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1Academic Journal
المؤلفون: Tian-li Yue, Weike Bao, Beat M. Jucker, Juan-li Gu, Anne M. Romanic, Peter J. Brown, Douglas T. Thudium, Rogely Boyce, Cynthia L. Burns-kurtis, Rosanna C. Mirabile, Karpagam Aravindhan, Eliot H. Ohlstein, Ms Rosanna, C. Mirabile, Ms Eliot, H. Ohlstein
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.325.2300; http://circ.ahajournals.org/content/108/19/2393.full.pdf
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2Academic Journal
المؤلفون: Susan Pickering, Juanli Gu, Evelyn Grau, Joyce Mao, Ganesh M. Sathe, Eliot H. Ohlstein, Tian-li Yue, Anne M. Romanic, Stephen M. Harrison, Weike Bao, Cynthia L. Burns-kurtis
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.335.6092; http://cardiovascres.oxfordjournals.org/content/54/3/549.full.pdf
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3
المؤلفون: Stefan Senger, Máire A. Convery, Robert J. Young, Stephanie Irvine, Iain M. McLay, Robert I. West, David J. Belton, Savvas Kleanthous, Carl Adams, John R. Toomey, Anne M. Exall, Anthony J. Pateman, Theresa J. Roethke, Caroline M. Whittaker, Laiq Chaudry, David E. Davies, Angela Patikis, Cynthia L. Burns-Kurtis, Nigel S. Watson, Gary J. Stelman, David W. Brown, John D. Harling, Wendy R. Irving, Chuen Chan, Ping Zhou
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:1588-1592
مصطلحات موضوعية: Serine Proteinase Inhibitors, medicine.drug_mechanism_of_action, Stereochemistry, Clinical Biochemistry, Coagulation Factor Xa, Factor Xa Inhibitor, Drug Evaluation, Preclinical, Administration, Oral, Pharmaceutical Science, Pharmacology, Crystallography, X-Ray, Biochemistry, Tissue plasminogen activator, Benzazepine, chemistry.chemical_compound, Tetrahydroisoquinolines, Drug Discovery, medicine, Animals, Molecular Biology, Molecular Structure, biology, Blood clotting, Tetrahydroisoquinoline, Organic Chemistry, Benzazepines, Rats, Long acting, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Factor Xa Inhibitors, medicine.drug
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4
المؤلفون: Shobha Senadhi, Joseph P. Marino, Cynthia L. Burns-Kurtis, Lorena A. Kallal, Dwight M. Morrow, Reema K. Thalji, Nambi Aiyar, Joseph A. Erhardt, Elizabeth A. Davenport
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:4104-4107
مصطلحات موضوعية: Bicyclic molecule, Chemistry, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Platelet Activation, Biochemistry, Chemical synthesis, In vitro, Receptors, Purinergic P2Y1, chemistry.chemical_compound, Drug Discovery, Purinergic P2Y Receptor Antagonists, Urea, Molecular Medicine, Potency, Platelet activation, Benzofuran, Receptor, Molecular Biology, Benzofurans
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5
المؤلفون: Savvas Kleanthous, Alan D. Borthwick, David Brown, Cynthia L. Burns-Kurtis, Matthew Campbell, Laiq Chaudry, Chuen Chan, Marie-Olive Clarte, Máire A. Convery, John D. Harling, Eric Hortense, Wendy R. Irving, Stephanie Irvine, Anthony J. Pateman, Angela N. Patikis, Ivan L. Pinto, Derek R. Pollard, Theresa J. Roethka, Stefan Senger, Gita P. Shah, Gary J. Stelman, John R. Toomey, Nigel S. Watson, Robert I. West, Caroline Whittaker, Ping Zhou, Robert J. Young
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:618-622
مصطلحات موضوعية: Binding Sites, Organic Chemistry, Clinical Biochemistry, Anticoagulants, Pharmaceutical Science, Crystallography, X-Ray, Biochemistry, Pyrrolidinones, Structure-Activity Relationship, Drug Design, Factor X, Drug Discovery, Molecular Medicine, Computer Simulation, Molecular Biology
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6
