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1
المؤلفون: Monica Patel, Mita Patel, Thomas Wai-Ho Lee, John Lord, Brian Christopher Raudenbush, Heather Grbic, Hossein Razavi, Darren Disalvo, David Joseph, Maryanne L. Brown, Alan David Swinamer, Della White, Siqi Lin, Karen Berg, Alison Kukulka, David S. Thomson, Christopher Ronald Sarko, Kim Fletcher, Pingrong Liu, Can Mao, Laura Amodeo, Christian Harcken
المصدر: Bioorganicmedicinal chemistry letters. 29(3)
مصطلحات موضوعية: CCR1, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Organic Chemistry, Clinical Biochemistry, Receptors, CCR1, Pharmaceutical Science, Pyrazole, 01 natural sciences, Biochemistry, Combinatorial chemistry, Amides, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, chemistry.chemical_compound, Chemokine receptor, Structure-Activity Relationship, chemistry, Drug Discovery, Molecular Medicine, Humans, Pyrazoles, Selectivity, Molecular Biology
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2
المؤلفون: Alison Kukulka, Qiang Zhang, Monica Patel, Can Mao, Melissa Canfield, Daniel Kuzmich, Darren Disalvo, Alan David Swinamer, Donald Souza, Hossein Razavi, Karen Berg, Donna Skow, David Joseph, Matthew S. Bogdanffy, Tara Sherry, Dustin Smith, Brain Cook, Maryanne L. Brown, Christian Harcken, Kimberly Fletcher, Pingrong Liu, Mita Patel
المصدر: Bioorganicmedicinal chemistry letters. 29(3)
مصطلحات موضوعية: Indazoles, Clinical Biochemistry, Receptors, CCR1, Pharmaceutical Science, Computational biology, Pyrazole, Scaffold hopping, 01 natural sciences, Biochemistry, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, Humans, Molecular Biology, Indazole, Aza Compounds, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Organic Chemistry, Antagonist, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, chemistry, Drug Design, Molecular Medicine
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3
المؤلفون: Christian Harcken, Morrison B. Mac, Melissa Hill-Drzewi, Debbie Studwell, Diva Sze-Ming Chan, Donna Terenzzio, Heather Xia, Mita Patel, Yu Hui, Brian Linehan, Pingrong Liu, Lynne Canne Bannen, Raymond A. Kemper, Louise K. Modis, Dustin Smith, Lemieux Rene M, Miller Craig Andrew, Darren Disalvo, Raj Betageri, Jeremy I. Levin, Kimberly Fletcher, Daniel Kuzmich, Lori Patenaude, Stephanie M. Ng, Yong Wang, Eugene R. Hickey, Wei Xu, John Lord, Monica Patel, Can Mao, Horan Joshua Courtney, Tamara Denise Hopkins
المصدر: Bioorganic & Medicinal Chemistry Letters. 26:466-471
مصطلحات موضوعية: 0301 basic medicine, Molecular charge, Clinical Biochemistry, Glutamic Acid, Pharmaceutical Science, Pharmacology, Biochemistry, Structure-Activity Relationship, 03 medical and health sciences, Thiadiazoles, Drug Discovery, Animals, Humans, Potency, Solubility, Molecular Biology, Oxadiazoles, S1p1 receptor, Chemistry, Organic Chemistry, Late stage, Brain, Hydrogen Bonding, Hep G2 Cells, Rats, Kinetics, Receptors, Lysosphingolipid, 030104 developmental biology, Molecular Medicine
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4
المؤلفون: Andrew D. Bolig, Maurice Brookhart, Thomas W. Lyons, Darren Disalvo
المصدر: Polyhedron. 103:51-57
مصطلحات موضوعية: chemistry.chemical_classification, Olefin fiber, 010405 organic chemistry, Chemistry, Alkene, Regioselectivity, Silyl enol ether, Nuclear magnetic resonance spectroscopy, 010402 general chemistry, 01 natural sciences, Medicinal chemistry, Article, 0104 chemical sciences, Catalysis, Inorganic Chemistry, chemistry.chemical_compound, Intramolecular force, Materials Chemistry, Organic chemistry, Dehydrogenation, Physical and Theoretical Chemistry
