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1
المؤلفون: David O. Calligaro, Paul L. Ornstein, Renhua Li, Phillips K, David L. McKinzie, Allen D, Jun-Xu Li, James A. Monn, Bryan G. Johnson, Stephon C. Smith, Jeffrey M. Witkin, Charles H. Mitch, Beverly A. Heinz, Steven Swanson, Gilmour G, Xushan Wang
المصدر: Pharmacology Biochemistry and Behavior. 155:43-55
مصطلحات موضوعية: Male, 0301 basic medicine, Agonist, Substance-Related Disorders, medicine.drug_class, Clinical Biochemistry, AMPA receptor, Motor Activity, Pharmacology, Receptors, Metabotropic Glutamate, Toxicology, Biochemistry, Rats, Sprague-Dawley, 03 medical and health sciences, Behavioral Neuroscience, Cognition, 0302 clinical medicine, Neurochemical, Cyclohexanes, medicine, Animals, Ketamine, Phencyclidine, Biological Psychiatry, Antagonist, Spontaneous alternation, Receptor antagonist, Rats, 030104 developmental biology, Psychology, Excitatory Amino Acid Antagonists, 030217 neurology & neurosurgery, medicine.drug
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2
المؤلفون: Chuanxi Xiang, Steven Swanson, Joan H. Carter, Paul L. Ornstein, Lisa M. Broad, Charles H. Mitch, Xu Shan Wang, Wesley H. Anderson, Helen E. Sanger, Renhua Li, Jeffrey M. Witkin, Stephon C. Smith, Stephen M. Fitzjohn, Francesca Pasqui, Xia Li, Jodi L. Smith, James A. Monn, Beverly A. Heinz, John T. Catlow
المصدر: Neuropharmacology. 115:100-114
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, medicine.drug_class, Metabotropic glutamate receptor 5, Metabotropic glutamate receptor 7, Metabotropic glutamate receptor 6, Biology, Receptor antagonist, 03 medical and health sciences, Cellular and Molecular Neuroscience, 030104 developmental biology, 0302 clinical medicine, Metabotropic receptor, Metabotropic glutamate receptor, medicine, Metabotropic glutamate receptor 1, Long-term depression, 030217 neurology & neurosurgery
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3
المؤلفون: Wesley H. Anderson, Paul L. Ornstein, Vladamir Tolstikov, Guy Carter, Renhua Li, Brian J. Eastwood, Carl D Overshiner, Alexander Nikolayev, Kurt Rasmussen, Stephen Smith, Gary Gilmour, Stephen Swanson, Linda M. Rorick-Kehn, Xia Li, Keith A. Wafford, John T. Catlow, Jeffrey M. Witkin, Stephen N. Mitchell, Charles H. Mitch, Ming-Shang Kuo, Jennifer Li, James A. Monn
المصدر: Journal of Pharmacology and Experimental Therapeutics. 361:68-86
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, medicine.drug_class, Chemistry, Antagonist, Glutamate receptor, Receptor antagonist, Ventral tegmental area, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, Metabotropic receptor, medicine.anatomical_structure, Dopamine, medicine, Molecular Medicine, Ketamine, Receptor, 030217 neurology & neurosurgery, medicine.drug
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4
المؤلفون: Charles H. Mitch, Aiping Zhang, Mercedes Carpintero, Bradley Condon, C. Groshong, Shane Atwell, John W. Koss, Carl D Overshiner, Jeffrey M. Schkeryantz, Stephon C. Smith, Mark G. Bures, James E. Matt, S.R. Wasserman, Adam M. Fivush, Wesley Seidel, Carlos Jaramillo, K. Conners, David W. Bedwell, Jeffrey M. Witkin, Maria-Jesus Blanco, Daniel Ray Mayhugh, Steven James Quimby, Bruce A. Dressman, Keith A. Wafford, John T. Catlow, Allie Edward Tripp, Paul L. Ornstein, Mario Barberis, José Francisco Soriano, Steven Swanson, Beverly A. Heinz, Jon A. Erickson, Xia Li, Iain MacEwan, Thomas C. Britton, James A. Monn, Susana García-Cerrada, Jing Wang, Mark Donald Chappell, Eric George Tromiczak, Renhua Li, José Eugenio de Diego, Christine Sougias, Tatiana Natali Vetman, Xushan Wang, Stephen Antonysamy
المصدر: Journal of Medicinal Chemistry. 59:10974-10993
