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المؤلفون: William A Carroll, Chengmin Zhong, Stephen Werness, Jinrong Liu, Matthew S Johnson, Lei Shi, Michael F Jarvis, James B. Thomas, Xu-Feng Zhang, Mark L. Chapman, Michael F. Gross, Shailen Joshi, Michael E. Kort, Marc J. C. Scanio, Dong Liu, Robert J Gregg, Rosemarie Roeloffs, Prisca Honore, Gricelda Hernandez, Gregory J Pacofsky, Douglas S. Krafte, Robert N. Atkinson, Brian E. Marron, Irene I. Drizin, Kennan C Marsh, Joseph P Mikusa, Michael J. Krambis, Bernard P Murray, Char-Chang Shieh, Connie R. Faltynek
المصدر: Journal of Medicinal Chemistry. 51:407-416
مصطلحات موضوعية: Male, Patch-Clamp Techniques, Stereochemistry, Analgesic, hERG, Pain, Nerve Tissue Proteins, Inflammation, In Vitro Techniques, Pharmacology, Sodium Channels, Cell Line, NAV1.8 Voltage-Gated Sodium Channel, Rats, Sprague-Dawley, Mice, Structure-Activity Relationship, Cricetulus, Sodium channel blocker, Cricetinae, Ganglia, Spinal, Drug Discovery, medicine, Animals, Humans, Furans, Neurons, Analgesics, biology, Chemistry, Sodium channel, Anti-Inflammatory Agents, Non-Steroidal, Chronic pain, Peripheral Nervous System Diseases, medicine.disease, Amides, Recombinant Proteins, Rats, Neuropathic pain, Systemic administration, biology.protein, Molecular Medicine, medicine.symptom, Sodium Channel Blockers
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المؤلفون: S A Buckner, Irene I. Drizin, Fatima Z. Basha, Robert J. Altenbach, T.M. Zydowsky, Crowell D, Boyd Steven A, Martin Winn, Michael E. Brune, Biswanath De
المصدر: Journal of Medicinal Chemistry. 36:2676-2688
مصطلحات موضوعية: Male, Pyrimidine, Pyrazine, Stereochemistry, Carboxylic acid, Biological Availability, Tetrazoles, Ring (chemistry), Niacin, Iodine Radioisotopes, Rats, Sprague-Dawley, Pyridazine, Angiotensin Receptor Antagonists, chemistry.chemical_compound, Rats, Inbred SHR, Drug Discovery, Pyridine, Animals, Antihypertensive Agents, Aorta, Alkyl, chemistry.chemical_classification, Receptors, Angiotensin, Angiotensin II, Nicotinic Acids, Rats, Liver, chemistry, Molecular Medicine, Rabbits, Muscle Contraction