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1
المؤلفون: Mary Jane Cullen, Qian Xiang, Jeffrey A. Robl, Philip M. Sher, Brian J. Murphy, Keith J. Miller, Timothy M. Harper, Andrew Alt, Emily Luk, Sarah E. Malmstrom, Dean A. Wacker, Ginger Wu, Kimberly A. Foster, John M. Fevig, Joseph Carpenter, Robert L. Bertekap, Mary F. Grubb, Ying Wang, Karen A. Rossi, Gang Wu, Christian L. Morales, Jianxin Feng, Xiang Yang Ye, Anthony V. Azzara, Matthias Broekema
المصدر: Journal of Medicinal Chemistry. 60:6166-6190
مصطلحات موضوعية: 0301 basic medicine, Agonist, biology, medicine.drug_class, Chemistry, Mutant, HEK 293 cells, Active site, ATP-binding cassette transporter, Pharmacology, 5-HT2C receptor, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, Biochemistry, Drug Discovery, biology.protein, medicine, Molecular Medicine, Structure–activity relationship, Receptor, 030217 neurology & neurosurgery
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2
المؤلفون: Joseph, Carpenter, Ying, Wang, Gang, Wu, Jianxin, Feng, Xiang-Yang, Ye, Christian L, Morales, Matthias, Broekema, Karen A, Rossi, Keith J, Miller, Brian J, Murphy, Ginger, Wu, Sarah E, Malmstrom, Anthony V, Azzara, Philip M, Sher, John M, Fevig, Andrew, Alt, Robert L, Bertekap, Mary Jane, Cullen, Timothy M, Harper, Kimberly, Foster, Emily, Luk, Qian, Xiang, Mary F, Grubb, Jeffrey A, Robl, Dean A, Wacker
المصدر: Journal of medicinal chemistry. 60(14)
مصطلحات موضوعية: Male, Mice, Knockout, Cell Membrane Permeability, Brain, Membranes, Artificial, Feeding Behavior, Arginine, Flavones, Rats, Sprague-Dawley, Structure-Activity Relationship, HEK293 Cells, Mutation, Receptor, Serotonin, 5-HT2B, Microsomes, Liver, Receptor, Serotonin, 5-HT2C, ATP Binding Cassette Transporter, Subfamily G, Member 2, Animals, Humans, Receptor, Serotonin, 5-HT2A, ATP Binding Cassette Transporter, Subfamily B, Member 1, Caco-2 Cells, Serotonin 5-HT2 Receptor Agonists
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3
المصدر: Tetrahedron. 63:8774-8780
مصطلحات موضوعية: Aluminate, Organic Chemistry, chemistry.chemical_element, Biochemistry, Medicinal chemistry, chemistry.chemical_compound, Stereospecificity, chemistry, Alkynylation, Phenylacetylene, Reagent, Yield (chemistry), Drug Discovery, Carbon, Geraniol
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4
المؤلفون: Atsu Apedo, Xiang-Yang Ye, Christian L. Morales, John Krupinski, Mojgan Abousleiman, Dean A. Wacker, Karen A. Rossi, Keith J. Miller, Sarah E. Malmstrom, Ying Wang, Jeffrey A. Robl, Larisa Sereda
المصدر: Bioorganicmedicinal chemistry letters. 24(11)
مصطلحات موضوعية: Agonist, Models, Molecular, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Substituent, Pharmaceutical Science, Biochemistry, Cell Line, Receptors, G-Protein-Coupled, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, medicine, Structure–activity relationship, Humans, Molecular Biology, Benzofurans, Dose-Response Relationship, Drug, Molecular Structure, Organic Chemistry, Metabolic stability, Piperazine, GPR119, chemistry, Ion channel activity, Molecular Medicine, Piperidine
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المؤلفون: Christian L. Morales, Brian L. Pagenkopf
المصدر: ChemInform. 39
مصطلحات موضوعية: Indole test, chemistry.chemical_compound, Nitrile, Chemistry, Yield (chemistry), Total synthesis, Goniomitine, General Medicine, Donor acceptor, Combinatorial chemistry, Cycloaddition, Cyclopropane
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6
المؤلفون: Christian L. Morales, Brian L. Pagenkopf
المصدر: Chemistry Publications
مصطلحات موضوعية: Indole test, Cyclopropanes, Nitrile, Lactams, Molecular Structure, Organic Chemistry, Total synthesis, Stereoisomerism, Biochemistry, Combinatorial chemistry, Cycloaddition, Cyclopropane, Indole Alkaloids, Chemistry, chemistry.chemical_compound, chemistry, Cyclization, Yield (chemistry), Nitriles, Molecule, Organic chemistry, Physical and Theoretical Chemistry, Microwaves
وصف الملف: application/pdf
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المصدر: ChemInform. 38
مصطلحات موضوعية: Aluminate, chemistry.chemical_element, General Medicine, Medicinal chemistry, chemistry.chemical_compound, Stereospecificity, chemistry, Alkynylation, Phenylacetylene, Reagent, Yield (chemistry), Organic chemistry, Carbon, Geraniol
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8
المؤلفون: H Jang, Brian L. Pagenkopf, Xin Wang, Jian Wang, Nicholas A. Morra, Christian L. Morales, Barbora Bajtos, Ming Yu
المصدر: ChemInform. 38
مصطلحات موضوعية: chemistry.chemical_compound, Annulation, chemistry, Autoxidation, Pyridine, Organic chemistry, General Chemistry, General Medicine, Electron, Donor acceptor, Medicinal chemistry, Cycloaddition
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9Academic JournalTotal Synthesis of (±)-Goniomitine via a Formal Nitrile/Donor−Acceptor Cyclopropane 3 2 Cyclization.
المؤلفون: Christian L. Morales1, Brian L. Pagenkopf1
المصدر: Organic Letters. Jan2008, Vol. 10 Issue 2, p157-159. 3p.
مصطلحات موضوعية: *CYCLOALKANES, *CYCLOPROPANE, *REACTION time, *RING formation (Chemistry)