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1
المؤلفون: Shashidhar S. Jatiani, Balireddy Akula, E. Premkumar Reddy, Poornima Ramkumar, Rinku Jain, E. Vijaya Bharathi, Aneel K. Aggarwal, Stephen C. Cosenza, M. V. Ramana Reddy, Vinay K. Billa, Muralidhar R. Mallireddigari, D. R. C. Venkata Subbaiah, Rodrigo Vasquez-Del Carpio, Venkat R. Pallela
المصدر: Bioorganic & Medicinal Chemistry. 24:521-544
مصطلحات موضوعية: 0301 basic medicine, Indoles, Clinical Biochemistry, Pharmaceutical Science, Pyrimidinones, Polo-like kinase, Protein Serine-Threonine Kinases, Biochemistry, PLK1, Article, Gene product, Structure-Activity Relationship, 03 medical and health sciences, 0302 clinical medicine, Drug Discovery, Humans, ASK1, Protein Kinase Inhibitors, Molecular Biology, Mitosis, Dose-Response Relationship, Drug, Molecular Structure, Kinase, Chemistry, Organic Chemistry, Wild type, Biological activity, Cell biology, 030104 developmental biology, 030220 oncology & carcinogenesis, Molecular Medicine
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2
المؤلفون: M. V. Ramana Reddy, E. Premkumar Reddy, Venkat R. Pallela, Muralidhar R. Mallireddigari, Amol Padgaonkar, D. R. C. Venkata Subbaiah, Stacey J. Baker, Saikrishna Athuluri-Divakar, Rodrigo Vasquez-Del Carpio, Balireddy Akula, Vinay K. Billa, E. Vijaya Bharathi, Stephen C. Cosenza
المصدر: Journal of Medicinal Chemistry
مصطلحات موضوعية: Pyridines, Mice, Nude, Antineoplastic Agents, Apoptosis, Pharmacology, Article, Mice, Structure-Activity Relationship, Cyclin D1, In vivo, Cell Line, Tumor, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, biology, Chemistry, Cyclin-dependent kinase 4, Kinase, Cell Cycle, Cyclin-Dependent Kinase 4, AMPK, Imatinib, medicine.disease, Molecular Docking Simulation, Repressor Proteins, Pyrimidines, biology.protein, Heterografts, Molecular Medicine, Female, Drug Screening Assays, Antitumor, Protein Kinases, Neoplasm Transplantation, Chronic myelogenous leukemia, medicine.drug
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3
المؤلفون: M. Kashi Reddy, E. Vijaya Bharathi, Ahmed Kamal, Manika Pal Bhadra, T. Lakshminarayan Reddy, D. Dastagiri, S.N.C.V.L. Pushpavalli, M. Janaki Ramaiah, J. Surendranadha Reddy, A. Viswanath, T. Basha Shaik
المصدر: European Journal of Medicinal Chemistry. 46:691-703
مصطلحات موضوعية: Stereochemistry, Antineoplastic Agents, Stereoisomerism, chemistry.chemical_compound, Cell Line, Tumor, Drug Discovery, medicine, Humans, Isoxazole, Cytotoxicity, Quinazolinone, Cell Proliferation, Quinazolinones, Pharmacology, Dose-Response Relationship, Drug, Molecular Structure, biology, Chemistry, Cell Cycle, Organic Chemistry, Isoxazoles, General Medicine, Tubulin, Mechanism of action, biology.protein, Drug Screening Assays, Antitumor, medicine.symptom, Linker, Conjugate
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4
المؤلفون: Ahmed Kamal, Farheen Sultana, D. Dastagiri, Subrata Sen, M. Janaki Ramaiah, Aarti Juvekar, Surekha M. Zingde, A. Viswanath, J. Surendranadha Reddy, E. Vijaya Bharathi, Manika Pal-Bhadra, S.N.C.V.L. Pushpavalli
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:3310-3313
مصطلحات موضوعية: Clinical Biochemistry, Pharmaceutical Science, Pyrrolobenzodiazepine, Antineoplastic Agents, Apoptosis, Biochemistry, Chemical synthesis, Benzodiazepines, chemistry.chemical_compound, Cell Line, Tumor, Drug Discovery, medicine, Humans, Pyrroles, ortho-Aminobenzoates, Cytotoxicity, Molecular Biology, Caspase 3, Chemistry, Cell Cycle, Organic Chemistry, Cell cycle, Flow Cytometry, Mechanism of action, Cell culture, Cancer cell, Molecular Medicine, Tumor Suppressor Protein p53, medicine.symptom
