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1Academic Journal
المؤلفون: Diana Donnelly-Roberts, Steve Mcgaraughty, Char-Chang Shieh, Prisca Honore, Michael F Jarvis
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.1082.2233; http://jpet.aspetjournals.org/content/jpet/324/2/409.full.pdf
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المؤلفون: Brett Antonio, Robert J. Gregg, Gricelda H. Simler, Matthew S Johnson, Yi Liu, Dong Liu, Marc J. C. Scanio, Prisca Honore, Alison Knox, James B. Thomas, Shailen K. Joshi, Mark L. Chapman, Brian E. Marron, Irene Drizin, Douglas S. Krafte, Connie R. Faltynek, Robert N. Atkinson, Xu-Feng Zhang, Michael J. Krambis, Kort Michael E, Michael F. Jarvis, Stephen Werness, Kennan C. Marsh, Lei Shi, Char-Chang Shieh
المصدر: Bioorganic & Medicinal Chemistry. 18:7816-7825
مصطلحات موضوعية: Clinical Biochemistry, Analgesic, Drug Evaluation, Preclinical, Administration, Oral, Pharmaceutical Science, Pharmacology, Biochemistry, Sodium Channels, NAV1.8 Voltage-Gated Sodium Channel, Structure-Activity Relationship, Sodium channel blocker, Oral administration, In vivo, Ganglia, Spinal, Microsomes, Drug Discovery, Animals, Humans, Molecular Biology, Neurons, Chemistry, Sodium channel, Organic Chemistry, Rats, Blockade, Disease Models, Animal, Nociception, Pyrazines, Neuropathic pain, Neuralgia, Molecular Medicine, Sodium Channel Blockers
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المؤلفون: Rosemarie Roeloffs, Stephen Werness, Brian E. Marron, Chengmin Zhong, Brett Antonio, Ahmed H. Hakeem, Irene Drizin, Char-Chang Shieh, Mark L. Chapman, Joseph P. Mikusa, Marc J. C. Scanio, James B. Thomas, Shailen K. Joshi, Dong Liu, Mark A. Matulenko, Douglas S. Krafte, Robert N. Atkinson, Lei Shi, Kennan C. Marsh, Gricelda H. Simler, Matthew S Johnson, Michael J. Krambis, Kort Michael E, Michael F. Jarvis, Xu-Feng Zhang, Robert J. Gregg, Connie R. Faltynek, Matthew A. Secrest, Prisca Honore
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:6812-6815
مصطلحات موضوعية: Niacinamide, Stereochemistry, Clinical Biochemistry, Administration, Oral, Biological Availability, Pharmaceutical Science, Pharmacology, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Sodium channel blocker, Furan, Drug Discovery, Animals, Structure–activity relationship, Molecular Biology, Nicotinamide, Sodium channel, Organic Chemistry, Rats, Bioavailability, chemistry, Neuropathic pain, Molecular Medicine, Linker, Sodium Channel Blockers
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المؤلفون: Brian E. Marron, Kort Michael E, Michael F. Jarvis, Prisca Honore, Mark L. Chapman, Char-Chang Shieh, Ahmed H. Hakeem, Mark A. Matulenko, Xu-Feng Zhang, Connie R. Faltynek, Shailen K. Joshi, Douglas S. Krafte, Robert N. Atkinson
المصدر: Neuropharmacology. 59:201-207
مصطلحات موضوعية: Male, Niacinamide, Pain Threshold, Patch-Clamp Techniques, Sensory Receptor Cells, Morpholines, Biophysics, Tetrodotoxin, Pharmacology, Transfection, Sodium Channels, Membrane Potentials, NAV1.8 Voltage-Gated Sodium Channel, Rats, Sprague-Dawley, Cellular and Molecular Neuroscience, chemistry.chemical_compound, Sodium channel blocker, Dorsal root ganglion, Ganglia, Spinal, medicine, Animals, Humans, Channel blocker, Patch clamp, Cells, Cultured, Spinal Cord Injuries, Membrane potential, Dose-Response Relationship, Drug, Chemistry, Sodium channel, Electric Stimulation, Rats, Disease Models, Animal, Allodynia, medicine.anatomical_structure, nervous system, Hyperalgesia, Neuralgia, medicine.symptom, Sodium Channel Blockers
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المؤلفون: Matthew S Johnson, Dong Liu, Robert J. Gregg, Irene Drizin, Michael F. Gross, Gricelda Hernandez, Kennan C. Marsh, James B. Thomas, Mark L. Chapman, Chang Z. Zhu, Brian E. Marron, Connie R. Faltynek, Shailen K. Joshi, Prisca Honore, Stephen Werness, Michael E. Kort, Douglas S. Krafte, Robert N. Atkinson, Rosemarie Roeloffs, William A. Carroll, Marc J. C. Scanio, Xu-Feng Zhang, Donna M. Gauvin, Michael J. Krambis, Michael F. Jarvis, Char-Chang Shieh, Lei Shi, Joseph P. Mikusa
