المؤلفون: Intagliata, Sebastiano, Ciaffaglione, Valeria, Consoli, Valeria, D'Amico, Agata Grazia, Vanella, Luca, Pittalà, Valeria, Sodano, Federica, Schiano, Marica Erminia, Sorrenti, Valeria, Salerno, Loredana

المساهمون: Intagliata, Sebastiano, Ciaffaglione, Valeria, Consoli, Valeria, D'Amico, Agata Grazia, Vanella, Luca, Pittalà, Valeria, Sodano, Federica, Schiano, Marica Erminia, Sorrenti, Valeria, Salerno, Loredana

مصطلحات موضوعية: Anticancer propertie, Codrug, Glioblastoma, HO-1 inhibitor, Temozolomide

Relation: volume:12; journal:EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY REPORTS; https://hdl.handle.net/11588/990211

الاتاحة: https://hdl.handle.net/11588/990211
https://doi.org/10.1016/j.ejmcr.2024.100227

المؤلفون: Albertini C., Naldi M., Petralla S., Strocchi S., Grifoni D., Monti B., Bartolini M., Bolognesi M. L.

المساهمون: Albertini C., Naldi M., Petralla S., Strocchi S., Grifoni D., Monti B., Bartolini M., Bolognesi M.L.

مصطلحات موضوعية: Alzheimer’s disease, Anti-amyloid, Anti-inflammatory, Codrug, Drug combination, Polypharmacology, Alzheimer Disease, Amyloid beta-Peptide, Animal, Behavior, Cell Survival, Cromolyn Sodium, Drosophila, Drug Design, Endocytosi, Ibuprofen, Immunomodulation, Mice, Microglia, Neuron, Neuroprotective Agent, Neurotoxin, Protein Aggregate, Rats, Wistar

وصف الملف: ELETTRONICO

Relation: info:eu-repo/semantics/altIdentifier/pmid/33669839; info:eu-repo/semantics/altIdentifier/wos/WOS:000624195100001; volume:26; issue:4; firstpage:1; lastpage:22; numberofpages:22; journal:MOLECULES; http://hdl.handle.net/11585/843407; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85102711388; https://www.mdpi.com/1420-3049/26/4/1112

الاتاحة: http://hdl.handle.net/11585/843407
https://doi.org/10.3390/molecules26041112
https://www.mdpi.com/1420-3049/26/4/1112

المؤلفون: Violet Eng Yee Lee (10004241), Zhi Chiaw Lim (10004244), Suet Li Chew (10004247), Wee Han Ang (1505530)

مصطلحات موضوعية: Biochemistry, Medicine, Molecular Biology, Neuroscience, Pharmacology, Biotechnology, Infectious Diseases, Space Science, Astronomical and Space Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, coumarin payload, self-immolative linkers, Pt, prodrug, coumarin derivatives, unconjugated cinnamate, bioactive payload, Traceless Codrug Delivery, self-immolative 4- aminobenzyl linkers, payload release, linker artifact

Relation: https://figshare.com/articles/journal_contribution/_b_Strategy_for_Traceless_Codrug_Delivery_with_Platinum_IV_Prodrug_Complexes_Using_Self-Immolative_Linkers_b_/13607754

الاتاحة: https://doi.org/10.1021/acs.inorgchem.0c03299.s001

المؤلفون: A. V. Sosnov, F. M. Semchenko, M. I. Vlasov, V. N. Tohmahchi, A. A. Sosnova

المصدر: Разработка и регистрация лекарственных средств, Vol 0, Iss 2, Pp 176-187 (2019)

مصطلحات موضوعية: opioid, non-narcotic analgesic, biological target, multitargeted formulation, multimodal analgesia, pharmaceutical composition, fixed-dose combination, codrug, Pharmaceutical industry, HD9665-9675

وصف الملف: electronic resource

Relation: https://www.pharmjournal.ru/jour/article/view/427; https://doaj.org/toc/2305-2066; https://doaj.org/toc/2658-5049

URL الوصول: https://doaj.org/article/a1a51f4d3b7c4081aefebb2131a13303

المؤلفون: Verdugo-Escamilla, Cristóbal, Acebedo Martínez, Francisco Javier, Domínguez Martín, Alicia, Gómez Morales, Jaime, Choquesillo Lazarte, Duane

مصطلحات موضوعية: Cocrystal, Codrug, Hydrochlorothiazide, Caffeine, Mechanochemical synthesis