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5
المؤلفون: D. Dastagiri, E. Vijaya Bharathi, Ahmed Kamal, J. Surendranadha Reddy
المصدر: Tetrahedron Letters. 49:348-353
مصطلحات موضوعية: chemistry.chemical_compound, Tosyl, chemistry, Methanesulfonyl chloride, Organic Chemistry, Drug Discovery, Base free, medicine, P-toluenesulfonyl chloride, Organic chemistry, Biochemistry, Chloride, medicine.drug
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6
المؤلفون: E. Vijaya Bharathi, A. Hari Babu, K. Venkata Ramana, A. Venkata Ramana, Ahmed Kamal, M. Shiva Kumar
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:2621-2623
مصطلحات موضوعية: Electrophoresis, Agar Gel, Azides, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Pyrrolobenzodiazepine, Biological activity, General Medicine, DNA, Affinity binding, Combinatorial chemistry, Biochemistry, Chemical synthesis, Benzodiazepines, chemistry.chemical_compound, chemistry, Reagent, Drug Discovery, Lactam, Molecular Medicine, Azide, Molecular Biology, Conjugate
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7
المؤلفون: E. Premkumar Reddy, E. Vijaya Bharathi, Amol Padgaonkar, Muralidhar R. Mallireddigari, Venkat R. Pallela, Vinay K. Billa, Hua Lv, James M. Gallo, D. R. C. Venkata Subbaiah, Balaiah Akula, Stephen C. Cosenza, M. V. Ramana Reddy
المصدر: Journal of medicinal chemistry. 56(13)
مصطلحات موضوعية: Cell Survival, Administration, Oral, Biological Availability, Mice, Nude, Antineoplastic Agents, Pharmacology, Blood–brain barrier, Microtubules, Article, Polymerization, Mice, Microtubule, In vivo, Tubulin, Cell Line, Tumor, Neoplasms, Drug Discovery, medicine, Animals, Humans, Cytotoxicity, Sulfonamides, biology, Chemistry, Cell Cycle Checkpoints, HCT116 Cells, Xenograft Model Antitumor Assays, In vitro, Tumor Burden, medicine.anatomical_structure, Drug development, Blood-Brain Barrier, Drug Resistance, Neoplasm, Drug Design, biology.protein, MCF-7 Cells, Molecular Medicine, Antimitotic Agent, K562 Cells
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8
المؤلفون: Pranjal Sarma, Farheen Sultana, Ahmed Kamal, E. Vijaya Bharathi, M. Janaki Ramaiah, S.N.C.V.L. Pushpavalli, Arutla Viswanath, Manika Pal Bhadra, G. Ramakrishna, A. Lavanya, Jayanti Naga Srirama Chandra Murty
المصدر: Anti-cancer agents in medicinal chemistry. 13(10)
مصطلحات موضوعية: Cancer Research, Poly ADP ribose polymerase, Pyrrolobenzodiazepine, Antineoplastic Agents, Apoptosis, Mitochondrion, Resting Phase, Cell Cycle, chemistry.chemical_compound, Benzodiazepines, Inhibitory Concentration 50, Structure-Activity Relationship, Cell Line, Tumor, Structure–activity relationship, Humans, Pyrroles, Mammary Glands, Human, Cell Proliferation, Pharmacology, Membrane Potential, Mitochondrial, Molecular Structure, Chemistry, Cell growth, Caspase 3, Epithelial Cells, Cell cycle, Mitochondria, Gene Expression Regulation, Neoplastic, Biochemistry, Cell culture, Molecular Medicine, Female, Drug Screening Assays, Antitumor, Poly(ADP-ribose) Polymerases, Ethers, Signal Transduction
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9
المؤلفون: M. Janaki Ramaiah, Ahmed Kamal, T. Lakshminarayan Reddy, M. Victor Prem Sagar, M. Kashi Reddy, Manika Pal-Bhadra, E. Vijaya Bharathi, D. Dastagiri, J. Surendranadha Reddy, S.N.C.V.L. Pushpavalli
