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1
المؤلفون: Neeta Soni, Eric P. Westra, Giuseppe Allegretta, André L. S. Araujo, Camila F. de Pinho, Sarah Morran, Jens Lerchl, Franck E. Dayan, Philip Westra, Todd A. Gaines
المصدر: Pest Management Science. 78:5080-5089
مصطلحات موضوعية: Acetolactate Synthase, Herbicides, Bromus, Secale, Insect Science, Humans, General Medicine, Agronomy and Crop Science, Herbicide Resistance, Plant Proteins
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2
المؤلفون: Giuseppe Allegretta, Christine K. Maurer, Jens Eberhard, Damien Maura, Rolf W. Hartmann, Laurence Rahme, Martin Empting
المساهمون: Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS),Saarland 9 University, 66123 Saarbrücken, Germany.
المصدر: Frontiers in Microbiology, Vol 8 (2017)
مصطلحات موضوعية: 0301 basic medicine, Microbiology (medical), Multidrug tolerance, Mutant, Regulator, lcsh:QR1-502, MvfR, Biology, medicine.disease_cause, 01 natural sciences, Microbiology, Virulence factor, lcsh:Microbiology, 03 medical and health sciences, medicine, Quorum Sensing Inhibitors, dihydroxyquinoline, 2′-aminoacetophenone, 010405 organic chemistry, Pseudomonas aeruginosa, Biofilm, persistence, Small molecule, 0104 chemical sciences, Quorum sensing, 030104 developmental biology, Biochemistry, quinolones, 2' -aminoacetophenone
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3Academic Journal
المؤلفون: Giuseppe Allegretta, Christine K. Maurer, Jens Eberhard, Damien Maura, Rolf W. Hartmann, Laurence Rahme, Martin Empting
المصدر: Frontiers in Microbiology, Vol 8 (2017)
مصطلحات موضوعية: Pseudomonas aeruginosa, quinolones, 2′-aminoacetophenone, dihydroxyquinoline, persistence, Quorum Sensing Inhibitors, Microbiology, QR1-502
وصف الملف: electronic resource
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4
المؤلفون: Kiran V. Mahasenan, Jeshina Janardhanan, Sara Tejera, Elena Lastochkin, Shahriar Mobashery, Yuanyuan Qian, William R. Wolter, Giuseppe Allegretta, Zhihong Peng, Melissa Malia N. Gozun, Mayland Chang, Rhona Feltzer, Valerie A. Schroeder
المصدر: Journal of Medicinal Chemistry. 63:5287-5296
مصطلحات موضوعية: 0303 health sciences, biology, Chemistry, medicine.drug_class, Antibiotics, Allosteric regulation, In vitro toxicology, Active site, biochemical phenomena, metabolism, and nutrition, medicine.disease_cause, 01 natural sciences, 0104 chemical sciences, Microbiology, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, chemistry.chemical_compound, Staphylococcus aureus, In vivo, Drug Discovery, medicine, biology.protein, Molecular Medicine, Structure–activity relationship, Quinazolinone, 030304 developmental biology
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5Academic Journal
المؤلفون: Emanuele M Gargano, Giuseppe Allegretta, Enrico Perspicace, Angelo Carotti, Chris Van Koppen, Martin Frotscher, Sandrine Marchais-Oberwinkler, Rolf W Hartmann
المصدر: PLoS ONE, Vol 10, Iss 7, p e0134754 (2015)
وصف الملف: electronic resource
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المؤلفون: Yuanyuan, Qian, Giuseppe, Allegretta, Jeshina, Janardhanan, Zhihong, Peng, Kiran V, Mahasenan, Elena, Lastochkin, Melissa Malia N, Gozun, Sara, Tejera, Valerie A, Schroeder, William R, Wolter, Rhona, Feltzer, Shahriar, Mobashery, Mayland, Chang
المصدر: J Med Chem
مصطلحات موضوعية: Mice, Mice, Inbred ICR, Staphylococcus aureus, Structure-Activity Relationship, Neutropenia, Animals, Female, Microbial Sensitivity Tests, biochemical phenomena, metabolism, and nutrition, Article, Anti-Bacterial Agents, Quinazolinones
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7
المؤلفون: Xabier Murgia, Verena Fetz, Felix Beckmann, Sarah Gordon, Giuseppe Allegretta, Chiara De Rossi, Florian Graef, Walid A. M. Elgaher, Martin Empting, Nicole Schneider-Daum, Robert Richter, Claus-Michael Lehr, Mark Brönstrup, Rolf W. Hartmann, Jörg Haupenthal
المصدر: ACS infectious diseases. 4(8)
مصطلحات موضوعية: 0301 basic medicine, RM, Chemistry, 030106 microbiology, Cell Membrane, Optical Imaging, Biological Transport, Periplasmic space, Permeation, Models, Theoretical, Bacterial cell structure, Permeability, Anti-Bacterial Agents, 03 medical and health sciences, 030104 developmental biology, Infectious Diseases, Membrane, Gram-Negative Bacteria, Periplasm, Biophysics, Inner membrane, Cell envelope, Bacterial outer membrane, Intracellular, Fluorescent Dyes
وصف الملف: application/pdf
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8
المؤلفون: Rolf W. Hartmann, Isabell Schnorr, Scott G. Franzblau, Ahmed A. M. Kamal, Giuseppe Allegretta, Alexander Schifrin, Joerg Haupenthal, Andreas Thomann, Martin Empting, Sang-Hyun Cho, Jens Eberhard, Christian Brengel
المساهمون: HIPS, Helmholtz-Institut für pharmazeutische Forschung Saarland, Universitätscampus 8.1, 66123 Saarbrücken, Germany.
