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1
المؤلفون: Catherine I. Soderstrom, Jennifer Larsen, Carolina Owen, David Gifondorwa, David Beidler, Florence H. Yong, Patricia Conrad, Hendrik Neubert, Steven A. Moore, Mohamed Hassanein
المصدر: The AAPS journal. 25(1)
مصطلحات موضوعية: Male, Dystrophin, Muscular Dystrophy, Duchenne, Biopsy, Blotting, Western, Infant, Newborn, Pharmaceutical Science, Humans, Muscle, Skeletal
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2
المؤلفون: Caterina P Minniti, Lanetta Bronte-Hall, Shannon Marraffino, Jason Healy, Denis Rybin, David Beidler, Lori Huang, Dana Shelton, Steven Taylor, Colet Goossens, Steven Arkin
المصدر: Blood. 140:2564-2565
مصطلحات موضوعية: Immunology, Cell Biology, Hematology, Biochemistry
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3
المؤلفون: Xiufeng Gao, Alan D. Michelson, Andrew L. Frelinger, Denis Rybin, Ke Liu, Michael U. Callaghan, David Beidler, Jennell White, Robert J Charnigo, Patrick C. Hines, Debra D. Pittman, Ahmar U. Zaidi
المصدر: Blood. 137(15)
مصطلحات موضوعية: Adult, Male, medicine.medical_specialty, Adolescent, Immunology, Pain, Disease, Anemia, Sickle Cell, Biochemistry, 03 medical and health sciences, Young Adult, 0302 clinical medicine, Patient Self-Report, Antisickling Agents, Internal medicine, Health care, Medicine, Humans, Hydroxyurea, Longitudinal Studies, Patient Reported Outcome Measures, Baseline values, business.industry, Daily function, Actigraphy, Cell Biology, Hematology, Blood collection, Middle Aged, Clinical trial, 030220 oncology & carcinogenesis, Female, business, Biomarkers, 030215 immunology
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4
المؤلفون: Alan D. Michelson, Nick Clarke, Denis Rybin, Debra D. Pittman, Beesan Tan, Jo Howard, Andrew L. Frelinger, David Beidler, Robert J Charnigo
المصدر: Clinical and Translational Science
مصطلحات موضوعية: Male, 030213 general clinical medicine, Platelet Aggregation, Phosphodiesterase Inhibitors, Placebo-controlled study, 030226 pharmacology & pharmacy, Gastroenterology, law.invention, Placebos, 0302 clinical medicine, Randomized controlled trial, law, Hydroxyurea, General Pharmacology, Toxicology and Pharmaceutics, General Neuroscience, General Medicine, Articles, Middle Aged, Dose–response relationship, Treatment Outcome, Drug Therapy, Combination, Female, E-Selectin, Adult, medicine.medical_specialty, Adolescent, Anemia, Anemia, Sickle Cell, Pyrimidinones, Placebo, General Biochemistry, Genetics and Molecular Biology, Drug Administration Schedule, Article, 03 medical and health sciences, Young Adult, Pharmacokinetics, Double-Blind Method, Internal medicine, medicine, Humans, Adverse effect, Aged, Dose-Response Relationship, Drug, business.industry, Research, medicine.disease, 3',5'-Cyclic-AMP Phosphodiesterases, Pharmacodynamics, Pyrazoles, business, Biomarkers
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5
المؤلفون: Richard D. Head, Ruo-Hua Song, Ruteja A. Barve, David Beidler, David J. Weiss, Marc D. Zack
المصدر: Cytokine. 63:10-17
مصطلحات موضوعية: CCR2, Receptors, CCR2, medicine.medical_treatment, CD14, Immunology, Biology, Biochemistry, Monocytes, Gene expression, medicine, Humans, Immunology and Allergy, Molecular Biology, Gene Expression Profiling, Interleukins, Macrophage Colony-Stimulating Factor, Macrophages, Monocyte, Reproducibility of Results, Cell Differentiation, Hematology, Flow Cytometry, Molecular biology, Tissue Donors, Cell biology, Cytokine, medicine.anatomical_structure, Monocyte differentiation, DNA microarray, Signal transduction, Biomarkers, Signal Transduction
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6
المؤلفون: Ron Sarver, Christopher Whitehead, Heidi Baum, James Hicks, Richard Gowan, Brian Sanchez, Xiao Kang Lu, Susan E. Bove, Joseph A. Cornicelli, Howard Miller, Sandra Lightle, Aurash B Shahripour, Katherine Welch, Craig Banotai, Jayvardhan Pandit, Mark S. Plummer, Timothy Braden, David Beidler, Adam Ogden, Skalitzky Donald James, Annise Paige Goodman, Howard Roark, Nalini Sadagopan, Charles J. Stankovic, Cindy Spessard, Xi Qiang Shen
