نتائج البحث - "Gavara L."

1

Conference

1,2,4-TRIAZOLE-3-THIONE COMPOUNDS POTENTLY INHIBIT VIM AND NDM-1 METALLO-b-LACTAMASES AND RE-SENSITIZE MULTI-RESISTANT CLINICAL ISOLATES TO MEROPENEM

المؤلفون: Legru, A., Gavara L., Verdirosa F., Vo-Hoang Y., Tassone G., Corsica G., Vascone F., Thomas C., Feller, Georges, Crowder M., Cendron L., Pozzi C., Mangani S., Docquier, Jean-Denis, Hernandez J.-F.

المصدر: International Symposium on Medicinal Chemistry, Nice, France [FR], 4-8 septembre

مصطلحات موضوعية: Life sciences, Biochemistry, biophysics & molecular biology, Sciences du vivant, Biochimie, biophysique & biologie moléculaire

URL الوصول: https://orbi.uliege.be/handle/2268/294502

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2

Academic Journal

4-(N-alkyl-and-acyl-amino)-1,2,4-triazole-3-thione analogs as metallo-β-lactamase inhibitors: Impact of 4-linker on potency and spectrum of inhibition

المؤلفون: Gavara L., Verdirosa F., Legru A., Mercuri P. S., Nauton L., Sevaille L., Feller G., Berthomieu D., Sannio F., Marcoccia F., Tanfoni S., Luca F. D., Gresh N., Galleni M., Docquier J. D., Hernandez J. -F.

المساهمون: Gavara, L., Verdirosa, F., Legru, A., Mercuri, P. S., Nauton, L., Sevaille, L., Feller, G., Berthomieu, D., Sannio, F., Marcoccia, F., Tanfoni, S., Luca, F. D., Gresh, N., Galleni, M., Docquier, J. D., Hernandez, J. -F.

مصطلحات موضوعية: 1,2,4-triazole-3-thione, Bacterial resistance, Enzyme inhibitors, Metallo-β-lactamase, β-lactam antibiotics

وصف الملف: ELETTRONICO

Relation: info:eu-repo/semantics/altIdentifier/pmid/32717907; info:eu-repo/semantics/altIdentifier/wos/WOS:000577788700001; volume:10; issue:8; numberofpages:18; journal:BIOMOLECULES; https://hdl.handle.net/11365/1125144; https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7465886/

الاتاحة: https://hdl.handle.net/11365/1125144
https://doi.org/10.3390/biom10081094
https://www.mdpi.com/2218-273X/10/8/1094
https://www.ncbi.nlm.nih.gov/pmc/articles/PMC7465886/

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3

Academic Journal

4-Alkyl-1,2,4-triazole-3-thione analogues as metallo-β-lactamase inhibitors

المؤلفون: Gavara, L., Legru, A., Verdirosa, F., Sevaille, L., Nauton, L., Corsica, G., Mercuri, Paola, Sannio, F., Feller, Georges, Coulon, R., De Luca, F., Cerboni, G., Tanfoni, S., Chelini, G., Galleni, Moreno, Docquier, Jean-Denis, Hernandez, J.-F.

المصدر: Bioorganic Chemistry, 113, 105024 (2021)

مصطلحات موضوعية: Bacterial resistance, Metallo-β-Lactamase, Life sciences, Microbiology, Human health sciences, Pharmacy, pharmacology & toxicology, Physical, chemical, mathematical & earth Sciences, Chemistry, Sciences du vivant, Microbiologie, Sciences de la santé humaine, Pharmacie, pharmacologie & toxicologie, Physique, chimie, mathématiques & sciences de la terre, Chimie

Relation: urn:issn:0045-2068; urn:issn:1090-2120

URL الوصول: https://orbi.uliege.be/handle/2268/261224

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4

Academic Journal

4-(N-Alkyl- and -Acyl-amino)-1,2,4-triazole-3-thione Analogs as Metallo-Beta-Lactamase Inhibitors: Impact of 4-Linker on Potency and Spectrum of Inhibition

المؤلفون: Gavara, L., Verdirosa, F., Legru, A., Mercuri, Paola, Nauton, L., Sevaille, L., Feller, Georges, Berthomieu, D., Sannio, F., Marcoccia, F., Tanfoni, S., De Luca, F., Gresh, N., Galleni, Moreno, Docquier, Jean-Denis, Hernandez, J.-F.

المصدر: Biomolecules, 10 (8), 1094 (2020)

مصطلحات موضوعية: Life sciences, Biochemistry, biophysics & molecular biology, Microbiology, Sciences du vivant, Biochimie, biophysique & biologie moléculaire, Microbiologie

Relation: urn:issn:2218-273X

URL الوصول: https://orbi.uliege.be/handle/2268/249795

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5

Academic Journal

4-Amino-1,2,4-triazole-3-thione-derived Schiff bases as metallo-beta-lactamase inhibitors

المصدر: European Journal of Medicinal Chemistry, 208, 112720 (2020)

مصطلحات موضوعية: Life sciences, Biochemistry, biophysics & molecular biology, Microbiology, Sciences du vivant, Biochimie, biophysique & biologie moléculaire, Microbiologie

Relation: urn:issn:0223-5234; urn:issn:1768-3254

URL الوصول: https://orbi.uliege.be/handle/2268/249902

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6

Academic Journal

Zidovudine-β-lactam pronucleoside strategy for selective delivery into Gram-negative bacteria triggered by β-lactamases

المؤلفون: ROSALES-HURTADO, M., Sannio, F., Lari, L., Verdirosa, F., Feller, Georges, Carretero, E., Vo Hoang, Y., Licznar-Fajardo, P., Docquier, Jean-Denis, Gavara, L.

