نتائج البحث - "Camper, Demarco V."

1

Academic Journal

High-throughput screening identifies small molecules that bind to the RAS:SOS:RAS complex and perturb RAS signaling

المؤلفون: Burns, Michael C., Howes, Jennifer E., Sun, Qi, Little, Andrew J., Camper, DeMarco V., Abbott, Jason R., Phan, Jason, Lee, Taekyu, Waterson, Alex G., Rossanese, Olivia W., Fesik, Stephen W.

المساهمون: Ann Melly Scholarship in Oncology, Public Health Service, National Institute of General Medical Studies, Vanderbilt Medical-Scientist Training Program, National Cancer Institute Specialized Program of Research Excellence award, Research Investigator Award from the Lustgarten Foundation, US Department of Energy Office of Science by the Argonne National Laboratory, US Department of Energy, Michigan Economic Development Corporation, Michigan Technology Tri- Corridor, Vanderbilt Institute of Chemical Biology, Vanderbilt Ingram Center

المصدر: Analytical Biochemistry ; volume 548, page 44-52 ; ISSN 0003-2697

الاتاحة: http://dx.doi.org/10.1016/j.ab.2018.01.025
https://api.elsevier.com/content/article/PII:S0003269718300587?httpAccept=text/xml
https://api.elsevier.com/content/article/PII:S0003269718300587?httpAccept=text/plain

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2

Academic Journal

Discovery and biological characterization of potent myeloid cell leukemia‐1 inhibitors

المساهمون: National Institutes of Health, National Cancer Institute, Vanderbilt University, U.S. Department of Energy

المصدر: FEBS Letters ; volume 591, issue 1, page 240-251 ; ISSN 0014-5793 1873-3468

الاتاحة: http://dx.doi.org/10.1002/1873-3468.12497
https://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1002%2F1873-3468.12497
https://onlinelibrary.wiley.com/doi/pdf/10.1002/1873-3468.12497
https://onlinelibrary.wiley.com/doi/full-xml/10.1002/1873-3468.12497
https://febs.onlinelibrary.wiley.com/doi/am-pdf/10.1002/1873-3468.12497
https://febs.onlinelibrary.wiley.com/doi/pdf/10.1002/1873-3468.12497

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3

Discovery of 2-Indole-acylsulfonamide Myeloid Cell Leukemia 1 (Mcl-1) Inhibitors Using Fragment-Based Methods

المؤلفون: Pelz, Nicholas F., Bian, Zhiguo, Zhao, Bin, Shaw, Subrata, Tarr, James C., Belmar, Johannes, Gregg, Claire, Camper, DeMarco V., Goodwin, Craig M., Arnold, Allison L., Sensintaffar, John L., Friberg, Anders, Rossanese, Olivia W., Lee, Taekyu, Olejniczak, Edward T., Fesik, Stephen W.

مصطلحات موضوعية: 60 APPLIED LIFE SCIENCES

وصف الملف: application/pdf

Relation: http://www.osti.gov/servlets/purl/1247370; https://www.osti.gov/biblio/1247370; https://doi.org/10.1021/acs.jmedchem.5b01660

الاتاحة: http://www.osti.gov/servlets/purl/1247370
https://www.osti.gov/biblio/1247370
https://doi.org/10.1021/acs.jmedchem.5b01660

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4

Academic Journal

Optimization of Potent and Selective Tricyclic Indole Diazepinone Myeloid Cell Leukemia-1 Inhibitors Using Structure-Based Design

المؤلفون: Shaw, Subrata, Bian, Zhiguo, Zhao, Bin, Tarr, James C., Veerasamy, Nagarathanam, Jeon, Kyu Ok, Belmar, Johannes, Arnold, Allison L., Fogarty, Stuart A., Perry, Evan, Sensintaffar, John L., Camper, DeMarco V., Rossanese, Olivia W., Lee, Taekyu, Olejniczak, Edward T., Fesik, Stephen W.

