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المؤلفون: Katlin B. Massirer, Lewis E. Pennicott, Fiona Scott, Jonathan M. Elkins, Simon E. Ward, Tristan Reuillon, A.M. Fala
المصدر: Bioorganic & Medicinal Chemistry Letters
مصطلحات موضوعية: Models, Molecular, HATU, hexafluorophosphate azabenzotriazole tetramethyl uronium, PARP, poly(ADP-ribose) polymerase, Chemical tool, Clinical Biochemistry, Pharmaceutical Science, IC50, half maximal inhibitory concentration, Chemical probe, PRK, protein kinase C-related kinase, DMSO, dimethyl sulfoxide, Crystallography, X-Ray, PRO2, glutamate 5-kinase Pro2, EGTA, egtazic acid, Benzimidazole, 01 natural sciences, Biochemistry, GST, glutathione S-transferase, CDI, 1,1′-carbonyldiimidazole, AGC, protein kinase A/G/C families, DNA, deoxyribonucleic acid, Neoplasms, CLK, CDC2-like kinase, DMF, N,N-dimethyl-formamide, Drug Discovery, PDB, protein databank, Kinome, Ki, inhibitor constant, Protein Kinase C, Cancer, ChEMBL, European Molecular Biology Laboratory Chemical database, Molecular Structure, Kinase, Chemistry, PRK2, KD, dissociation constant, PAK2, p21 activated kinase 2, DCM, dichloromethane, SFM, scanning force microscopy, Agc kinase, Molecular Medicine, THF, tetrahydrofuran, EtOH, ethanol, SDS, sodium dodecyl sulfate, ATP, adenosine triphosphate, TCEP, tris(2-carboxyethyl)phosphine, Antineoplastic Agents, Kinases, Heart failure, STK, serine/threonine kinase, Article, Structure-Activity Relationship, Protein kinase N2, Drug Development, TR-FRET, time resolved fluorescence resonance energy transfer, AcOH, acetic acid, PKC, protein kinase C, DIPEA, N,N-diisopropylethylamine, medicine, Humans, NMR, nuclear magnetic resonance, Protein kinase A, Protein Kinase Inhibitors, Molecular Biology, PAGE, polyacrylamide gel electrophoresis, ComputingMethodologies_COMPUTERGRAPHICS, PKN2, Inflammation, Dose-Response Relationship, Drug, EDTA, ethylenediaminetetraacetic acid, 010405 organic chemistry, Organic Chemistry, HEPES, 4-(2-hydroxyethyl)-1-piperazineethanesulfonic acid, AGC kinase, medicine.disease, SAR, structure activity relationship, 0104 chemical sciences, Abl, Abelson murine leukemia viral oncogene, 010404 medicinal & biomolecular chemistry, CV, column volumes, Benzimidazoles, MeOH, methanol, PKN, protein kinase N
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