المصدر: ACS Infectious Diseases, 9, 1546-1557 (2023)

مصطلحات موضوعية: Life sciences, Biochemistry, biophysics & molecular biology, Sciences du vivant, Biochimie, biophysique & biologie moléculaire

Relation: urn:issn:2373-8227; https://orbi.uliege.be/handle/2268/304845; info:hdl:2268/304845; info:pmid:37439673

الاتاحة: https://orbi.uliege.be/handle/2268/304845
https://doi.org/10.1021/acsinfecdis.3c00110

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7

Academic Journal

Optimization of 1,2,4-triazole-3-thiones towards broad-spectrum metallo-β-lactamase inhibitors showing potent synergistic activity on VIM- and NDM-1-producing clinical isolates

المصدر: Journal of Medicinal Chemistry (2022)

مصطلحات موضوعية: Life sciences, Biochemistry, biophysics & molecular biology, Sciences du vivant, Biochimie, biophysique & biologie moléculaire

Relation: urn:issn:0022-2623; urn:issn:1520-4804; https://orbi.uliege.be/handle/2268/296522; info:hdl:2268/296522

الاتاحة: https://orbi.uliege.be/handle/2268/296522

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8

Academic Journal

Intermolecular interactions of the extended recognition site of VIM-2 metallo-β-lactamase with 1,2,4-triazole-3-thione inhibitors. Validations of a polarizable molecular mechanics potential by ab initio QC

المؤلفون: Kwapien K., Gavara L., Docquier J. D., Berthomieu D., Hernandez J. -F., Gresh N.

المساهمون: Kwapien, K., Gavara, L., Docquier, J. D., Berthomieu, D., Hernandez, J. -F., Gresh, N.

مصطلحات موضوعية: 1,2,4-triazole-3-thione inhibitor, ab initio quantum chemistry, intermolecular interaction, metallo-β-lactamase, polarizable molecular mechanics

وصف الملف: STAMPA

Relation: info:eu-repo/semantics/altIdentifier/pmid/33169865; info:eu-repo/semantics/altIdentifier/wos/WOS:000587727200001; volume:42; issue:2; firstpage:86; lastpage:106; numberofpages:21; journal:JOURNAL OF COMPUTATIONAL CHEMISTRY; http://hdl.handle.net/11365/1125161; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85096766562

الاتاحة: http://hdl.handle.net/11365/1125161
https://doi.org/10.1002/jcc.26437
https://onlinelibrary.wiley.com/doi/10.1002/jcc.26437

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9

Academic Journal

4-Amino-1,2,4-triazole-3-thione-derived Schiff bases as metallo-β-lactamase inhibitors

المؤلفون: Gavara L., Sevaille L., De Luca F., Mercuri P., Bebrone C., Feller G., Legru A., Cerboni G., Tanfoni S., Baud D., Cutolo G., Bestgen B., Chelini G., Verdirosa F., Sannio F., Pozzi C., Benvenuti M., Kwapien K., Fischer M., Becker K., Frere J. -M., Mangani S., Gresh N., Berthomieu D., Galleni M., Docquier JD, Hernandez J. -F.

المساهمون: Gavara, L., Sevaille, L., De Luca, F., Mercuri, P., Bebrone, C., Feller, G., Legru, A., Cerboni, G., Tanfoni, S., Baud, D., Cutolo, G., Bestgen, B., Chelini, G., Verdirosa, F., Sannio, F., Pozzi, C., Benvenuti, M., Kwapien, K., Fischer, M., Becker, K., Frere, J. -M., Mangani, S., Gresh, N., Berthomieu, D., Galleni, M., Docquier, Jd, Hernandez, J. -F.

مصطلحات موضوعية: Metallo-b-Lactamase, 1,2,4-Triazole-3-thione, Schiff bases, Bacterial resistance, b-lactam antibiotic

وصف الملف: ELETTRONICO

Relation: info:eu-repo/semantics/altIdentifier/pmid/32937203; info:eu-repo/semantics/altIdentifier/wos/WOS:000600384300009; volume:208; numberofpages:22; journal:EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY; https://hdl.handle.net/11365/1120638; https://www.sciencedirect.com/science/article/pii/S0223523420306929

الاتاحة: https://hdl.handle.net/11365/1120638
https://doi.org/10.1016/j.ejmech.2020.112720
https://www.sciencedirect.com/science/article/pii/S0223523420306929

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