المصدر: European journal of medicinal chemistry. 46(12)
مصطلحات موضوعية: Pyrimidine, Down-Regulation, Antineoplastic Agents, Apoptosis, chemistry.chemical_compound, Cyclin D1, Cell Line, Tumor, Neoplasms, Drug Discovery, Humans, Protein kinase B, Caspase, Pharmacology, Sulfonamides, biology, Chemistry, Organic Chemistry, G1 Phase, NF-kappa B, General Medicine, Pyrimidines, Biochemistry, biology.protein, Phosphorylation, G1 phase, K562 cells
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10
المؤلفون: Ahmed Kamal, Pranjal Sarma, M. Janaki Ramaiah, Y. V. V. Srikanth, J. Surendranadha Reddy, D. Dastagiri, Rajender, Manika Pal-Bhadra, S.N.C.V.L. Pushpavalli, M. Kashi Reddy, E. Vijaya Bharathi
المصدر: Bioorganicmedicinal chemistry. 19(8)
مصطلحات موضوعية: Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Triazole, Pharmaceutical Science, Pyrrolobenzodiazepine, Antineoplastic Agents, Breast Neoplasms, Biochemistry, Chemical synthesis, Steroid, chemistry.chemical_compound, Benzodiazepines, Structure-Activity Relationship, Tubulin, Cell Line, Tumor, Drug Discovery, medicine, Moiety, Humans, Pyrroles, Molecular Biology, Estradiol, Organic Chemistry, Cell Cycle, Biological activity, Estrogens, chemistry, Mechanism of action, Molecular Medicine, Female, medicine.symptom, Linker
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11
المؤلفون: Dhananjaya Pal, Manika Pal-Bhadra, M. Janaki Ramaiah, Ahmed Kamal, Chatla Srinivas, E. Vijaya Bharathi, D. Dastagiri, J. Surendranadha Reddy, S.N.C.V.L. Pushpavalli
المصدر: ChemMedChem. 5(11)
مصطلحات موضوعية: Chalcone, Imidazothiazole, Stereochemistry, Antineoplastic Agents, Apoptosis, Biochemistry, chemistry.chemical_compound, Cell Line, Tumor, Cyclins, Drug Discovery, Humans, General Pharmacology, Toxicology and Pharmaceutics, Thiazole, Pharmacology, Biological studies, Organic Chemistry, Cell Cycle, Imidazoles, NF-kappa B, NF-κB, Caspase 9, Cyclin-Dependent Kinases, Thiazoles, chemistry, Cell culture, Molecular Medicine, Female
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12
المؤلفون: Aarti Juvekar, Subrata Sen, G. Balakishan, E. Vijaya Bharathi, J. Surendranadha Reddy, S.N.C.V.L. Pushpavalli, Surekha M. Zingde, Manika Pal-Bhadra, Pranjal Sarma, D. Dastagiri, M. Janaki Ramaiah, Ahmed Kamal
المصدر: Bioorganicmedicinal chemistry. 18(18)
مصطلحات موضوعية: Male, Clinical Biochemistry, Pharmaceutical Science, Pyrrolobenzodiazepine, Antineoplastic Agents, Apoptosis, Biochemistry, chemistry.chemical_compound, Benzodiazepines, Mice, Bcl-2-associated X protein, Cyclin-dependent kinase, Mice, Inbred NOD, Cell Line, Tumor, Neoplasms, Drug Discovery, medicine, Animals, Humans, Cytotoxicity, Molecular Biology, Caspase, bcl-2-Associated X Protein, Oxadiazoles, biology, Organic Chemistry, Cell Cycle, Cyclin-Dependent Kinase 2, Xenograft Model Antitumor Assays, In vitro, Mitochondria, Mechanism of action, chemistry, Caspases, biology.protein, Molecular Medicine, medicine.symptom, Tumor Suppressor Protein p53
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13
المؤلفون: Aarti Juvekar, M. Janaki Ramaiah, E. Vijaya Bharathi, Manika Pal-Bhadra, S.N.C.V.L. Pushpavalli, Farheen Sultana, M. Ameruddin Azhar, Surekha M. Zingde, Ahmed Kamal, D. Dastagiri, J. Surendranadha Reddy, Subrata Sen
المصدر: European journal of medicinal chemistry. 45(9)