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5
المؤلفون: Christian Harcken, Richard M. Nelson, Daniel Kuzmich, Tazmeen Fadra-Khan, Edward Pack, Jörg Bentzien, Donald Souza, Darren Disalvo, Alison Kukulka, David S. Thomson, Raj Betageri, Gerald Nabozny
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:6640-6644
مصطلحات موضوعية: Agonist, medicine.drug_class, Clinical Biochemistry, Anti-Inflammatory Agents, Pharmaceutical Science, Pharmacology, Biochemistry, Mice, Structure-Activity Relationship, Receptors, Glucocorticoid, Glucocorticoid receptor, In vivo, Drug Discovery, medicine, Enzyme-linked receptor, Animals, Molecular Biology, chemistry.chemical_classification, Sulfonamides, Binding Sites, Chemistry, Arthritis, Organic Chemistry, Tryptamines, Protein Structure, Tertiary, Sulfonamide, Molecular Docking Simulation, Nuclear receptor, Molecular Medicine, Estrogen-related receptor gamma, Pharmacophore, Protein Binding
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6
المؤلفون: Kathy O’Shea, Denice M. Spero, Ronald L. Magolda, Mario G. Cardozo, Lisa H. Liu, Hanbo Hu, Derek Cogan, Heather Grbic, Thomas M. Farrell, John P. Wolak, John D. Ginn, Della White, Deborah D. Jeanfavre, Mohammed A. Kashem, Maryanne L. Brown, Anthony S. Prokopowicz, Carol Ann Homon, Erick R. R. Young, Joseph R. Woska, Paul Kaplita, Darren Disalvo, Georg Dahmann, Charles L. Cywin
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:225-230
مصطلحات موضوعية: CD4-Positive T-Lymphocytes, Models, Molecular, Protein Conformation, Clinical Biochemistry, Protein Kinase C-theta, Substituent, Pharmaceutical Science, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Humans, Structure–activity relationship, Homology modeling, Protein Kinase Inhibitors, Molecular Biology, Protein Kinase C, Protein kinase C, Molecular Structure, Chemistry, Kinase, Organic Chemistry, Hit to lead, Combinatorial chemistry, Isoenzymes, Pyrimidines, Interleukin-2, Molecular Medicine, Selectivity
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7
المؤلفون: Gerald Nabozny, Tazmeen Fadra-Khan, David S. Thomson, Christian Harcken, John R. Regan, Darren Disalvo, Richard M. Nelson, Daniel Kuzmich, Alison Kukulka, Jörg Bentzien
المصدر: Bioorganicmedicinal chemistry letters. 23(24)
مصطلحات موضوعية: Agonist, medicine.drug_class, Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Ligands, Biochemistry, Partial agonist, Steroid, Structure-Activity Relationship, Glucocorticoid receptor, Receptors, Glucocorticoid, Drug Discovery, medicine, Inverse agonist, Molecular Biology, Glucocorticoids, Sulfonamides, Binding Sites, Chemistry, Organic Chemistry, Hydrogen Bonding, Protein Structure, Tertiary, Molecular Docking Simulation, Nuclear receptor, Molecular Medicine, Estrogen-related receptor gamma, Steroids, Glucocorticoid, medicine.drug, Protein Binding
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8
المؤلفون: M. Mar Díaz-Requejo, Maurice Brookhart, Darren Disalvo
المصدر: ChemInform. 34
مصطلحات موضوعية: Reaction mechanism, Intramolecular reaction, Chemistry, chemistry.chemical_element, Hydrogen transfer, Homogeneous catalysis, General Chemistry, General Medicine, Alkenes, Silanes, Biochemistry, Combinatorial chemistry, Catalysis, Rhodium, Colloid and Surface Chemistry, Intramolecular force, Catalyst selectivity, Organometallic Compounds, Organic chemistry, Amines, Ethers, Hydrogen