Relation: Verdugo-Escamilla, C.; Alarcón-Payer, C.; Frontera, A.; Acebedo-Martínez, F.J.; Domínguez-Martín, A.; Gómez-Morales, J.; Choquesillo-Lazarte, D. Interconvertible Hydrochlorothiazide–Caffeine Multicomponent Pharmaceutical Materials: A Solvent Issue. Crystals 2020, 10, 1088. https://doi.org/10.3390/cryst10121088; http://hdl.handle.net/10481/66592

الاتاحة: http://hdl.handle.net/10481/66592
https://doi.org/10.3390/cryst10121088

المؤلفون: Rossi M., Petralla S., Protti M., Baiula M., Kobrlova T., Soukup O., Spampinato S. M., Mercolini L., Monti B., Bolognesi M. L.

المساهمون: Rossi M., Petralla S., Protti M., Baiula M., Kobrlova T., Soukup O., Spampinato S.M., Mercolini L., Monti B., Bolognesi M.L.

مصطلحات موضوعية: Codrug, Polypharmacology, Valproic acid, α-linolenic acid

وصف الملف: ELETTRONICO

Relation: info:eu-repo/semantics/altIdentifier/pmid/33329762; info:eu-repo/semantics/altIdentifier/wos/WOS:000599586900005; volume:11; issue:12; firstpage:2406-2413; lastpage:2413; numberofpages:8; journal:ACS MEDICINAL CHEMISTRY LETTERS; https://hdl.handle.net/11585/786566; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85095879511

الاتاحة: https://hdl.handle.net/11585/786566
https://doi.org/10.1021/acsmedchemlett.0c00375
https://pubs.acs.org/doi/10.1021/acsmedchemlett.0c00375

المؤلفون: Yazici, Aysenur, Marinelli, Lisa, Cacciatore, Ivana, Emsen, Bugrahan, Eusepi, Piera, Di Biase, Giuseppe, Di Stefano, Antonio, Mardinoglu, Adil, Turkez, Hasan

المصدر: Current Drug Delivery. 18(3):350-356

مصطلحات موضوعية: Anti-proliferative action, codrug strategy, carvacrol codrug, glioblastoma multiforme, gene expression

وصف الملف: print

URL الوصول: https://urn.kb.se/resolve?urn=urn:nbn:se:kth:diva-296450

المؤلفون: A. V. Sosnov, F. M. Semchenko, M. I. Vlasov, V. N. Tohmahchi, A. A. Sosnova, А. В. Соснов, Ф. М. Семченко, М. И. Власов, В. Н. Тохмахчи, А. А. Соснова

المصدر: Drug development & registration; № 2 (2017); 176-187 ; Разработка и регистрация лекарственных средств; № 2 (2017); 176-187 ; 2658-5049 ; 2305-2066

مصطلحات موضوعية: солекарство, non-narcotic analgesic, biological target, multitargeted formulation, multimodal analgesia, pharmaceutical composition, fixed-dose combination, codrug, ненаркотический анальгетик, биомишень, мультитаргетный препарат, мультимодальная анальгезия, фармацевтическая композиция, комбинация фиксированного состава

وصف الملف: application/pdf

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الاتاحة: https://www.pharmjournal.ru/jour/article/view/427

المؤلفون: Violet Eng Yee Lee, Zhi Chiaw Lim, Suet Li Chew, Wee Han Ang

المصدر: Inorganic Chemistry. 60:1823-1831

مصطلحات موضوعية: Aqueous solution, Codrug, 010405 organic chemistry, Decarboxylation, Chemistry, chemistry.chemical_element, Prodrug, 010402 general chemistry, Coumarin, 01 natural sciences, Combinatorial chemistry, 0104 chemical sciences, Inorganic Chemistry, chemistry.chemical_compound, Molecule, Physical and Theoretical Chemistry, Platinum, Linker

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::ccea6e5c9b4822ee4425742b951143a4
https://doi.org/10.1021/acs.inorgchem.0c03299

المؤلفون: Arunava Dasgupta, Kakasaheb R. Mahadik, Suneela Dhaneshwar, Neha V. Bhilare