مصطلحات موضوعية: Stereochemistry, Pyrrolobenzodiazepine, Antineoplastic Agents, Apoptosis, Cell Cycle Proteins, Chemical synthesis, chemistry.chemical_compound, Benzodiazepines, Inhibitory Concentration 50, Cell Line, Tumor, Drug Discovery, Humans, Isoxazole, Cell Proliferation, Pharmacology, biology, Cytochrome c, Organic Chemistry, Biological activity, General Medicine, Isoxazoles, Cell cycle, In vitro, Gene Expression Regulation, Neoplastic, chemistry, Drug Design, biology.protein
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14
المؤلفون: M. Janaki Ramaiah, Manika Pal-Bhadra, M. Kashi Reddy, E. Vijaya Bharathi, D. Dastagiri, S.N.C.V.L. Pushpavalli, Ahmed Kamal, J. Surendranadha Reddy
المصدر: Bioorganicmedicinal chemistry letters. 20(17)
مصطلحات موضوعية: Pyrimidine, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Pyrrolobenzodiazepine, Carboxamide, behavioral disciplines and activities, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Benzodiazepines, Cell Line, Tumor, Drug Discovery, medicine, Humans, Cytotoxicity, Molecular Biology, Aniline Compounds, biology, Cytochrome c, Organic Chemistry, Biological activity, Pyrimidines, Mechanism of action, chemistry, biology.protein, Molecular Medicine, medicine.symptom, Drug Screening Assays, Antitumor
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15
المؤلفون: Manika Pal-Bhadra, Farheen Sultana, Hemant Kumar Srivastava, E. Vijaya Bharathi, A. Viswanath, Aarti Juvekar, Subrata Sen, M. Janaki Ramaiah, J. Surendranadha Reddy, S.N.C.V.L. Pushpavalli, D. Dastagiri, G. Narahari Sastry, Ahmed Kamal, Surekha M. Zingde
المصدر: Bioorganicmedicinal chemistry. 18(2)
مصطلحات موضوعية: Models, Molecular, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Pyrrolobenzodiazepine, Antineoplastic Agents, Molecular Dynamics Simulation, Biochemistry, chemistry.chemical_compound, Benzodiazepines, Drug Discovery, medicine, Tumor Cells, Cultured, Moiety, Humans, Pyrroles, Molecular Biology, Quinazolinone, Biological evaluation, Cell Proliferation, Quinazolinones, Benzodiazepine, Molecular Structure, Organic Chemistry, Stereoisomerism, chemistry, Design synthesis, Drug Design, Molecular Medicine, Drug Screening Assays, Antitumor, Human cancer, Conjugate
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16
المؤلفون: Ahmed Kamal, E. Vijaya Bharathi, D. Dastagiri, J. Surendranadha Reddy
المصدر: ChemInform. 39
مصطلحات موضوعية: chemistry.chemical_compound, Tosyl, chemistry, Base free, medicine, General Medicine, Medicinal chemistry, Chloride, medicine.drug
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17
المؤلفون: Chatla Srinivas, Y. V. V. Srikanth, Arutla Viswanath, Ranjita Nayak, M. Janaki Ramaiah, E. Vijaya Bharathi, S.N.C.V.L. Pushpavalli, Ahmed Kamal, Farheen Sultana, Manika Pal-Bhadra
المصدر: MedChemComm. 4:575
مصطلحات موضوعية: Pharmacology, Senescence, Organic Chemistry, Pharmaceutical Science, Biology, Biochemistry, Molecular biology, Telomere, chemistry.chemical_compound, chemistry, Drug Discovery, Ic50 values, SKP2, Molecular Medicine, Inducer, Cytotoxicity, G1 phase, Quinazolinone
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18
المؤلفون: Paramita Ray, Ahmed Kamal, E. Vijaya Bharathi, S.N.C.V.L. Pushpavalli, M. Janaki Ramaiah, M. Victor Prem Sagar, D. Dastagiri, J. Surendranadha Reddy, Manika Pal-Bhadra
المصدر: MedChemComm. 1:355
مصطلحات موضوعية: Pharmacology, Imidazopyridine, Chalcone, Pyrimidine, biology, Stereochemistry, Organic Chemistry, Cyclin-dependent kinase 2, Pharmaceutical Science, Biochemistry, chemistry.chemical_compound, Cyclin D1, chemistry, Cell culture, Apoptosis, Drug Discovery, biology.protein, Molecular Medicine, G1 phase