المؤلفون: Elizabeth A. Davenport, Reema K. Thalji, Nambi Aiyar, Todd L. Graybill, Peng Li, Allyn T. Londregan, Dwight M. Morrow, Angel I. Morales-Ramos, Terry Kiesow, Steve Zhao, John S. Mecom, Shobha Senadhi, Gregory D. Brown, Lorena A. Kallal, Beth Anne Knapp-Reed, Joseph P. Marino, Cynthia L. Burns-Kurtis
المصدر: Bioorganic & Medicinal Chemistry Letters. 18:6222-6226
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Stereoisomerism, Biochemistry, Chemical synthesis, Receptors, Purinergic P2Y1, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Purinergic P2 Receptor Antagonists, Combinatorial Chemistry Techniques, Humans, Structure–activity relationship, Receptor, Molecular Biology, chemistry.chemical_classification, Molecular Structure, Receptors, Purinergic P2, Chemistry, Organic Chemistry, Antagonist, Aromatic amine, Thrombosis, Aminoquinolines, Molecular Medicine, Platelet aggregation inhibitor, Piperidine, Platelet Aggregation Inhibitors
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7
المصدر: Journal of Pharmacology and Experimental Therapeutics. 328:231-239
مصطلحات موضوعية: Male, Agonist, medicine.drug_class, Thromboxane, Guinea Pigs, Receptors, Thromboxane, TRPV Cation Channels, Aorta, Thoracic, Vasodilation, Arachidonic Acids, Pharmacology, Rats, Sprague-Dawley, Thromboxane receptor, Mice, chemistry.chemical_compound, 8,11,14-Eicosatrienoic Acid, Hydroxyeicosatetraenoic Acids, medicine, Animals, Splanchnic Circulation, Receptor, Mice, Knockout, Leukotriene, Chemistry, Prostanoid, Rats, Trachea, Biochemistry, Vasoconstriction, 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid, cardiovascular system, Molecular Medicine, Vascular Resistance, lipids (amino acids, peptides, and proteins), Arachidonic acid
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8
المؤلفون: Anthony J. Pateman, John R. Toomey, Paul F. Koster, Augustin Amour, Saul Needle, Laiq Chaudry, Melanie A Abboud, Champa Patel, Angela Patikis, Cynthia L. Burns-Kurtis, Robert J. Young, Richard E. Valocik, David Brown, Ping Zhou, Chuen Chan, Nigel S. Watson
المصدر: Journal of Cardiovascular Pharmacology. 52:66-71
مصطلحات موضوعية: Male, Bleeding Time, medicine.drug_mechanism_of_action, Factor Xa Inhibitor, Administration, Oral, Vena Cava, Inferior, Pharmacology, Inferior vena cava, Rats, Sprague-Dawley, Fibrinolytic Agents, In vivo, Prothrombinase, Antithrombotic, Animals, Medicine, Carotid Artery Thrombosis, Receptor, Venous Thrombosis, Sulfonamides, Dose-Response Relationship, Drug, business.industry, Pyrrolidinones, Rats, Disease Models, Animal, medicine.vein, Hemostasis, Blood Coagulation Tests, Rabbits, Jugular Veins, Cardiology and Cardiovascular Medicine, business, Ex vivo, Factor Xa Inhibitors
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9
المؤلفون: Alan D. Borthwick, Marie Charbaut, Robert J. Young, Máire A. Convery, Ivan Leo Pinto, Andrew M. Mason, Weston Helen Elisabeth, Matthew Campbell, David W. Brown, Anthony J. Pateman, Henry Anderson Kelly, Derek Pollard, Shah Gita Punjabhai, John R. Toomey, N. Paul King, Stefan Senger, Eric Hortense, Ping Zhou, Hawa Diallo, Nigel S. Watson, Wendy R. Irving, Angela Patikis, Cynthia L. Burns-Kurtis, Savvas Kleanthous, Chuen Chan
المصدر: Bioorganic & Medicinal Chemistry Letters. 18:28-33
