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1Academic Journal
المؤلفون: Greco, Rosaria, Demartini, Chiara, Zanaboni, Anna Maria, Francavilla, Miriam, Reggiani, Angelo, Realini, Natalia, Scarpelli, Rita, Piomelli, Daniele, Tassorelli, Cristina
المصدر: The Journal of Headache and Pain. 23(1)
مصطلحات موضوعية: Pharmacology and Pharmaceutical Sciences, Biomedical and Clinical Sciences, Neurosciences, Clinical Sciences, Headaches, Pain Research, Migraines, Chronic Pain, Drug Abuse (NIDA only), Substance Misuse, Dental/Oral and Craniofacial Disease, 5.1 Pharmaceuticals, Development of treatments and therapeutic interventions, Amides, Amidohydrolases, Animals, Disease Models, Animal, Endocannabinoids, Hyperalgesia, Inflammation, Male, Migraine Disorders, Nitroglycerin, Pain, Rats, Rats, Sprague-Dawley, FAAH inhibitors, NTG, Trigeminal hyperalgesia, Lipid-derived mediators, Genetics, Neurology & Neurosurgery, Clinical sciences
وصف الملف: application/pdf
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2Academic Journal
المؤلفون: Bala Krishna Prabhala, Jiwan Chettri, Nagalakshmi Irrinki, Abhroop Garg, Rosa Jersie-Christensen, Håvard Jenssen, Biljana Mojsoska, Neeraj Soni, Kristi A. Kohlmeier
المصدر: European Journal of Medicinal Chemistry Reports, Vol 9, Iss , Pp 100111- (2023)
مصطلحات موضوعية: LDT, FAAH inhibitors, FAAH, Lipids, ex vivo model, Oleyl trifluoro methyl ketone, Pharmacy and materia medica, RS1-441, Other systems of medicine, RZ201-999
وصف الملف: electronic resource
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3Academic Journal
المؤلفون: Rosaria Greco, Chiara Demartini, Anna Maria Zanaboni, Miriam Francavilla, Angelo Reggiani, Natalia Realini, Rita Scarpelli, Daniele Piomelli, Cristina Tassorelli
المصدر: The Journal of Headache and Pain, Vol 23, Iss 1, Pp 1-10 (2022)
مصطلحات موضوعية: FAAH inhibitors, NTG, Trigeminal hyperalgesia, Lipid-derived mediators, Medicine
وصف الملف: electronic resource
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4Academic Journal
المؤلفون: Mangiatordi, Giuseppe, Felice, Cavalluzzi, Maria, Maddalena, Delre, Pietro, Lamanna, Giuseppe, Lumuscio, Maria, Cristina, Saviano, Michele, Majoral, Jean-Pierre, Mignani, Serge, Duranti, Andrea, Lentini, Giovanni
المساهمون: Institute of Crystallography (CNR-IC), National Research Council of Italy, Università degli studi di Bari Aldo Moro = University of Bari Aldo Moro (UNIBA), Laboratoire de chimie de coordination (LCC), Institut de Chimie de Toulouse (ICT), Institut de Recherche pour le Développement (IRD)-Université Toulouse III - Paul Sabatier (UT3), Université de Toulouse (UT)-Université de Toulouse (UT)-Institut de Chimie - CNRS Chimie (INC-CNRS)-Centre National de la Recherche Scientifique (CNRS)-Institut National Polytechnique (Toulouse) (Toulouse INP), Université de Toulouse (UT)-Institut de Recherche pour le Développement (IRD)-Université Toulouse III - Paul Sabatier (UT3), Université de Toulouse (UT)-Centre National de la Recherche Scientifique (CNRS), Centre d'Etudes et de Recherche sur le Médicament de Normandie (CERMN), Université de Caen Normandie (UNICAEN), Normandie Université (NU)-Normandie Université (NU), Centro de Química da Madeira, Universidade da Madeira (UMA), Università degli Studi di Urbino 'Carlo Bo', University of Bari Aldo Moro, FCT-Fundação para a Ciência e a Tecnologia, ARDITI-Agência Regional para o Desenvolvimento da Investigação Tecnologia e Inovação, University of Urbino Carlo Bo
المصدر: ISSN: 2227-9059 ; Biomedicines ; https://hal.science/hal-04174953 ; Biomedicines, 2023, 11 (2), pp.469. ⟨10.3390/biomedicines11020469⟩.
