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1Academic Journal
المؤلفون: Tokalı F. S., Taslimi P., Sadeghi M., Şenol H.
المساهمون: ŞENOL, HALIL
مصطلحات موضوعية: AChE, BChE, hCA I-II, molecular docking, quinazolin-4(3H)-one
وصف الملف: application/pdf
Relation: CHEMISTRYSELECT; Tokalı F. S., Taslimi P., Sadeghi M., Şenol H., "Synthesis and Evaluation of Quinazolin-4(3H)-one Derivatives as Multitarget Metabolic Enzyme Inhibitors: A Biochemistry-Oriented Drug Design", CHEMISTRYSELECT, cilt.8, sa.25, ss.1-14, 2023; 14; 25; https://hdl.handle.net/20.500.12645/38383; WOS:001018020800001
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2Academic Journal
المؤلفون: Atteeque Ahmed, Imran Shafique, Aamer Saeed, Ghulam Shabir, Arslan Saleem, Parham Taslimi, Tugba Taskin Tok, Mahinur Kirici, Eda Mehtap Üç, Muhammad Zaffar Hashmi
المصدر: European Journal of Medicinal Chemistry Reports, Vol 6, Iss , Pp 100082- (2022)
مصطلحات موضوعية: Nimesulide analogues, Acyl thiourea, Molecular hybridization, Synthetic approaches, hCA I, II, α-amylase inhibitor, Pharmacy and materia medica, RS1-441, Other systems of medicine, RZ201-999
وصف الملف: electronic resource
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3Academic Journal
المؤلفون: Songül KARAKAYA, Zeynebe BİNGÖL, İlhami GÜLÇİN, Fatmagül DELİMUSTAFAOĞLU, Hayri DUMAN, Ceyda Sibel KILIÇ
المصدر: Bezmiâlem Science, Vol 9, Iss 2, Pp 153-157 (2021)
مصطلحات موضوعية: apiaceae, carbonic anhydrase, ferulago, leiotulus, hca i, hca ii, Medicine (General), R5-920
وصف الملف: electronic resource
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4Academic Journal
المؤلفون: Demet Uzun, Ebru Erdoğdu, Ayla Balaban Gündüzalp, Ümmühan Özmen Özdemir, Ali Öztürk, Neslihan Özbek, Kerem Kaya, Olkar Abdulmajet
المصدر: Macedonian Journal of Chemistry and Chemical Engineering, Vol 40, Iss 2 (2021)
مصطلحات موضوعية: sulfonylhydrazones, hCA I isoenzyme, cyclic voltammetry (CV), minimum inhibitory concentrations (MICs), Chemical engineering, TP155-156, Biochemistry, QD415-436
وصف الملف: electronic resource
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5Academic Journal
المصدر: Antibiotics, Vol 12, Iss 1, p 128 (2023)
مصطلحات موضوعية: antibacterial, antibiofilm, anti-QS activity, gamma radiation, hCA-I and -II inhibition, molecular docking, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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6Academic Journal
المؤلفون: Aggul, Ahmet Gokhan, Taslimi, Parham, Kuzu, Muslum, Uzun, Naim, Bilginer, Sinan, Gulcin, Ilhami
المساهمون: Belirlenecek
مصطلحات موضوعية: oleuropein, verbascoside, carbonic anhydrase, enzyme inhibition, molecular docking, Phenolic-Compounds, Antioxidant Activity, Isoenzymes I, Hca I, Proteins
Relation: Journal Of Oleo Science; Makale - Uluslararası Hakemli Dergi - Kurum Öğretim Elemanı; https://doi.org/10.5650/jos.ess21106; https://hdl.handle.net/20.500.12501/3157; 70; 1275; 1283; WOS:000709764400010; 2-s2.0-85114624383
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7Academic Journal
المؤلفون: Mohammad M. Al-Sanea, Ahmed Elkamhawy, Sora Paik, Silvia Bua, So Ha Lee, Mohamed A. Abdelgawad, Eun Joo Roh, Wagdy M. Eldehna, Claudiu T. Supuran
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 34, Iss 1, Pp 1457-1464 (2019)
مصطلحات موضوعية: benzenesulfonamides, carbonic anhydrase, quinolines, synthesis, cytosolic isoforms hca i and ii, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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8Academic Journal
المؤلفون: Kesari Lakshmi Manasa, Sravya Pujitha, Aaftaab Sethi, Mohammed Arifuddin, Mallika Alvala, Andrea Angeli, Claudiu T. Supuran
المصدر: Metabolites; Volume 10; Issue 4; Pages: 136
مصطلحات موضوعية: carbonic anhydrase, hCA I, hCA II, hCA IX, hCA XII, imidazo[2,1- b ]thiazole, sulfonyl piperazine
وصف الملف: application/pdf
Relation: Pharmacology and Drug Metabolism; https://dx.doi.org/10.3390/metabo10040136
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9Academic Journal
المؤلفون: Aydın T., Yurtvermez B., Şentürk M., Kazaz C., Çakır A.