المصدر: Bioorganic & Medicinal Chemistry. 16:6379-6386
مصطلحات موضوعية: Male, Clinical Biochemistry, Analgesic, Pharmaceutical Science, Lamotrigine, Pharmacology, Biochemistry, Piperazines, Sodium Channels, Rats, Sprague-Dawley, Mice, Structure-Activity Relationship, Sodium channel blocker, Mexiletine, Drug Discovery, medicine, Animals, Humans, Potency, Furans, Molecular Biology, Voltage-gated ion channel, Chemistry, Sodium channel, Organic Chemistry, Analgesics, Non-Narcotic, Ether-A-Go-Go Potassium Channels, Rats, Neuropathic pain, Neuralgia, Molecular Medicine, Sodium Channel Blockers, medicine.drug
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المؤلفون: William A Carroll, Chengmin Zhong, Stephen Werness, Jinrong Liu, Matthew S Johnson, Lei Shi, Michael F Jarvis, James B. Thomas, Xu-Feng Zhang, Mark L. Chapman, Michael F. Gross, Shailen Joshi, Michael E. Kort, Marc J. C. Scanio, Dong Liu, Robert J Gregg, Rosemarie Roeloffs, Prisca Honore, Gricelda Hernandez, Gregory J Pacofsky, Douglas S. Krafte, Robert N. Atkinson, Brian E. Marron, Irene I. Drizin, Kennan C Marsh, Joseph P Mikusa, Michael J. Krambis, Bernard P Murray, Char-Chang Shieh, Connie R. Faltynek
المصدر: Journal of Medicinal Chemistry. 51:407-416
مصطلحات موضوعية: Male, Patch-Clamp Techniques, Stereochemistry, Analgesic, hERG, Pain, Nerve Tissue Proteins, Inflammation, In Vitro Techniques, Pharmacology, Sodium Channels, Cell Line, NAV1.8 Voltage-Gated Sodium Channel, Rats, Sprague-Dawley, Mice, Structure-Activity Relationship, Cricetulus, Sodium channel blocker, Cricetinae, Ganglia, Spinal, Drug Discovery, medicine, Animals, Humans, Furans, Neurons, Analgesics, biology, Chemistry, Sodium channel, Anti-Inflammatory Agents, Non-Steroidal, Chronic pain, Peripheral Nervous System Diseases, medicine.disease, Amides, Recombinant Proteins, Rats, Neuropathic pain, Systemic administration, biology.protein, Molecular Medicine, medicine.symptom, Sodium Channel Blockers
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المؤلفون: Diana L. Donnelly-Roberts, Steve McGaraughty, Prisca Honore, Michael F. Jarvis, Char-Chang Shieh
المصدر: Journal of Pharmacology and Experimental Therapeutics. 324:409-415
مصطلحات موضوعية: endocrine system, P2Y receptor, Purinergic Antagonists, Pain, Uridine Triphosphate, Pharmacology, P2 receptor, Purinergic Agonists, Adenosine Triphosphate, medicine, Animals, Humans, Receptor, Pain Measurement, urogenital system, Chemistry, musculoskeletal, neural, and ocular physiology, Purinergic receptor, Receptors, Purinergic, Purinergic signalling, Allodynia, Molecular Medicine, medicine.symptom, Neuroscience
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المؤلفون: Ivan Milicic, Steven A. Buckner, A Parihar, Murali Gopalakrishnan, X.-F Zhang, Sean C. Turner, J Wilkins, Char-Chang Shieh, Jinkerson T
المصدر: British Journal of Pharmacology. 151:798-806
مصطلحات موضوعية: Pharmacology, medicine.medical_specialty, Chemistry, Smooth muscle contraction, Iberiotoxin, Sensory neuron, Potassium channel, Contractility, Electrophysiology, medicine.anatomical_structure, Endocrinology, Internal medicine, medicine, Biophysics, Premovement neuronal activity, medicine.symptom, Muscle contraction
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المؤلفون: Char-Chang Shieh, William A. Carroll, Michael E. Brune, Matsushita K, Yoshihisa Kurachi, Kristi L. Whiteaker, Adebola Fabiyi, Jorge D. Brioni, Anthony V. Daza, Murali Gopalakrishnan, Eduardo J. Molinari, Steven A. Buckner, Mitsuhiko Yamada, Milicic Ia
المصدر: British Journal of Pharmacology. 151:467-475
مصطلحات موضوعية: Pharmacology, Urinary bladder, medicine.diagnostic_test, business.industry, Pig bladder, Cystometry, medicine.disease, Potassium channel, chemistry.chemical_compound, Muscle relaxation, medicine.anatomical_structure, Overactive bladder, chemistry, Anesthesia, Pinacidil, Medicine, Potassium channel opener, business
