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1Academic Journal
المؤلفون: Jolita Bruzgulienė, Greta Račkauskienė, Aurimas Bieliauskas, Vaida Milišiūnaitė, Miglė Dagilienė, Gita Matulevičiūtė, Vytas Martynaitis, Sonata Krikštolaitytė, Frank A. Sløk, Algirdas Šačkus
المصدر: Beilstein Journal of Organic Chemistry, Vol 18, Iss 1, Pp 102-109 (2022)
مصطلحات موضوعية: β-enamino ketoesters, heterocyclic amino acids, 15n-labeled 1,2-oxazole, nmr (1h, 13c, 15n), 1,2-oxazole (isoxazole), x-ray structure analysis, Science, Organic chemistry, QD241-441
وصف الملف: electronic resource
Relation: https://doaj.org/toc/1860-5397
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2Academic Journal
المؤلفون: Emilis Gudelis, Sonata Krikštolaitytė, Monika Stančiauskaitė, Urtė Šachlevičiūtė, Aurimas Bieliauskas, Vaida Milišiūnaitė, Rokas Jankauskas, Neringa Kleizienė, Frank A. Sløk, Algirdas Šačkus
المصدر: Molecules, Vol 28, Iss 3, p 1091 (2023)
مصطلحات موضوعية: azetidine, oxetane, heterocyclic amines, heterocyclic amino acids, aza-Michael addition, Suzuki–Miyaura cross-coupling reaction, Organic chemistry, QD241-441
وصف الملف: electronic resource
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3Academic Journal
المؤلفون: Karolina Dzedulionytė, Paulina Voznikaitė, Aurimas Bieliauskas, Vida Malinauskienė, Frank A. Sløk, Algirdas Šačkus
المصدر: Molbank, Vol 2021, Iss 2, p M1207 (2021)
مصطلحات موضوعية: azetidine, 1,3-selenazole, heterocyclic amino acids, Hantzsch synthesis, Inorganic chemistry, QD146-197
وصف الملف: electronic resource
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4Academic Journal
المؤلفون: Gita Matulevičiūtė, Eglė Arbačiauskienė, Neringa Kleizienė, Vilija Kederienė, Greta Ragaitė, Miglė Dagilienė, Aurimas Bieliauskas, Vaida Milišiūnaitė, Frank A. Sløk, Algirdas Šačkus
المصدر: Molecules, Vol 26, Iss 13, p 3808 (2021)
مصطلحات موضوعية: heterocyclic amino acids, pyrazoles, piperidines, β-keto esters, enamines, hydrazines, Organic chemistry, QD241-441
وصف الملف: electronic resource
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5Academic Journal
المؤلفون: Lars K. Petersen (10136877), Allan B. Christensen (10136880), Jacob Andersen (1368906), Charlotta G. Folkesson (5704343), Ole Kristensen (258994), Charlotte Andersen (769079), Amaya Alzu (10136883), Frank A. Sløk (3013266), Peter Blakskjær (1265859), Daniel Madsen (6105128), Carlos Azevedo (3964760), Iolanda Micco (2020078), Nils J. V. Hansen (10136886)
مصطلحات موضوعية: Biophysics, Biochemistry, Cell Biology, Genetics, Molecular Biology, Pharmacology, Biotechnology, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, oocyte, screening, 100 000 times, Living Cell DNA-encoded, digit nanomolar potencies, 1 μ L, protein targets, ACSS, frog Xenopus laevis, DEL members binding, target protein
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6
المؤلفون: Algirdas Šačkus, Vilija Kederienė, Eglė Arbačiauskienė, Greta Ragaitė, Neringa Kleizienė, Aurimas Bieliauskas, Gita Matulevičiūtė, Vaida Milišiūnaitė, Frank A. Sløk, Miglė Dagilienė
المساهمون: MDPI AG (Basel, Switzerland)
المصدر: Molecules, Vol 26, Iss 3808, p 3808 (2021)
Molecules
Volume 26
Issue 13مصطلحات موضوعية: β-keto esters, Hydrazine, Pharmaceutical Science, Halide, Organic chemistry, Pyrazole, 010402 general chemistry, 01 natural sciences, Medicinal chemistry, Analytical Chemistry, building blocks, Dimethyl acetal, chemistry.chemical_compound, QD241-441, heterocyclic amino acids, Drug Discovery, piperidines, Physical and Theoretical Chemistry, enamines, Alkyl, chemistry.chemical_classification, hydrazines, 010405 organic chemistry, Tautomer, pyrazoles, 0104 chemical sciences, Amino acid, chemistry, Chemistry (miscellaneous), Molecular Medicine, Hydrate
وصف الملف: application/pdf
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7
المؤلفون: Charlotte Andersen, Iolanda Micco, Daniel Madsen, Peter Blakskjaer, Amaya Alzu, Jacob Andersen, Ole Kristensen, Lars Kjerulf Petersen, Charlotta G. Folkesson, Frank Abildgaard Sløk, Carlos Azevedo, Allan Beck Christensen, Nils Jakob Vest Hansen
المصدر: Journal of the American Chemical Society. 143(7)
