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1
المؤلفون: Min Hee Oh, Jiayu Wen, Barbara S. Slusher, Ian A. Bettencourt, Im Hong Sun, Jesse Alt, Richard L. Blosser, Jonathan D. Powell, Robert Leone, Judson Englert, Chirag H. Patel, Im Meng Sun, Ada Tam, Eva Prchalova, Liang Zhao, Matthew L. Arwood, Rana Rais
المصدر: Science. 366:1013-1021
مصطلحات موضوعية: Male, Glutamine, medicine.medical_treatment, Citric Acid Cycle, CD8-Positive T-Lymphocytes, Lymphocyte Activation, Immunotherapy, Adoptive, Lymphocytes, Tumor-Infiltrating, Immune system, Cancer immunotherapy, Tumor Microenvironment, medicine, Animals, Caproates, Mice, Inbred BALB C, Tumor microenvironment, Multidisciplinary, Effector, Chemistry, Neoplasms, Experimental, Immunotherapy, Mice, Inbred C57BL, Glucose, Tumor Escape, Cancer cell, Cancer research, Female, Energy Metabolism, Azo Compounds, Immunologic Memory
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2
المؤلفون: Arindom Pal, Barbara S. Slusher, Jenny Lam, Eva Prchalova, Run-Duo Gao, Rana Rais, Niyada Hin, Takashi Tsukamoto
المصدر: Bioorg Med Chem Lett
مصطلحات موضوعية: Molecular Structure, Stereochemistry, Glutamine, Organic Chemistry, Clinical Biochemistry, Diazooxonorleucine, Antagonist, Pharmaceutical Science, Nitroso, Prodrug, Biochemistry, 6-Diazo-5-oxo-L-norleucine, Article, chemistry.chemical_compound, chemistry, Drug Stability, Amide, Drug Design, Drug Discovery, Molecular Medicine, Moiety, Diazo, Prodrugs, Molecular Biology
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3
المؤلفون: Eva Prchalova, Michael T. Nedelcovych, Atsushi Saito, Ying Wu, Wade Coomer, Atsushi Kamiya, Yuto Hasegawa, Jesse Alt, Ajit G. Thomas, Barbara S. Slusher, Rana Rais, Gabriel Perez, Aisa Moreno-Megui, Lukáš Tenora, Camilo Rojas, Xiaolei Zhu, Varun Vohra, Pavel Majer
المصدر: Neuropsychopharmacology. 44:683-694
مصطلحات موضوعية: Pharmacology, business.industry, Glutaminase, Glutamate receptor, Hippocampus, medicine.disease, Glutaminase activity, 030227 psychiatry, Social defeat, 03 medical and health sciences, Psychiatry and Mental health, 0302 clinical medicine, Medicine, Major depressive disorder, Signal transduction, business, Prefrontal cortex, Neuroscience, 030217 neurology & neurosurgery
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4
المؤلفون: Carolyn Tallon, Kevin Liaw, Kristen R. Hollinger, Ajit G. Thomas, Camilo Rojas, Sujatha Kannan, Ying Wu, Barbara S. Slusher, Xiaolei Zhu, Eva Prchalova, Atsushi Kamiya, Elizabeth S Khoury
المصدر: J Alzheimers Dis
مصطلحات موضوعية: 0301 basic medicine, Glutamine, Apolipoprotein E4, Mice, Transgenic, Pharmacology, Hippocampal formation, Glutaminase activity, Hippocampus, Article, Cell Line, 03 medical and health sciences, Mice, 0302 clinical medicine, Cognition, Glutaminase, Alzheimer Disease, medicine, Animals, Humans, Enzyme Inhibitors, Caproates, Cells, Cultured, Microglia, Dose-Response Relationship, Drug, General Neuroscience, Antagonist, General Medicine, Barnes maze, Mice, Inbred C57BL, Psychiatry and Mental health, Clinical Psychology, 030104 developmental biology, medicine.anatomical_structure, Blood chemistry, Female, Geriatrics and Gerontology, Azo Compounds, 030217 neurology & neurosurgery