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المؤلفون: Joseph P. Mikusa, Prisca Honore, Gricelda Hernandez, Karen Kage, Wende Niforatos, Char-Chang Shieh, Torben R. Neelands, Michael F. Jarvis, S.K. Joshi, Xu-Feng Zhang, Ping Han, Connie R. Faltynek, James P. Sullivan, Scott J. Baker, Douglas S. Krafte
المصدر: Pain. 123:75-82
مصطلحات موضوعية: Male, Patch-Clamp Techniques, Freund's Adjuvant, Drug Evaluation, Preclinical, Nerve Tissue Proteins, Tetrodotoxin, Sodium Channels, Oligodeoxyribonucleotides, Antisense, NAV1.8 Voltage-Gated Sodium Channel, Rats, Sprague-Dawley, Pressure, medicine, Animals, Neurons, Afferent, Ligation, Injections, Spinal, Inflammation, Pain, Postoperative, Ion Transport, Behavior, Animal, business.industry, Sodium, Nerve injury, medicine.disease, Sciatic Nerve, Rats, Spinal Nerves, Anesthesiology and Pain Medicine, Peripheral neuropathy, Allodynia, Nociception, Neurology, Hyperalgesia, Vincristine, Anesthesia, Spinal nerve, Neuropathic pain, Neuralgia, Stress, Mechanical, Neurology (clinical), Sciatic nerve, medicine.symptom, business
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المؤلفون: Sean C. Turner, Char-Chang Shieh
المصدر: Voltage-Gated Ion Channels as Drug Targets, Volume 29
مصطلحات موضوعية: Chemistry, Ca2 activated k channel, Medicinal chemistry, Potassium channel
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المؤلفون: Jun Chen, Char-Chang Shieh, Murali Gopalakrishnan
المصدر: Voltage-Gated Ion Channels as Drug Targets
مصطلحات موضوعية: Stereochemistry, Computational chemistry, Chemistry, Crystal structure, Potassium channel
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المؤلفون: Kennan C. Marsh, Lee C. Preusser, Linda L. King, Bryan F. Cox, Ryan M. Fryer, Pamela A. Rakestraw, Murali Gopalakrishnan, Steven A. Buckner, William A. Carroll, Glenn A. Reinhart, Char-Chang Shieh, Michael E. Brune
المصدر: Journal of Cardiovascular Pharmacology. 46:232-240
مصطلحات موضوعية: Male, Dihydropyridines, Mean arterial pressure, medicine.medical_specialty, Patch-Clamp Techniques, Potassium Channels, Vascular smooth muscle, Muscle Relaxation, Guinea Pigs, Urinary Bladder, Aorta, Thoracic, Blood Pressure, In Vitro Techniques, Pharmacology, Ligands, Rats, Sprague-Dawley, Radioligand Assay, Adenosine Triphosphate, Dogs, Heart Rate, In vivo, Internal medicine, medicine, Animals, Anesthesia, Patch clamp, Dose-Response Relationship, Drug, Portal Vein, Chemistry, Hemodynamics, Dihydropyridine, Muscle, Smooth, Potassium channel, Rats, Muscle relaxation, Endocrinology, Pyrones, Potassium channel opener, Cardiology and Cardiovascular Medicine, Ion Channel Gating, medicine.drug
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المؤلفون: David G. McKenna, Connie R. Faltynek, Char-Chang Shieh, Xu-Feng Zhang, Jay F. Sarthy, Jonathan D. Trumbull, Murali Gopalakrishnan, Ashutosh S. Parihar
المصدر: ASSAY and Drug Development Technologies. 1:655-663
مصطلحات موضوعية: Patch-Clamp Techniques, Computer science, Test station, Cell Culture Techniques, Drug Evaluation, Preclinical, Control software, Ligands, Sensitivity and Specificity, Ion Channels, Membrane Potentials, User-Computer Interface, Xenopus laevis, Drug Discovery, medicine, Animals, Cells, Cultured, Ion channel, Reproducibility of Results, Equipment Design, Robotics, Oocyte, Cell biology, Electrophysiology, Equipment Failure Analysis, medicine.anatomical_structure, Oocytes, Feasibility Studies, Molecular Medicine, Ligand-gated ion channel, Ion Channel Gating, Microelectrodes, Algorithms
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المؤلفون: Ivan Milicic, Char-Chang Shieh, Gary A. Gintant, Rachel Davis-Taber, Murali Gopalakrishnan, John Malysz, Eduardo J. Molinari, Jeffrey S. McDermott, Robert J. Altenbach, Victoria E. Scott, Michael J. Coghlan, Kristi L. Whiteaker, William A. Carroll, Steven A. Buckner, Gary A. Rotert
