 12 , pp. 8486-8509 . https://doi.org/10.1021/acs.jmedchem.1c00420; ORCID: /0000-0002-8139-5950/work/108068897; ORCID: /0000-0002-0886-9769/work/108069455; ORCID: /0000-0002-7780-482X/work/108071474; ORCID: /0000-0002-0816-8241/work/108071505; http://hdl.handle.net/10138/339824; 029ef40b-9fac-4846-9454-0953b466cff6; 000668340800034
الاتاحة: http://hdl.handle.net/10138/339824
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3Academic Journal
المؤلفون: Erdogan, Fettah, Radu, Tudor Bogdan, Orlova, Anna, Qadree, Abdul Khawazak, de Araujo, Elvin Dominic, Israelian, Johan, Valent, Peter, Mustjoki, Satu M., Herling, Marco, Moriggl, Richard, Gunning, Patrick Thomas
المساهمون: HUS Comprehensive Cancer Center, Department of Clinical Chemistry and Hematology, Clinicum, Digital Precision Cancer Medicine (iCAN), TRIMM - Translational Immunology Research Program, Hematologian yksikkö
مصطلحات موضوعية: blood cancer, breast cancer, colorectal cancers, JAK, STAT pathway in cancers, liver cancers, lung cancer, protein-protein interactions, systems medicine, COLORECTAL-CANCER, DISEASE GENES, HUMAN BREAST, APOPTOSIS, ACTIVATION, MUTATIONS, CELLS, INHIBITION, TUMORS, EGFR, Biomedicine, Biochemistry, cell and molecular biology
وصف الملف: application/pdf
Relation: NSERC, Grant/Award Number: RGPIN-2014-05767; CIHR, Grant/Award Number: MOP-130424 and MOP-137036; Canada Research Chair, Grant/Award Number: 950-232042; Canadian Cancer Society, Grant/Award Number: 703963; Canadian Breast Cancer Foundation, Grant/ Award Number: 705456; CFI, Grant/ Award Number: 33536; Ontario Research Fund, Grant/Award Number: 34876; EU consortia ERAPerMed `JAKSTAT--TARGET'; ERANETPLL; European Research Council; Austrian Science Fund, Grant/Award Number: SFB- -F04707 and SFB--F06105; Erdogan , F , Radu , T B , Orlova , A , Qadree , A K , de Araujo , E D , Israelian , J , Valent , P , Mustjoki , S M , Herling , M , Moriggl , R & Gunning , P T 2022 , ' JAK-STAT core cancer pathway : An integrative cancer interactome analysis ' , Journal of Cellular and Molecular Medicine , vol. 26 , no. 7 , pp. 2049-2062 . https://doi.org/10.1111/jcmm.17228; ORCID: /0000-0002-0816-8241/work/111921364; http://hdl.handle.net/10138/342896; 15527420-f381-4be3-988d-a8e64fa37b30; 000762358800001
الاتاحة: http://hdl.handle.net/10138/342896
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4Academic Journal
المؤلفون: de Araujo, Elvin D., Erdogan, Fettah, Neubauer, Heidi A., Meneksedag-Erol, Deniz, Manaswiyoungkul, Pimyupa, Eram, Mohammad S., Seo, Hyuk-Soo, Qadree, Abdul K., Israelian, Johan, Orlova, Anna, Suske, Tobias, Pham, Ha T. T., Boersma, Auke, Tangermann, Simone, Kenner, Lukas, Rülicke, Thomas, Dong, Aiping, Ravichandran, Manimekalai, Brown, Peter J., Audette, Gerald F., Rauscher, Sarah, Dhe-Paganon, Sirano, Moriggl, Richard, Gunning, Patrick T.
المساهمون: Austrian Science Fund, Gouvernement du Canada | Natural Sciences and Engineering Research Council of Canada, Gouvernement du Canada | Canadian Institutes of Health Research, Canada Research Chairs, Canadian Cancer Society Research Institute, Canadian Breast Cancer Foundation, Canada Foundation for Innovation, Ontario Research Foundation
المصدر: Nature Communications ; volume 10, issue 1 ; ISSN 2041-1723
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5Academic Journal
المؤلفون: Erdogan, Fettah, Qadree, Abdul K., Radu, Tudor B., Orlova, Anna, de Araujo, Elvin D., Israelian, Johan, Valent, Peter, Mustjoki, Satu M., Herling, Marco, Moriggl, Richard, Gunning, Patrick T.