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5
المؤلفون: Vijayabhaskar Veeravalli, Eva Prchalova, Ajit G. Thomas, Rana Rais, Jesse Alt, Xinzhong Dong, Sheena Chatrath, Theresa A. Kopajtic, Qin Liu, Barbara S. Slusher, Tomoki Nishioka, Kyoko Yoshizawa, Shuichi Suzuki, Justin Ng, Hiroe Hihara, Zhe Li, Camilo Rojas, Takashi Tsukamoto, Niyada Hin, Mika Aoki
المصدر: J Med Chem
مصطلحات موضوعية: Agonist, Male, Magnetic Resonance Spectroscopy, medicine.drug_class, Pharmacology, 01 natural sciences, Benzamidine, Article, Receptors, G-Protein-Coupled, 03 medical and health sciences, chemistry.chemical_compound, Mice, Drug Discovery, medicine, Moiety, Animals, Humans, Receptor, 030304 developmental biology, G protein-coupled receptor, Neurons, 0303 health sciences, Analgesics, Chemistry, HEK 293 cells, Transfection, Isoquinolines, 0104 chemical sciences, Benzamidines, 010404 medicinal & biomolecular chemistry, HEK293 Cells, Opioid, Drug Design, Molecular Medicine, Chronic Pain, medicine.drug
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6
المؤلفون: Atsushi Kamiya, Michael T. Nedelcovych, Ranjeet Prasad Dash, Rana Rais, Barbara S. Slusher, Eran Hadas, Ying Wu, Lyndah Lovell, Arena A. Manning, Jesse Alt, Eva Prchalova, Ajit G. Thomas, David J. Volsky, Boe-Hyun Kim, Xiaolei Zhu, Jennifer Kelschenbach, Wei Chao
المصدر: J Neuroimmune Pharmacol
مصطلحات موضوعية: 0301 basic medicine, Male, AIDS Dementia Complex, Glutamine, Immunology, Central nervous system, Conditioning, Classical, Neuroscience (miscellaneous), Spatial Learning, Pharmacology, Article, 03 medical and health sciences, Glutamatergic, Mice, 0302 clinical medicine, Glutamates, Norleucine, medicine, Immunology and Allergy, Animals, Prodrugs, Maze Learning, Caproates, CD11b Antigen, Microglia, Glutaminase, business.industry, Glutamate receptor, Antagonist, Fear, Leukemia Virus, Murine, Mice, Inbred C57BL, 030104 developmental biology, medicine.anatomical_structure, Memory, Short-Term, HIV-1, business, Cognition Disorders, Neurocognitive, Azo Compounds, 030217 neurology & neurosurgery, Reassortant Viruses
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7
المؤلفون: Ying Wu, Barbara S. Slusher, Michael T. Nedelcovych, Atsushi Kamiya, Ranjeet Prasad Dash, Arena A. Manning, David J. Volsky, Lyndah Lovell, Xiaolei Zhu, Rana Rais, Jesse Alt, Jennifer Kelschenbach, Eva Prchalova, Wei Chao, Ajit G. Thomas, Eran Hadas, Boe-Hyun Kim
المصدر: Journal of Neuroimmune Pharmacology. 16:693-693
مصطلحات موضوعية: Pharmacology, business.industry, Immunology, Neuroscience (miscellaneous), Antagonist, Human immunodeficiency virus (HIV), Glutamate receptor, Cognition, medicine.disease_cause, Glutamine, Murine model, Immunology and Allergy, Medicine, business, Neurocognitive
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8