المساهمون: National Cancer Institute, NIH Office of the Director

المصدر: Journal of Medicinal Chemistry ; volume 61, issue 6, page 2410-2421 ; ISSN 0022-2623 1520-4804

الاتاحة: http://dx.doi.org/10.1021/acs.jmedchem.7b01155
https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.7b01155

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5

Discovery and Biological Characterization of Potent Myeloid Cell Leukemia-1 (Mcl-1) Inhibitors

مصطلحات موضوعية: Membrane Potential, Mitochondrial, Bcl-2-Like Protein 11, Cell Survival, bcl-X Protein, Antineoplastic Agents, Article, Mice, immune system diseases, hemic and lymphatic diseases, Cell Line, Tumor, Drug Design, Drug Discovery, Animals, Humans, Immunoprecipitation, Myeloid Cell Leukemia Sequence 1 Protein, neoplasms, Cell Proliferation

URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::61f63bca4d4ca92a0e75918334e75055
https://europepmc.org/articles/PMC5381274/

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6

Academic Journal

Identification and Optimization of Anthranilic Acid Based Inhibitors of Replication Protein A

المؤلفون: Patrone, James D., Pelz, Nicholas F., Bates, Brittney S., Souza‐Fagundes, Elaine M., Vangamudi, Bhavatarini, Camper, Demarco V., Kuznetsov, Alexey G., Browning, Carrie F., Feldkamp, Michael D., Frank, Andreas O., Gilston, Benjamin A., Olejniczak, Edward T., Rossanese, Olivia W., Waterson, Alex G., Chazin, Walter J., Fesik, Stephen W.

المساهمون: Vanderbilt High-Throughput Screening Core, US National Institutes of Health (NIH), American Recovery and Reinvestment Act (ARRA), National Council for Scientific and Technological Development (CNPq), Federal University of Minas Gerais (Brazil), Deutscher Akademischer Austauschdienst (DAAD), NIH National Research Service Award (NRSA), NIH NRSA

المصدر: ChemMedChem ; volume 11, issue 8, page 893-899 ; ISSN 1860-7179 1860-7187

الاتاحة: http://dx.doi.org/10.1002/cmdc.201500479
https://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1002%2Fcmdc.201500479
http://onlinelibrary.wiley.com/wol1/doi/10.1002/cmdc.201500479/fullpdf

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7

Academic Journal

Discovery of Tricyclic Indoles That Potently Inhibit Mcl-1 Using Fragment-Based Methods and Structure-Based Design

المؤلفون: Burke, Jason P., Bian, Zhiguo, Shaw, Subrata, Zhao, Bin, Goodwin, Craig M., Belmar, Johannes, Browning, Carrie F., Vigil, Dominico, Friberg, Anders, Camper, DeMarco V., Rossanese, Olivia W., Lee, Taekyu, Olejniczak, Edward T., Fesik, Stephen W.

المساهمون: NIH Office of the Director, Basic Energy Sciences, American Cancer Society, National Institutes of Health

المصدر: Journal of Medicinal Chemistry ; volume 58, issue 9, page 3794-3805 ; ISSN 0022-2623 1520-4804

الاتاحة: http://dx.doi.org/10.1021/jm501984f
https://pubs.acs.org/doi/pdf/10.1021/jm501984f

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8

Academic Journal

A method for the second-site screening of K-Ras in the presence of a covalently attached first-site ligand

المؤلفون: Sun, Qi, Phan, Jason, Friberg, Anders R., Camper, DeMarco V., Olejniczak, Edward T., Fesik, Stephen W.

المصدر: Journal of Biomolecular NMR ; volume 60, issue 1, page 11-14 ; ISSN 0925-2738 1573-5001

الاتاحة: http://dx.doi.org/10.1007/s10858-014-9849-8
http://link.springer.com/content/pdf/10.1007/s10858-014-9849-8.pdf
http://link.springer.com/article/10.1007/s10858-014-9849-8/fulltext.html
http://link.springer.com/content/pdf/10.1007/s10858-014-9849-8

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9

Academic Journal

Discovery of a Potent Inhibitor of Replication Protein A Protein–Protein Interactions Using a Fragment-Linking Approach

المؤلفون: Frank, Andreas O., Feldkamp, Michael D., Kennedy, J. Phillip, Waterson, Alex G., Pelz, Nicholas F., Patrone, James D., Vangamudi, Bhavatarini, Camper, DeMarco V., Rossanese, Olivia W., Chazin, Walter J., Fesik, Stephen W.