المصدر: Drug and Chemical Toxicology. 45:850-860

مصطلحات موضوعية: Male, Drug, Tuberculosis, Antioxidant, Health, Toxicology and Mutagenesis, media_common.quotation_subject, medicine.medical_treatment, Antitubercular Agents, 010501 environmental sciences, Pharmacology, Toxicology, 01 natural sciences, Antioxidants, Mice, 03 medical and health sciences, 0302 clinical medicine, Isoniazid, medicine, Animals, Rats, Wistar, Adverse effect, 0105 earth and related environmental sciences, media_common, Liver injury, Chemical Health and Safety, Codrug, business.industry, Public Health, Environmental and Occupational Health, General Medicine, bacterial infections and mycoses, medicine.disease, Sulfur containing, Rats, Pharmaceutical Preparations, Chemical and Drug Induced Liver Injury, Rifampin, business, Sulfur, 030217 neurology & neurosurgery, medicine.drug

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cd5d2d5e524e4bfbd6b976f190e60d9c
https://doi.org/10.1080/01480545.2020.1778021

المؤلفون: Yan-Tuan Li, Fan-Zhi Bu, Zhi-Yong Wu, Ling-Yang Wang, Cui-Wei Yan

المصدر: Crystal Growth & Design. 20:3236-3246

مصطلحات موضوعية: Codrug, 010405 organic chemistry, Chemistry, medicine.drug_class, Amantadine Hydrochloride, General Chemistry, 010402 general chemistry, Condensed Matter Physics, 01 natural sciences, Combinatorial chemistry, Cocrystal, 0104 chemical sciences, Sulfathiazole, medicine, General Materials Science, Antiviral drug, medicine.drug

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::597c96198214be2c7b1663f5a6643cca
https://doi.org/10.1021/acs.cgd.0c00075

المؤلفون: Jaime Gómez-Morales, Duane Choquesillo-Lazarte, Alicia Domínguez-Martín, Antonio Frontera, Carolina Alarcón-Payer, Francisco Javier Acebedo-Martínez, Cristóbal Verdugo-Escamilla

المساهمون: European Commission, Agencia Estatal de Investigación (España), Ministerio de Ciencia, Innovación y Universidades (España), [Verdugo-Escamilla, Cristobal] Univ Granada, Lab Estudios Cristalog, IACT, CSIC, Avda Palmeras 4, Armilla 18100, Spain, [Javier Acebedo-Martinez, Francisco] Univ Granada, Lab Estudios Cristalog, IACT, CSIC, Avda Palmeras 4, Armilla 18100, Spain, [Gomez-Morales, Jaime] Univ Granada, Lab Estudios Cristalog, IACT, CSIC, Avda Palmeras 4, Armilla 18100, Spain, [Choquesillo-Lazarte, Duane] Univ Granada, Lab Estudios Cristalog, IACT, CSIC, Avda Palmeras 4, Armilla 18100, Spain, [Alarcon-Payer, Carolina] Hosp Univ Jaen, Serv Farm, Jaen 23007, Spain, [Frontera, Antonio] Univ Illes Balears, Dept Chem, Crta Valldemossa Km 7-5, Palma De Mallorca 07122, Baleares, Spain, [Dominguez-Martin, Alicia] Univ Granada, Fac Pharm, Dept Inorgan Chem, Granada 18071, Spain, Spanish Agencia Estatal de Investigacion of the Ministerio de Ciencia, Innovacion y Universidades (MICIU), FEDER, UE, MICIU/AEI from SPAIN

المصدر: Crystals, Vol 10, Iss 1088, p 1088 (2020)
Digibug: Repositorio Institucional de la Universidad de Granada
Universidad de Granada (UGR)
Digital.CSIC. Repositorio Institucional del CSIC
instname
Digibug. Repositorio Institucional de la Universidad de Granada
Crystals
Volume 10
Issue 12

مصطلحات موضوعية: Thermogravimetric analysis, Design, Codrug, General Chemical Engineering, Stacking, codrug, 02 engineering and technology, 010402 general chemistry, 01 natural sciences, Cocrystal, Inorganic Chemistry, Cocrystals, Differential scanning calorimetry, Caffeine, lcsh:QD901-999, General Materials Science, Mechanochemicals synthesis, Solubility, cocrystal, caffeine, Active ingredient, Program, Synthon, Chemistry, Co-crystals, mechanochemical synthesis, 021001 nanoscience & nanotechnology, Condensed Matter Physics, Combinatorial chemistry, hydrochlorothiazide, 0104 chemical sciences, Solvent, Hydrochlorothiazide, lcsh:Crystallography, 0210 nano-technology, Mechanochemical synthesis, Dissolution

وصف الملف: application/pdf

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5cf04e08269f5a67815ef77110a6e43e
https://www.mdpi.com/2073-4352/10/12/1088

