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1Academic Journal
المؤلفون: Romain Pierre, Anne Brethon, Sylvain A. Jacques, Aurélie Blond, Sandrine Chambon, Sandrine Talano, Catherine Raffin, Branislav Musicki, Claire Bouix-Peter, Loic Tomas, Gilles Ouvry, Rémy Morgentin, Laurent F. Hennequin, Craig S. Harris
المصدر: Beilstein Journal of Organic Chemistry, Vol 17, Iss 1, Pp 156-165 (2021)
مصطلحات موضوعية: 7-azabenzotriazole, hinge-binder, ionic hydrogenation, library, pyridine-2(1h)-one, Science, Organic chemistry, QD241-441
وصف الملف: electronic resource
Relation: https://doaj.org/toc/1860-5397
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2
المؤلفون: Stéphan, Billié, Kevin, Reversé, Sandrine, Chambon, Tony, Cachot, Romain, Pierre, Thibaud, Gerfaud, Davide, Longoni, Massimiliano, Gennari, Héloïse, Raynard, Eric, Talbot, Karine, Charras, Didier, Bertin, Marine, Joly-Battaglini, Gerald, Pedrassi, Jean-Guy, Boiteau, Cécile, Cren, Craig S, Harris
المصدر: Journal of Pharmaceutical and Biomedical Analysis. 220:114993
مصطلحات موضوعية: Clinical Biochemistry, Drug Discovery, Lymecycline, Pharmaceutical Science, Capsules, Drug Contamination, Chromatography, High Pressure Liquid, Spectroscopy, Analytical Chemistry
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3
المؤلفون: Jean-Guy Boiteau, Jing Jing, Vanina Cosenza, Tamiris Vilas Boas Figueiredo, Isabelle Jeacomine, Thibaud Gerfaud, Rachel Auzély-Velty, Johan Olsson, Craig S. Harris, Yu Ogawa
المساهمون: Centre de Recherches sur les Macromolécules Végétales (CERMAV), Institut de Chimie du CNRS (INC)-Université Grenoble Alpes (UGA)-Centre National de la Recherche Scientifique (CNRS)
المصدر: Polymer Chemistry
Polymer Chemistry, Royal Society of Chemistry-RSC, 2020, 11, pp.3800-3811. ⟨10.1039/D0PY00308E⟩مصطلحات موضوعية: Polymers and Plastics, Organic Chemistry, Diol, Rational design, Bioengineering, 02 engineering and technology, 010402 general chemistry, 021001 nanoscience & nanotechnology, Ring (chemistry), 01 natural sciences, Biochemistry, Combinatorial chemistry, 0104 chemical sciences, chemistry.chemical_compound, Molecular dynamics, chemistry, Self-healing hydrogels, Molecule, [CHIM]Chemical Sciences, 0210 nano-technology, [SDV.IB.BIO]Life Sciences [q-bio]/Bioengineering/Biomaterials, Boronic acid, Conjugate
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المؤلفون: Jean-Guy Boiteau, Yu Ogawa, Johan Olsson, Raphael Michel, Craig S. Harris, Jing Jing, Thibaud Gerfaud, Rachel Auzély-Velty, Sonia Ortega, Tamiris Vilas Boas Figueiredo, Vanina Cosenza, Alicia Vallet, Isabelle Jeacomine
المساهمون: Centre de Recherches sur les Macromolécules Végétales (CERMAV), Institut de Chimie du CNRS (INC)-Centre National de la Recherche Scientifique (CNRS)-Université Grenoble Alpes (UGA), Institut de biologie structurale (IBS - UMR 5075), Centre National de la Recherche Scientifique (CNRS)-Institut de Recherche Interdisciplinaire de Grenoble (IRIG), Direction de Recherche Fondamentale (CEA) (DRF (CEA)), Commissariat à l'énergie atomique et aux énergies alternatives (CEA)-Commissariat à l'énergie atomique et aux énergies alternatives (CEA)-Direction de Recherche Fondamentale (CEA) (DRF (CEA)), Commissariat à l'énergie atomique et aux énergies alternatives (CEA)-Commissariat à l'énergie atomique et aux énergies alternatives (CEA)-Université Grenoble Alpes (UGA), Nestle Skin Health GALDERMA R&D, Institut de Chimie du CNRS (INC)-Université Grenoble Alpes (UGA)-Centre National de la Recherche Scientifique (CNRS)
المصدر: Soft Matter
Soft Matter, 2020, 16 (15), pp.3628-3641. ⟨10.1039/D0SM00178C⟩
