-
1Academic Journal
المؤلفون: Due-Hansen, Maria E, Pandey, Sunil K, Christiansen, Elisabeth, Andersen, Rikke, Hansen, Steffen V F, Ulven, Trond
المصدر: Due-Hansen , M E , Pandey , S K , Christiansen , E , Andersen , R , Hansen , S V F & Ulven , T 2016 , ' A protocol for amide bond formation with electron deficient amines and sterically hindered substrates ' , Organic & Biomolecular Chemistry , vol. 14 , no. 2 , pp. 430-433 . https://doi.org/10.1039/c5ob02129d
وصف الملف: application/pdf
-
2Academic Journal
المصدر: Journal of Loss Prevention in the Process Industries ; volume 73, page 104614 ; ISSN 0950-4230
-
3Academic Journal
المؤلفون: Hudson, Brian D, Due-Hansen, Maria E, Christiansen, Elisabeth, Hansen, Anna M, Mackenzie, Amanda E, Murdoch, Hannah, Pandey, Sunil K, Ward, Richard J, Marquez, Rudi, Tikhonova, Irina G, Ulven, Trond, Milligan, Graeme
المصدر: Hudson , B D , Due-Hansen , M E , Christiansen , E , Hansen , A M , Mackenzie , A E , Murdoch , H , Pandey , S K , Ward , R J , Marquez , R , Tikhonova , I G , Ulven , T & Milligan , G 2013 , ' Defining the molecular basis for the first potent and selective orthosteric agonists of the FFA2 free fatty acid receptor ' , Journal of Biological Chemistry , vol. 288 , no. 24 , pp. 17296-17312 . https://doi.org/10.1074/jbc.M113.455337
مصطلحات موضوعية: /dk/atira/pure/subjectarea/asjc/1300/1303, name=Biochemistry, /dk/atira/pure/subjectarea/asjc/1300/1307, name=Cell Biology, /dk/atira/pure/subjectarea/asjc/1300/1312, name=Molecular Biology
وصف الملف: application/pdf
-
4Academic Journal
المؤلفون: Schmidt, Johannes, Liebscher, Kathrin, Merten, Nicole, Grundmann, Manuel, Mielenz, Manfred, Sauerwein, Helga, Christiansen, Elisabeth, Due-Hansen, Maria E., Ulven, Trond, Ullrich, Susanne, Gomeza, Jesús, Drewke, Christel, Kostenis, Evi
المصدر: Journal of Biological Chemistry ; volume 286, issue 14, page 11890-11894 ; ISSN 0021-9258
-
5Academic Journal
المؤلفون: Due-Hansen, Maria E., Dullum, Ove
المصدر: Safety Science ; volume 96, page 33-40 ; ISSN 0925-7535
-
6Academic Journal
المؤلفون: Hansen, Steffen Vissing Fahnøe, Christiansen, Elisabeth, Urban, Christian, Hudson, Brian D, Stocker, Claire J, Due-Hansen, Maria E, Wargent, Ed T, Shimpukade, Bharat, Almeida, Reinaldo, Ejsing, Christer S, Cawthorne, Michael A, Kassack, Matthias U, Milligan, Graeme, Ulven, Trond
المصدر: Hansen , S V F , Christiansen , E , Urban , C , Hudson , B D , Stocker , C J , Due-Hansen , M E , Wargent , E T , Shimpukade , B , Almeida , R , Ejsing , C S , Cawthorne , M A , Kassack , M U , Milligan , G & Ulven , T 2016 , ' Discovery of a Potent Free Fatty Acid 1 Receptor Agonist with Low Lipophilicity, Low Polar Surface Area and Robust in Vivo Efficacy ' , Journal of Medicinal Chemistry , vol. 59 , ....