مصطلحات موضوعية: 0301 basic medicine, chemistry.chemical_classification, Metabotropic glutamate receptor 5, Hydrochloride, medicine.drug_class, Stereochemistry, Antagonist, Receptor antagonist, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, Dicarboxylic acid, Metabotropic receptor, chemistry, APICA, Drug Discovery, medicine, Molecular Medicine, Structure–activity relationship, 030217 neurology & neurosurgery
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5
المؤلفون: Bruce A. Dressman, Charles H. Mitch, Mercedes Carpintero, Susana García-Cerrada, John T. Catlow, Tatiana Natali Vetman, Wesley Seidel, Mark Donald Chappell, Jeffrey M. Schkeryantz, Albert Khilevich, Xushan Wang, Allie Edward Tripp, Jeffrey M. Witkin, Maria-Jesus Blanco, Renhua Li, Stephon C. Smith, José Francisco Soriano, Mario Barberis, Steven Swanson, Xia Li, Carlos Jaramillo, Beverly A. Heinz, Thomas C. Britton, Carl D Overshiner, Keith A. Wafford, Eric George Tromiczak, José Eugenio de Diego, James E. Matt, David W. Bedwell, Steven James Quimby, Adam M. Fivush, Paul L. Ornstein
المصدر: Bioorganic & Medicinal Chemistry Letters. 26:5663-5668
مصطلحات موضوعية: 0301 basic medicine, Clinical Biochemistry, Glutamic Acid, Pharmaceutical Science, Pharmacology, Receptors, Metabotropic Glutamate, Biochemistry, Cell Line, Madin Darby Canine Kidney Cells, Bridged Bicyclo Compounds, Mice, 03 medical and health sciences, Dogs, 0302 clinical medicine, In vivo, Drug Discovery, Animals, Hexanes, Humans, Receptor, Molecular Biology, Depressive Disorder, Major, Metabotropic glutamate receptor 5, Chemistry, Organic Chemistry, Glutamate receptor, Haplorhini, Glutamic acid, Antidepressive Agents, Rats, 030104 developmental biology, Metabotropic receptor, Molecular Medicine, Metabotropic glutamate receptor 2, 030217 neurology & neurosurgery, Behavioural despair test
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6
المؤلفون: Mark D, Chappell, Renhua, Li, Stephon C, Smith, Bruce A, Dressman, Eric G, Tromiczak, Allie E, Tripp, Maria-Jesus, Blanco, Tatiana, Vetman, Steven J, Quimby, James, Matt, Thomas C, Britton, Adam M, Fivush, Jeffrey M, Schkeryantz, Daniel, Mayhugh, Jon A, Erickson, Mark G, Bures, Carlos, Jaramillo, Mercedes, Carpintero, José Eugenio de, Diego, Mario, Barberis, Susana, Garcia-Cerrada, José F, Soriano, Stephen, Antonysamy, Shane, Atwell, Iain, MacEwan, Bradley, Condon, Christine, Sougias, Jing, Wang, Aiping, Zhang, Kris, Conners, Chris, Groshong, Stephen R, Wasserman, John W, Koss, Jeffrey M, Witkin, Xia, Li, Carl, Overshiner, Keith A, Wafford, Wesley, Seidel, Xu-Shan, Wang, Beverly A, Heinz, Steven, Swanson, John T, Catlow, David W, Bedwell, James A, Monn, Charles H, Mitch, Paul L, Ornstein
المصدر: Journal of medicinal chemistry. 59(24)
مصطلحات موضوعية: Male, Models, Molecular, Behavior, Animal, Dose-Response Relationship, Drug, Molecular Structure, Brain, Mice, Inbred Strains, Motor Activity, Receptors, Metabotropic Glutamate, Antidepressive Agents, Mice, Structure-Activity Relationship, Cyclohexanes, Drug Discovery, Animals, Humans, Swimming
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7
المؤلفون: Alma Jiménez, Marta Garcia De La Torre, Nuria Diaz, Emily Jane Canada, David L. McKinzie, Concepción Pedregal, Charles H. Mitch, Qing Shi, Michael A. Statnick, Steven James Quimby, Steven D. Kahl, Dana Rae Benesh, Vanessa N. Barth, Karen S. Rash
المصدر: Journal of Medicinal Chemistry. 54:8000-8012
مصطلحات موضوعية: Pyrrolidines, medicine.drug_class, CHO Cells, Pharmacology, Radioligand Assay, Structure-Activity Relationship, chemistry.chemical_compound, Cricetulus, Tandem Mass Spectrometry, Opioid receptor, Cricetinae, Opioid Receptor Binding, Drug Discovery, medicine, Animals, Humans, Benzamide, Receptor, Receptors, Opioid, kappa, Chinese hamster ovary cell, Antagonist, Brain, Stereoisomerism, JDTic, Rats, HEK293 Cells, chemistry, Opioid, Benzamides, Molecular Medicine, Chromatography, Liquid, medicine.drug