المساهمون: Belirlenecek
مصطلحات موضوعية: 1-(4'-methoxyphenyl)-1,2,3-trihydroxypropane, Artemisia dracunculus L, Enzyme inhibition, HCA I, HCA II, 1 (4' methoxyphenyl) 1,2,3 trihydroxypropane, 1 (piperidin 1 yl)undeca 2,4 diene 8,10 diyn 1 one, acetazolamide, alcohol, anethole, Artemisia dracunculus extract, carbonate dehydratase I, carbonate dehydratase II, dichloromethane, herniarin, hexane, methanol, n isobutylundeca 2,4 dien 8,10 diynamide, plant extract, stigmasterol, unclassified drug, affinity chromatography, Artemisia dracunculus, Article, chemical structure, column chromatography, drug activity, IC50, isolation, metabolite
Relation: Records of Natural Products; Makale - Ulusal Hakemli Dergi - Kurum Öğretim Elemanı; https://doi.org/10.25135/rnp.102.18.07.329; https://hdl.handle.net/20.500.12501/2547; 13; 216; 225; 2-s2.0-85067581913
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10Academic Journal
المؤلفون: Aydin, Tuba, Yurtvermez, Bayram, Senturk, Murat, Kazaz, Cavit, Cakir, Ahmet
المساهمون: ##Belirlenecek##
مصطلحات موضوعية: Artemisia dracunculus L, 1-(4 '-methoxyphenyl)-1,2,3-trihydroxypropane, enzyme inhibition, hCA I, hCA II
Relation: RECORDS OF NATURAL PRODUCTS; Makale - Uluslararası Hakemli Dergi - Kurum Öğretim Elemanı; https://dx.doi.org/10.1016/j.heliyon.2019.e01422; https://hdl.handle.net/20.500.12501/692; 13; 216; 225; 000466970300091
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11Academic Journal
المؤلفون: Tan, Ayse, Kızılkaya, Serap, Ates, Burhan, Kara, Yunus
المساهمون: Bursa Uludağ Üniversitesi/Fen Edebiyat Fakültesi/Kimya Bölümü., Noma, Samir A. A., NOMA, Samir Abbas Ali, ABH-1773-2021
مصطلحات موضوعية: Carbonic-anhydrase, Inhibitory properties, Anticancer activity, Uric-acid, Derivatives, Tetrazole, 1h-tetrazole, 3(2h)-dione, Anhydrase isoenzymes (hca i and ii), Hybrid molecules, Isoindole-1, Molecular docking, Xanthine oxidase, Science & technology, Life sciences & biomedicine, Biochemistry & molecular biology, Toxicology
Relation: Makale - Uluslararası Hakemli Dergi; Journal Of Biochemical And Molecular Toxicology; https://doi.org/10.1002/jbt.23015; https://hdl.handle.net/11452/48393; 000765579300001; 36
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12Academic Journal
المؤلفون: Polat, M. Fatih, Anil, Derya Aktas, Saglamtas, Ruya, Tarikogullari, Ayse H., Alagoz, M. Abdullah, Gulcin, Ilhami, Algul, Oztekin
مصطلحات موضوعية: Acetylcholinesterase, Chalcone, Butyrylcholinesterase, Carbonic anhydrase, Enzyme inhibition, Molecular docking, Anhydrase Isoenzymes I, Carbonic-Anhydrase, Acetylcholinesterase Inhibitors, Biological Evaluation, Alpha-Glycosidase, Hca-I, Design, Esterase, Anticancer
