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1Academic Journal
المؤلفون: Haruto Kurata, Hiroki Shioya, Hiromu Habashita, Kazutoyo Sato, Kenji Hiraizumi, Shinji Nakade, Tomohiro Hoshino, Yuichi Inagaki
المصدر: Biological and Pharmaceutical Bulletin. 2021, 44(2):188
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2Academic Journal
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3
المؤلفون: Masaharu Komeno, Yuka Takada, Takaki Komiya, Tatsuo Maeda, Haruto Kurata, Ryo Suzuki, Tetsu Kondo, Norikazu Matsunaga, Hiroshi Hagiya, Takeji Ono, Kazuhiro Otsuki, Ken-ici Nunoya, Sachiko Tominaga, Shinji Nakade, Hirotaka Mizuno, Kensuke Kusumi, Hidekazu Kiyoshi, Hiroki Shioya, Masakuni Kurono, Hiromu Habashita
المصدر: Journal of Medicinal Chemistry. 60:9508-9530
مصطلحات موضوعية: 0301 basic medicine, Agonist, chemistry.chemical_classification, biology, Stereochemistry, Chemistry, medicine.drug_class, Sphingosine-1-phosphate receptor, Pharmacology, biology.organism_classification, Amino acid, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, 030220 oncology & carcinogenesis, Drug Discovery, medicine, Molecular Medicine, Moiety, Cricetulus, Sphingosine-1-phosphate, Receptor, Lead compound
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4Academic Journal
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5Academic Journal
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6
المؤلفون: Haruto, Kurata, Kensuke, Kusumi, Kazuhiro, Otsuki, Ryo, Suzuki, Masakuni, Kurono, Takaki, Komiya, Hiroshi, Hagiya, Hirotaka, Mizuno, Hiroki, Shioya, Takeji, Ono, Yuka, Takada, Tatsuo, Maeda, Norikazu, Matsunaga, Tetsu, Kondo, Sachiko, Tominaga, Ken-Ici, Nunoya, Hidekazu, Kiyoshi, Masaharu, Komeno, Shinji, Nakade, Hiromu, Habashita
المصدر: Journal of medicinal chemistry. 60(23)
مصطلحات موضوعية: Male, Mice, Inbred BALB C, Administration, Oral, CHO Cells, Naphthalenes, Autoimmune Diseases, Rats, Sprague-Dawley, Macaca fascicularis, Mice, Receptors, Lysosphingolipid, Cricetulus, Rats, Inbred Lew, Animals, Azetidines, Humans, Female, Lymphocytes
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7
المؤلفون: Masaya Kokubo, Natsuko Tokuda, Kazuhiko Takeda, Tetsuya Sugiyama, Hiromu Habashita, Hiroshi Ochiai, Shiro Shibayama, Noriki Watanabe, Masamichi Imai, Takaki Komiya
المصدر: European Journal of Pharmacology. 720:335-343
مصطلحات موضوعية: Male, Receptors, CCR4, Ovalbumin, C-C chemokine receptor type 6, Biology, Ligands, CCL5, Cell Line, Mice, Chemokine receptor, Th2 Cells, Cell Movement, Anti-Allergic Agents, Sulfanilamides, Animals, Humans, CCL17, Antigens, CCL13, CXCL16, Chemokine CCL22, Pharmacology, Mice, Inbred BALB C, Pneumonia, Adoptive Transfer, Cell biology, HEK293 Cells, Mice, Inbred DBA, CC chemokine receptors, Spleen, CCL21
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8
المؤلفون: Masashi Gohda, Kenji Tanaka, Hiromu Habashita, Sho Koyama, Tetsuya Hagio, Kazuhito Kawabata, Akira Imagawa, Hidekazu Matsuya, Masaru Sakai, Yasushi Hirota, Yasuo Yonetomi, Taihei Nishiyama, Ai Hashimoto, Takehiro Ono, Shinya Sakimoto
المصدر: Stroke. 48
مصطلحات موضوعية: Advanced and Specialized Nursing, Intracerebral hemorrhage, Prothrombin time, medicine.diagnostic_test, medicine.drug_class, business.industry, Anticoagulant, 030204 cardiovascular system & hematology, medicine.disease, Thrombosis, Argatroban, 03 medical and health sciences, 0302 clinical medicine, medicine.artery, Anesthesia, Middle cerebral artery, medicine, Neurology (clinical), Cardiology and Cardiovascular Medicine, business, Stroke, 030215 immunology, Partial thromboplastin time, medicine.drug
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9
المؤلفون: Motoyuki Tanaka, Taku Fujimoto, Hiromu Habashita, Shinji Nakade, Hideyuki Ueda, Takuya Seko, Yoshikazu Takaoka, Hiroshi Saga, Hiroshi Kohno, Kazuya Hashimura, Hidehiro Suzuki, Masahiko Terakado
