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1
المؤلفون: Ute Gerhard, Gregory John Hollingworth, Steven R. Thomas, Richard H. Herbert, Russell J. Mortishire-Smith
المصدر: Magnetic Resonance in Chemistry. 43:658-661
مصطلحات موضوعية: Models, Molecular, Magnetic Resonance Spectroscopy, Stereochemistry, Aryl, Molecular Conformation, Stereoisomerism, General Chemistry, Fluorine-19 NMR, Crystallography, X-Ray, Ring (chemistry), Structure-Activity Relationship, chemistry.chemical_compound, Neurokinin-1 Receptor Antagonists, chemistry, Proton NMR, Spiro Compounds, General Materials Science, Protons, Tetrahydrofuran, Binding affinities
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2
المؤلفون: Gary G. Chicchi, Mark Peter Ridgill, Gregory John Hollingworth, Angela Williams, W. Rycroft, Kwei-Lan Tsao, Christopher John Swain, Kevin Dinnell, Jason Matthew Elliott, Madhumeeta J Dhar, Marc M. Kurtz
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:1237-1240
مصطلحات موضوعية: Indoles, Nitrogen, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Molecular Conformation, Substituent, Pharmaceutical Science, chemistry.chemical_element, Electrons, Carboxamide, CHO Cells, Substance P, Binding, Competitive, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Neurokinin-1 Receptor Antagonists, Cricetinae, Drug Discovery, medicine, Animals, Molecular Biology, Indole test, Behavior, Animal, Bicyclic molecule, Aryl, Organic Chemistry, Recombinant Proteins, chemistry, Molecular Medicine, Gerbillinae, Selectivity, Palladium
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3
المؤلفون: Christopher John Swain, Christopher Thomson, Kevin Dinnell, Jason Matthew Elliott, Laura C. Dickinson, Gregory John Hollingworth, Janusz Jozef Kulagowski
المصدر: Tetrahedron Letters. 40:2633-2636
مصطلحات موضوعية: chemistry.chemical_compound, General method, chemistry, Aryl, Organic Chemistry, Drug Discovery, Organic chemistry, Phenol, Phenols, Alkylation, Biochemistry, Cyclopropane
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4
المؤلفون: Michael B. Hursthouse, Gregory John Hollingworth, Jeremy D. Kilburn, Peter N. Horton, Jonathan J. Underwood
المصدر: Tetrahedron Letters. 45:2223-2225
مصطلحات موضوعية: chemistry.chemical_compound, Samarium diiodide, Chemistry, Organic Chemistry, Drug Discovery, Methylenecyclopropane, Biochemistry, Medicinal chemistry
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5ChemInform Abstract: A Convenient Method for the Preparation of Aryl Cyclopropyl Ethers from Phenols
المؤلفون: Laura C. Dickinson, Janusz Jozef Kulagowski, Christopher Thomson, Christopher John Swain, Kevin Dinnell, Gregory John Hollingworth, Jason Matthew Elliott
المصدر: ChemInform. 30
مصطلحات موضوعية: chemistry.chemical_compound, General method, Chemistry, Aryl, Organic chemistry, Phenol, General Medicine, Phenols, Alkylation, Cyclopropane
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6
المؤلفون: Kwei-Lan Tsao, Gregory John Hollingworth, Jason Matthew Elliott, Christopher John Swain, W. Rycroft, Gary G. Chicchi, Jerry Di Salvo, Natalie Clark, Marc M. Kurtz, F. David Tattersall, Laura Catherine Cooper, José L. Castro, Ruth Kilburn, Emma J. Carlson, Olivier Dirat
المصدر: Bioorganicmedicinal chemistry letters. 16(5)
مصطلحات موضوعية: Lactams, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Substance P, Cyclohexylamine, Biochemistry, Chemical synthesis, Methylation, chemistry.chemical_compound, Inhibitory Concentration 50, Structure-Activity Relationship, In vivo, Tachykinins, Drug Discovery, Animals, Humans, Molecular Biology, Molecular Structure, Organic Chemistry, Antagonist, Receptors, Neurokinin-1, Amides, In vitro, chemistry, Lactam, Molecular Medicine, Antiemetics, Penetrant (biochemical), Gerbillinae
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7
المؤلفون: Peter N. Horton, Jeremy D. Kilburn, Jonathan J. Underwood, Michael B. Hursthouse, Gregory John Hollingworth
المصدر: ChemInform. 35
مصطلحات موضوعية: Samarium diiodide, Chemistry, Organic chemistry, General Medicine
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8
المؤلفون: Zahid Ali, Susan Boyce, Natalie Clark, Gregory J. Kaczorowski, Simon Teague, J.K. Webb, Guy R. Seabrook, Richard E. Middleton, Wolfgang Jarolimek, Gregory John Hollingworth, Kathy G. Sutton, Margaret Z Chou, A. Brian Jones, Julie Kerby
المصدر: The Journal of pharmacology and experimental therapeutics. 303(3)
مصطلحات موضوعية: Male, medicine.drug_class, Receptors, Drug, TRPV1, Resiniferatoxin, Action Potentials, CHO Cells, Pharmacology, Rats, Sprague-Dawley, chemistry.chemical_compound, Mice, In vivo, Cricetinae, medicine, Animals, Humans, Receptor, Mice, Knockout, Dose-Response Relationship, Drug, Cannabinoids, Antagonist, Receptor antagonist, Rats, Mice, Inbred C57BL, chemistry, Capsaicin, Molecular Medicine, Diterpenes, Capsazepine
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9
المؤلفون: Alan P. Watt, Gary G. Chicchi, Laura Catherine Cooper, Denise Morrison, Duncan Shaw, Angela Williams, Karen L Locker, Kwei-Lan Tsao, Christopher John Swain, Kevin Dinnell, Gregory John Hollingworth, Marc M. Kurtz, Jason Matthew Elliott
المصدر: Bioorganicmedicinal chemistry letters. 11(9)
مصطلحات موضوعية: Indoles, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, CHO Cells, Substance P, Biochemistry, Chemical synthesis, Binding, Competitive, chemistry.chemical_compound, Structure-Activity Relationship, Neurokinin-1 Receptor Antagonists, Cricetinae, Drug Discovery, medicine, Animals, Receptor, Molecular Biology, Indole test, Brain Chemistry, Bicyclic molecule, Behavior, Animal, Chemistry, Aryl, Organic Chemistry, In vitro, Rats, Molecular Medicine, Indicators and Reagents, Selectivity, Gerbillinae