Relation: Computational Biology And Chemistry; Makale - Uluslararası Hakemli Dergi - Kurum Öğretim Elemanı; https://hdl.handle.net/11454/76484; https://doi.org/10.1016/j.compbiolchem.2022.107748; Anıl, Derya Aktas/0000-0003-2584-275X; POLAT, M. Fatih/0000-0002-2838-163X; 100
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13Academic Journal
المؤلفون: Osmaniye, Derya, Türkeş, Cüneyt, Demir, Yeliz, Özkay, Yusuf, Kaplancıklı, Zafer Asım, Beydemir, Şükrü
المساهمون: Beydemir, Şükrü
مصطلحات موضوعية: Dithiocarbamate, hCA I, hCA II, Methysulfonyl, Molecular Docking
وصف الملف: application/pdf
Relation: Archiv der Pharmazie; Makale - Uluslararası Hakemli Dergi - Kurum Öğretim Elemanı; PubMed; Scopus; WoS; WoS - Index Chemicus; WoS - Science Citation Index Expanded; Osmaniye D, Türkeş C, Demir Y, Özkay Y, Beydemir Ş, Kaplancıklı ZA. Design, synthesis, and biological activity of novel dithiocarbamate-methylsulfonyl hybrids as carbonic anhydrase inhibitors. Arch Pharm (Weinheim). 2022 Aug;355(8):e2200132. doi:10.1002/ardp.202200132. Epub 2022 May 3. PMID: 35502846.; https://doi.org/10.1002/ardp.202200132; https://hdl.handle.net/11552/2968; 355
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14Academic Journal
المؤلفون: Burmaoglu, Serdar, Kazancioglu, Elif Akin, Kazancioglu, Mustafa Z., Saglamtas, Ruya, Yalcin, Gozde, Gulcin, Ilhami, Algul, Oztekin
المساهمون: Belirlenecek
مصطلحات موضوعية: Chalcone, Acetylcholinesterase, Carbonic anhydrase, Butyrylcholinesterase, Enzyme inhibition, Anhydrase Isoenzymes I, Trout Oncorhynchus-Mykiss, Carbonic-Anhydrase, Crystal-Structure, Hca I, Biological Evaluation, Alpha-Glycosidase, Mannich-Bases
Relation: Journal Of Molecular Structure; Makale - Uluslararası Hakemli Dergi - Kurum Öğretim Elemanı; https://doi.org/10.1016/j.molstruc.2022.132358; https://hdl.handle.net/20.500.12501/2816; 1254; WOS:000791803000012; 2-s2.0-85122631523
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15Academic Journal
المؤلفون: Aggul, Ahmet Gokhan, Uzun, Naim, Kuzu, Muslum, Taslimi, Parham, Gulcin, Ilhami
المساهمون: Belirlenecek
مصطلحات موضوعية: carbonic anhydrase, enzyme inhibition, molecular docking, olive leaf, phenolic compound, Isozymes I, Hca I, Isoenzymes I, Derivatives, Oleuropein, Hydroxytyrosol, Products, Proteins
Relation: Archiv Der Pharmazie; Makale - Uluslararası Hakemli Dergi - Kurum Öğretim Elemanı; https://doi.org/10.1002/ardp.202100476; https://hdl.handle.net/20.500.12501/2630; 355; WOS:000770784600001; 2-s2.0-85126563829
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16Academic Journal
المصدر: Open Chemistry, Vol 7, Iss 4, Pp 909-922 (2009)
مصطلحات موضوعية: quantitative structure-activity relationship (qsar), inhibition activities of sulfonamide and sulfamate derivatives for human carbonic anhydrases (hca i and hca ii) and α-carbonic anhydrase from helicobacter pylori (hpca), combinatorial protocol in multiple linear regression (cp-mlr) analysis, dragon descriptors, Chemistry, QD1-999