مصطلحات موضوعية: 0301 basic medicine, medicine.medical_specialty, Chemistry, Organic Chemistry, Antagonist, Hit to lead, Pharmacology, Biochemistry, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, Endocrinology, Blood pressure, In vivo, Tamsulosin, 030220 oncology & carcinogenesis, Internal medicine, Drug Discovery, Lysophosphatidic acid, medicine, Potency, Receptor, medicine.drug
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10
المؤلفون: Ryo Suzuki, Kazuhiro Otsuki, Takaki Komiya, Masakuni Kurono, Hiromu Habashita, Takeji Ono, Masashi Minami, Hiroshi Hagiya, Shinji Nakade, Kensuke Kusumi, Natsuko Tokuda, Yuka Takada, Hirotaka Mizuno, Hiroki Shioya, Haruto Kurata
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:144-148
مصطلحات موضوعية: Stereochemistry, Chemistry, Pharmaceutical, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Naphthalenes, Ligands, Ring (chemistry), Biochemistry, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Sphingosine, In vivo, Drug Discovery, Animals, Humans, Structure–activity relationship, Benzene, Receptor, Molecular Biology, Chemistry, Organic Chemistry, In vitro, Rats, Receptors, Lysosphingolipid, Models, Chemical, Drug Design, Molecular Medicine, Chlorine, Lysophospholipids, Selectivity, Linker
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11
المؤلفون: Takeji Ono, Kazuhiro Otsuki, Ryo Suzuki, Masakuni Kurono, Takaki Komiya, Hiroki Shioya, Masashi Minami, Hirotaka Mizuno, Yuka Takada, Haruto Kurata, Hiroshi Hagiya, Hiromu Habashita, Shinji Nakade, Kensuke Kusumi
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:3885-3889
مصطلحات موضوعية: Agonist, Propanols, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, CHO Cells, Naphthalenes, Biochemistry, Chemical synthesis, Mice, Structure-Activity Relationship, Cricetulus, Sphingosine, In vivo, Cricetinae, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Lymphocytes, Receptor, Molecular Biology, G protein-coupled receptor, Molecular Structure, Fingolimod Hydrochloride, Chemistry, organic chemicals, Organic Chemistry, In vitro, Receptors, Lysosphingolipid, Propylene Glycols, Molecular Medicine, lipids (amino acids, peptides, and proteins), Selectivity
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12
المؤلفون: Kenji Maeda, Shiro Shibayama, Katsuya Hisaichi, Hideaki Tada, Yoshikazu Takaoka, Chiaki Minamoto, Toshihiko Nishiyama, Kenji Sagawa, Hiromu Habashita, Masaaki Toda, Rena Nishizawa, Naoki Matsunaga, Daikichi Fukushima, Hiroaki Mitsuya
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:727-731
مصطلحات موضوعية: Magnetic Resonance Spectroscopy, Anti-HIV Agents, Stereochemistry, Metabolite, Clinical Biochemistry, Pharmaceutical Science, CHO Cells, Oxidative phosphorylation, In Vitro Techniques, Hydroxylation, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Cricetulus, Isomerism, Cricetinae, Drug Discovery, Animals, Combinatorial Chemistry Techniques, Humans, Chemokine CCL4, Molecular Biology, Chromatography, High Pressure Liquid, Active metabolite, Chemokine CCL3, chemistry.chemical_classification, Dipeptide, Chemistry, Organic Chemistry, Antagonist, Biological activity, Macrophage Inflammatory Proteins, Cyclic peptide, Rats, Drug Design, CCR5 Receptor Antagonists, Microsomes, Liver, Molecular Medicine, Indicators and Reagents, Oxidation-Reduction, Protein Binding
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13
المؤلفون: Masahiro Ikura, Tsuneyuki Sugiura, Shingo Nakatani, Shingo Yamamoto, Satoshi Itadani, Hiroyuki Ohno, Yoshitaka Nishita, Hiromu Habashita, Masaaki Toda, Kanji Takahashi, Koji Ogawa, Hisao Nakai
المصدر: Bioorganic & Medicinal Chemistry. 14:5402-5422
مصطلحات موضوعية: Matrix metalloproteinase inhibitor, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Stereoisomerism, Matrix Metalloproteinase Inhibitors, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Humans, Organic chemistry, Structure–activity relationship, Enzyme Inhibitors, Molecular Biology, Benzofurans, chemistry.chemical_classification, Hydroxamic acid, Molecular Structure, biology, Organic Chemistry, Chemical modification, Tissue Inhibitor of Metalloproteinases, Butyrates, Enzyme, chemistry, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine
