نتائج البحث - "Burke, Terrence R., Jr."

1

Academic Journal

Mono-Anionic Phosphopeptides Produced by Unexpected Histidine Alkylation Exhibit High Plk1 Polo-Box Domain-Binding Affinities and Enhanced Antiproliferative Effects in HeLa Cells

المؤلفون: Qian, Wen-Jian, Park, Jung-Eun, Lim, Dan, Lai, Christopher C., Kelley, James A., PARK, SUK YOUL, Lee, Ki Won, Yaffe, Michael B., Lee, Kyung S., Burke, Terrence R., Jr.

المساهمون: PARK, SUK YOUL

مصطلحات موضوعية: SMALL-MOLECULE INHIBITOR, KINASE 1, PEPTIDE, TARGET, PRODRUGS, PHOSPHOTHREONINE, FRAGMENTATION, DISCOVERY, INSIGHTS, POSITION, Plk1, polo kinase, polo-box domain, crystal structure, cationic dialkyl histidine, intramolecular charge masking, phosphopeptides

Relation: BIOPOLYMERS; Biochemistry & Molecular Biology; Biophysics; https://oasis.postech.ac.kr/handle/2014.oak/107103; 45982; BIOPOLYMERS, v.102, no.6, pp.444 - 455; 000345364900004

الاتاحة: https://oasis.postech.ac.kr/handle/2014.oak/107103
https://doi.org/10.1002/bip.22569

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2

Academic Journal

An Allosteric Mechanism for Inhibiting HIV-1 Integrase with a Small Molecule

المؤلفون: Kessl, Jacques J., Eidahl, Jocelyn O., Shkriabai, Nikolozi, Zhao, Zhuojun, McKee, Christopher J., Hess, Sonja, Burke, Terrence R., Jr., Kvaratskhelia, Mamuka

المصدر: Molecular Pharmacology, 76(4), 824-832, (2009-10)

Relation: https://doi.org/10.1124/mol.109.058883; eprintid:16299

الاتاحة: https://doi.org/10.1124/mol.109.058883

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3

Academic Journal

HIV-1 Integrase-Targeted Short Peptides Derived from a Viral Protein R Sequence

المؤلفون: Zhao, Xue Zhi, Métifiot, Mathieu, Kiselev, Evgeny, Kessl, Jacques, Maddali, Kasthuraiah, Marchand, Christophe, Kvaratskhelia, Mamuka, Pommier, Yves, Burke, Terrence R., Jr.

المصدر: Faculty Publications

مصطلحات موضوعية: HIV-1 integrase, viral protein R, photoaffinity probe, inhibitor, Chemistry, Medicinal-Pharmaceutical Chemistry, Physical Sciences and Mathematics

وصف الملف: application/pdf

Relation: https://aquila.usm.edu/fac_pubs/15369; https://aquila.usm.edu/context/fac_pubs/article/16686/viewcontent/HIV_1_Integrase.pdf

الاتاحة: https://aquila.usm.edu/fac_pubs/15369
https://aquila.usm.edu/context/fac_pubs/article/16686/viewcontent/HIV_1_Integrase.pdf

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4

Academic Journal

Structural basis for strand-transfer inhibitor binding to HIV intasomes.

المؤلفون: Oliveira Passos, Dario, Min Li, Jóźwik, Ilona K., Xue Zhi Zhao, Santos-Martins, Diogo, Renbin Yang, Smith, Steven J., Youngmin Jeon, Forli, Stefano, Hughes, Stephen H., Burke, Terrence R. Jr., Craigie, Robert, Lyumkis, Dmitry

المصدر: Science; 2/14/2020, Vol. 367 Issue 6479, p810-814, 5p, 4 Diagrams

5

Academic Journal

Design and Synthesis of Phosphonodifluoromethyl Phenylalanine (F 2 Pmp): A Useful Phosphotyrosyl Mimetic

المؤلفون: Burke, Terrence R. Jr.

