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1Academic Journal
المؤلفون: Baburajeev, C.P., Mohan, C.D., Rangappa, S., Mason, D.J., Fuchs, J.E., Bender, A., Barash, U., Vlodavsky, I., Basappa, ., Rangappa, K.S.
مصطلحات موضوعية: Chemistry
وصف الملف: text
Relation: http://eprints-bangaloreuniversity.in/8213/1/baburajeev2017.pdf; Baburajeev, C.P. and Mohan, C.D. and Rangappa, S. and Mason, D.J. and Fuchs, J.E. and Bender, A. and Barash, U. and Vlodavsky, I. and Basappa, . and Rangappa, K.S. (2017) Identification of Novel Class of Triazolo-Thiadiazoles as Potent Inhibitors of Human Heparanase and their Anticancer Activity. BMC Cancer, 17 (1). ISSN 14712407
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2Academic Journal
المؤلفون: Subramanian, G., Babu Rajeev, C.P., Mohan, C.D., Sinha, A., Chu, T.T., Anusha, S., Ximei, H., Fuchs, J.E.
مصطلحات موضوعية: Chemistry
وصف الملف: text
Relation: http://eprints-bangaloreuniversity.in/7505/1/GOWTHAM.pdf; Subramanian, G. and Babu Rajeev, C.P. and Mohan, C.D. and Sinha, A. and Chu, T.T. and Anusha, S. and Ximei, H. and Fuchs, J.E. (2016) Synthesis and in vitro evaluation of hydrazinyl phthalazines against malaria parasite, Plasmodium falciparum. Bioorganic & Medicinal Chemistry Letters, 26 (14). pp. 3300-3306. ISSN 1464-3405
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3Academic Journal
المؤلفون: Keerthy, H.K., Vivek, H.K., Bharathkumar, H., Rangappa, S., Bulusu, K.C., Mervin, L.H., Fuchs, J.E., Priya, B.S., Basappa, N., Swamy, A.S., Bender, A., Rangappa, K.S.
مصطلحات موضوعية: Chemistry
وصف الملف: text
Relation: http://eprints-bangaloreuniversity.in/3972/1/MOLPRINT%202D%20based%20identification%20and%20synthesis%20of%20n.pdf; Keerthy, H.K. and Vivek, H.K. and Bharathkumar, H. and Rangappa, S. and Bulusu, K.C. and Mervin, L.H. and Fuchs, J.E. and Priya, B.S. and Basappa, N. and Swamy, A.S. and Bender, A. and Rangappa, K.S. (2016) Molprint 2D-Based Identification and Synthesis of Novel Chromene Based Small Molecules that Target Pla2: Validation through Chemo-And Bioinformatics Approaches. RSC Advances, 5 (109). pp. 89797-89808. ISSN 20462069
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4Academic Journal
المؤلفون: Neelgundmath, M., Dinesh, K.R., Mohan, C.D., Li, F., Dai, X., Siveen, K.S., Paricharak, S., Mason, D.J., Fuchs, J.E., Sethi, G., Bender, A., Rangappa, K.S., Kotresh, O., Basappa
Relation: http://www.sciencedirect.com/science/article/pii/S0960894X14013730; lucris-id: 12731651; https://hdl.handle.net/1887/3197451
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5Academic Journal
المؤلفون: Baburajeev, C.P, Dhananjaya Mohan, C, Ananda, H, Rangappa, S, Fuchs, J.E, Jagadish, S, Sivaraman Siveen, K, Chinnathambi, A, Ali Alharbi, S, Zayed, M.E, Zhang, J, Li, F, Sethi, G, Girish, K.S, Bender, A, Basappa, Rangappa, K.S
المساهمون: DEPT OF PHARMACOLOGY, CANCER SCIENCE INSTITUTE OF SINGAPORE
المصدر: Unpaywall 20200831
مصطلحات موضوعية: 6-(2-benzylphenyl)-3-phenyl-(1,2,4)triazolo(3)(1,3,4)thiadiazole, antineoplastic agent, benzofuran derivative, BIRC5 protein, human, caspase 3, chromone derivative, cyclin D1, inhibitor of apoptosis protein, nicotinamide adenine dinucleotide adenosine diphosphate ribosyltransferase, protein bcl 2, protein tyrosine phosphatase 1B, PTPN1 protein, sanggenone C, STAT3 protein, thiadiazole derivative, triazole derivative, animal, antagonists and inhibitors, biosynthesis, Carcinoma, Ehrlich Tumor, Hepatocellular, cell motion, disease model, dose response, drug effects, female, G1 phase cell cycle checkpoint, Hep-G2 cell line