المساهمون: Canadian Cancer Society, Ontario Research Foundation, Sigrid Juséliuksen Säätiö, European Commission, Canadian Institutes of Health Research, Syöpäsäätiö, European Research Council, Natural Sciences and Engineering Research Council of Canada, Canada Research Chairs, Academy of Finland, Canada Foundation for Innovation, Austrian Science Fund
المصدر: Biochimica et Biophysica Acta (BBA) - General Subjects ; volume 1866, issue 3, page 130058 ; ISSN 0304-4165
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6Academic Journal
المؤلفون: Nawar, Nabanita, Bukhari, Shazreh, Adile, Ashley A., Suk, Yujin, Manaswiyoungkul, Pimyupa, Toutah, Krimo, Olaoye, Olasunkanmi O., Raouf, Yasir S., Sedighi, Abootaleb, Garcha, Harsimran Kaur, Hassan, Muhammad Murtaza, Gwynne, William, Israelian, Johan, Radu, Tudor B., Geletu, Mulu, Abdeldayem, Ayah, Gawel, Justyna M., Cabral, Aaron D., Venugopal, Chitra, de Araujo, Elvin D., Singh, Sheila K., Gunning, Patrick T.
المساهمون: Canadian Institutes of Health Research, Canada Foundation for Innovation, Canada Research Chairs, Natural Sciences and Engineering Research Council of Canada, Leukemia and Lymphoma Society of Canada, Canadian Breast Cancer Foundation, Canadian Cancer Society, McMaster University, Government of Ontario, Ontario Ministry of Research, Innovation and Science, Ontario Institute for Cancer Research, Jesse’s Journey
المصدر: Journal of Medicinal Chemistry ; volume 65, issue 4, page 3193-3217 ; ISSN 0022-2623 1520-4804
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7Academic Journal
المؤلفون: Toutah, Krimo, Nawar, Nabanita, Timonen, Sanna, Sorger, Helena, Raouf, Yasir S., Bukhari, Shazreh, von Jan, Jana, Ianevski, Aleksandr, Gawel, Justyna M., Olaoye, Olasunkanmi O., Geletu, Mulu, Abdeldayem, Ayah, Israelian, Johan, Radu, Tudor B., Sedighi, Abootaleb, Bhatti, Muzaffar N., Hassan, Muhammad Murtaza, Manaswiyoungkul, Pimyupa, Shouksmith, Andrew E., Neubauer, Heidi A., de Araujo, Elvin D., Aittokallio, Tero, Kraemer, Oliver H., Moriggl, Richard, Mustjoki, Satu, Herling, Marco, Gunning, Patrick T.
مصطلحات موضوعية: ddc:no
Relation: Toutah, Krimo, Nawar, Nabanita, Timonen, Sanna orcid:0000-0002-8139-5950 , Sorger, Helena, Raouf, Yasir S., Bukhari, Shazreh, von Jan, Jana, Ianevski, Aleksandr orcid:0000-0002-7780-482X , Gawel, Justyna M., Olaoye, Olasunkanmi O., Geletu, Mulu, Abdeldayem, Ayah, Israelian, Johan, Radu, Tudor B., Sedighi, Abootaleb, Bhatti, Muzaffar N., Hassan, Muhammad Murtaza, Manaswiyoungkul, Pimyupa, Shouksmith, Andrew E., Neubauer, Heidi A., de Araujo, Elvin D., Aittokallio, Tero orcid:0000-0002-0886-9769 , Kraemer, Oliver H., Moriggl, Richard orcid:0000-0003-0918-9463 , Mustjoki, Satu orcid:0000-0002-0816-8241 , Herling, Marco and Gunning, Patrick T. (2021). Development of HDAC Inhibitors Exhibiting Therapeutic Potential in T-Cell Prolymphocytic Leukemia. J. Med. Chem., 64 (12). S. 8486 - 8510. WASHINGTON: AMER CHEMICAL SOC. ISSN 1520-4804
الاتاحة: https://kups.ub.uni-koeln.de/59959/
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8Academic Journal
المؤلفون: Olaoye, Olasunkanmi O., Watson, Paris R., Nawar, Nabanita, Geletu, Mulu, Sedighi, Abootaleb, Bukhari, Shazreh, Raouf, Yasir S., Manaswiyoungkul, Pimyupa, Erdogan, Fettah, Abdeldayem, Ayah, Cabral, Aaron D., Hassan, Muhammad Murtaza, Toutah, Krimo, Shouksmith, Andrew E., Gawel, Justyna M., Israelian, Johan, Radu, Tudor B., Kachhiyapatel, Niyati, de Araujo, Elvin D., Christianson, David W., Gunning, Patrick T.
المساهمون: Canadian Institutes of Health Research, Canada Research Chairs, U.S. Department of Energy, Natural Sciences and Engineering Research Council of Canada, National Institute of General Medical Sciences, Canadian Breast Cancer Foundation, Canadian Cancer Society, Jesse's Journey, Ontario Research Fund
المصدر: Journal of Medicinal Chemistry ; volume 64, issue 5, page 2691-2704 ; ISSN 0022-2623 1520-4804
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9Academic Journal
المؤلفون: Nitschke, Felix, Wang, Peixiang, Schmieder, Peter, Girard, Jean-Marie, Awrey, Donald E., Wang, Tony, Israelian, Johan, Zhao, XiaoChu, Turnbull, Julie, Heydenreich, Matthias, Kleinpeter, Erich, Steup, Martin, Minassian, Berge A.