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2391-5420
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17
المؤلفون: Derya Aktas Anil, M. Fatih Polat, Ruya Saglamtas, Ayse H. Tarikogullari, M. Abdullah Alagoz, Ilhami Gulcin, Oztekin Algul, Serdar Burmaoglu
المساهمون: Belirlenecek
مصطلحات موضوعية: Alpha-Glycosidase, Design, Acetylcholinesterase Inhibitors, Esterase, Biochemistry, Structure-Activity Relationship, Chalcones, Chalcone, Structural Biology, Humans, Anhydrase Isoenzymes I, Carbonic Anhydrase Inhibitors, Carbonic anhydrase, Molecular Structure, Organic Chemistry, Carbonic-Anhydrase, Hca-I, Molecular Docking Simulation, Computational Mathematics, Enzyme inhibition, Anticancer, Butyrylcholinesterase, Molecular docking, Acetylcholinesterase, Cholinesterase Inhibitors, Biological Evaluation
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18
المؤلفون: Ayse Tan, Serap Kizilkaya, Samir A. A. Noma, Burhan Ates, Yunus Kara
المصدر: Journal of biochemical and molecular toxicologyREFERENCES. 36(5)
مصطلحات موضوعية: Molecular Structure, Health, Toxicology and Mutagenesis, Allopurinol, 1H-tetrazole, 3(2H)-dione, anhydrase isoenzymes (hCA I and II), hybrid molecules, isoindole-1, molecular docking, xanthine oxidase, Tetrazoles, General Medicine, Isoindoles, Toxicology, Biochemistry, Isoenzymes, Molecular Docking Simulation, Structure-Activity Relationship, Molecular Medicine, Carbonic-Anhydrase, Inhibitory Properties, Anticancer Activity, Uric-Acid, Derivatives, Tetrazole, Carbonic Anhydrase Inhibitors, Molecular Biology, Carbonic Anhydrases
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19Academic Journal
المؤلفون: Demir, N., Nadaroglu, H., Gungor, A. A., Demir, Y.
المساهمون: MÜ
مصطلحات موضوعية: Tumor Markers, Carbonic Anhydrase, HCA-I, HCA-II, BCA, CA-IV, Zn2+
Relation: Bratislava Medical Journal-Bratislavske Lekarske Listy; Makale - Uluslararası Hakemli Dergi - Kurum Öğretim Elemanı; https://doi.org/10.4149/BLL_2015_062; https://hdl.handle.net/20.500.12809/3248; 116; 330; 333
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20Academic Journal
المؤلفون: Kazanci, Ali, Gok, Yetkin, Kaya, Ruya, Aktas, Aydin, Taslimi, Parham, Gulcin, Ilhami
المساهمون: Belirlenecek
مصطلحات موضوعية: Dative donor ligand, Enzyme inhibition, Carbonic anhydrase, N-phthalimidomethyl, Silver(I)NHC complex, Anhydrase Inhibitory Properties, Peppsi Complexes Synthesis, Bis-Benzimidazolium Salts, Potent Carbonic-Anhydrase, Erythrocytes In-Vitro, Crystal-Structure, Catalytic-Activity, Ii Inhibition, Isoenzymes I, Hca I
Relation: Polyhedron; Makale - Uluslararası Hakemli Dergi - Kurum Öğretim Elemanı; https://doi.org/10.1016/j.poly.2020.114866; https://hdl.handle.net/20.500.12501/2834; 193; WOS:000598080700006; 2-s2.0-85095707422