المصدر: Journal of Medicinal Chemistry ; volume 56, issue 22, page 9242-9250 ; ISSN 0022-2623 1520-4804

الاتاحة: http://dx.doi.org/10.1021/jm401333u
https://pubs.acs.org/doi/pdf/10.1021/jm401333u

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10

Academic Journal

Fully automated protein purification

المؤلفون: Camper, DeMarco V., Viola, Ronald E.

المصدر: Analytical Biochemistry ; volume 393, issue 2, page 176-181 ; ISSN 0003-2697

الاتاحة: http://dx.doi.org/10.1016/j.ab.2009.07.009
https://api.elsevier.com/content/article/PII:S0003269709004710?httpAccept=text/xml
https://api.elsevier.com/content/article/PII:S0003269709004710?httpAccept=text/plain

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11

Academic Journal

Zirconium tungstate hydroxide hydrate revisited: Crystallization dependence on halide and hydronium ions

المؤلفون: Colin, Julie A., Camper, DeMarco V., Gates, Stacy D., Simon, Monty D., Witker, Karen L., Lind, Cora

المصدر: Journal of Solid State Chemistry ; volume 180, issue 12, page 3504-3509 ; ISSN 0022-4596

الاتاحة: http://dx.doi.org/10.1016/j.jssc.2007.10.012
https://api.elsevier.com/content/article/PII:S0022459607004252?httpAccept=text/xml
https://api.elsevier.com/content/article/PII:S0022459607004252?httpAccept=text/plain

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12

Academic Journal

Discovery and biological characterization of potent myeloid cell leukemia-1 inhibitors.

المصدر: FEBS Letters; Jan2017, Vol. 591 Issue 1, p240-251, 12p

مصطلحات موضوعية: MYELOID leukemia, APOPTOSIS, GENETIC overexpression, PROTEIN expression, RNA interference

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13

Academic Journal

Discovery of 2-Indole-acylsulfonamide Myeloid Cell Leukemia 1 (Mcl-1) Inhibitors Using Fragment-Based Methods.

المؤلفون: Pelz, Nicholas F., Bian, Zhiguo, Zhao, Bin, Shaw, Subrata, Tarr, James C., Belmar, Johannes, Gregg, Claire, Camper, DeMarco V., Goodwin, Craig M., Arnold, Allison L., Sensintaffar, John L., Friberg, Anders, Rossanese, Olivia W., Lee, Taekyu, Olejniczak, Edward T., Fesik, Stephen W.

المصدر: Journal of Medicinal Chemistry; Mar2016, Vol. 59 Issue 5, p2054-2066, 13p

14

Academic Journal

Discovery of a Potent Inhibitorof Replication ProteinA Protein–Protein Interactions Using a Fragment-Linking Approach.

المؤلفون: Frank, Andreas O., Feldkamp, Michael D., Kennedy, J. Phillip, Waterson, Alex G., Pelz, Nicholas F., Patrone, James D., Vangamudi, Bhavatarini, Camper, DeMarco V., Rossanese, Olivia W., Chazin, Walter J., Fesik, Stephen W.

المصدر: Journal of Medicinal Chemistry; Nov2013, Vol. 56 Issue 22, p9242-9250, 9p

15

Identification and Optimization of Anthranilic Acid-Based Inhibitors of Replication Protein A ; ChemMedChem

المساهمون: Patrone, James D., Pelz, Nicholas F., Bates, Brittney S., Souza-Fagundes, Elaine M., Vangamudi, Bhavatarini, Camper, Demarco V., Kuznetsov, Alexey G., Browning, Carrie F., Feldkamp, Michael D., Frank, Andreas O., Gilston, Benjamin A., Olejniczak, Edward T., Rossanese, Olivia W., Waterson, Alex G., Chazin, Walter J., Fesik, Stephen W.

المصدر: ChemMedChem. 11(8):893-899.

مصطلحات موضوعية: Article, Replication Protein A, High throughput screening, Protein protein interactions, Medicinal chemistry, Hit optimization, Anisotropy, Dose-Response Relationship, Drug, Fluorescence Polarization, High-Throughput Screening Assays, Models, Molecular, Molecular Structure, Structure-Activity Relationship, ortho-Aminobenzoates

Relation: cdc:40995; http://stacks.cdc.gov/view/cdc/40995/

الاتاحة: http://stacks.cdc.gov/view/cdc/40995/

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