مصطلحات موضوعية: African clawed frog, Somatic cell, Cell, Xenopus, Acetate-CoA Ligase, 010402 general chemistry, 01 natural sciences, Biochemistry, Catalysis, Mitogen-Activated Protein Kinase 14, Small Molecule Libraries, chemistry.chemical_compound, Xenopus laevis, Colloid and Surface Chemistry, medicine, Animals, Humans, biology, Chemistry, Dock5, General Chemistry, DNA, biology.organism_classification, 0104 chemical sciences, Cell biology, medicine.anatomical_structure, biology.protein, Oocytes, Target protein
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8
المؤلفون: Vida Malinauskienė, Aurimas Bieliauskas, Aistė Kveselytė, Karolina Dzedulionytė, Frank A. Sløk, Saulius Burinskas, Algirdas Šačkus
المصدر: Chemistry of Heterocyclic Compounds. 54:469-473
مصطلحات موضوعية: chemistry.chemical_classification, 010405 organic chemistry, Stereochemistry, Carboxylic acid, Selenourea, Organic Chemistry, Substituent, Nuclear magnetic resonance spectroscopy, 010402 general chemistry, Ring (chemistry), 01 natural sciences, 0104 chemical sciences, Amino acid, chemistry.chemical_compound, chemistry, Functional group, N-Bromosuccinimide
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9
المؤلفون: Paulina Voznikaitė, Vida Malinauskienė, Karolina Dzedulionytė, Algirdas Šačkus, Aurimas Bieliauskas, Frank A. Sløk
المساهمون: MDPI AG (Basel, Switzerland)
المصدر: Molbank, Vol 2021, Iss M1207, p M1207 (2021)
مصطلحات موضوعية: chemistry.chemical_classification, 010405 organic chemistry, Stereochemistry, Organic Chemistry, Azetidine, 010402 general chemistry, 01 natural sciences, Biochemistry, Cycloaddition, 0104 chemical sciences, Amino acid, chemistry.chemical_compound, 1,3-selenazole, chemistry, Elemental analysis, heterocyclic amino acids, Carboxylate, azetidine, Physical and Theoretical Chemistry, Inorganic chemistry, QD146-197, Hantzsch synthesis
وصف الملف: application/pdf
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10
المؤلفون: Diana Bričkutė, Osvaldas Paliulis, Algirdas Šačkus, Frank A. Sløk
المصدر: Journal of Heterocyclic Chemistry. 52:1032-1036
مصطلحات موضوعية: chemistry.chemical_compound, Hydrolysis, Chiral auxiliary, Propanoic acid, Malonate, chemistry, Stereochemistry, Organic Chemistry, Halogenation, Ring (chemistry), Thiazole
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11
المؤلفون: Ulla Geneser, Tine B. Stensbøl, Jeremy R. Greenwood, Birgitte Nielsen, Jan Egebjerg, Mikael Begtrup, Frank A. Sløk, Hans Bräuner-Osborne, Mai Marie Holm, Povl Krogsgaard-Larsen, Lotte Brehm
المصدر: Chirality. 16:452-466
مصطلحات موضوعية: musculoskeletal diseases, Pharmacology, Agonist, Kainic acid, Stereochemistry, medicine.drug_class, Organic Chemistry, AMPA receptor, Catalysis, Analytical Chemistry, Chiral column chromatography, chemistry.chemical_compound, Metabotropic receptor, chemistry, immune system diseases, Drug Discovery, medicine, Enantiomer, Metabotropic glutamate receptor 2, skin and connective tissue diseases, Receptor, Spectroscopy
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12
المؤلفون: Algirdas akus, Diana Brikutė, Frank A. Sløk, Christian Rømming
المصدر: Journal of the Chemical Society, Perkin Transactions 1. :652-656
مصطلحات موضوعية: chemistry.chemical_compound, Hydrolysis, Nucleophile, Thiourea, chemistry, Bromide, Organic chemistry, Molecule, Azide, Crystal structure, Medicinal chemistry, Ion
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13
المصدر: Tetrahedron. 57:2195-2201
مصطلحات موضوعية: Chemistry, Organic Chemistry, Biochemistry, Medicinal chemistry, Coupling reaction, Stille reaction, Benzaldehyde, chemistry.chemical_compound, Benzoyl chloride, Bromide, Heck reaction, Drug Discovery, Palladium-catalyzed coupling reactions, Isoxazole
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14
المؤلفون: Tommy N. Johansen, Tine B. Stensbøl, Hans Brünum, Karla Frydenvang, Birgitte Nielsen, Stine B. Vogensen, Ulf Madsen, Povl Krogsgaard-Larsen, uner‐Osborne, Frank A. Sløk
المصدر: Chirality. 13:523-532
مصطلحات موضوعية: musculoskeletal diseases, Pharmacology, Agonist, Eudysmic ratio, Kainic acid, Stereochemistry, medicine.drug_class, Organic Chemistry, AMPA receptor, Catalysis, Analytical Chemistry, Chiral column chromatography, chemistry.chemical_compound, Metabotropic receptor, chemistry, immune system diseases, Drug Discovery, medicine, NMDA receptor, skin and connective tissue diseases, Receptor, Spectroscopy
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15