مصطلحات موضوعية: Male, Models, Molecular, Serine Proteinase Inhibitors, medicine.drug_mechanism_of_action, Antithrombotic Agent, Tertiary amine, Stereochemistry, Clinical Biochemistry, Factor Xa Inhibitor, Coagulation Factor Xa, Pharmaceutical Science, Biochemistry, Chemical synthesis, Rats, Sprague-Dawley, Structure-Activity Relationship, Drug Discovery, medicine, Animals, Molecular Biology, chemistry.chemical_classification, biology, Chemistry, Organic Chemistry, Anticoagulants, Stereoisomerism, Bridged Bicyclo Compounds, Heterocyclic, Thiophene derivatives, Pyrrolidinones, Rats, Sulfonamide, Enzyme inhibitor, biology.protein, Molecular Medicine, Hydrophobic and Hydrophilic Interactions, Factor Xa Inhibitors
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10
المؤلفون: Robert J. Young, David W. Brown, Stefan Senger, Chuen Chan, Máire A. Convery, Anthony J. Pateman, Nigel S. Watson, John R. Toomey, Ping Zhou, Henry Anderson Kelly, Shah Gita Punjabhai, Julia A. Hubbard, Angela Patikis, Cynthia L. Burns-Kurtis
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:2927-2930
مصطلحات موضوعية: Models, Molecular, medicine.drug_class, Stereochemistry, Morpholines, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Biochemistry, Structure-Activity Relationship, Dogs, Thrombin, Fibrinolytic Agents, Oral administration, Drug Discovery, medicine, Animals, Molecular Biology, chemistry.chemical_classification, Sulfonamides, Molecular Structure, biology, Organic Chemistry, Rats, Sulfonamide, Bioavailability, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Factor Xa Inhibitors, Discovery and development of direct thrombin inhibitors, medicine.drug
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11
المؤلفون: Terry P. Kenakin, David W. Gray, Jim Coote, Alan Wise, Heather Giles, Cynthia L. Burns-Kurtis, Sara Pritchard, Noel Lloyd Staton, Jason D. Brown, Richard J. Wilson, Valerie Morrison, Susan Roomans, Sharron A. Rhodes, Kerri Ann Cartwright, Gerard Martin Paul Giblin, Jannatara Chowdhury, Vanessa J. Shield
المصدر: British Journal of Pharmacology. 148:326-339
مصطلحات موضوعية: Pharmacology, Agonist, Chemistry, medicine.drug_class, Stereochemistry, Prostaglandin E2 receptor, Antagonist, Prostanoid, musculoskeletal system, chemistry.chemical_compound, Competitive antagonist, cardiovascular system, medicine, Radioligand, lipids (amino acids, peptides, and proteins), Platelet, Receptor
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12
المؤلفون: Cynthia L. Burns-Kurtis, Josephine H. Fox, Saul Needle, Elizabeth A. Capper, Anne M. Romanic, Alan R. Olzinski, Michael S. McQueney, Fiona M. Kelly
المصدر: Cardiovascular Research. 62:610-620
مصطلحات موضوعية: Male, Neointima, Pathology, medicine.medical_specialty, Physiology, Blotting, Western, Hypercholesterolemia, Constriction, Pathologic, Biology, Polymerase Chain Reaction, Basement Membrane, Collagen Type I, Monocytes, Muscle, Smooth, Vascular, Extracellular matrix, Andrology, Cell Movement, Laminin, Physiology (medical), medicine, Animals, Humans, Cystatin C, Cathepsin S, Foam cell, Cathepsin, Extracellular Matrix Proteins, CATS, Macrophages, Cathepsins, Cystatins, Immunohistochemistry, Fibronectins, Femoral Artery, Lipoproteins, LDL, Fibronectin, biology.protein, Rabbits, Cardiology and Cardiovascular Medicine, Angioplasty, Balloon
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13
المؤلفون: Weike Bao, Juan-Li Gu, Eliot H. Ohlstein, Tian-Li Yue, Douglas T. Thudium, Anne M. Romanic, Cynthia L. Burns-Kurtis, Beat M. Jucker, Jianqi Cui, Rogely W. Boyce, Karpagam Aravindhan, Peter Brown, Rosanna C. Mirabile
المصدر: Circulation. 108:2393-2399