المؤلفون: LASERRA, SARA, A. Basit, SOZIO, Piera, MARINELLI, LISA, FORNASARI, ERIKA, CACCIATORE, Ivana, CIULLA, MICHELE, TURKEZ, HASAN, F. Geyikoglu, DI STEFANO, Antonio

المساهمون: Laserra, Sara, A., Basit, Sozio, Piera, Marinelli, Lisa, Fornasari, Erika, Cacciatore, Ivana, Ciulla, Michele, Turkez, Hasan, F., Geyikoglu, DI STEFANO, Antonio

مصطلحات موضوعية: Alzheimer's disease, Codrug, Lipoic acid, Memantine, Solid lipid nanoparticles

وصف الملف: STAMPA

Relation: info:eu-repo/semantics/altIdentifier/pmid/25747452; info:eu-repo/semantics/altIdentifier/wos/WOS:000353730400021; volume:485; issue:1-2; firstpage:183; lastpage:191; numberofpages:9; journal:INTERNATIONAL JOURNAL OF PHARMACEUTICS; http://hdl.handle.net/11564/630910; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-84924939569

الاتاحة: http://hdl.handle.net/11564/630910
https://doi.org/10.1016/j.ijpharm.2015.03.001

المؤلفون: Hanju Lee, Soojin Kim, Jin-Wook Yoo, Yunjin Jung, Seongkeun Jeong, Hyun Young Kim, In-Soo Yoon, Wooseong Kim, Sanghyun Ju, Eunok Im, Heeyeong Cho, Gwangbeom Heo

المصدر: Molecular Pharmaceutics. 17:167-179

مصطلحات موضوعية: Male, Agonist, Aminosalicylic acid, Colon, medicine.drug_class, Pharmaceutical Science, 02 engineering and technology, Pharmacology, 030226 pharmacology & pharmacy, Inflammatory bowel disease, Receptors, G-Protein-Coupled, Rats, Sprague-Dawley, Mice, 03 medical and health sciences, chemistry.chemical_compound, Drug Delivery Systems, 0302 clinical medicine, Sulfasalazine, Cell Line, Tumor, Drug Discovery, medicine, Animals, Humans, Colitis, Mesalamine, Codrug, Anti-Inflammatory Agents, Non-Steroidal, NF-kappa B, Nicotinic Acids, Antagonist, Prodrug, Inflammatory Bowel Diseases, 021001 nanoscience & nanotechnology, medicine.disease, digestive system diseases, Interleukin-10, Rats, surgical procedures, operative, chemistry, Molecular Medicine, 0210 nano-technology, Chromatography, Liquid, medicine.drug

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8f418accd69a722351db8afb8e19f630
https://doi.org/10.1021/acs.molpharmaceut.9b00872

المؤلفون: Sebastiano Miscia, Emanuela Ricciotti, Ivana Cacciatore, Sara Franceschelli, Daniela Maria Pia Gatta, Antonio Di Stefano, Paola Lanuti, Mirko Pesce, Mario Felaco, Antonia Patruno, Lorenza Speranza, Alessio Ferrone, Alfredo Grilli

مصطلحات موضوعية: chemistry.chemical_classification, Reactive oxygen species, Codrug, Neurotoxicity, Substantia nigra, Glutathione, Pharmacology, medicine.disease, medicine.disease_cause, Neuroprotection, chemistry.chemical_compound, chemistry, medicine, Protein kinase B, Oxidative stress

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::9ecb2671349805a5bba90f3e9252ab6a
https://doi.org/10.9734/bpi/cacb/v9/10081d

المؤلفون: In-Soo Yoon, Jin-Wook Yoo, Sohee Park, Sanghyun Ju, Soojin Kim, Do Sik Min, Yunjin Jung, Hanju Lee

المصدر: Molecular pharmaceutics. 18(4)

مصطلحات موضوعية: Agonist, Male, Indoles, medicine.drug_class, Colon, Metabolite, Drug Compounding, Anti-Inflammatory Agents, Pharmaceutical Science, Administration, Oral, 02 engineering and technology, Pharmacology, 030226 pharmacology & pharmacy, Receptors, G-Protein-Coupled, 03 medical and health sciences, chemistry.chemical_compound, Cecum, Mice, 0302 clinical medicine, In vivo, Sulfasalazine, Drug Discovery, medicine, Animals, Humans, Prodrugs, Colitis, Intestinal Mucosa, skin and connective tissue diseases, Codrug, Nicotinic Acids, Prodrug, bacterial infections and mycoses, 021001 nanoscience & nanotechnology, medicine.disease, respiratory tract diseases, Rats, Disease Models, Animal, medicine.anatomical_structure, RAW 264.7 Cells, chemistry, Molecular Medicine, Dinitrofluorobenzene, Propionates, 0210 nano-technology, medicine.drug