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8
المؤلفون: Allison E. Sahr, Michael A. Statnick, Charles H. Mitch, Dana Sindelar, Jesline T. Alexander-Chacko, Brian J. Eastwood
المصدر: American Journal of Physiology-Regulatory, Integrative and Comparative Physiology. 295:R463-R471
مصطلحات موضوعية: Male, medicine.medical_specialty, Time Factors, Physiology, medicine.drug_class, Dopamine, Microdialysis, Narcotic Antagonists, Nucleus accumbens, Biology, Nucleus Accumbens, Rats, Sprague-Dawley, Eating, Food Preferences, chemistry.chemical_compound, Piperidines, Cyclohexanes, In vivo, Physiology (medical), Internal medicine, medicine, Animals, Potency, Neurotransmitter, Receptor, Neurons, Behavior, Animal, Appetite Regulation, Antagonist, Rats, Endocrinology, chemistry, Receptors, Opioid, Catecholamine, Reinforcement, Psychology, Opioid antagonist, medicine.drug
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9
المؤلفون: Elizabeth Marie Thomas, Paul J. Emmerson, Todd M. Suter, Michael A. Statnick, Kumiko Takeuchi, Jamie H. McKinzie, Charles H. Mitch, William Glen Holloway, Miles Goodman Siegel, Steven James Quimby, Peggy L. Surface
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:6841-6846
مصطلحات موضوعية: medicine.drug_class, Stereochemistry, Narcotic Antagonists, Clinical Biochemistry, Acrylic Resins, Carboxylic Acids, Pharmaceutical Science, Biochemistry, Chemical synthesis, δ-opioid receptor, Structure-Activity Relationship, chemistry.chemical_compound, Opioid receptor, Drug Discovery, polycyclic compounds, medicine, Structure–activity relationship, Receptor, Molecular Biology, Molecular Structure, Nicotinamide, Chemistry, Organic Chemistry, Antagonist, Amides, In vitro, Receptors, Opioid, Molecular Medicine, Ethers
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10
المؤلفون: Jeffrey M, Witkin, Paul L, Ornstein, Charles H, Mitch, Renhua, Li, Stephon C, Smith, Beverly A, Heinz, Xu-Shan, Wang, Chuanxi, Xiang, Joan H, Carter, Wesley H, Anderson, Xia, Li, Lisa M, Broad, Francesca, Pasqui, Stephen M, Fitzjohn, Helen E, Sanger, Jodi L, Smith, John, Catlow, Steven, Swanson, James A, Monn
المصدر: Neuropharmacology. 115
مصطلحات موضوعية: Cerebral Cortex, Male, Rats, Sprague-Dawley, Dose-Response Relationship, Drug, Cyclohexanes, Animals, Humans, Receptors, Metabotropic Glutamate, Excitatory Amino Acid Antagonists, Cell Line, Rats
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11
المؤلفون: Miles Goodman Siegel, Peggy L. Surface, Nuria Diaz, Jamie H. McKinzie, Ryan Favors, Mark J. Benvenga, Joseph M. Woodland, Michael A. Statnick, Nita J. Patel, Elizabeth Marie Thomas, Paul J. Emmerson, Steven C. Peters, Michael Mangold, Charles H. Mitch, Harlan E. Shannon, Steven James Quimby
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:3844-3848
مصطلحات موضوعية: medicine.drug_class, Stereochemistry, Narcotic Antagonists, Clinical Biochemistry, Drug Evaluation, Preclinical, Administration, Oral, Pain, Pharmaceutical Science, Carboxamide, Ligands, Biochemistry, Chemical synthesis, Radioligand Assay, Structure-Activity Relationship, chemistry.chemical_compound, Phenols, Piperidines, Cyclohexanes, In vivo, Opioid receptor, Drug Discovery, medicine, Animals, Molecular Biology, Chemistry, Organic Chemistry, Biological activity, Feeding Behavior, Rats, Liver, Opioid, Molecular Medicine, Opioid antagonist, medicine.drug
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12
المؤلفون: Michael A. Statnick, Jamie H. McKinzie, Todd M. Suter, Paul J. Emmerson, Peggy L. Surface, Charles H. Mitch
المصدر: European Journal of Pharmacology. 494:121-130