مصطلحات موضوعية: Male, Agonist, medicine.medical_specialty, medicine.drug_class, Premedication, Drug Evaluation, Preclinical, Myocardial Infarction, Myocardial Ischemia, Ischemia, Down-Regulation, Receptors, Cytoplasmic and Nuclear, Peroxisome proliferator-activated receptor, Myocardial Reperfusion Injury, Mice, NF-KappaB Inhibitor alpha, Physiology (medical), Internal medicine, Animals, Medicine, RNA, Messenger, Myocardial infarction, Receptor, Ligation, Beta oxidation, Mice, Knockout, Cardioprotection, chemistry.chemical_classification, business.industry, Myocardium, Phenylurea Compounds, Fatty Acids, NF-kappa B, medicine.disease, Matrix Metalloproteinases, Butyrates, Chemotaxis, Leukocyte, Endocrinology, chemistry, Cytokines, I-kappa B Proteins, Cardiology and Cardiovascular Medicine, business, Oxidation-Reduction, Reperfusion injury, Transcription Factors
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14
المؤلفون: Eliot H. Ohlstein, Anne M. Romanic, Cynthia L. Burns-Kurtis, Anthony J. Arleth, Zhaohui Ao
المصدر: American Journal of Physiology-Renal Physiology. 281:F309-F317
مصطلحات موضوعية: Adult, Male, medicine.medical_specialty, Adolescent, Matrix Metalloproteinases, Membrane-Associated, Physiology, Tubular atrophy, Immunoblotting, Matrix metalloproteinase, Biology, Kidney, Polymerase Chain Reaction, Nephropathy, Extracellular matrix, Downregulation and upregulation, Internal medicine, medicine, Loop of Henle, Humans, RNA, Messenger, Aged, Tissue Extracts, Proteolytic enzymes, Metalloendopeptidases, Middle Aged, medicine.disease, Immunohistochemistry, Up-Regulation, Cell biology, Diabetes Mellitus, Type 1, Endocrinology, medicine.anatomical_structure, Matrix Metalloproteinase 2, Female
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15
المؤلفون: Máire A. Convery, Stephanie Irvine, Graham Foster, Mike Blows, Robert J. Young, Steve Jackson, Stefan Senger, Angela Patikis, Eric Hortense, Cynthia L. Burns-Kurtis, John R. Toomey, Carl Adams, Savvas Kleanthous, Gary J. Stelman, David W. Brown, John D. Harling, Nigel S. Watson, Ping Zhou, Robert I. West, Wendy R. Irving, Anne M. Exall, Theresa J. Roethka, David E. Davies, Anthony J. Pateman, Chuen Chan, Laiq Chaudry, Caroline M. Whittaker
المصدر: Bioorganicmedicinal chemistry letters. 21(6)
مصطلحات موضوعية: Models, Molecular, Pyrrolidines, Serine Proteinase Inhibitors, medicine.drug_mechanism_of_action, Stereochemistry, Clinical Biochemistry, Coagulation Factor Xa, Factor Xa Inhibitor, Pharmaceutical Science, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Drug Discovery, medicine, Molecular Biology, biology, Blood clotting, Chemistry, Organic Chemistry, Rational design, Thiophene derivatives, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, Factor Xa Inhibitors
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16
المؤلفون: Mark Pullen, David J. Behm, Charlene Wu, Cynthia L. Burns-Kurtis, Stephen A. Douglas, Andrea Ogbonna
المصدر: Circulation. 118
مصطلحات موضوعية: biology, business.industry, Cytochrome P450, Vasodilation, Endogeny, Pharmacology, Epoxyeicosatrienoic acid, Thromboxane receptor, chemistry.chemical_compound, chemistry, Physiology (medical), cardiovascular system, biology.protein, Medicine, lipids (amino acids, peptides, and proteins), Arachidonic acid, Cardiology and Cardiovascular Medicine, Receptor, business, Function (biology)
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17Structure and property based design of factor Xa inhibitors: pyrrolidin-2-ones with biaryl P4 motifs
المؤلفون: N. Paul King, Stefan Senger, Matthew Campbell, Henry Anderson Kelly, Máire A. Convery, David W. Brown, Shah Gita Punjabhai, Angela Patikis, Cynthia L. Burns-Kurtis, Savvas Kleanthous, Marie Charbaut, Alan D. Borthwick, Ivan Leo Pinto, Weston Helen Elisabeth, John R. Toomey, Chuen Chan, Chun-wa Chung, Robert J. Young, Nigel S. Watson, Derek Pollard, Andrew M. Mason, Anthony J. Pateman
المصدر: Bioorganicmedicinal chemistry letters. 18(1)