المؤلفون: Ajit G. Thomas, Rana Rais, Atsushi Saito, Atsushi Kamiya, Yuto Hasegawa, Aisa Moreno-Megui, Gabriel Perez, Barbara S. Slusher, Wade Coomer, Jesse Alt, Xiaolei Zhu, Lukáš Tenora, Camilo Rojas, Eva Prchalova, Ying Wu, Michael T. Nedelcovych, Varun Vohra, Pavel Majer
المصدر: Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology. 44(6)
مصطلحات موضوعية: Male, Diazooxonorleucine, Prefrontal Cortex, Hippocampus, Glutaminase activity, Article, Social defeat, Mice, Glutaminase, Animals, Medicine, Prodrugs, Depression (differential diagnoses), Inflammation, Pharmacology, CD11b Antigen, Behavior, Animal, biology, Depression, business.industry, Correction, Mice, Inbred C57BL, Neuropsychopharmacology, Disease Models, Animal, Psychiatry and Mental health, Integrin alpha M, biology.protein, business, Neuroscience, Stress, Psychological, Signal Transduction
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9
المؤلفون: Susan K. Pierce, Louis H. Miller, Jeeva Munasinghe, Sanhita Sinharay, William Schreiber-Stainthorp, Eva Prchalova, Jonathan D. Powell, Dragan Maric, Dima A. Hammoud, Barbara S. Slusher, Brittany A. Riggle
المصدر: Proceedings of the National Academy of Sciences. 115
مصطلحات موضوعية: Adult, 0301 basic medicine, Pathology, medicine.medical_specialty, Glutamine, Diazooxonorleucine, Plasmodium falciparum, Malaria, Cerebral, Brain Edema, Antimalarials, Mice, 03 medical and health sciences, In vivo, Edema, medicine, Animals, Humans, Malaria, Falciparum, Child, Multidisciplinary, biology, business.industry, Antagonist, Brain, biology.organism_classification, Magnetic Resonance Imaging, Mice, Inbred C57BL, Disease Models, Animal, 030104 developmental biology, PNAS Plus, Blood-Brain Barrier, Cerebral Malaria, Adjunctive treatment, Disease Progression, Female, medicine.symptom, Complication, business, Biomarkers
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10
المؤلفون: Andrej Jančařík, Rana Rais, Lenka Monincová, Ranjeet Prasad Dash, Sarah C. Zimmermann, Barbara S. Slusher, Gregory J. Riggins, Jan Vávra, Pavel Majer, Alexandra J. Gadiano, Ying Wu, Lukáš Tenora, C. Ethan Slusher, Tomáš Tichý, Eva Prchalova
المصدر: Journal of medicinal chemistry. 61(9)
مصطلحات موضوعية: 0301 basic medicine, Male, Nitrogen, Mebendazole, Administration, Oral, Biological Availability, 03 medical and health sciences, Mice, Structure-Activity Relationship, 0302 clinical medicine, Dogs, Drug Stability, Drug Discovery, Aqueous solubility, medicine, Structure–activity relationship, Animals, Prodrugs, Tissue Distribution, Anthelmintic, Solubility, Anthelmintics, Chemistry, Water, Prodrug, Bioavailability, 030104 developmental biology, 030220 oncology & carcinogenesis, Molecular Medicine, medicine.drug, Nuclear chemistry, Biological availability
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11eBook
المؤلفون: David Drábek, Petra Hůlová, Eva Prchalová, Kateřina Rudčenková, S.d.Ch, Anna Saavedra, Roman Sikora, Tomáš Vůjtek, David Zábranský, Matthias Naumann, Barbora Schnelle
Resource Type: eBook.