المصدر: Cell Metabolism ; volume 17, issue 5, page 756-767 ; ISSN 1550-4131
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10Academic Journal
المؤلفون: Tiberia, Erica, Turnbull, Julie, Wang, Tony, Ruggieri, Alessandra, Zhao, Xiao-Chu, Pencea, Nela, Israelian, Johan, Wang, Yin, Ackerley, Cameron A., Wang, Peixiang, Liu, Yan, Minassian, Berge A.
المصدر: Journal of Biological Chemistry ; volume 287, issue 30, page 25650-25659 ; ISSN 0021-9258
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11Academic Journal
المؤلفون: Gawel, Justyna M., Shouksmith, Andrew E., Raouf, Yasir S., Nawar, Nabanita, Toutah, Krimo, Bukhari, Shazreh, Manaswiyoungkul, Pimyupa, Olaoye, Olasunkanmi O., Israelian, Johan, Radu, Tudor B., Cabral, Aaron D., Sina, Diana, Sedighi, Abootaleb, de Araujo, Elvin D., Gunning, Patrick T.
المساهمون: NSERC, CIHR, Canada Research Chair, Canadian Cancer Society, Canadian Breast Cancer Foundation, Leukaemia and Lymphoma Society of Canada and infrastructure grants, Ontario Research Foundation
المصدر: European Journal of Medicinal Chemistry ; volume 201, page 112411 ; ISSN 0223-5234
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12Academic Journal
المؤلفون: Hassan, Muhammad Murtaza, Israelian, Johan, Nawar, Nabanita, Ganda, Giovanni, Manaswiyoungkul, Pimyupa, Raouf, Yasir S., Armstrong, David, Sedighi, Abootaleb, Olaoye, Olasunkanmi O., Erdogan, Fettah, Cabral, Aaron D., Angeles, Fabrizio, Altintas, Rabia, de Araujo, Elvin D., Gunning, Patrick T.
المساهمون: Canadian Institutes of Health Research, Canada Foundation for Innovation, Ontario Research Foundation, Canada Research Chairs, Natural Sciences and Engineering Research Council of Canada, Canadian Cancer Society Research Institute, Canadian Breast Cancer Foundation
المصدر: Journal of Medicinal Chemistry ; volume 63, issue 15, page 8634-8648 ; ISSN 0022-2623 1520-4804
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13
المؤلفون: de Araujo, Elvin D., Erdogan, Fettah, Neubauer, Heidi A., Meneksedag-Erol, Deniz, Manaswiyoungkul, Pimyupa, Eram, Mohammad S., Seo, Hyuk-Soo, Qadree, Abdul K., Israelian, Johan, Orlova, Anna, Suske, Tobias, Pham, Ha T. T., Boersma, Auke, Tangermann, Simone, Kenner, Lukas, Rülicke, Thomas, Dong, Aiping, Ravichandran, Manimekalai, Brown, Peter J., Audette, Gerald F., Rauscher, Sarah, Dhe-Paganon, Sirano, Moriggl, Richard, Gunning, Patrick T.
Relation: https://doi.org/10.5281/zenodo.2648567; https://doi.org/10.5281/zenodo.2648568; oai:zenodo.org:2648568
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14
المؤلفون: de Araujo, Elvin D., Erdogan, Fettah, Neubauer, Heidi A., Meneksedag-Erol, Deniz, Manaswiyoungkul, Pimyupa, Eram, Mohammad S., Seo, Hyuk-Soo, Qadree, Abdul K., Israelian, Johan, Orlova, Anna, Suske, Tobias, Pham, Ha T. T., Boersma, Auke, Tangermann, Simone, Kenner, Lukas, Rülicke, Thomas, Dong, Aiping, Ravichandran, Manimekalai, Brown, Peter J., Audette, Gerald F., Rauscher, Sarah, Dhe-Paganon, Sirano, Moriggl, Richard, Gunning, Patrick T.
Relation: https://doi.org/10.5281/zenodo.2648609; https://doi.org/10.5281/zenodo.2648610; oai:zenodo.org:2648610
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15
المؤلفون: de Araujo, Elvin D, Erdogan, Fettah, Neubauer, Heidi A, Meneksedag-Erol, Deniz, Eram, Mohammad S, Seo, Hyuk-Soo, Qadree, Abdul K, Israelian, Johan, Orlova, Anna, Suske, Tobias, Pham, Ha T. T., Boersma, Auke, Tangermann, Simone, Kenner, Lukas, Rülicke, Thomas, Dong, Aiping, Ravichandran, Manimekalai, Brown, Peter J, Audette, Gerald F, Rauscher, Sarah, Dhe-Paganon, Sirano, Moriggl, Richard, Gunning, Patrick T.