Soft Matter, Royal Society of Chemistry, 2020, 16 (15), pp.3628-3641. ⟨10.1039/D0SM00178C⟩مصطلحات موضوعية: Diol, Kinetics, 02 engineering and technology, 010402 general chemistry, 01 natural sciences, chemistry.chemical_compound, Rheology, Hyaluronic Acid, [SDV.IB.BIO]Life Sciences [q-bio]/Bioengineering/Biomaterials, Nuclear Magnetic Resonance, Biomolecular, ComputingMilieux_MISCELLANEOUS, chemistry.chemical_classification, technology, industry, and agriculture, Rational design, Hydrogels, General Chemistry, Polymer, [CHIM.MATE]Chemical Sciences/Material chemistry, Hydrogen-Ion Concentration, 021001 nanoscience & nanotechnology, Condensed Matter Physics, Combinatorial chemistry, Boronic Acids, 0104 chemical sciences, [CHIM.POLY]Chemical Sciences/Polymers, chemistry, Covalent bond, Self-healing hydrogels, 0210 nano-technology, [PHYS.COND.CM-SCM]Physics [physics]/Condensed Matter [cond-mat]/Soft Condensed Matter [cond-mat.soft], Boronic acid
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المؤلفون: Craig S. Harris, Romain Pierre, Rodolphe Vatinel, Jean-Marie Arlabosse, Veronique Parnet, Catherine Raffin, Claire Bouix-Peter, Thibaud Gerfaud, Sebastien Daver, Jean-Guy Boiteau, Branislav Musicki, Guillaume Lafitte, Loïc Tomas, Gilles Ouvry
المصدر: Tetrahedron. 74:5974-5986
مصطلحات موضوعية: 010405 organic chemistry, Chemistry, Organic Chemistry, Topical treatment, Pharmacology, 010402 general chemistry, medicine.disease, 01 natural sciences, Biochemistry, 0104 chemical sciences, RAR-related orphan receptor gamma, Psoriasis, Drug Discovery, medicine, Inverse agonist
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المؤلفون: Corinne Millois, Loïc Tomas, Catherine Comino, Laurence Dumais, Sandrine Talano, Kevin Reverse, Céline Mathieu, Craig S. Harris, Nicolas Vanthuyne, Grégoire Mouis, Anne-Laurence Ghilini, Laurent F. Hennequin, Claire Bouix-Peter, Vincent Rodeschini, Ghizlane El-Bazbouz, Laurence Clary, Sandrine Chambon, Romain Pierre, Jean-François Fournier, Anne Brethon
المساهمون: Nestle Skin Health GALDERMA R&D, Institut des Sciences Moléculaires de Marseille (ISM2), Aix Marseille Université (AMU)-École Centrale de Marseille (ECM)-Institut de Chimie du CNRS (INC)-Centre National de la Recherche Scientifique (CNRS), edelris
المصدر: Tetrahedron
Tetrahedron, Elsevier, 2018, 74 (37), pp.4805-4822. ⟨10.1016/j.tet.2018.07.029⟩
Tetrahedron, 2018, 74 (37), pp.4805-4822. ⟨10.1016/j.tet.2018.07.029⟩مصطلحات موضوعية: 0301 basic medicine, Drug, Peptidomimetic, media_common.quotation_subject, Caspase 1, 01 natural sciences, Biochemistry, 03 medical and health sciences, chemistry.chemical_compound, Drug Discovery, [CHIM]Chemical Sciences, media_common, 010405 organic chemistry, Drug discovery, Organic Chemistry, Acetal, Uracil, Combinatorial chemistry, 0104 chemical sciences, 3. Good health, 030104 developmental biology, chemistry, Caspase-1 inhibitors 1, Hemiacetal, 5-Trisubstitued uracil Peptidomimetics Topical application Excipient stability Chiral stability
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المؤلفون: Catherine Soulet, Laurent F. Hennequin, Nicolas Fleury-Brégeot, Craig S. Harris, Blanche Gauthier, Gwenaëlle Duvert, Etienne Thoreau, Laurent Chantalat, Karine Grisendi, Jean-François Fournier, Jerome Aubert, Michèle Aurelly, Rémy Morgentin, Claire Bouix-Peter, Bénédicte Drean, Guillaume Lafitte, Yushma Bhurruth-Alcor, Florence Joly, Jonathan Pascau, Branislav Musicki, Yves Rival, David Piwnica, Karinne Bouquet, Marion Delorme, T. Isabet, Corinne Millois, Loïc Tomas
المصدر: Bioorganic & Medicinal Chemistry Letters. 28:2985-2992
