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1
المؤلفون: Andrew D. Cansfield, Mark A. Ator, Joydeep Banerjee, Michael Bestwick, Andrea Bortolato, Giles A. Brown, Jason Brown, Kristina Butkovic, Julie E. Cansfield, John A. Christopher, Miles Congreve, Gabriella Cseke, Francesca Deflorian, Benjamin Dugan, Martina Petrovic Hunjadi, Antun Hutinec, Trinadh Kumar Inturi, Goran Landek, Jonathan Mason, Alistair O’Brien, Gregory R. Ott, Renata Rupcic, Gordon Saxty, Stacey M. Southall, Rahela Zadravec, Stephen P. Watson
المصدر: ACS Chemical Neuroscience. 13:751-765
مصطلحات موضوعية: GPCR CGRP CGRPR macrocycle macrocyclic antagonist, Physiology, Cognitive Neuroscience, Calcitonin Receptor-Like Protein, Cell Biology, General Medicine, Crystallography, X-Ray, Ligands, Biochemistry, Receptors, Calcitonin Gene-Related Peptide, Receptors, G-Protein-Coupled
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2
المؤلفون: Radan Spaventi, Santiago Ferrer, Sulejman Alihodžić, Goran Landek, Kristina Starčević, Esperanza Herreros, Ana Toplak, Dijana Pesic, Mihaela Perić
المصدر: European Journal of Medicinal Chemistry. 49:365-378
مصطلحات موضوعية: Plasmodium falciparum, Azithromycin, Pharmacology, Azalide, Cell Line, Antimalarials, Chloroquine, malaria, antimalarial, azalide, quinoline, hybrid molecules, synthesis, parasitic diseases, Drug Discovery, medicine, Humans, Antimalarial Agent, biology, Chemistry, Organic Chemistry, General Medicine, biology.organism_classification, medicine.disease, In vitro, Malaria, Aminoquinolines, Macrolides, Antibacterial activity, medicine.drug
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3
المؤلفون: Mihaela Perić, Wilbur K. Milhous, Nedjeljko Kujundžić, Jasna Padovan, Zrinka Ivezić Schönfeld, Andrea Fajdetić, Kirsten S. Smith, Dubravko Jelić, Colin Ohrt, Wolfgang Schönfeld, William Y. Ellis, Arba L. Ager, Radan Spaventi, Dinko Žiher, Mirjana Bukvić Krajačić, Goran Landek
المصدر: Journal of Medicinal Chemistry. 54:3595-3605
مصطلحات موضوعية: Stereochemistry, Chemistry, Pharmaceutical, Plasmodium falciparum, Azithromycin, Azalide, Ring (chemistry), Antimalarials, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Drug Discovery, medicine, Animals, Humans, Urea, Structure–activity relationship, Aromatic moiety, Chemistry, Thiourea, SAR, antimalarial acivity, urea, thiourea, azalides, In vitro, Models, Chemical, Drug Design, Lipophilicity, Molecular Medicine, Macrolides, medicine.drug
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4
المؤلفون: Marijana Vinković, Vladimir Vinković, Darko Kontrec, Goran Landek
المصدر: Chromatographia. 64:469-473
مصطلحات موضوعية: Bicyclic molecule, Chemistry, Organic Chemistry, Clinical Biochemistry, Diol, Nuclear magnetic resonance spectroscopy, Biochemistry, High-performance liquid chromatography, Analytical Chemistry, NMR spectra database, Crystallography, chemistry.chemical_compound, Phase (matter), Organic chemistry, Enantiomer, Chiral derivatizing agent
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5
المؤلفون: Dijana Pesic, Goran Landek, Ivana Ozimec Landek, Milan Mesic, Vitomir Šunjić
مصطلحات موضوعية: Ring flip, Resolution (mass spectrometry), Stereochemistry, General Chemistry, Nuclear magnetic resonance spectroscopy, High-performance liquid chromatography, Chiral resolution, Chiral column chromatography, chemistry.chemical_compound, Crystallography, chemistry, Thiepine, fused oxepine, fused thiepene, NMR spectroscopy, conformational isomers, Enantiomer
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6
المؤلفون: Kristina Starčević, Esperanza Herreros, Radan Spaventi, Santiago Ferrer, Mihaela Perić, Goran Landek, Sulejman Alihodzic, Ana Toplak, Dijana Pesic
المصدر: ChemInform. 43
مصطلحات موضوعية: Chemistry, Covalent bond, medicine, Moiety, Molecule, General Medicine, Antimalarial Agent, Azalide, Combinatorial chemistry, medicine.drug
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7
المؤلفون: Andrea Fajdetić, Dubravko Jelić, Mirjana Bukvić Krajačić, Jasna Padovan, Sulejman Alihodžić, Arba L. Ager, Wilbur K. Milhous, Kirsten S. Smith, Milan Mesic, Dinko Žiher, Radan Spaventi, Antun Hutinec, William Y. Ellis, Mihaela Perić, Goran Landek, Zrinka Ivezić-Schönfeld, Renata Rupčić, Colin Ohrt
المصدر: Journal of medicinal chemistry. 55(3)
مصطلحات موضوعية: Male, Plasmodium berghei, Plasmodium falciparum, Drug Resistance, Pharmacology, Azalide, Azithromycin, Antimalarials, Mice, Structure-Activity Relationship, Parasitic Sensitivity Tests, In vivo, Chloroquine, Cell Line, Tumor, Drug Discovery, medicine, Structure–activity relationship, Potency, Animals, Humans, Amines, biology, Chemistry, biology.organism_classification, Amides, Bioavailability, Erythromycin, Malaria, Rats, Aminoquinolines, Microsomes, Liver, Molecular Medicine, Macrolides, medicine.drug
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8
المؤلفون: Irena Dokli, Vladimir Vinković, Goran Landek, Anamarija Knezevic
المصدر: ChemInform. 42
مصطلحات موضوعية: chemistry.chemical_compound, Enantiopure drug, Novozym 435, Chemistry, Aryl, General Medicine, Combinatorial chemistry
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9
المؤلفون: Anamarija Knežević, Irena Dokli, Goran Landek, Vladimir Vinković
مصطلحات موضوعية: chemistry.chemical_classification, biology, Aryl, Organic Chemistry, Lipase b, aryl-allylamines, Candida antarctica B, Overman rearrangement, enantioselectivity, biology.organism_classification, Catalysis, Inorganic Chemistry, Hydrolysis, chemistry.chemical_compound, Enzyme, chemistry, Organic chemistry, Candida antarctica, Knoevenagel condensation, Physical and Theoretical Chemistry
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10Electronic Resource
المصدر: Croatica Chemica Acta; ISSN 0011-1643 (Print); ISSN 1334-417X (Online); Volume 77; Issue 4
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11
المؤلفون: Irena Dokli, Anamarija Knežević, Vladimir Vinković, Goran Landek
المصدر: Tetrahedron: Asymmetry. 22:1594
مصطلحات موضوعية: Inorganic Chemistry, chemistry.chemical_compound, chemistry, Computational chemistry, Aryl, media_common.quotation_subject, Organic Chemistry, Tetrahedron, Addendum, Physical and Theoretical Chemistry, Asymmetry, Catalysis, media_common