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:3438-3442
مصطلحات موضوعية: Dihydropyridines, Phosphodiesterase Inhibitors, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Osteoarthritis, Plasma protein binding, Pharmacology, Crystallography, X-Ray, Biochemistry, Structure-Activity Relationship, Catalytic Domain, Drug Discovery, medicine, Animals, Structure–activity relationship, Binding site, Molecular Biology, chemistry.chemical_classification, Binding Sites, biology, Azirines, Chemistry, fungi, Organic Chemistry, Active site, medicine.disease, Cyclic Nucleotide Phosphodiesterases, Type 2, Cyclic Nucleotide Phosphodiesterases, Type 4, Disease Models, Animal, Transformation (genetics), Enzyme, biology.protein, Molecular Medicine, Phosphodiesterase 2, Phosphodiesterase 4 Inhibitors, Protein Binding
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7
المؤلفون: Skalitzky Donald James, Craig Banotai, Jayvardhan Pandit, Adam Ogden, James Hicks, Annise Paige Goodman, Xiao Kang Lu, Howard Miller, Howard Roark, Susan E. Bove, Sandra Lightle, Aurash B Shahripour, Timothy Braden, Mark S. Plummer, Katherine Welch, Charles J. Stankovic, Ron Sarver, Joseph A. Cornicelli, Christopher Whitehead, Brian Sanchez, Nalini Sadagopan, Heidi Baum, Richard Gowan, David Beidler, Xi Qiang Shen, Cindy Spessard
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:3443-3447
مصطلحات موضوعية: Dihydropyridines, Phosphodiesterase Inhibitors, Clinical Biochemistry, Analgesic, Drug Evaluation, Preclinical, Pharmaceutical Science, Pharmacology, Crystallography, X-Ray, Biochemistry, law.invention, Structure-Activity Relationship, Pharmacokinetics, law, In vivo, Catalytic Domain, Osteoarthritis, Drug Discovery, Animals, Structure–activity relationship, Molecular Biology, chemistry.chemical_classification, Analgesics, Binding Sites, Azirines, fungi, Organic Chemistry, Azepines, Cyclic Nucleotide Phosphodiesterases, Type 2, Rats, Bioavailability, Disease Models, Animal, Enzyme, chemistry, Recombinant DNA, Pyrazoles, Molecular Medicine, Phosphodiesterase 2, Phosphodiesterase 4 Inhibitors, Half-Life, Protein Binding
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8
المؤلفون: David Beidler, Hiroyuki Eda, Hideaki Shimada, Joseph B. Monahan
المصدر: Rheumatology International. 31:1525-1530
مصطلحات موضوعية: MAPK/ERK pathway, MAP Kinase Signaling System, p38 mitogen-activated protein kinases, Interleukin-1beta, Immunology, Proinflammatory cytokine, chemistry.chemical_compound, Rheumatology, Humans, Immunology and Allergy, Medicine, RNA, Messenger, Enzyme Inhibitors, Extracellular Signal-Regulated MAP Kinases, Cells, Cultured, Osteoblasts, Tumor Necrosis Factor-alpha, Kinase, business.industry, Interleukins, Macrophage Colony-Stimulating Factor, JNK Mitogen-Activated Protein Kinases, NF-kappa B, NF-κB, Molecular biology, Gene Expression Regulation, chemistry, Interleukin 34, Cytokines, Tumor necrosis factor alpha, Mitogen-Activated Protein Kinases, Signal transduction, business, Signal Transduction
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9
المؤلفون: Kay Ahn, Benjamin F. Cravatt, Cory Michael Stiff, Yuntao Song, Sarah E. Smith, Mark Morris, Douglas S. Johnson, Tyzoon K. Nomanbhoy, James B. Dunbar, David Beidler, Lorraine Kathleen Fay, Marya Liimatta, Lazerwith Scott E, Tracy Fay Gregory, Suzanne Ross Kesten
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:2865-2869
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Thiophenes, Biochemistry, Article, Piperazines, Amidohydrolases, Amidase, Serine, Structure-Activity Relationship, chemistry.chemical_compound, Piperidines, Fatty acid amide hydrolase, Drug Discovery, Animals, Humans, Urea, Computer Simulation, Enzyme Inhibitors, Molecular Biology, biology, Organic Chemistry, Activity-based proteomics, Benzothiophene, Biological activity, Rats, Piperazine, Models, Chemical, nervous system, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, lipids (amino acids, peptides, and proteins), psychological phenomena and processes