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Skin Neoplasms, Clinical Biochemistry, Histone Deacetylase 2, Pharmaceutical Science, Antineoplastic Agents, Apoptosis, Histone Deacetylase 1, Pharmacology, Crystallography, X-Ray, Biochemistry, Structure-Activity Relationship, 03 medical and health sciences, 0302 clinical medicine, Cell Line, Tumor, Drug Discovery, Hydrolase, medicine, Humans, Solubility, Molecular Biology, Cell Proliferation, chemistry.chemical_classification, Mycosis fungoides, Dose-Response Relationship, Drug, Molecular Structure, Quinine, Organic Chemistry, Cutaneous T-cell lymphoma, Squaramide, medicine.disease, Lymphoma, T-Cell, Cutaneous, Histone Deacetylase Inhibitors, 030104 developmental biology, Enzyme, chemistry, Cell culture, 030220 oncology & carcinogenesis, Molecular Medicine, Histone deacetylase, Drug Screening Assays, Antitumor
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المؤلفون: Laurence Dumais, Emeric Varvier, Guillaume Lafitte, Kana Kunihiro, Loïc Tomas, Craig S. Harris
المصدر: Advanced Synthesis & Catalysis. 360:2757-2761
مصطلحات موضوعية: 010405 organic chemistry, Chemistry, One-pot synthesis, General Chemistry, 010402 general chemistry, Heterogeneous catalysis, 01 natural sciences, Combinatorial chemistry, 0104 chemical sciences
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المؤلفون: Ghizlane El-Bazbouz, Loïc Tomas, Romain Pierre, Grégoire Mouis, Gilles Ouvry, Frédéric Gaigne, Craig S. Harris
المصدر: Synlett. 29:1102-1106
مصطلحات موضوعية: Steric effects, Hydroxamic acid, Drug discovery, Organic Chemistry, 010402 general chemistry, 01 natural sciences, Combinatorial chemistry, 0104 chemical sciences, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, chemistry, 030220 oncology & carcinogenesis, Identification (biology), Polystyrene
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المؤلفون: Didier M. Roche, Danielle Orfila, Ghizlane El-Bazbouz, Laurence Dumais, Laurent F. Hennequin, Céline Mathieu, Michèle Aurelly, Jerome Aubert, Claude Lardy, Etienne Thoreau, Anne-Pascale Luzy, Claire Bouix-Peter, Kenny Mebrouk, T. Isabet, Jean-François Fournier, Kevin Reverse, Catherine Comino, Corinne Millois, Anne-Laurence Ghilini, Jonathan Pascau, Sandrine Talano, Anne Brethon, Craig S. Harris, Romain Pierre, Sandrine Chambon, Laurence Clary, Olivier Christin, Laurent Chantalat, Vincent Rodeschini
المصدر: Journal of Medicinal Chemistry. 61:4030-4051
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Protein Conformation, Administration, Topical, medicine.medical_treatment, Caspase 1, Drug design, Pharmacology, 01 natural sciences, Cell Line, Mice, 03 medical and health sciences, chemistry.chemical_compound, Acne Vulgaris, Drug Discovery, medicine, Animals, Humans, Tissue Distribution, Caspase, Acne, Protease, biology, 010405 organic chemistry, Uracil, medicine.disease, Caspase Inhibitors, 0104 chemical sciences, 030104 developmental biology, chemistry, Drug Design, Solvents, biology.protein, Molecular Medicine, Pharmacophore, Phototoxicity
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المؤلفون: Craig S. Harris, Isabelle Cardinaud, Feriel Hacini-Rachinel, Nicolas Rodeville, Audrey Beillard, Arnaud Reitz, Marilyne Bourotte, Benoit Deprez, Laetitia Bonnary, Catherine Comino, Corinne Millois, Delphine Spiesse, Claire Bouix-Peter, Denis Duvert, Jean-Guy Boiteau, Jean-Marie Arlabosse, Yushma Bhurruth-Alcor, Anne-Pascale Luzy, Laurent F. Hennequin, Gaëlle Polge, Emmanuel Vial, Loïc Tomas, Samuel Tabet, Kevin Reverse, Arnaud Mathieu, Artur Pinto, Angélique Feret, Karine Bouquet, Gilles Ouvry, Stéphanie Astri, Nicolas Orsini, Jonathan Pascau, Nathalie Taquet, David Piwnica, Patricia Rossio
المصدر: Bioorganic & Medicinal Chemistry. 26:945-956