مصطلحات موضوعية: Endocannabinoid system, FAAH inhibitors, MGL inhibitors, Repositioning, Drug-likeness, hERG, Ligand efficiency metrics, [CHIM.THER]Chemical Sciences/Medicinal Chemistry, [SDV.NEU.NB]Life Sciences [q-bio]/Neurons and Cognition [q-bio.NC]/Neurobiology
Relation: hal-04174953; https://hal.science/hal-04174953; https://hal.science/hal-04174953/document; https://hal.science/hal-04174953/file/Mangiatordi,%20Endocannabinoid%20Degradation%20Enzyme%20Inhibitors,%202023.pdf
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5Academic Journal
المؤلفون: Duranti, Andrea, Beldarrain González, Gorane, Álvarez Díaz, Antonia Ángeles, Sbriscia, Matilde, Carloni, Silvia, Balduini, Walter, Alonso-Alconada, Daniel
مصطلحات موضوعية: endocannabinoid system, cannabinoid receptors, FAAH inhibitors, MGL inhibitors, neonatal brain injury, hypoxia–ischemia, neuroprotection, neurogenesis
وصف الملف: application/pdf
Relation: https://www.mdpi.com/2227-9059/11/1/28; Biomedicines 11(1) : (2023) // Article ID 28; http://hdl.handle.net/10810/59449
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6Academic Journal
المؤلفون: Greco, Rosaria, Demartini, Chiara, Zanaboni, Anna M, Piomelli, Daniele, Tassorelli, Cristina
المصدر: Frontiers in Neuroscience. 12(MAR)
مصطلحات موضوعية: Pharmacology and Pharmaceutical Sciences, Biomedical and Clinical Sciences, Neurosciences, Clinical Sciences, Substance Misuse, Drug Abuse (NIDA only), Chronic Pain, Cannabinoid Research, Dental/Oral and Craniofacial Disease, Neurodegenerative, Headaches, Migraines, Pain Research, Neurological, migraine, inflammation, trigeminal hyperalgesia, endocannabinoid system, FAAH inhibitors, Psychology, Cognitive Sciences, Biological psychology
وصف الملف: application/pdf
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7Academic Journal
المؤلفون: Rømer Thomsen, Kristine, Thylstrup, Birgitte, Kenyon, Emily A., Lees, Rachel, Baandrup, Lone, Feldstein Ewing, Sarah W., Freeman, Tom P.