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10
المؤلفون: Mauro Mileni, Stephen Swaney, Eranthie Weerapana, Benjamin F. Cravatt, Marya Liimatta, Michele K. McKinney, Sarah E. Smith, Lazerwith Scott E, Nalini Sadagopan, David Beidler, Cory Michael Stiff, Satwik Kamtekar, Douglas S. Johnson, Keri Van Becelaere, Keshab Bhattacharya, Yanhua Zhang, Jonathan Z. Long, Kay Ahn, Raymond C. Stevens
المصدر: Chemistry & Biology. 16:411-420
مصطلحات موضوعية: Male, Polyunsaturated Alkamides, medicine.medical_treatment, Clinical Biochemistry, Pain, Arachidonic Acids, Pharmacology, Crystallography, X-Ray, Biochemistry, MOLNEURO, Article, Piperazines, Amidohydrolases, Rats, Sprague-Dawley, Structure-Activity Relationship, chemistry.chemical_compound, Piperidines, Fatty acid amide hydrolase, In vivo, Drug Discovery, medicine, Animals, Humans, Urea, Enzyme Inhibitors, Receptors, Cannabinoid, Piperazine, Molecular Biology, JZL184, Brain, General Medicine, Anandamide, Lipid signaling, ABHD6, Endocannabinoid system, Rats, CHEMBIO, nervous system, chemistry, Molecular Medicine, lipids (amino acids, peptides, and proteins), Cannabinoid, psychological phenomena and processes, Endocannabinoids
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11
المؤلفون: Ke Liu, Michael U. Callaghan, Robert J Charnigo, David Beidler, Alan D. Michelson, Melanie Simmons, Martin David, Andreas M. Pleil, Bryan Hannan, Denis Rybin, Alexandra I. Barsdorf, Ahmar U. Zaidi, Debra D. Pittman, Nick Clarke, Jennell White, Patrick C. Hines, Xiufeng Gao, Andrew L. Frelinger
المصدر: Blood. 130:973-973
مصطلحات موضوعية: medicine.medical_specialty, Longitudinal study, business.operation, business.industry, Surrogate endpoint, Immunology, Actigraphy, Cell Biology, Hematology, Emergency department, Octapharma, Biochemistry, Clinical trial, Emergency medicine, Health care, Clinical endpoint, medicine, business
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12
المؤلفون: Sarah E. Smith, Scott J. Bowen, Scott A. Long, David Beidler, Marvin J. Meyers, Atli Thorarensen, Heather M. Madsen, Joseph J. McDonald, Susan Foltin, Barbara A. Schweitzer, Tenbrink Ruth E, Jane L. Wang, Mark C. Walker, Matthew James Pelc
المصدر: Bioorganicmedicinal chemistry letters. 21(21)
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Decane, Biochemistry, Amidohydrolases, chemistry.chemical_compound, Structure-Activity Relationship, Fatty acid amide hydrolase, Drug Discovery, Potency, Structure–activity relationship, Spiro Compounds, Enzyme Inhibitors, Molecular Biology, Aza Compounds, Drug discovery, Organic Chemistry, Endocannabinoid system, nervous system, chemistry, Molecular Medicine, lipids (amino acids, peptides, and proteins), Nonane, Selectivity, psychological phenomena and processes
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13
المؤلفون: Sarah E. Smith, Marvin J. Meyers, Young-Sun Yang, Joseph J. McDonald, David Beidler, Atli Thorarensen, Matthew James Pelc, Jeanne M. Rumsey, Mark V. Wilcox, Satwik Kamtekar, Scott A. Long, Scott J. Bowen, Jane L. Wang, Mark C. Walker, Susan Foltin, Barbara A. Schweitzer
المصدر: Bioorganicmedicinal chemistry letters. 21(21)
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Administration, Oral, Biological Availability, Pain, Biochemistry, Amidase, Amidohydrolases, chemistry.chemical_compound, Fatty acid amide hydrolase, In vivo, Drug Discovery, Animals, Spiro Compounds, Enzyme Inhibitors, Molecular Biology, Chromatography, High Pressure Liquid, Analgesics, Aza Compounds, Fatty acid amide, biology, Chemistry, Organic Chemistry, Serine hydrolase, Anandamide, Endocannabinoid system, Rats, Enzyme inhibitor, biology.protein, Molecular Medicine
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14
المؤلفون: David T. Dudley, Tyzoon K. Nomanbhoy, Benjamin F. Cravatt, Nalini Sadagopan, Stephen J. Kesten, Shobha N. Bhattachar, David Beidler, Lorraine Kathleen Fay, Cory Michael Stiff, Marya Liimatta, Mark Morris, Lazerwith Scott E, Douglas S. Johnson, Kay Ahn, Suzanne Ross Kesten, Sarah E. Smith