مصطلحات موضوعية: medicine.medical_specialty, medicine.drug_class, Narcotic Antagonists, Diprenorphine, CHO Cells, Pharmacology, Ligands, Binding, Competitive, κ-opioid receptor, Naltrexone, δ-opioid receptor, Eating, Radioligand Assay, Piperidines, Cyclohexanes, Opioid receptor, Cricetinae, Receptors, Opioid, delta, Internal medicine, Appetite Depressants, medicine, Animals, Inverse agonist, Dose-Response Relationship, Drug, Chemistry, Cell Membrane, Sodium, Enkephalin, Ala(2)-MePhe(4)-Gly(5), Rats, Rats, Zucker, Endocrinology, Opioid, Guanosine 5'-O-(3-Thiotriphosphate), Receptors, Opioid, Anorectic, μ-opioid receptor, medicine.drug
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13
المؤلفون: Michael A. Statnick, Brian J. Eastwood, Frank C. Tinsley, Todd M. Suter, Mark L. Heiman, Charles H. Mitch
المصدر: American Journal of Physiology-Regulatory, Integrative and Comparative Physiology. 284:R1399-R1408
مصطلحات موضوعية: Drug, medicine.medical_specialty, Food intake, Physiology, Chemistry, media_common.quotation_subject, Lipid metabolism, medicine.disease, Obesity, Dose–response relationship, Endocrinology, Opioid, Physiology (medical), Internal medicine, medicine, Receptor, Antagonism, media_common, medicine.drug
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14
المؤلفون: Dana Rae Benesh, Lee A. Phebus, Zhaogen Chen, Charles H. Mitch, Anne B. Need, John Mehnert Schaus, Elizabeth M. Joshi, Thomas J. Raub, Vanessa N. Barth, Stuart Morton
المصدر: ACS chemical neuroscience. 5(12)
مصطلحات موضوعية: Physiology, Cognitive Neuroscience, Standardized uptake value, Mass spectrometry, Biochemistry, Mice, In vivo, Tandem Mass Spectrometry, TRACER, medicine, Animals, Humans, Pet tracer, medicine.diagnostic_test, Chemistry, business.industry, Binding potential, Brain, Cell Biology, General Medicine, Small molecule, Rats, Positron emission tomography, Positron-Emission Tomography, Biophysics, Radiopharmaceuticals, Nuclear medicine, business, Biomarkers, Chromatography, Liquid
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15
المؤلفون: Michael Kapinos, Karen S. Rash, Shu-fei Lin, Vanessa N. Barth, Daniel Holden, Antonio Navarro, Ming-Qiang Zheng, Yiyun Huang, Charles H. Mitch, Richard E. Carson, Jim Ropchan, Su Jin Kim, Anne B. Need, Kathleen Maloney
مصطلحات موضوعية: Male, Stereochemistry, medicine.drug_class, Pyridines, (+)-Naloxone, Chemistry Techniques, Synthetic, Pharmacology, Article, Rats, Sprague-Dawley, In vivo, Opioid receptor, Radioligand, medicine, Animals, Radiology, Nuclear Medicine and imaging, Radioactive Tracers, Binding selectivity, Temporal cortex, Radiochemistry, Chemistry, Receptors, Opioid, kappa, Binding potential, Macaca mulatta, Rats, Positron-Emission Tomography, Benzamides, Radiopharmaceuticals, Ex vivo
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16
المؤلفون: Charles H. Mitch, David O. Calligaro, Celia Ann Whitesitt, Frank P. Bymaster, Barry D. Sawyer, John S. Ward, Julie F. Falcone, Harlan E. Shannon
المصدر: General Pharmacology: The Vascular System. 32:445-452
مصطلحات موضوعية: Male, medicine.medical_specialty, Carbachol, Aorta, Thoracic, Muscarinic Antagonists, Muscarinic Agonists, Muscle, Smooth, Vascular, Internal medicine, medicine.artery, Muscarinic acetylcholine receptor, medicine, Animals, Thoracic aorta, Receptor, Receptor, Muscarinic M3, Pharmacology, Aorta, Chemistry, Muscarinic acetylcholine receptor M3, Receptors, Muscarinic, Vasodilation, Endocrinology, Vasoconstriction, Pilocarpine, cardiovascular system, Endothelium, Vascular, Rabbits, medicine.symptom, medicine.drug, Muscle contraction
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17
المؤلفون: Anders Fink-Jensen, John S. Ward, Lone Jeppesen, Harlan E. Shannon, Per Sauerberg, Frank P. Bymaster, Steven C. Peters, Wei Zhang, Petra A. Carter, Karin Rimvall, Malcolm J. Sheardown, Charles H. Mitch, Celia Ann Whitesitt, Neil DeLapp, David O. Calligaro
المصدر: Brain Research. 795:179-190