-
7Academic Journal
المؤلفون: Due‐Hansen, Maria E., Pandey, Sunil K., Christiansen, Elisabeth, Andersen, Rikke, Hansen, Steffen V. F., Ulven, Trond
المصدر: ChemInform ; volume 47, issue 20 ; ISSN 0931-7597 1522-2667
-
8Academic Journal
المؤلفون: Christiansen, Elisabeth, Due-Hansen, Maria E, Urban, Christian, Grundmann, Manuel, Schmidt, Johannes, Hansen, Steffen V F, Hudson, Brian D, Zaibi, Mohamed, Markussen, Stine B, Hagesaether, Ellen, Milligan, Graeme, Cawthorne, Michael A, Kostenis, Evi, Kassack, Matthias U, Ulven, Trond
المصدر: Christiansen , E , Due-Hansen , M E , Urban , C , Grundmann , M , Schmidt , J , Hansen , S V F , Hudson , B D , Zaibi , M , Markussen , S B , Hagesaether , E , Milligan , G , Cawthorne , M A , Kostenis , E , Kassack , M U & Ulven , T 2013 , ' Discovery of a potent and selective free fatty acid receptor 1 agonist with low lipophilicity and high oral bioavailability ' , Journal of Medicinal Chemistry , vol. 56 , no. ....
مصطلحات موضوعية: Administration, Oral, Animals, Biological Availability, Drug Discovery, Magnetic Resonance Spectroscopy, Mice, Models, Molecular, Receptors, G-Protein-Coupled, Spectrometry, Mass, Electrospray Ionization, Structure-Activity Relationship
-
9Academic Journal
المؤلفون: Christiansen, Elisabeth, Due-Hansen, Maria E, Urban, Christian, Grundmann, Manuel, Schröder, Ralf, Hudson, Brian D, Milligan, Graeme, Cawthorne, Michael A, Kostenis, Evi, Kassack, Matthias U, Ulven, Trond
المصدر: Christiansen , E , Due-Hansen , M E , Urban , C , Grundmann , M , Schröder , R , Hudson , B D , Milligan , G , Cawthorne , M A , Kostenis , E , Kassack , M U & Ulven , T 2012 , ' Free Fatty Acid Receptor 1 (FFA1/GPR40) Agonists : Mesylpropoxy Appendage Lowers Lipophilicity and Improves ADME Properties ' , Journal of Medicinal Chemistry , vol. 55 , no. 14 , pp. 6624-8 . https://doi.org/10.1021/jm3002026
-
10Academic Journal
المؤلفون: Christiansen, Elisabeth, Urban, Christian, Grundmann, Manuel, Due-Hansen, Maria E., Hagesaether, Ellen, Schmidt, Johannes, Pardo, Leonardo, Ullrich, Susanne, Kostenis, Evi, Kassack, Matthias, Ulven, Trond
المصدر: Journal of Medicinal Chemistry ; volume 54, issue 19, page 6691-6703 ; ISSN 0022-2623 1520-4804
-
11Academic Journal
المؤلفون: Christiansen, Elisabeth, Due-Hansen, Maria E, Ulven, Trond
المصدر: Christiansen , E , Due-Hansen , M E & Ulven , T 2010 , ' A Rapid and Efficient Sonogashira Protocol and Improved Synthesis of Free Fatty Acid 1 (FFA1) Receptor Agonists ' , Journal of Organic Chemistry , vol. 75 , no. 4 , pp. 1301-4 . https://doi.org/10.1021/jo902533p
-
12Academic Journal
المؤلفون: Christiansen, Elisabeth, Due-Hansen, Maria E., Urban, Christian, Merten, Nicole, Pfleiderer, Michael, Karlsen, Kasper K., Rasmussen, Sanne S., Steensgaard, Mette, Hamacher, Alexandra, Schmidt, Johannes, Drewke, Christel, Petersen, Rasmus Koefoed, Kristiansen, Karsten, Ullrich, Susanne, Kostenis, Evi, Kassack, Matthias U., Ulven, Trond
المصدر: Christiansen , E , Due-Hansen , M E , Urban , C , Merten , N , Pfleiderer , M , Karlsen , K K , Rasmussen , S S , Steensgaard , M , Hamacher , A , Schmidt , J , Drewke , C , Petersen , R K , Kristiansen , K , Ullrich , S , Kostenis , E , Kassack , M U & Ulven , T 2010 , ' Structure−Activity Study of Dihydrocinnamic Acids and Discovery of the Potent FFA1 (GPR40) Agonist TUG-469 ' , ACS Medicinal Chemistry Letters , vol. 1 , ....