مصطلحات موضوعية: 0301 basic medicine, Process development, Administration, Topical, Clinical Biochemistry, Druggability, Pharmaceutical Science, Topical treatment, ADAM17 Protein, Pharmacology, Hydroxamic Acids, Skin Diseases, 01 natural sciences, Biochemistry, Mice, 03 medical and health sciences, In vivo, Psoriasis, Drug Discovery, medicine, Animals, Humans, Enzyme Inhibitors, Molecular Biology, Mice, Hairless, Sulfonamides, Tumor Necrosis Factor-alpha, 010405 organic chemistry, Chemistry, Organic Chemistry, Oxazolone, medicine.disease, Tace inhibitor, 0104 chemical sciences, 030104 developmental biology, Solubility, Drug Design, Microsomes, Liver, Molecular Medicine, Female
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المؤلفون: Marcus Gastreich, Laurence Clary, Jonathan Pascau, Anne Brethon, Laurent Chantalat, Olivier Christin, Etienne Thoreau, Jean-François Fournier, Craig S. Harris, Didier Roche, T. Isabet, Vincent Rodeschini
المصدر: Bioorganic & Medicinal Chemistry Letters. 27:5373-5377
مصطلحات موضوعية: 0301 basic medicine, Scaffold, Stereochemistry, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, CASPASE 1 INHIBITOR, Crystallography, X-Ray, Scaffold hopping, 01 natural sciences, Biochemistry, Inhibitory Concentration 50, 03 medical and health sciences, chemistry.chemical_compound, 4-Butyrolactone, Drug Discovery, Molecular Biology, Biological Products, Binding Sites, Natural product, 010405 organic chemistry, Caspase 1, Organic Chemistry, Hydrogen Bonding, Dipeptides, Caspase Inhibitors, Combinatorial chemistry, Protein Structure, Tertiary, 0104 chemical sciences, Molecular Docking Simulation, 030104 developmental biology, chemistry, Docking (molecular), Molecular Medicine, Azabicyclo Compounds
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المؤلفون: Arnaud Reitz, Corinne Millois, Marilyne Bourotte, Feriel Hacini-Rachinel, Carine Rosignoli, Arnaud Mathieu, Sandrine Chambon, Denis Duvert, Anne-Pascale Luzy, Laetitia Bonnary, Gwenaëlle Duvert, Gilles Ouvry, Jonathan Pascau, Craig S. Harris, Benoit Deprez, Laurent F. Hennequin, Catherine Comino, Yushma Bhurruth-Alcor, Yaël Berton, Nathalie Taquet, Claire Bouix-Peter, Gaëlle Polge, Kevin Reverse, Artur Pinto, Karine Bouquet
المصدر: Bioorganic & Medicinal Chemistry Letters. 27:1848-1853
مصطلحات موضوعية: 0301 basic medicine, Cellular activity, Side effect, Administration, Topical, Clinical Biochemistry, Pharmaceutical Science, Context (language use), ADAM17 Protein, Pharmacology, Hydroxamic Acids, 01 natural sciences, Biochemistry, 03 medical and health sciences, Psoriasis, Drug Discovery, medicine, Humans, Enzyme Inhibitors, Molecular Biology, Tumor necrosis factor α, ADME, chemistry.chemical_classification, 010405 organic chemistry, Organic Chemistry, medicine.disease, 0104 chemical sciences, 030104 developmental biology, Enzyme, chemistry, Molecular Medicine
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المؤلفون: Etienne Thoreau, Loïc Tomas, T. Isabet, Laurent Chantalat, Craig S. Harris, Sophie Deret, Alessandro Taddei, Emmanuel Vial, Emeric Varvier, Emilie Borde, Laurent Lamy, Claire Defoin-Platel, Catherine Soulet, Nathalie Taquet, Laetitia Bonnary, Anne-Pascale Luzy, Michèle Aurelly, Laurence Clary, Claire Bouix-Peter, Gilles Ouvry, Laurent F. Hennequin, Mathieu Forissier, Jonathan Pascau
المصدر: ACS Med Chem Lett
مصطلحات موضوعية: Chemistry, Kinase, Organic Chemistry, Drug Discovery, Biophysics, sense organs, Discovery and development of mTOR inhibitors, skin and connective tissue diseases, Biochemistry, Sapanisertib, PI3K/AKT/mTOR pathway
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15Academic Journal
المؤلفون: Craig S. Harris, O Craig, S. Hams, Simon Fraser University, Canada Camda, Van Volr Tvbmo
