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1
المؤلفون: Xinchun Tong, Melanie Latham, Ying Chen, Denise P. Milot, Milton L. Hammond, Amjad Ali, Eugene Tan, Sheryl A. Hyland, Carl P. Sparrow, Qiu Guo, Joann B. Napolitano, Laurence B. Peterson, Samuel D. Wright, Suoyu S. Xu, Qiaolin Deng, Yi-Heng Chen, Gayle E. Taylor, Zhijian Lu, Peter J. Sinclair, Suzanne S. Eveland, Matt S. Anderson
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:199-203
مصطلحات موضوعية: Stereochemistry, Chemistry, Pharmaceutical, Clinical Biochemistry, Pharmaceutical Science, Mice, Transgenic, Ring (chemistry), Biochemistry, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Anacetrapib, Drug Discovery, Animals, Humans, Molecular Biology, Oxazolidinones, Biological evaluation, Biphenyl, Trifluoromethyl, Dose-Response Relationship, Drug, Cholesterol, HDL, Organic Chemistry, Cetp inhibition, In vitro, Cholesterol Ester Transfer Proteins, carbohydrates (lipids), Models, Chemical, chemistry, Drug Design, Molecular Medicine, lipids (amino acids, peptides, and proteins)
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2
المؤلفون: Milton L. Hammond, Anne-Marie Cumiskey, Sheryl A. Hyland, Ray Rosa, Christopher F. Thompson, Amjad Ali, Ying Chen, Suoyu S. Xu, James V. Pivnichny, Xinchun Tong, Qiu Guo, Hong Li, Carl P. Sparrow, Peter J. Sinclair, Joann B. Napolitano, Melanie Latham, Zhijian Lu, Samuel D. Wright, Laurence B. Peterson, Matt S. Anderson, Suzanne S. Eveland, Cameron J. Smith, Gayle E. Taylor, Denise P. Milot
المصدر: Journal of Medicinal Chemistry. 54:4880-4895
مصطلحات موضوعية: Male, Stereochemistry, Mice, Transgenic, Ring (chemistry), Mice, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Anacetrapib, Drug Discovery, Cholesterylester transfer protein, Animals, Humans, Oxazolidinones, Biphenyl, biology, Cholesterol, HDL, Stereoisomerism, Recombinant Proteins, Cholesterol Ester Transfer Proteins, Mice, Inbred C57BL, Macaca fascicularis, chemistry, biology.protein, Molecular Medicine, lipids (amino acids, peptides, and proteins), Methyl group
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3
المؤلفون: Gool F. Patel, Ronald E. Painter, Wayne M. Geissler, Gayle E. Taylor, Georgianna Harris, Lynn L. Silver, Kenneth P. Ellsworth, Richard L. Tolman, Donald W. Graham, Amjad Ali, Katherine Young, Susan D. Aster
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:2185-2188
مصطلحات موضوعية: Staphylococcus aureus, DNA polymerase, Clinical Biochemistry, Pharmaceutical Science, Microbial Sensitivity Tests, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Drug Discovery, Enzyme Inhibitors, Molecular Biology, DNA Polymerase III, Antibacterial agent, chemistry.chemical_classification, Aniline Compounds, biology, DNA synthesis, Organic Chemistry, biology.organism_classification, In vitro, Anti-Bacterial Agents, Pyrimidines, Enzyme, chemistry, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, Bacteria
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4
المؤلفون: Paul Mazur, Michael J. Forrest, Joann Williamson, Georgianna Harris, Mark L. Greenlee, Karen Lowitz, Gayle E. Taylor, Silvi Luell, Monica Einstein, Shilpa Pandit, Joseph C. Santoro, Milton L. Hammond, Lan Ge, Greg Rouen, Amjad Ali, Chuanlin Wang, Ester Carballo-Jane, James M. Balkovec, Ayesha Sitlani, Terri M. Kelly, Denise M. Visco
المصدر: Bioorganicmedicinal chemistry. 16(16)
مصطلحات موضوعية: Blood Glucose, Clinical Biochemistry, Anti-Inflammatory Agents, Pharmaceutical Science, Biochemistry, Betamethasone, Transactivation, Glucocorticoid receptor, Tyrosine aminotransferase, Receptors, Glucocorticoid, Glutamate-Ammonia Ligase, Glutamine synthetase, Drug Discovery, medicine, Animals, Insulin, Muscle, Skeletal, Molecular Biology, Triglycerides, Transrepression, Tyrosine Transaminase, Chemistry, Organic Chemistry, Body Weight, Biological activity, Ligand (biochemistry), Rats, Liver, Molecular Medicine, Carbamates, Matrix Metalloproteinase 1, medicine.drug
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5
المؤلفون: Katherine Young, Georgianna Harris, Lynn L. Silver, Gayle E. Taylor, Ken Ellsworth, Amjad Ali, Ronald E. Painter
المصدر: Journal of medicinal chemistry. 46(10)
مصطلحات موضوعية: Staphylococcus aureus, Pyrimidine, DNA polymerase, Enterococcus faecium, Microbial Sensitivity Tests, medicine.disease_cause, RNA polymerase III, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, medicine, Enzyme Inhibitors, Antibacterial agent, DNA Polymerase III, chemistry.chemical_classification, Aniline Compounds, biology, Chemistry, Anti-Bacterial Agents, Enzyme, Pyrimidines, Streptococcus pneumoniae, Biochemistry, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, Pyrazoles, DNA, Bacillus subtilis