Relation: Baburajeev, C.P, Dhananjaya Mohan, C, Ananda, H, Rangappa, S, Fuchs, J.E, Jagadish, S, Sivaraman Siveen, K, Chinnathambi, A, Ali Alharbi, S, Zayed, M.E, Zhang, J, Li, F, Sethi, G, Girish, K.S, Bender, A, Basappa, Rangappa, K.S (2015). Development of novel triazolo-thiadiazoles from heterogeneous "green" catalysis as protein tyrosine phosphatase 1B inhibitors. Scientific Reports 5 : 14195. ScholarBank@NUS Repository. https://doi.org/10.1038/srep14195; https://scholarbank.nus.edu.sg/handle/10635/175483
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6Academic Journal
المؤلفون: Bharathkumar, H., Mohan, C.D., Ananda, H., Li, F., Fuchs, J.E., Rangappa, S., Surender, M., Bulusu, K.C., Girish, K.S., Sethi, G., Bender, A., Basappab, ., Rangappa, K.S.
مصطلحات موضوعية: Chemistry
وصف الملف: text
Relation: http://eprints-bangaloreuniversity.in/6934/1/bharath%20kumar.pdf; Bharathkumar, H. and Mohan, C.D. and Ananda, H. and Li, F. and Fuchs, J.E. and Rangappa, S. and Surender, M. and Bulusu, K.C. and Girish, K.S. and Sethi, G. and Bender, A. and Basappab, . and Rangappa, K.S. (2015) Microwave-assisted synthesis, characterization and cytotoxic studies of novel estrogen receptor alpha ligands towards human breast cancer cells. Bioorganic and Medicinal Chemistry Letters, 25 (8). pp. 1804-1807. ISSN 0960-894X
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7Academic Journal
المؤلفون: Anilkumar, N.C., Sundaram, M.S., Mohan, C.D., Rangappa, S., Bulusu, K.C., Fuchs, J.E., Girish, K.S., Bender, A., Basappa, ., Rangappa, K.S.
مصطلحات موضوعية: Chemistry
وصف الملف: text
Relation: http://eprints-bangaloreuniversity.in/4031/1/A%20One%20Pot%20Synthesis%20of%20Novel%20Bioactive%20Tri-.pdf; Anilkumar, N.C. and Sundaram, M.S. and Mohan, C.D. and Rangappa, S. and Bulusu, K.C. and Fuchs, J.E. and Girish, K.S. and Bender, A. and Basappa, . and Rangappa, K.S. (2015) A One Pot Synthesis of Novel Bioactive Tri-Substitute-Condensed-Imidazopyridines that Targets Snake Venom Phospholipase A2. PLoS ONE. p. 20131896. ISSN 19326203
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8Academic Journal
المؤلفون: Anusha, S., Baburajeev, C.P., Mohan, C.D., Mathai, J., Rangappa, S., Mohan, S., Chandra, ., Paricharak, S., Mervin, L., Fuchs, J.E., Mahedra, M., Bender, A., Rangappa, K.S.
مصطلحات موضوعية: Chemistry
وصف الملف: text
Relation: http://eprints-bangaloreuniversity.in/3973/1/A%20Nano-MgO%20and%20Ionic%20Liquid-Catalyzed.pdf; Anusha, S. and Baburajeev, C.P. and Mohan, C.D. and Mathai, J. and Rangappa, S. and Mohan, S. and Chandra, . and Paricharak, S. and Mervin, L. and Fuchs, J.E. and Mahedra, M. and Bender, A. and Rangappa, K.S. (2015) A Nano-Mgo and Ionic Liquid-Catalyzed ‘Green’ Synthesis Protocol for the Development of Adamantyl-Imidazolo-Thiadiazoles as Anti-Tuberculosis Agents Targeting Sterol 14α-Demethylase (CYP51). PLoS ONE, 10 (10). pp. 1-12. ISSN 19326203
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9Academic Journal
المؤلفون: Anusha, S., Sinha, A., Babu Rajeev, C.P., Chu, T.T.T., Mathai, J., Ximei, H., Fuchs, J.E., Shivananju, N., Bender, A., Preiser, P.R., Rangappa, K.S., Basappa, S., Chandramohanadas, R.