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14
المؤلفون: Masaaki Toda, Shin Ichi Hamano, Hiroaki Mitsuya, Shiro Shibayama, Daikichi Fukushima, Kenji Sagawa, Nobuyuki Hamanaka, Kenji Maeda, Masaya Kokubo, Hideaki Tada, Hiromu Habashita
المصدر: Journal of Medicinal Chemistry. 49:4140-4152
مصطلحات موضوعية: Models, Molecular, Scaffold, Receptors, CCR5, Anti-HIV Agents, Stereochemistry, CHO Cells, Virus Replication, Cleavage (embryo), Chemical synthesis, Piperazines, Drug Resistance, Multiple, Viral, Cricetinae, Drug Discovery, Animals, Combinatorial Chemistry Techniques, Humans, Spiro Compounds, Chemokine CCL4, Receptor, Chemokine CCL3, G protein-coupled receptor, Chemistry, Biological activity, Macrophage Inflammatory Proteins, Combinatorial chemistry, Molecular Weight, Design synthesis, Drug Design, CCR5 Receptor Antagonists, HIV-1, Molecular Medicine, Ugi reaction, Calcium
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15
المؤلفون: Akane Omagari, Shinya Oishi, Hirokazu Tamamura, Kenichi Hiramatsu, Hiromu Habashita, Nobutaka Fujii, Hideki Nakashima, Akira Otaka, Kazuyo Gotoh, Naoki Yamamoto, Taisei Kanamoto
المصدر: Bioorganic & Medicinal Chemistry. 10:1417-1426
مصطلحات موضوعية: Receptors, CXCR4, CXCR4 Inhibitor, Anti-HIV Agents, Cell Survival, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Naphthalenes, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Chemokine receptor, Drug Discovery, Tumor Cells, Cultured, Peptide synthesis, medicine, Aromatic amino acids, Humans, Structure–activity relationship, Amino Acid Sequence, Calcium Signaling, Molecular Biology, Peptide sequence, Alanine, Organic Chemistry, chemistry, HIV-1, Molecular Medicine, Oligopeptides
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16
المصدر: The Journal of Organic Chemistry. 63:2392-2396
مصطلحات موضوعية: Computational chemistry, Chemistry, Organic Chemistry, Substructure
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17
المؤلفون: Nobutaka Fujii, Hiromu Habashita, Takeshi Kawasaki, Hirokazu Tamamura, Masako Akaji, Tetsutaro Kimachi, Toshiro Ibuka
المصدر: Tetrahedron Letters. 38:8307-8310
مصطلحات موضوعية: Allylic rearrangement, Organic Chemistry, chemistry.chemical_element, Epoxy, Zinc, Iodine, Biochemistry, chemistry.chemical_compound, chemistry, visual_art, Drug Discovery, visual_art.visual_art_medium, Organic chemistry, Ammonium chloride
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18
المؤلفون: Nobutaka Fujii, Hiromu Habashita, Masaki Noda, Toshiro Ibuka
المصدر: Chemical and Pharmaceutical Bulletin. 45:1259-1264
مصطلحات موضوعية: chemistry.chemical_classification, Dipeptide, Alkene, Stereochemistry, Isostere, General Chemistry, General Medicine, Alkylation, Chemical synthesis, chemistry.chemical_compound, Stereospecificity, chemistry, Drug Discovery, Lewis acids and bases, Chirality (chemistry)
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19
المؤلفون: Masayuki Imamura, Takatomo Koshiba, Toshiro Ibuka, Jeon-Uk Lee, Michihiko Wada, Hiromu Habashita, Ryuichiro Doi, Nobutaka Fujii, Ryo Hosotani, Koji Fujimoto, Kazuo Nakai
المصدر: Life Sciences. 60:29-34
مصطلحات موضوعية: Male, Agonist, Isostere, Stereochemistry, medicine.drug_class, Partial agonist, General Biochemistry, Genetics and Molecular Biology, Rats, Sprague-Dawley, Structure-Activity Relationship, chemistry.chemical_compound, medicine, Animals, Structure–activity relationship, General Pharmacology, Toxicology and Pharmaceutics, Pancreas, Dose-Response Relationship, Drug, Antagonist, Bombesin, Biological activity, General Medicine, Peptide Fragments, Rats, Bombesin receptor, chemistry, Amylases
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20
المؤلفون: Toshiro Ibuka, Yoshinori Yamamoto, Hirokazu Tamamura, Norio Mimura, Nobutaka Fujii, Kazuo Nakai, Masako Akaji, Hiromu Habashita
المصدر: Tetrahedron Letters. 37:2849-2852
مصطلحات موضوعية: chemistry.chemical_compound, Dipeptide, Chemistry, Group (periodic table), Stereochemistry, Organic Chemistry, Drug Discovery, Biochemistry, Catalysis