المصدر: Molecular Pharmacology. 64:143-153
مصطلحات موضوعية: Male, Dihydropyridines, Potassium Channels, Pyridines, Purkinje fibers, Guinea Pigs, Urinary Bladder, Thiophenes, Pharmacology, Iodine Radioisotopes, Guinea pig, Radioligand Assay, chemistry.chemical_compound, Adenosine Triphosphate, medicine, Diazoxide, Animals, Channel blocker, Binding site, Binding Sites, Myocardium, Dihydropyridine, Membrane Proteins, Heart, Potassium channel, Kinetics, medicine.anatomical_structure, chemistry, Pinacidil, Molecular Medicine, Radiopharmaceuticals, medicine.drug
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المصدر: European Journal of Pharmacology. 471:157-164
مصطلحات موضوعية: Male, Charybdotoxin, Pharmacology, Apamin, Potassium Channels, Calcium-Activated, chemistry.chemical_compound, Cell Line, Tumor, Scyllatoxin, LNCaP, Humans, Medicine, Riluzole, Dose-Response Relationship, Drug, business.industry, Prostatic Neoplasms, Iberiotoxin, Calcium Channel Blockers, Calcium Channel Agonists, chemistry, Cancer cell, Benzimidazoles, Efflux, business, Cell Division, medicine.drug
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المؤلفون: Xu-Feng Zhang, Char-Chang Shieh, James P. Sullivan, Ivan Milicic, Steven A. Buckner, Tammie K. White, William A. Carroll, Ashutosh S. Parihar, Michael J. Coghlan, Murali Gopalakrishnan, Sean C. Turner
المصدر: Bioorganic & Medicinal Chemistry Letters. 13:2003-2007
مصطلحات موضوعية: Indoles, Swine, Stereochemistry, Muscle Relaxation, Urinary Bladder, Clinical Biochemistry, Pharmaceutical Science, chemistry.chemical_element, In Vitro Techniques, Calcium, Transfection, Biochemistry, Chemical synthesis, Cell Line, Potassium Channels, Calcium-Activated, Structure-Activity Relationship, Drug Discovery, medicine, Animals, Humans, Amines, Molecular Biology, Aza Compounds, Smooth muscle tissue, Organic Chemistry, HEK 293 cells, Urinary Bladder Diseases, Muscle, Smooth, Urination Disorders, In vitro, medicine.anatomical_structure, chemistry, Biophysics, Molecular Medicine, Efflux, medicine.symptom, Muscle contraction
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المؤلفون: Jonathan D. Trumbull, Eugene S. Maslana, David G. Mckenna, Thomas A. Nemcek, Wende Niforatos, Jeffrey Y. Pan, Ashutosh S. Parihar, Char-Chang Shieh, Julie A. Wilkins, Clark A. Briggs, Daniel Bertrand
المصدر: Receptors and Channels. 9:19-28
مصطلحات موضوعية: Pharmacology, Endocrinology, Clinical Biochemistry, Cell Biology
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المؤلفون: Victoria E. Scott, Char-Chang Shieh, Murali Gopalakrishnan, Sujatha M. Gopalakrishnan, Usha Warrior, Michael J. Coghlan, David J. Burns, Kristi L. Whiteaker, Duncan R. Groebe
المصدر: SLAS Discovery. 6:305-312
مصطلحات موضوعية: Male, 0301 basic medicine, Patch-Clamp Techniques, Potassium Channels, High-throughput screening, Guinea Pigs, Analytical chemistry, 01 natural sciences, Biochemistry, Membrane Potentials, Analytical Chemistry, 03 medical and health sciences, Animals, Patch clamp, Coloring Agents, Cells, Cultured, Rapid response, Membrane potential, Quenching (fluorescence), Chemistry, Muscle, Smooth, Fluorescence, Potassium channel, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 030104 developmental biology, Time course, Biophysics, Molecular Medicine, Biotechnology
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المؤلفون: Victoria E. Scott, Eduardo J. Molinari, Lisa M. Monteggia, Jorge D. Brioni, Jean M. Roch, Kristi L. Whiteaker, Char Chang Shieh, James P. Sullivan, Murali Gopalakrishnan
المصدر: British Journal of Pharmacology. 129:1323-1332
مصطلحات موضوعية: Pharmacology, Membrane potential, endocrine system, ATP-sensitive potassium channel, Chemistry, Inward-rectifier potassium ion channel, Kir6.2, Potassium channel, Biochemistry, Biophysics, Diazoxide, medicine, Sulfonylurea receptor, Patch clamp, medicine.drug