مصطلحات موضوعية: Chemistry
وصف الملف: text
Relation: http://eprints-bangaloreuniversity.in/3323/1/c5ob01479d.pdf; Anusha, S. and Sinha, A. and Babu Rajeev, C.P. and Chu, T.T.T. and Mathai, J. and Ximei, H. and Fuchs, J.E. and Shivananju, N. and Bender, A. and Preiser, P.R. and Rangappa, K.S. and Basappa, S. and Chandramohanadas, R. (2015) Synthesis, characterization and in vitro evaluation of novel enantiomerically-pure sulphonamide antimalarials. Organic and Biomolecular Chemistry, 13 (43). pp. 10681-10690. ISSN 14770520
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10Academic Journal
المؤلفون: Srinivas, V., Mohan, C.D., Baburajeev, C.P., Rangappa, S., Jagadish, S., Fuchs, J.E., Sukhorukov, A.Y., Chandra, ., Mason, D.J., Sharath Kumar, K.S., Madegowda, M., Bender, A., Basappa, ., Rangappa, K.S.
مصطلحات موضوعية: Chemistry
وصف الملف: text
Relation: http://eprints-bangaloreuniversity.in/3302/1/Synthesis%20and%20characterization%20of%20novel%20oxazines%20and%20demonstration.pdf; Srinivas, V. and Mohan, C.D. and Baburajeev, C.P. and Rangappa, S. and Jagadish, S. and Fuchs, J.E. and Sukhorukov, A.Y. and Chandra, . and Mason, D.J. and Sharath Kumar, K.S. and Madegowda, M. and Bender, A. and Basappa, . and Rangappa, K.S. (2015) Synthesis and characterization of novel oxazines and demonstration that they specifically target cyclooxygenase 2. Bioorganic and Medicinal Chemistry Letters, 25 (15). pp. 2931-2936. ISSN 0960-894X
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11Academic Journal
المؤلفون: Bharathkumar, H., Mohan, C.D., Ananda, H., Fuchs, J.E., Li, F., Rangappa, S., Surender, M., Bulusu, K.C., Girish, K.S., Sethi, G., Bender, A., Basappa, ., Rangappa, K.S.
مصطلحات موضوعية: Chemistry
وصف الملف: text
Relation: http://eprints-bangaloreuniversity.in/3293/1/Microwave-assisted%20synthesis,%20characterization%20and%20cytotoxic%20studies.pdf; Bharathkumar, H. and Mohan, C.D. and Ananda, H. and Fuchs, J.E. and Li, F. and Rangappa, S. and Surender, M. and Bulusu, K.C. and Girish, K.S. and Sethi, G. and Bender, A. and Basappa, . and Rangappa, K.S. (2015) Microwave-assisted synthesis, characterization and cytotoxic studies of novel estrogen receptor α ligands towards human breast cancer cells. Bioorganic and Medicinal Chemistry Letters, 25 (8). pp. 1804-1807. ISSN 0960-894X
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12Academic Journal
المؤلفون: Bharathkumar, H., Mohan, C.D., Rangappa, S., Kang, T., Keerthy, H.K., Fuchs, J.E., Kwon, N.H., Bender, A., Kim, S., Basappaa, ., Rangappa, K.S.