مصطلحات موضوعية: Male, Dihydropyridines, Quinuclidines, Pyridines, Physostigmine, Cholinergic Agents, Tetrazoles, Hypothermia, Pharmacology, Phosphatidylinositols, Mice, Radioligand Assay, chemistry.chemical_compound, Oximes, Tremor, Muscarinic acetylcholine receptor, Muscarinic acetylcholine receptor M4, Hydrolysis, General Neuroscience, Pilocarpine, Muscarinic acetylcholine receptor M1, Parasympathomimetics, Tacrine, Imines, Salivation, medicine.drug, Agonist, medicine.medical_specialty, medicine.drug_class, Mice, Inbred Strains, Lithium, Muscarinic Agonists, Binding, Competitive, Muscarinic agonist, Internal medicine, Thiadiazoles, Oxotremorine, medicine, Animals, Molecular Biology, Brain Chemistry, Dose-Response Relationship, Drug, Milameline, Bridged Bicyclo Compounds, Heterocyclic, Endocrinology, chemistry, Cholinesterase Inhibitors, Neurology (clinical), Xanomeline, Developmental Biology
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18
المؤلفون: Su Wu, Charles H. Mitch, Christian Thomsen, Shelia Little, Frank P. Bymaster, John S. Ward, Edward M. Johnstone, Celia Ann Whitesitt, David O. Calligaro, Harlan E. Shannon, Anders Fink-Jensen, Malcolm J. Sheardown, Rama M. Belagaje, Lone Jeppesen, Per Sauerberg, Neil DeLapp
المصدر: Biochemical and Biophysical Research Communications. 244:156-160
مصطلحات موضوعية: Agonist, medicine.medical_specialty, Carbachol, Pyridines, medicine.drug_class, Blotting, Western, Biophysics, Peptide, CHO Cells, Muscarinic Agonists, Biology, Transfection, Biochemistry, Muscarinic agonist, Amyloid beta-Protein Precursor, chemistry.chemical_compound, Alzheimer Disease, Cricetinae, Internal medicine, Thiadiazoles, mental disorders, medicine, Animals, Humans, Cloning, Molecular, Beta (finance), Molecular Biology, Sweden, chemistry.chemical_classification, Amyloid beta-Peptides, Chinese hamster ovary cell, Receptor, Muscarinic M1, Cell Biology, Receptors, Muscarinic, Molecular biology, Peptide Fragments, Endocrinology, chemistry, Mutation, Xanomeline, Protein Processing, Post-Translational, medicine.drug
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19
المؤلفون: David Brunsting, Celia Ann Whitesitt, Michael D. B. Swedberg, John S. Ward, David O. Calligaro, Per Sauerberg, Charles H. Mitch, Preben H. Olesen, Lone Jeppesen, Harlan E. Shannon, Malcolm J. Sheardown, Leander Merritt, Franklin Porter Bymaster
المصدر: Journal of Medicinal Chemistry. 41:379-392
مصطلحات موضوعية: Male, Models, Molecular, Agonist, Quinuclidines, Stereochemistry, medicine.drug_class, Static Electricity, Substituent, Muscarinic Agonists, Phosphatidylinositols, Muscarinic agonist, Cell Line, Rats, Sprague-Dawley, Mice, Radioligand Assay, chemistry.chemical_compound, Thiadiazoles, Drug Discovery, Muscarinic acetylcholine receptor, medicine, Animals, Aceclidine, Hydrolysis, Brain, Muscarinic acetylcholine receptor M1, Rats, chemistry, Molecular Medicine, Xanomeline, medicine.drug
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20
المؤلفون: Frank P. Bymaster, Preben H. Olesen, Neil C. Bodick, Lars Farde, Lisa A. Shipley, Celia Ann Whitesitt, Malcolm J. Sheardown, Michael D. B. Swedberg, Neil DeLapp, Per Sauerberg, Judith L. Buelke-Sam, Charles H. Mitch, David O. Calligaro, John S. Ward, Kristian Tage Hansen, Harlan E. Shannon, Peter D. Suzdak
المصدر: Drug Development Research. 40:158-170
مصطلحات موضوعية: Agonist, medicine.medical_specialty, business.industry, medicine.drug_class, Muscarinic antagonist, Muscarinic acetylcholine receptor M3, Muscarinic acetylcholine receptor M2, Muscarinic acetylcholine receptor M1, Muscarinic agonist, chemistry.chemical_compound, Endocrinology, chemistry, Internal medicine, Drug Discovery, Muscarinic acetylcholine receptor, medicine, business, Xanomeline, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::ff3821f6b98caef6e2110b1e363be351
https://doi.org/10.1002/(sici)1098-2299(199702)40:2<158::aid-ddr6>3.0.co;2-k