مصطلحات موضوعية: Male, Models, Molecular, Quantitative structure–activity relationship, Serine Proteinase Inhibitors, medicine.drug_mechanism_of_action, Stereochemistry, Clinical Biochemistry, Factor Xa Inhibitor, Pharmaceutical Science, Biochemistry, Chemical synthesis, Sulfone, Rats, Sprague-Dawley, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, medicine, Animals, Molecular Biology, Sulfonamides, Blood clotting, biology, Chemistry, Organic Chemistry, Anticoagulants, Pyrrolidinones, Rats, Enzyme inhibitor, Drug Design, Lipophilicity, biology.protein, Lactam, Molecular Medicine, Factor Xa Inhibitors
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18
المؤلفون: Robert J. Young, Alan D. Borthwick, Nigel S. Watson, Weston Helen Elisabeth, Chun-wa Chung, J. Nicole Hamblin, Chuen Chan, Anthony J. Pateman, Savvas Kleanthous, Laiq Chaudry, Shah Gita Punjabhai, David W. Brown, Matthew Campbell, Champa Patel, Máire A. Convery, Stefan Senger, Lisa Johnstone, Angela Patikis, Cynthia L. Burns-Kurtis, Henry Anderson Kelly, Caroline Whitworth, Ping Zhou, John R. Toomey
المصدر: Journal of medicinal chemistry. 50(7)
مصطلحات موضوعية: Male, Models, Molecular, Pyrrolidines, Molecular model, medicine.drug_mechanism_of_action, Stereochemistry, medicine.drug_class, Morpholines, Factor Xa Inhibitor, Carboxamide, Crystallography, X-Ray, Ligands, Rats, Sprague-Dawley, Structure-Activity Relationship, Dogs, Drug Discovery, medicine, Animals, Humans, Binding site, Serum Albumin, Sulfonamides, Bicyclic molecule, biology, Molecular Structure, Chemistry, Anticoagulants, Stereoisomerism, Human serum albumin, Rats, Enzyme inhibitor, Lipophilicity, Factor Xa, biology.protein, Prothrombin Time, Molecular Medicine, Female, medicine.drug, Factor Xa Inhibitors, Protein Binding
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19
المؤلفون: Joseph A. Erhardt, Richard E. Valocik, Kodandaram Pillarisetti, John R. Toomey, Cynthia L. Burns-Kurtis, Paul F. Koster, T. M. Danoff, Melanie A Abboud
المصدر: Journal of thrombosis and haemostasis : JTH. 4(9)
مصطلحات موضوعية: Protamine sulfate, Drug Evaluation, Preclinical, Hemorrhage, Vena Cava, Inferior, Pharmacology, Inferior vena cava, Antithrombotic, medicine, Animals, cardiovascular diseases, Glycosides, Protamines, Thrombus, Glycosaminoglycans, Venous Thrombosis, Dose-Response Relationship, Drug, business.industry, Antithrombin, Warfarin, Anticoagulants, Hematology, medicine.disease, Thrombosis, Rats, Venous thrombosis, Disease Models, Animal, medicine.vein, Heparin Cofactor II, business, medicine.drug
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20
المؤلفون: Matthew Campbell, Ping Zhou, Robert J. Young, Weston Helen Elisabeth, Savvas Kleanthous, David W. Brown, Champa Patel, Satish Dayal, Shah Gita Punjabhai, Alan D. Borthwick, N. Paul King, Cynthia L. Burns-Kurtis, Stefan Senger, Hawa Diallo, Máire A. Convery, Nigel S. Watson, Paul W. Smith, Henry Anderson Kelly, Miriam Crowe, Chuen Chan, Anthony J. Pateman, Jackie E. Mordaunt, Andrew M. Mason
المصدر: Bioorganicmedicinal chemistry letters. 16(23)
مصطلحات موضوعية: Models, Molecular, medicine.drug_mechanism_of_action, Molecular model, Stereochemistry, Clinical Biochemistry, Factor Xa Inhibitor, Antithrombin III, Substituent, Pharmaceutical Science, Crystallography, X-Ray, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Structure-Activity Relationship, Amide, Drug Discovery, Hydrolase, medicine, Pyrroles, Molecular Biology, chemistry.chemical_classification, Alanine, Binding Sites, Molecular Structure, Organic Chemistry, Anticoagulants, Amides, Sulfonamide, chemistry, Drug Design, Lipophilicity, Factor Xa, Molecular Medicine