مصطلحات موضوعية: Chemistry
وصف الملف: text
Relation: http://eprints-bangaloreuniversity.in/3271/1/Screening%20of%20Quinoline,%201,3-Benzoxazine,%20and%201,3-Oxazine-based%20Small%20Molecules%20Against.pdf; Bharathkumar, H. and Mohan, C.D. and Rangappa, S. and Kang, T. and Keerthy, H.K. and Fuchs, J.E. and Kwon, N.H. and Bender, A. and Kim, S. and Basappaa, . and Rangappa, K.S. (2015) Screening of quinoline, 1,3-benzoxazine, and 1,3-oxazine-based small molecules against isolated methionyl-tRNA synthetase and A549 and HCT116 cancer cells including an in silico binding mode analysis. Organic and Biomolecular Chemistry, 13 (36). pp. 9381-9387. ISSN 14770520
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13Academic Journal
المؤلفون: Ashwini, N., Garg, M., Mohan, C.D., Fuchs, J.E., Rangappa, S., Anusha, S., Swaroop, T.R., Rakesh, K.S., Kanojia, D, Madan, V., Bender, A., Koeffler, H.P., Basappa, ., Rangappa, K.S.
مصطلحات موضوعية: Chemistry
وصف الملف: text
Relation: http://eprints-bangaloreuniversity.in/3250/1/Synthesis%20of%201,2-Benzisoxazole%20Tethered%201,2,3-Triazoles%20That%20Exhibit.pdf; Ashwini, N. and Garg, M. and Mohan, C.D. and Fuchs, J.E. and Rangappa, S. and Anusha, S. and Swaroop, T.R. and Rakesh, K.S. and Kanojia, D and Madan, V. and Bender, A. and Koeffler, H.P. and Basappa, . and Rangappa, K.S. (2015) Synthesis of 1,2-benzisoxazole tethered 1,2,3-triazoles that exhibit anticancer activity in acute myeloid leukemia cell lines by inhibiting histone deacetylases, and inducing p21 and tubulin acetylation. Bioorganic and Medicinal Chemistry, 23 (18). pp. 6157-6165. ISSN 09680896
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14Academic Journal
المؤلفون: Baburajeev, C.P., Dhananjaya Mohan, C., Ananda, H., Rangappa, S., Fuchs, J.E., Jagadish, S., Sivaraman Siveen, K., Chinnathambi, A., Ali Alharbi, S., Zayed, M.E., Zhang, J., Li, F., Sethi, G., Girish, K.S., Bender, A., Basappaa, ., Rangappa, K.S.
مصطلحات موضوعية: Chemistry
وصف الملف: text
Relation: http://eprints-bangaloreuniversity.in/3248/1/Development%20of%20Novel%20TriazoloThiadiazoles.pdf; Baburajeev, C.P. and Dhananjaya Mohan, C. and Ananda, H. and Rangappa, S. and Fuchs, J.E. and Jagadish, S. and Sivaraman Siveen, K. and Chinnathambi, A. and Ali Alharbi, S. and Zayed, M.E. and Zhang, J. and Li, F. and Sethi, G. and Girish, K.S. and Bender, A. and Basappaa, . and Rangappa, K.S. (2015) Development of novel triazolo-thiadiazoles from heterogeneous "green" catalysis as protein tyrosine phosphatase 1B inhibitors. Scientific Reports, 5. ISSN 20452322
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15
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16Academic Journal
المؤلفون: Bharathkumar, H, Paricharak, S, Dinesh, K.R, Siveen, K.S, Fuchs, J.E, Rangappa, S, Mohan, C.D, Mohandas, N, Kumar, A.P, Sethi, G, Bender, A, Basappa, Laboratory of Chemical Biology, Department of Chemistry, Bangalore University, Palace Road, Bangalore, 560001, India, Rangappa, K.S
المساهمون: CANCER SCIENCE INSTITUTE OF SINGAPORE, ANATOMY, PHARMACOLOGY
المصدر: Unpaywall 20200831
مصطلحات موضوعية: Biological evaluation, In-silico, In-vitro
Relation: Bharathkumar, H, Paricharak, S, Dinesh, K.R, Siveen, K.S, Fuchs, J.E, Rangappa, S, Mohan, C.D, Mohandas, N, Kumar, A.P, Sethi, G, Bender, A, Basappa, Laboratory of Chemical Biology, Department of Chemistry, Bangalore University, Palace Road, Bangalore, 560001, India, Rangappa, K.S (2014). Synthesis, biological evaluation and in silico and in vitro mode-of-action analysis of novel dihydropyrimidones targeting PPAR-γ. RSC Advances 4 (85) : 45143-45146. ScholarBank@NUS Repository. https://doi.org/10.1039/c4ra08713e; https://scholarbank.nus.edu.sg/handle/10635/176019
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17Academic Journal
المؤلفون: Bharathkumar, H., Paricharak, S., Dinesh, K.R., Siveen, K.S, Fuchs, J.E, Rangappa, S., Mohan, C.D., Mohandas, N., Kumar, A.P., Sethi, G., Bender, A., Basappa, ., Rangappa, K.S.
