-
1
المؤلفون: Peter J. Tummino, C.M. Jacobs, Elizabeth A. Lunney, Bradley Dean Tait, D. Ferguson, L. Hupe, D. Hupe
المصدر: Archives of Biochemistry and Biophysics. 316:523-528
مصطلحات موضوعية: Models, Molecular, Stereochemistry, medicine.medical_treatment, Carboxylic acid, Molecular Sequence Data, Carboxylic Acids, Biophysics, Biochemistry, Sulfone, chemistry.chemical_compound, Non-competitive inhibition, HIV-1 protease, medicine, Phenyl group, Computer Simulation, Amino Acid Sequence, Molecular Biology, chemistry.chemical_classification, Biphenyl, Binding Sites, Protease, biology, Biphenyl Compounds, HIV Protease Inhibitors, Recombinant Proteins, Kinetics, Solubility, chemistry, Drug Design, HIV-1, biology.protein, Lineweaver–Burk plot
-
2
المؤلفون: E A, Lunney, S E, Hagen, J M, Domagala, C, Humblet, J, Kosinski, B D, Tait, J S, Warmus, M, Wilson, D, Ferguson, D, Hupe
المصدر: Journal of Medicinal Chemistry. 37:2664-2677
مصطلحات موضوعية: Models, Molecular, Protein Conformation, Stereochemistry, medicine.medical_treatment, Molecular Conformation, Crystallography, X-Ray, HIV Protease, HIV-1 protease, Coumarins, Drug Discovery, medicine, Humans, Mass screening, chemistry.chemical_classification, Acquired Immunodeficiency Syndrome, Binding Sites, Protease, Molecular Structure, biology, Active site, Biological activity, 4-Hydroxycoumarins, HIV Protease Inhibitors, Enzyme, chemistry, Docking (molecular), Enzyme inhibitor, Drug Design, HIV-1, biology.protein, Molecular Medicine, Monte Carlo Method, Oligopeptides
-
3
المؤلفون: C J, Donahue, M, Santoro, D, Hupe, J M, Jones, B, Pollok, R, Heim, D, Giegel
المصدر: Cytometry. 45(3)
مصطلحات موضوعية: Green Fluorescent Proteins, Statistics as Topic, G1 Phase, Antibodies, Monoclonal, Gene Expression, Apoptosis, Flow Cytometry, Transfection, Resting Phase, Cell Cycle, Substrate Specificity, Antibodies, Monoclonal, Murine-Derived, Jurkat Cells, Luminescent Proteins, Tandem Repeat Sequences, Caspases, Humans
-
4Academic Journal
المؤلفون: Y Song, D Hupe, P J Tummino, P J Harvey, T Mcquade, J Domagala, R Gogliotti
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.601.6547; http://aac.asm.org/content/41/2/394.full.pdf
-
5
المؤلفون: J M, Domagala, R, Gogliotti, J P, Sanchez, M A, Stier, K, Musa, Y, Song, J, Loo, M, Reily, P, Tummino, P, Harvey, D, Hupe, L, Sharmeen, D, Mack, J, Scholten, J, Saunders, T, McQuade
المصدر: Drug design and discovery. 15(1)
مصطلحات موضوعية: Thioamides, Mice, Structure-Activity Relationship, Thiazoles, Alkylation, Anti-HIV Agents, Benzamides, HIV-1, Animals, Humans, Disulfides, Nucleocapsid Proteins, Cell Line
-
6
المؤلفون: J V, Prasad, E A, Lunney, K S, Para, P J, Tummino, D, Ferguson, D, Hupe, J M, Domagala, J W, Erickson
المصدر: Drug design and discovery. 13(3-4)
مصطلحات موضوعية: Models, Molecular, Structure-Activity Relationship, Cell Membrane Permeability, Molecular Structure, Drug Design, Drug Evaluation, Preclinical, Humans, HIV Protease Inhibitors, Caco-2 Cells, Crystallography, X-Ray, Protein Binding, Pyrans
-
7
المؤلفون: B D, Tait, J, Domagala, E L, Ellsworth, D, Ferguson, C, Gajda, D, Hupe, E A, Lunney, P J, Tummino
المصدر: Journal of molecular recognition : JMR. 9(2)
مصطلحات موضوعية: Models, Molecular, Structure-Activity Relationship, Binding Sites, HIV Protease, Protein Conformation, Pyridones, Pyrones, Drug Design, HIV Protease Inhibitors, Furans