Relation: https://doi.org/10.5281/zenodo.2654891; https://doi.org/10.5281/zenodo.2654892; oai:zenodo.org:2654892
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16
المؤلفون: de Araujo, Elvin D., Univ. of Toronto, ON, Erdogan, Fettah Univ. of Toronto, ON, Neubauer, Heidi A., University of Veterinary Medicine, Vienna, Ludwig Boltzmann Institute for Cancer Research, Vienna, Meneksedag-Erol, Deniz Univ. of Toronto, ON, Manaswiyoungkul, Pimyupa Univ. of Toronto, Eram, Mohammad S., Univ. of Toronto, Mississauga, ON, Seo, Hyuk-Soo Dana-Farber Cancer Institute, Boston, MA, Harvard Medical School, Boston, MA, Qadree, Abdul K. Univ. of Toronto, ON, Israelian, Johan Univ. of Toronto, ON, Orlova, Anna University of Veterinary Medicine, Suske, Tobias University of Veterinary Medicine, Pham, Ha T., T. University of Veterinary Medicine, Vienna, Boersma, Auke University of Veterinary Medicine, Tangermann, Simone University of Veterinary Medicine, Kenner, Lukas Ludwig Boltzmann Institute for Cancer Research, University of Veterinary Medicine, Medical University of Vienna, Rülicke, Thomas University of Veterinary Medicine, Dong, Aiping Univ. of Toronto, ON, Ravichandran, Manimekalai Univ. of Toronto, Brown, Peter J. Univ. of Toronto, ON, Audette, Gerald F. York Univ., Toronto, ON, Rauscher, Sarah Univ. of Toronto, ON, Dhe-Paganon, Sirano Dana-Farber Cancer Institute, Moriggl, Richard University of Veterinary Medicine, Gunning, Patrick T.
مصطلحات موضوعية: 59 BASIC BIOLOGICAL SCIENCES, envir, socio
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17Academic Journal
المؤلفون: Atikian, Haig A., Meesala, Srujan, Burek, Michael J., Sohn, Young-Ik, Israelian, Johan, Patri, Adarsh S., Clarke, Nigel, Sipahigil, Alp, Evans, Ruffin E., Sukachev, Denis D., Westervelt, Robert, Lukin, Mikhail D., Lončar, Marko
المصدر: SPIE Newsroom ; ISSN 1818-2259
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18Academic Journal
المؤلفون: de Araujo, Elvin D., Manaswiyoungkul, Pimyupa, Israelian, Johan, Park, Jisung, Yuen, Karen, Farhangi, Shiva, Berger-Becvar, Angelika, Abu-Jazar, Lubna, Gunning, Patrick T.
المساهمون: Mitacs Inc., Natural Sciences and Engineering Research Council of Canada, Canadian Institutes of Health Research, Canada Research Chair, Canadian Foundation for Innovation and the Ontario Research Fund
المصدر: Journal of Pharmaceutical and Biomedical Analysis ; volume 143, page 159-167 ; ISSN 0731-7085
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19Periodical
المؤلفون: Nawar, Nabanita, Bukhari, Shazreh, Adile, Ashley A., Suk, Yujin, Manaswiyoungkul, Pimyupa, Toutah, Krimo, Olaoye, Olasunkanmi O., Raouf, Yasir S., Sedighi, Abootaleb, Garcha, Harsimran Kaur, Hassan, Muhammad Murtaza, Gwynne, William, Israelian, Johan, Radu, Tudor B., Geletu, Mulu, Abdeldayem, Ayah, Gawel, Justyna M., Cabral, Aaron D., Venugopal, Chitra, de Araujo, Elvin D., Singh, Sheila K., Gunning, Patrick T.
المصدر: Journal of Medicinal Chemistry; 20220101, Issue: Preprints
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20Academic Journal
المؤلفون: de Araujo, Elvin D., Erdogan, Fettah, Neubauer, Heidi A., Meneksedag-Erol, Deniz, Manaswiyoungkul, Pimyupa, Eram, Mohammad S., Seo, Hyuk-Soo, Qadree, Abdul K., Israelian, Johan, Orlova, Anna, Suske, Tobias, Pham, Ha T. T., Boersma, Auke, Tangermann, Simone, Kenner, Lukas, Rülicke, Thomas, Dong, Aiping, Ravichandran, Manimekalai, Brown, Peter J., Audette, Gerald F.
المصدر: Nature Communications; 6/7/2019, Vol. 10 Issue 1, pN.PAG-N.PAG, 1p