المؤلفون: Lisbeth Eriksen, Frank A. Sløk, Ulf Madsen, Miguel V. Poulsen, Povl Krogsgaard-Larsen, Hans Bräuner-Osborne, Tine B. Stensbøl, Hans-Christian H Lützhøft
المصدر: European Journal of Medicinal Chemistry. 35:69-76
مصطلحات موضوعية: Agonist, N-Methylaspartate, medicine.drug_class, Stereochemistry, AMPA receptor, Pharmacology, Receptors, N-Methyl-D-Aspartate, Quinoxalines, Drug Discovery, medicine, Animals, Receptors, AMPA, alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid, Cerebral Cortex, Chemistry, Organic Chemistry, Antagonist, Isoxazoles, General Medicine, Rats, Electrophysiology, Metabotropic receptor, Receptors, Glutamate, Competitive antagonist, Excitatory Amino Acid Antagonists, NMDA receptor, Propionates, Ionotropic effect
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16
المؤلفون: Connie Kjøller, Nils Henrik Diemer, Povl Krogsgaard-Larsen, Tine B. Stensbøl, Ulf Madsen, Joseph D. Trometer, Jan Egebjerg, Stephen D. Hurt, Bjarke Ebert, Frank A. Sløk
المصدر: European Journal of Pharmacology. 373:251-262
مصطلحات موضوعية: musculoskeletal diseases, Pharmacology, Agonist, Kainic acid, education.field_of_study, medicine.drug_class, Stereochemistry, Population, AMPA receptor, Dissociation constant, chemistry.chemical_compound, nervous system, chemistry, Mechanism of action, Biochemistry, medicine, Radioligand, medicine.symptom, skin and connective tissue diseases, Receptor, education
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17
المؤلفون: Tommy N. Johansen, Ulf Madsen, Tine B. Stensbøl, Povl Krogsgaard-Larsen, Frank A. Sløk, Haleh Ahmadian, Birgitte Nielsen, Naohiro Sekiyama, Hans Bräuner-Osborne, Shigetada Nakanishi
المصدر: Journal of Medicinal Chemistry. 40:3700-3705
مصطلحات موضوعية: Agonist, Magnetic Resonance Spectroscopy, medicine.drug_class, Stereochemistry, CHO Cells, AMPA receptor, In Vitro Techniques, Phosphatidylinositols, Receptors, Metabotropic Glutamate, Membrane Potentials, Cricetinae, Drug Discovery, Cyclic AMP, Excitatory Amino Acid Agonists, medicine, Animals, Receptor, alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid, Chromatography, High Pressure Liquid, Chemistry, Hydrolysis, Stereoisomerism, Glutamic acid, Receptor antagonist, Recombinant Proteins, Rats, Chiral column chromatography, Metabotropic receptor, Molecular Medicine, Enantiomer
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18
المؤلفون: Y. Lang, P. Krogsgaard-Larsen, Frank A. Sløk, Sibylle M. Lenz, Ulf Madsen, Bjarke Ebert
المصدر: European Journal of Medicinal Chemistry. 32:329-338
مصطلحات موضوعية: Pharmacology, Agonist, chemistry.chemical_classification, medicine.drug_class, Stereochemistry, musculoskeletal, neural, and ocular physiology, Organic Chemistry, General Medicine, AMPA receptor, Chemical synthesis, Amino acid, chemistry.chemical_compound, nervous system, chemistry, Drug Discovery, medicine, NMDA receptor, NBQX, Isoxazole, Receptor
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19
المؤلفون: Frank A. Sløk, Bjarke Ebert, Povl Krogsgaard-Larsen, Niels Skjærbæk, Naohiro Sekiyama, Hans Bräuner-Osborne, Shigetada Nakanishi
المصدر: Journal of Medicinal Chemistry. 39:3188-3194
مصطلحات موضوعية: Agonist, Magnetic Resonance Spectroscopy, N-Methylaspartate, Stereochemistry, medicine.drug_class, CHO Cells, AMPA receptor, Receptors, Metabotropic Glutamate, Butyric acid, chemistry.chemical_compound, Cricetinae, Drug Discovery, Aspartic acid, Excitatory Amino Acid Agonists, medicine, Animals, Excitatory Amino Acid Agonist, alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid, Alanine, Hexanoic acid, chemistry.chemical_classification, Dose-Response Relationship, Drug, Molecular Structure, Amino acid, chemistry, Molecular Medicine
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20
المؤلفون: Lotte Brehm, Hans Bräuner-Osborne, Frank A. Sløk, T. N. Johansen, Bjarke Ebert, Trine Meldgaard Lund, Povl Krogsgaard-Larsen, Ulf Madsen
المصدر: European Journal of Medicinal Chemistry. 31:515-537
مصطلحات موضوعية: Pharmacology, chemistry.chemical_classification, Organic Chemistry, Kainate receptor, General Medicine, AMPA receptor, Partial agonist, Amino acid, chemistry.chemical_compound, Metabotropic receptor, chemistry, Drug Discovery, NMDA receptor, Glycine receptor, Ibotenic acid