المصدر: Rømer Thomsen , K , Thylstrup , B , Kenyon , E A , Lees , R , Baandrup , L , Feldstein Ewing , S W & Freeman , T P 2022 , ' Cannabinoids for the treatment of cannabis use disorder : New avenues for reaching and helping youth? ' , Neuroscience and Biobehavioral Reviews , vol. 132 , pp. 169-180 . https://doi.org/10.1016/j.neubiorev.2021.11.033
مصطلحات موضوعية: Cannabidiol, Cannabinoids, Cannabis, Cannabis use disorder, FAAH inhibitors, Pharmacotherapy, Treatment, Youth, Δ-9-Tetrahydrocannabinol, /dk/atira/pure/subjectarea/asjc/3200/3206, name=Neuropsychology and Physiological Psychology, /dk/atira/pure/subjectarea/asjc/2800/2805, name=Cognitive Neuroscience, /dk/atira/pure/subjectarea/asjc/2800/2802, name=Behavioral Neuroscience
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8Academic Journal
المؤلفون: Carmine Marco Morgillo, Antonio Lupia, Alessandro Deplano, Luciano Pirone, Bianca Fiorillo, Emilia Pedone, F. Javier Luque, Valentina Onnis, Federica Moraca, Bruno Catalanotti
المصدر: International Journal of Molecular Sciences; Volume 23; Issue 24; Pages: 15502
مصطلحات موضوعية: FAAH inhibitors, propanamide derivatives, molecular dynamics simulations
جغرافية الموضوع: agris
وصف الملف: application/pdf
Relation: Molecular Informatics; https://dx.doi.org/10.3390/ijms232415502
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9Academic Journal
المساهمون: Pharmaceutical Design and Discovery group, Division of Pharmaceutical Chemistry and Technology, Medicinal Chemistry research group
مصطلحات موضوعية: Biochemistry, cell and molecular biology, Pharmacy, 3D QSAR, ACID AMIDE HYDROLASE, COMFA, COMSIA, CoMFA model, CoMSIA model, FAAH inhibitors
وصف الملف: application/pdf
Relation: Zięba , A , Laitinen , T , Patel , J , Poso , A & Kaczor , A A 2021 , ' Docking-Based 3D-QSAR Studies for 1,3,4-oxadiazol-2-one Derivatives as FAAH Inhibitors ' , International Journal of Molecular Sciences , vol. 22 , no. 11 , 6108 . https://doi.org/10.3390/ijms22116108; ORCID: /0000-0002-2562-1888/work/98272619; http://hdl.handle.net/10138/332945; 45c6f22c-fb62-4229-a070-d506775415e0; 000660220600001
الاتاحة: http://hdl.handle.net/10138/332945
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10Academic Journal
المؤلفون: Robert Ramer, Felix Wittig, Burkhard Hinz
المصدر: Cancers; Volume 13; Issue 22; Pages: 5701
مصطلحات موضوعية: cannabinoids, endocannabinoid system, FAAH inhibitors, MAGL inhibitors, cancer, apoptosis, autophagy, tumour cell proliferation, tumour cell invasion, metastasis, angiogenesis, tumour-immune interactions
وصف الملف: application/pdf
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11Academic Journal
المؤلفون: Agata Zięba, Tuomo Laitinen, Jayendra Z. Patel, Antti Poso, Agnieszka A. Kaczor
المصدر: International Journal of Molecular Sciences; Volume 22; Issue 11; Pages: 6108
مصطلحات موضوعية: 3D QSAR, CoMFA model, CoMSIA model, FAAH inhibitors
جغرافية الموضوع: agris
وصف الملف: application/pdf
Relation: Molecular Informatics; https://dx.doi.org/10.3390/ijms22116108
الاتاحة: https://doi.org/10.3390/ijms22116108
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12Academic Journal
المؤلفون: Vacondio, Federica, Silva, Claudia, Lodola, Alessio, Carmi, Caterina, Rivara, Silvia, Duranti, Andrea, Tontini, Andrea, Sanchini, Silvano, Clapper, Jason R, Piomelli, Daniele, Tarzia, Giorgio, Mor, Marco
المصدر: European Journal of Medicinal Chemistry. 46(9)
مصطلحات موضوعية: Digestive Diseases, Liver Disease, Amidohydrolases, Animals, Area Under Curve, Blood, Carbamates, Enzyme Inhibitors, Liver, Male, Rats, Rats, Wistar, Alkylcarbamates, FAAH inhibitors, Liquid chromatography, SPR, Stability, Rat plasma, Medicinal and Biomolecular Chemistry, Organic Chemistry, Pharmacology and Pharmaceutical Sciences, Medicinal & Biomolecular Chemistry
وصف الملف: application/pdf
URL الوصول: https://escholarship.org/uc/item/6b11j7hx