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0007c9f412bfd01f6eef870fd3df8b90
https://pubmed.ncbi.nlm.nih.gov/33661643

المؤلفون: Maria Laura Bolognesi, Marina Naldi, Sabrina Petralla, Claudia Albertini, Barbara Monti, Manuela Bartolini, Daniela Grifoni, Silvia Strocchi

المساهمون: Albertini C., Naldi M., Petralla S., Strocchi S., Grifoni D., Monti B., Bartolini M., Bolognesi M.L.

المصدر: Molecules
Volume 26
Issue 4
Molecules, Vol 26, Iss 1112, p 1112 (2021)

مصطلحات موضوعية: Amyloid beta-Peptide, Polypharmacology, Pharmaceutical Science, Ibuprofen, Pharmacology, Analytical Chemistry, chemistry.chemical_compound, Anti-amyloid, Mice, 0302 clinical medicine, Drug Discovery, Ethanolamide, Drug combination, media_common, Neurons, 0303 health sciences, Microglia, Behavior, Animal, Endocytosi, Endocytosis, Neuroprotective Agents, medicine.anatomical_structure, Chemistry (miscellaneous), Molecular Medicine, Drosophila, Alzheimer’s disease, Drug, anti-amyloid, anti-inflammatory, codrugs, drug combinations, polypharmacology, Codrug, Amyloid, Cell Survival, media_common.quotation_subject, Neurotoxins, Neuroprotective Agent, Neuroprotection, Article, lcsh:QD241-441, Immunomodulation, Protein Aggregates, 03 medical and health sciences, lcsh:Organic chemistry, In vivo, Alzheimer Disease, Cromolyn Sodium, medicine, Animals, Physical and Theoretical Chemistry, Rats, Wistar, 030304 developmental biology, Amyloid beta-Peptides, business.industry, Animal, Organic Chemistry, Neurotoxicity, Neuron, medicine.disease, In vitro, chemistry, Drug Design, Protein Aggregate, Anti-inflammatory, business, Neurotoxin, 030217 neurology & neurosurgery

وصف الملف: ELETTRONICO; application/pdf

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6fa954cf3574dca02f20761e8fbd9d4b
http://hdl.handle.net/11585/843407

المؤلفون: Lucjusz Zaprutko, Dorota Olender, Justyna Żwawiak, Anna Pawełczyk

المصدر: Mini reviews in medicinal chemistry. 21(12)

مصطلحات موضوعية: Pharmacology, chemistry.chemical_classification, Drug, Codrug, media_common.quotation_subject, General Medicine, Combinatorial chemistry, Terpene, chemistry.chemical_compound, chemistry, Triterpene, Betulinic acid, Drug Discovery, Moiety, Animals, Humans, Prodrugs, Pentacyclic Triterpenes, Oleanolic acid, media_common

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0024a9fcb33cf9fa6a8c64c1b679f8b7
https://pubmed.ncbi.nlm.nih.gov/33402080

المؤلفون: Osayd Zohud, Raghad Adas, Naim Kittana, Doaa Abu Saleh, Asala Arar, Sahar Alhaj Qasem, Mohyeddin Assali

المصدر: RSC Advances. 9:1055-1061

مصطلحات موضوعية: biology, Codrug, Combination therapy, Chemistry, General Chemical Engineering, 02 engineering and technology, General Chemistry, Pharmacology, 010402 general chemistry, 021001 nanoscience & nanotechnology, biology.organism_classification, 01 natural sciences, Micelle, 0104 chemical sciences, HeLa, Critical micelle concentration, Cancer cell, medicine, 0210 nano-technology, Cytotoxicity, Camptothecin, medicine.drug

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2de46a92971d61458742f567a2fe49a8
https://doi.org/10.1039/c8ra08794f

المؤلفون: Amjad Qandil

المصدر: International Journal of Molecular Sciences; Volume 13; Issue 12; Pages: 17244-17274

مصطلحات موضوعية: anti-inflammatory, cyclooxygenase, codrug, mutual prodrug, NO-NSAIDs, NSAIDs, Phospho-NSAIDs, prodrug

جغرافية الموضوع: agris

وصف الملف: application/pdf

Relation: Biochemistry; https://dx.doi.org/10.3390/ijms131217244

الاتاحة: https://doi.org/10.3390/ijms131217244