المصدر: ACS medicinal chemistry letters. 2(2)
مصطلحات موضوعية: Fatty acid amide, Organic Chemistry, Serine hydrolase, Cannabinoid Receptor Agonists, Anandamide, Biology, Pharmacology, Biochemistry, Endocannabinoid system, Serine, chemistry.chemical_compound, nervous system, chemistry, Fatty acid amide hydrolase, Drug Discovery, lipids (amino acids, peptides, and proteins), PF-04457845, psychological phenomena and processes
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15
المؤلفون: David T. Dudley, Yanhua Zhang, Eranthie Weerapana, Kay Ahn, Benjamin F. Cravatt, Nalini Sadagopan, Tyzoon K. Nomanbhoy, Marya Liimatta, Jacqueline L. Blankman, Douglas S. Johnson, Sarah E. Smith, Shoba N. Bhattachar, David Beidler, Cory Michael Stiff, Daniel K. K. Nomura, Paul Bryan Wren, Steven Swaney, Keri Van Becelaere, Tim Young
المصدر: The Journal of pharmacology and experimental therapeutics. 338(1)
مصطلحات موضوعية: Male, Cannabinoid receptor, Pain, Pharmacology, Catalepsy, Amidohydrolases, Rats, Sprague-Dawley, chemistry.chemical_compound, Mice, Drug Discovery and Translational Medicine, Piperidines, In vivo, Fatty acid amide hydrolase, medicine, Animals, Humans, Urea, PF-04457845, Enzyme Inhibitors, IC50, Inflammation, Chemistry, Anandamide, medicine.disease, Endocannabinoid system, Rats, Mice, Inbred C57BL, Pyridazines, Molecular Medicine, lipids (amino acids, peptides, and proteins)
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16
المؤلفون: Robert H. Keith, Hiroyuki Eda, Marshall L. Michener, Jian Zhang, Joseph B. Monahan, David Beidler
المصدر: Cytokine. 52(3)
مصطلحات موضوعية: Macrophage colony-stimulating factor, Chemokine, biology, Chemistry, Interleukins, Macrophage Colony-Stimulating Factor, Immunology, Hematology, Anisoles, Biochemistry, Molecular biology, Monocytes, CXCL2, Pyrimidines, biology.protein, Immunology and Allergy, CCL17, CXCL10, XCL2, Humans, Interleukin 8, Chemokines, CCL13, Molecular Biology
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17
المؤلفون: Matthew James Pelc, Heather M. Madsen, Joseph J. McDonald, Scott J. Bowen, Barbara A. Schweitzer, David Beidler, Atli Thorarensen, Tenbrink Ruth E, Jane L. Wang
المصدر: Bioorganicmedicinal chemistry letters. 19(20)
مصطلحات موضوعية: Clinical Biochemistry, Azetidine, Pharmaceutical Science, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Amidase, Amidohydrolases, chemistry.chemical_compound, Structure-Activity Relationship, Fatty acid amide hydrolase, Drug Discovery, Hydrolase, Animals, Humans, Urea, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, Analgesics, Binding Sites, biology, Organic Chemistry, In vitro, Rats, Pyridazines, Enzyme, chemistry, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, Azetidines
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18Academic Journal
المؤلفون: Kay Ahn, Douglas S. Johnson, Mauro Mileni, David Beidler, Jonathan Z. Long, Michele K. Mckinney, Eranthie Weerapana, Nalini Sadagopan, Marya Liimatta, Sarah E. Smith, Scott Lazerwith, Cory Stiff, Satwik Kamtekar, Yanhua Zhang, Stephen Swaney, Keri Van Becelaere, Raymond C, Benjamin F. Cravatt
المساهمون: The Pennsylvania State University CiteSeerX Archives
المصدر: http://download.cell.com/chemistry-biology/mmcs/journals/1074-5521/piis1074552109000805.mmc1.pdf.
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.544.1758; http://download.cell.com/chemistry-biology/mmcs/journals/1074-5521/piis1074552109000805.mmc1.pdf
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19Academic Journal
المؤلفون: Kay Ahn, Douglas S. Johnson, Mauro Mileni, David Beidler, Jonathan Z. Long, Michele K. Mckinney, Eranthie Weerapana, Nalini Sadagopan, Marya Liimatta, Sarah E. Smith, Scott Lazerwith, Cory Stiff, Satwik Kamtekar, Keshab Bhattacharya, Yanhua Zhang, Stephen Swaney, Keri Van Becelaere, Raymond C. Stevens, Benjamin F. Cravatt
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.394.6171; http://www.scripps.edu/cravatt/pdf/Ahn2009.pdf