مصطلحات موضوعية: Chemistry
وصف الملف: text
Relation: http://eprints-bangaloreuniversity.in/3221/1/Synthesis,%20biological%20evaluation%20and%20in%20silico%20and%20in.pdf; Bharathkumar, H. and Paricharak, S. and Dinesh, K.R. and Siveen, K.S and Fuchs, J.E and Rangappa, S. and Mohan, C.D. and Mohandas, N. and Kumar, A.P. and Sethi, G. and Bender, A. and Basappa, . and Rangappa, K.S. (2014) Synthesis, biological evaluation and in silico and in vitro mode-of-action analysis of novel dihydropyrimidones targeting PPAR-γ. RSC Advances, 4 (85). pp. 45143-45146. ISSN 20462069
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18Academic Journal
المؤلفون: Kumar Keerthy, H., Mohan, C.D., Siveen, K.S., Fuchs, J.E., Rangappa, S., Sundaram, M.S., Li, F., Girish, K.S., Sethi, G., Basappaa, ., Bender, A., Rangappa, K.S.
مصطلحات موضوعية: Chemistry
وصف الملف: text
Relation: http://eprints-bangaloreuniversity.in/3109/1/novel.pdf; Kumar Keerthy, H. and Mohan, C.D. and Siveen, K.S. and Fuchs, J.E. and Rangappa, S. and Sundaram, M.S. and Li, F. and Girish, K.S. and Sethi, G. and Basappaa, . and Bender, A. and Rangappa, K.S. (2014) Novel Synthetic Biscoumarins Target Tumor Necrosis Factor- in Hepatocellular Carcinoma in Vitro and in Vivo*. Journal of Biological Chemistry, 289 (46). pp. 31879-31890. ISSN 1083-351X
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19Academic Journal
المؤلفون: Mohan, C.D., Bharathkumar, H., Bulusu, K.C., Pandey, V., Rangappa, S., Fuchs, J.E., Shanmugam, M.K., Dai, X., Li, F., Deivasigamani, A., Hui, K.M., Kumar, A.P., Lobie, P.E., Bender, A., Basappab, ., Sethi, G., Rangappa, K.S.
مصطلحات موضوعية: Chemistry
وصف الملف: text
Relation: http://eprints-bangaloreuniversity.in/3108/1/Development%20of%20a%20Novel%20Azaspirane%20That%20Targets%20the%20Janus.pdf; Mohan, C.D. and Bharathkumar, H. and Bulusu, K.C. and Pandey, V. and Rangappa, S. and Fuchs, J.E. and Shanmugam, M.K. and Dai, X. and Li, F. and Deivasigamani, A. and Hui, K.M. and Kumar, A.P. and Lobie, P.E. and Bender, A. and Basappab, . and Sethi, G. and Rangappa, K.S. (2014) Development of a novel azaspirane that targets the Janus Kinase-signal transducer and activator of transcription (STAT) pathway in hepatocellular carcinoma in vitro and in vivo. Journal of Biological Chemistry, 289 (49). pp. 34296-34307. ISSN 00219258
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20
المؤلفون: Ackaert, C., Kofler, S., Horejs-Hoeck, J., Zulehner, N., Asam, C., von Grafenstein, S., Fuchs, J.E., Briza, P., Liedl, K.R., Bohle, B., Ferreira, F., Brandstetter, H., Oostingh, G.J., Duschl, A.
المصدر: 'PloS One ', vol: 9, pages: e104520-1-e104520-11 (2014)
وصف الملف: application/pdf