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13Academic Journal
المؤلفون: Vacondio, Federica, Silva, Claudia, Lodola, Alessio, Fioni, Alessandro, Rivara, Silvia, Duranti, Andrea, Tontini, Andrea, Sanchini, Silvano, Clapper, Jason R, Piomelli, Daniele, Mor, Marco, Tarzia, Giorgio
المصدر: ChemMedChem. 4(9)
مصطلحات موضوعية: Medicinal and Biomolecular Chemistry, Chemical Sciences, Amidohydrolases, Animals, Carbamates, Drug Stability, Enzyme Inhibitors, Half-Life, Male, Rats, Rats, Wistar, Structure-Activity Relationship, cyclohexylcarbamic acid aryl esters, FAAH inhibitors, liquid chromatography, stability, structure-activity relationships, Organic Chemistry, Pharmacology and Pharmaceutical Sciences, Medicinal & Biomolecular Chemistry, Medicinal and biomolecular chemistry, Organic chemistry
وصف الملف: application/pdf
URL الوصول: https://escholarship.org/uc/item/1d5375nx
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14Academic Journal
المصدر: Frontiers in Neuroscience, Vol 12 (2018)
مصطلحات موضوعية: migraine, inflammation, trigeminal hyperalgesia, endocannabinoid system, FAAH inhibitors, Neurosciences. Biological psychiatry. Neuropsychiatry, RC321-571
وصف الملف: electronic resource
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15
المؤلفون: Andrea Duranti, Gorane Beldarrain, Antonia Álvarez, Matilde Sbriscia, Silvia Carloni, Walter Balduini, Daniel Alonso-Alconada
مصطلحات موضوعية: neurogenesis, cannabinoid receptors, neonatal brain injury, FAAH inhibitors, Medicine (miscellaneous), neuroprotection, MGL inhibitors, endocannabinoid system, hypoxia–ischemia, General Biochemistry, Genetics and Molecular Biology
وصف الملف: application/pdf
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16Academic Journal
المصدر: Medicines; Volume 5; Issue 3; Pages: 91
مصطلحات موضوعية: multiple sclerosis, endocannabinoid system, cannabinoid receptors, monoacylglycerol lipase (MAGL) inhibitors, fatty acid amide hydrolase (FAAH) inhibitors, arachidonoylethanolamine (AEA) reuptake inhibitors
وصف الملف: application/pdf
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17Academic Journal
المؤلفون: Dale Deutsch
المصدر: Frontiers in Pharmacology, Vol 7 (2016)
مصطلحات موضوعية: Fatty acid amide hydrolase, FABPs, FAAH, Fatty acid binding proteins, FAAH inhibitors, Anandamide transporter, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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18Academic Journal
المؤلفون: Dong-sheng Zhao, Hai-yan Wang, Zhi-hui Lian, Da-xiong Han, Xin Jin
المصدر: Acta Pharmaceutica Sinica B, Vol 1, Iss 1, Pp 27-35 (2011)
مصطلحات موضوعية: FAAH inhibitors, Pharmacophore, Virtual screening, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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19
المؤلفون: Greco Rosaria, Demartini Chiara, Zanaboni Anna Maria, Francavilla Miriam, Reggiani Angelo, Realini Natalia, Scarpelli Rita, Piomelli Daniele, Tassorelli Cristina
مصطلحات موضوعية: FAAH inhibitors, NTG, trigeminal hyperalgesia, lipid-derived mediators
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20
المؤلفون: Cristina Campestre, Giovanna Poce, Simone Carradori, Paolo Guglielmi
المصدر: Expert Opinion on Therapeutic Patents. 29:769-780
مصطلحات موضوعية: FAAH inhibitors, glaucoma, RNA interference, adenosine receptor, endocannabinoids, melatonin receptor agonists, Intraocular pressure, genetic structures, Glaucoma, Disease, Bioinformatics, 01 natural sciences, Medication Adherence, Patents as Topic, Structure-Activity Relationship, 03 medical and health sciences, 0302 clinical medicine, Drug Development, Risk Factors, Drug Discovery, Animals, Humans, Medicine, Patient compliance, Intraocular Pressure, Pharmacology, Blindness, business.industry, General Medicine, medicine.disease, eye diseases, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Prostaglandin analog, 030220 oncology & carcinogenesis, Expert opinion, business