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.454.6927; http://www.nlc-bnc.ca/obj/s4/f2/dsk2/ftp03/MQ51353.pdf
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المؤلفون: Jean-François Fournier, Didier Roche, Craig S. Harris, Sandrine Talano, Anne Brethon, Claude Lardy, Laurence Clary, Claire Bouix-Peter, Vincent Rodeschini
المصدر: Tetrahedron Letters. 57:5924-5927
مصطلحات موضوعية: 010405 organic chemistry, Chemistry, Peptidomimetic, Organic Chemistry, Drug Discovery, Alkylation, 010402 general chemistry, 01 natural sciences, Biochemistry, Combinatorial chemistry, 0104 chemical sciences, Stereocenter
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17
المؤلفون: Romain Pierre, Etienne Thoreau, Catherine Raffin, Claire Bouix-Peter, Laurent Chantalat, Gaëlle Polge, Jonathan Pascau, Gilles Ouvry, Nathalie Taquet, Catherine Comino, Denis Duvert, Danielle Orfila, Agnès Perrin, Yves Rival, Laurent Francois Andre Hennequin, Laurent Lamy, Christophe Feret, Branislav Musicki, Veronique Parnet, Anne-Pascale Luzy, Olivier Christin, Fabrice Ciesielski, Craig S. Harris
المصدر: Bioorganic & Medicinal Chemistry Letters. 26:5802-5808
مصطلحات موضوعية: 0301 basic medicine, Indazoles, Drug Inverse Agonism, Clinical Biochemistry, Allosteric regulation, Pharmaceutical Science, Topical treatment, Pharmacology, Biochemistry, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Drug Discovery, Humans, Inverse agonist, Molecular Biology, Organic Chemistry, Nuclear Receptor Subfamily 1, Group F, Member 3, Molecular Docking Simulation, 030104 developmental biology, Nuclear receptor, chemistry, 030220 oncology & carcinogenesis, Molecular Medicine, Lead compound
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18
المؤلفون: Nicolas Rodeville, Jean-Guy Boiteau, Sebastien Daver, Corinne Millois, Jean-François Fournier, Laurence Dumais, Loïc Tomas, Laurence Clary, Kenny Mebrouk, Sandrine Talano, Romain Pierre, Craig S. Harris, Claire Bouix-Peter, Sandrine Chambon
المصدر: Tetrahedron Letters. 57:2367-2371
مصطلحات موضوعية: chemistry.chemical_classification, 5-nitrouracil, 010405 organic chemistry, Component (thermodynamics), Stereochemistry, Organic Chemistry, Uracil, Alkylation, 010402 general chemistry, 01 natural sciences, Biochemistry, 0104 chemical sciences, Amino acid, chemistry.chemical_compound, chemistry, Drug Discovery, Protecting group
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19
المؤلفون: Craig S. Harris, Romain Pierre, Arnaud Reitz, Claire Bouix-Peter, Grégoire Mouis, Karinne Bouquet, Laurence Clary, Gilles Ouvry, Yushma Bhurruth-Alcor, Audrey Beillard, Sandrine Chambon, Loïc Tomas, Corinne Millois
المصدر: Tetrahedron Letters. 57:2165-2170
مصطلحات موضوعية: chemistry.chemical_classification, Base (chemistry), 010405 organic chemistry, Chemistry, Carboxylic acid, Organic Chemistry, food and beverages, 010402 general chemistry, 01 natural sciences, Biochemistry, Carbonyl group, 0104 chemical sciences, chemistry.chemical_compound, Yield (chemistry), Drug Discovery, Organic chemistry, Carboxylic ester
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المؤلفون: Loïc Tomas, Rodolphe Vatinel, Craig S. Harris, Veronique Parnet, Gilles Ouvry, Catherine Raffin, Bénédicte Drean, Claire Bouix-Peter, Kana Kunihiro, Guillaume Lafitte, Branislav Musicki, Jean-François Fournier, Frédéric Gaigne, Romain Pierre, Céline Bonneaud
المصدر: Tetrahedron Letters. 58:3757-3759
مصطلحات موضوعية: Scope (project management), 010405 organic chemistry, Chemistry, Organic Chemistry, Drug Discovery, One-pot synthesis, Substrate (chemistry), Organic chemistry, 010402 general chemistry, 01 natural sciences, Biochemistry, 0104 chemical sciences, Butyl lithium