-
13Electronic Resource
المؤلفون: Christiansen, Elisabeth, Due-Hansen, Maria E., Urban, Christian, Merten, Nicole, Pfleiderer, Michael, Karlsen, Kasper Kannegård, Rasmussen, Sanne S., Steensgaard, Mette, Hamacher, Alexandra, Schmidt, Johannes, Drewke, Christel, Petersen, Rasmus Koefoed, Kristiansen, Karsten, Ullrich, Susanne, Kostenis, Evi, Kassack, Matthias U., Ulven, Trond
المصدر: Christiansen , E , Due-Hansen , M E , Urban , C , Merten , N , Pfleiderer , M , Karlsen , K K , Rasmussen , S S , Steensgaard , M , Hamacher , A , Schmidt , J , Drewke , C , Petersen , R K , Kristiansen , K , Ullrich , S , Kostenis , E , Kassack , M U & Ulven , T 2010 , ' Structure-activity study of dihydrocinnamic acids and discovery of the potent FFA1 (GPR40) agonist TUG-469 ' , ACS Medicinal Chemistry Letters , vol. 1 , no. 7 , pp. 345-349 .
مصطلحات الفهرس: Diabetes, FFA1, FFAR1, GPR40, fatty acids, drug discovery, article
URL:
https://curis.ku.dk/portal/da/publications/structureactivity-study-of-dihydrocinnamic-acids-and-discovery-of-the-potent-ffa1-gpr40-agonist-tug469(1adfb575-0039-4f2b-9520-5e4c3989e744).html https://doi.org/10.1021/ml100106c -
14Academic Journal
المؤلفون: Hansen, Steffen V. F., Christiansen, Elisabeth, Urban, Christian, Hudson, Brian D., Stocker, Claire J., Due-Hansen, Maria E., Wargent, Ed T., Shimpukade, Bharat, Almeida, Reinaldo, Ejsing, Christer S., Cawthorne, Michael A., Kassack, Matthias U., Milligan, Graeme, Ulven, Trond
المصدر: Journal of Medicinal Chemistry; Mar2016, Vol. 59 Issue 6, p2841-2846, 6p
-
15Academic Journal
المؤلفون: Due-Hansen, Maria E., Pandey, Sunil K., Christiansen, Elisabeth, Andersen, Rikke, Hansen, Steffen V. F., Ulven, Trond
المصدر: Organic & Biomolecular Chemistry; 1/14/2016, Vol. 14 Issue 2, p430-433, 4p
-
16Academic Journal
المؤلفون: Wagner, Robert, Kaiser, Gabriele, Gerst, Felicia, Christiansen, Elisabeth, Due-Hansen, Maria E, Grundmann, Manuel, Machicao, Fausto, Peter, Andreas, Kostenis, Evi, Ulven, Trond, Fritsche, Andreas, Häring, Hans-Ulrich, Ullrich, Susanne
المصدر: Diabetes; Jun2013, Vol. 62 Issue 6, p2106-2111, 6p
-
17Academic Journal
المؤلفون: Christiansen, Elisabeth, Due-Hansen, Maria E., Urban, Christian, Grundmann, Manuel, Schmidt, Johannes, Hansen, Steffen V. F., Hudson, Brian D., Zaibi, Mohamed, Markussen, Stine B., Hagesaether, Ellen, Milligan, Graeme, Cawthorne, Michael A., Kostenis, Evi, Kassack, Matthias U., Ulven, Trond
المصدر: Journal of Medicinal Chemistry; Vol. 56 Issue 3, p982-992, 11p
-
18Academic Journal
المؤلفون: Christiansen, Elisabeth, Due-Hansen, Maria E., Urban, Christian, Grundmann, Manuel, SchroÌder, Ralf, Hudson, Brian D., Milligan, Graeme, Cawthorne, Michael A., Kostenis, Evi, Kassack, Matthias U., Ulven, Trond
المصدر: Journal of Medicinal Chemistry; Jul2012, Vol. 55 Issue 14, p6624-6628, 5p
-
19
المؤلفون: Due-Hansen, Maria E.
المصدر: Due-Hansen , M E 2013 , ' Development of potent and selective modulators of the free fatty acid 1 (FFA1/GPR40) receptor ' .