المصدر: ChemMedChem
مصطلحات موضوعية: 0301 basic medicine, Econazole, Antimycobacterial Agents, medicine.drug_class, Cell Survival, Antitubercular Agents, Computational biology, Heme, Microbial Sensitivity Tests, Pharmacology, Biology, Antimycobacterial, Biochemistry, Cell Line, Mycobacterium tuberculosis, Small Molecule Libraries, 03 medical and health sciences, Bacterial Proteins, Cytochrome P-450 Enzyme System, Biological profile, Drug Resistance, Multiple, Bacterial, biophysics, Drug Discovery, inhibitors, medicine, Humans, General Pharmacology, Toxicology and Pharmaceutics, Enzyme Inhibitors, Structural class, Toxicity profile, Binding Sites, screening, Organic Chemistry, Surface Plasmon Resonance, biology.organism_classification, Recombinant Proteins, Protein Structure, Tertiary, Multiple drug resistance, Molecular Docking Simulation, 030104 developmental biology, HEK293 Cells, anti-infectives, Molecular Medicine, Spectrophotometry, Ultraviolet, medicine.drug, Protein Binding
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9
المؤلفون: Gerhard Unteregger, Michael J. Hoffmann, Giuseppe Allegretta, Carsten-H. Ohlmann, Michael Stöckle, Rolf W. Hartmann, Jill A. van der Zee, Kerstin Junker, Jörg Haupenthal, Antonio G. Gomes de Mello Martins, Jens Eberhard, Rolf Müller
المصدر: The Journal of steroid biochemistry and molecular biology. 174
مصطلحات موضوعية: 0301 basic medicine, Male, endocrine system, medicine.medical_specialty, Neuroactive steroid, medicine.drug_class, Endocrinology, Diabetes and Metabolism, medicine.medical_treatment, Clinical Biochemistry, Dehydroepiandrosterone, Pregnanolone, Biology, urologic and male genital diseases, Biochemistry, 03 medical and health sciences, 0302 clinical medicine, Endocrinology, Internal medicine, Cell Line, Tumor, medicine, Humans, Gonadal Steroid Hormones, Molecular Biology, Testosterone, Prostatic Neoplasms, Steroid 17-alpha-Hydroxylase, Cell Biology, Androgen, body regions, Steroid hormone, 030104 developmental biology, CYP17A1, 030220 oncology & carcinogenesis, Dihydrotestosterone, Pregnenolone, Androgens, Molecular Medicine, Androstenes, human activities, medicine.drug
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10
المؤلفون: Ahmed A. M. Kamal, Christine K. Maurer, Martin Empting, Giuseppe Allegretta, Rolf W. Hartmann, Jörg Haupenthal
المصدر: Topics in Medicinal Chemistry ISBN: 9783319708386
مصطلحات موضوعية: 0301 basic medicine, 010405 organic chemistry, Drug discovery, Pseudomonas aeruginosa, medicine.drug_class, Antibiotics, Biofilm, Virulence, Biology, medicine.disease_cause, 01 natural sciences, 0104 chemical sciences, Microbiology, 03 medical and health sciences, Quorum sensing, 030104 developmental biology, Antibiotic resistance, medicine, Pathogen
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11
المصدر: ChemInform. 47
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Pyrimidine, Robustness (computer science), Leaving group, Organic chemistry, Tetrazole, General Medicine, Microwave assisted, Microwave, Catalysis
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المساهمون: Helmholtz Institute for Pharmaceutical Research Saarland (HIPS), Saarland University, Building A4.1, 66123 Saarbruecken, Germany., Helmholtz-Institute for Pharmaceutical Research Saarland, Saarland University
مصطلحات موضوعية: chemistry.chemical_compound, Pyrimidine, chemistry, Nucleophilic aromatic substitution, Robustness (computer science), Organic Chemistry, Leaving group, Tetrazole, Microwave assisted, Combinatorial chemistry, Microwave, Catalysis
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13
المساهمون: Helmholtz Institute for Pharmaceutical Research Saarland (HIPS), PO Box 15 11 50, D-66041 Saarbrücken, Germany.
المصدر: European journal of medicinal chemistry. 90
مصطلحات موضوعية: Pharmacology, chemistry.chemical_classification, Chalcone synthase, biology, Stereochemistry, Organic Chemistry, Catechols, Substrate (chemistry), Active site, Quorum Sensing, General Medicine, Substrate Specificity, chemistry.chemical_compound, Quorum sensing, Enzyme, chemistry, Bacterial Proteins, Drug Discovery, Pseudomonas aeruginosa, Anthranilic acid, biology.protein, Moiety, Enzyme Inhibitors, Linker, Acyltransferases
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14
المصدر: Organicbiomolecular chemistry. 12(32)
مصطلحات موضوعية: Quinolones, medicine.disease_cause, Biochemistry, law.invention, chemistry.chemical_compound, Structure-Activity Relationship, Biosynthesis, Bacterial Proteins, law, medicine, Structure–activity relationship, Physical and Theoretical Chemistry, Mode of action, chemistry.chemical_classification, 4-Quinolones, Pseudomonas aeruginosa, Chemistry, Methanol, Organic Chemistry, In vitro, Enzyme, Mutation, Recombinant DNA
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15
المؤلفون: C.H. Ohlmann, Gerhard Unteregger, Giuseppe Allegretta, Rolf W. Hartmann, A.G. Gomes De Mello Martins, Kerstin Junker, J. Van Der Zee, Michael Stöckle, Joerg Haupenthal, Jens Eberhard
المصدر: European Urology Supplements. 15:e137
مصطلحات موضوعية: Starvation, Oncology, Abiraterone, chemistry.chemical_compound, medicine.medical_specialty, chemistry, business.industry, Urology, Internal medicine, Prostate cancer cell, medicine, medicine.symptom, business