Categories: PERFORMING ARTS / Theater / Playwriting
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12
المؤلفون: Andrej Jančařík, Rana Rais, Caroline Garrett, Michael T. Nedelcovych, Ranjeet Prasad Dash, Alexandra J. Gadiano, Gerald Brandacher, Boe-Hyun Kim, Jennifer Kelschenbach, Georg J. Furtmüller, Eran Hadas, Eva Prchalova, Lukáš Tenora, Pavel Majer, Byoung Chol Oh, David J. Volsky, Wei Chao, Barbara S. Slusher, Jesse Alt, Sarah C. Zimmermann
مصطلحات موضوعية: 0301 basic medicine, Male, Swine, Diazooxonorleucine, Neurocognitive Disorders, Glutamic Acid, HIV Infections, Pharmacology, Neurotransmission, Article, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Drug Stability, Glutaminase, Drug Discovery, medicine, Animals, Humans, Prodrugs, Nootropic Agents, Aminocaproates, Microglia, Glutamate receptor, Antagonist, Brain, Prodrug, Viral Load, 6-Diazo-5-oxo-L-norleucine, Glutamine, Mice, Inbred C57BL, 030104 developmental biology, medicine.anatomical_structure, Blood, chemistry, Molecular Medicine, Female, Azo Compounds, 030217 neurology & neurosurgery, Isopropyl
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13
المؤلفون: Barbara S. Slusher, Peter A. Calabresi, Jesse Alt, Kristen R. Hollinger, Matthew D. Smith, Rana Rais, Eva Prchalova, Leslie Kirby
المصدر: Neurology® Neuroimmunology & Neuroinflammation
مصطلحات موضوعية: Male, 0301 basic medicine, Encephalomyelitis, Autoimmune, Experimental, Multiple Sclerosis, Glutamine, Pharmacology, Article, Flow cytometry, Mice, 03 medical and health sciences, 0302 clinical medicine, Immune system, In vivo, medicine, Animals, Cognitive Dysfunction, Caproates, Cells, Cultured, Behavior, Animal, medicine.diagnostic_test, Cell growth, business.industry, Experimental autoimmune encephalomyelitis, Antagonist, medicine.disease, 3. Good health, Barnes maze, Mice, Inbred C57BL, 030104 developmental biology, Neurology, Female, Neurology (clinical), business, Azo Compounds, 030217 neurology & neurosurgery
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14
المؤلفون: Cynthia A. Zahnow, Jonathan D. Powell, Min-Hee Oh, Stephen M. Brown, Maureen R. Horton, Samuel L. Collins, Meghan Travers, Rana Rais, Liang Zhao, Matthew L. Arwood, Wei Xu, Im-Meng Sun, Eva Prchalova, Robert Leone, Barbara S. Slusher, Im-Hong Sun
المصدر: Cancer Research. 79:LB-022
مصطلحات موضوعية: Cancer Research, Tumor microenvironment, Regulatory T cell, business.industry, Cancer, medicine.disease, Glutamine, medicine.anatomical_structure, Immune system, Oncology, Ascites, Cancer research, medicine, Myeloid-derived Suppressor Cell, medicine.symptom, Ovarian cancer, business
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15
المؤلفون: Ladislav Kniezo, Lukas Werner, Kamil Parkan, Eva Prchalova, Zuzana Lövyova
المصدر: Carbohydrate Research. 345:352-362
مصطلحات موضوعية: Glycosylation, Vinyl Compounds, Chemistry, Stereochemistry, Organic Chemistry, Stereoisomerism, General Medicine, Disaccharides, Mandelic acid, Biochemistry, Cycloaddition, Analytical Chemistry, chemistry.chemical_compound, Mandelic Acids, Stereoselectivity, Enantiomer
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16Academic Journal
المؤلفون: Kateřina Novotná, Lukáš Tenora, Eva Prchalová, James Paule, Jesse Alt, Vijay Veeravalli, Jenny Lam, Ying Wu, Ivan Šnajdr, Sadakatali Gori, Vijaya Saradhi Mettu, Takashi Tsukamoto, Pavel Majer, Barbara S. Slusher, Rana Rais
مصطلحات موضوعية: Biochemistry, Medicine, Cell Biology, Genetics, Physiology, Pharmacology, Cancer, Chemical Sciences not elsewhere classified, >- butyl -(<, glutamine antagonist 6, phenylpropanamido )- 5, high aqueous solubility, glutamine antagonist prodrugs, enhanced metabolic stability, improved solubility, >)- 6, high tumor, various ester, therapeutic potential, targeting profile, recently reported, pharmacokinetics studies, pharmacokinetic attributes, one prodrugs, new generation, intestinal homogenate, inactive m1, improved physicochemical, excellent efficacy, clinical trials