المصدر: ChemInform ; volume 38, issue 10 ; ISSN 0931-7597 1522-2667

الاتاحة: http://dx.doi.org/10.1002/chin.200710253
https://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1002%2Fchin.200710253
https://onlinelibrary.wiley.com/doi/pdf/10.1002/chin.200710253

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6

Academic Journal

Incorporation of Phosphotyrosyl Mimetic 4‐(Phosphonodifluoromethyl)phenyl Alanine (F2Pmp) into Signal Transduction‐Directed Peptides

المؤلفون: Yao, Zhu‐Jun, Lee, Kyeong, Burke, Terrence R. Jr.

المصدر: ChemInform ; volume 37, issue 10 ; ISSN 0931-7597 1522-2667

الاتاحة: http://dx.doi.org/10.1002/chin.200610260
https://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1002%2Fchin.200610260
https://onlinelibrary.wiley.com/doi/pdf/10.1002/chin.200610260

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7

Academic Journal

A One‐Step Synthesis of N α ‐Fmoc‐4‐O‐ [O′,O′′‐di‐tert‐butyl‐2‐(2‐fluoromalonyl)]‐L‐tyrosine from Commercially Available Starting Material.

المؤلفون: Kang, Sang Uk, Burke, Terrence R. Jr.

المصدر: ChemInform ; volume 36, issue 7 ; ISSN 0931-7597 1522-2667

الاتاحة: http://dx.doi.org/10.1002/chin.200507189
https://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1002%2Fchin.200507189
https://onlinelibrary.wiley.com/doi/pdf/10.1002/chin.200507189

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8

Academic Journal

Synthesis of the First α‐Fluoro‐phosphotyrosyl Mimetic.

المؤلفون: Shi, Zhen‐Dan, Liu, Hongpeng, Zhang, Manchao, Yang, Dajun, Burke, Terrence R. Jr.

المصدر: ChemInform ; volume 36, issue 12 ; ISSN 0931-7597 1522-2667

الاتاحة: http://dx.doi.org/10.1002/chin.200512194
https://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1002%2Fchin.200512194
https://onlinelibrary.wiley.com/doi/pdf/10.1002/chin.200512194

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9

Academic Journal

Design and Synthesis of Photoactivatable Aryl Diketo Acid‐Containing HIV‐1 Integrase Inhibitors (I) as Potential Affinity Probes.

المؤلفون: Zhang, Xuechun, Marchand, Christophe, Pommier, Yves, Burke, Terrence R. Jr.

المصدر: ChemInform ; volume 35, issue 23 ; ISSN 0931-7597 1522-2667

الاتاحة: http://dx.doi.org/10.1002/chin.200423100
https://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1002%2Fchin.200423100
https://onlinelibrary.wiley.com/doi/pdf/10.1002/chin.200423100

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10

Academic Journal

Phosphotyrosyl Mimetics in the Development of Signal Transduction Inhibitors

المؤلفون: Burke, Terrence R. Jr., Lee, Kyeong

المصدر: ChemInform ; volume 34, issue 36 ; ISSN 0931-7597 1522-2667

الاتاحة: http://dx.doi.org/10.1002/chin.200336266
https://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1002%2Fchin.200336266
https://onlinelibrary.wiley.com/doi/pdf/10.1002/chin.200336266

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11

Academic Journal

Acylsulfonamide‐Containing PTP1B Inhibitors Designed to Mimic an Enzyme‐Bound Water of Hydration.

المؤلفون: Liu, Ding‐Guo, Gao, Yang, Voigt, Johannes H., Lee, Kyeong, Nicklaus, Marc C., Wu, Li, Zhang, Zhong‐Yin, Burke, Terrence R. Jr.

المصدر: ChemInform ; volume 35, issue 1 ; ISSN 0931-7597 1522-2667

الاتاحة: http://dx.doi.org/10.1002/chin.200401212
https://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1002%2Fchin.200401212
https://onlinelibrary.wiley.com/doi/pdf/10.1002/chin.200401212

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12

Academic Journal

Azido‐Containing Aryl β‐Diketo Acid HIV‐1 Integrase Inhibitors.

المؤلفون: Zhang, Xuechun, Pais, Godwin C. G., Svarovskaia, Evguenia S., Marchand, Christophe, Johnson, Allison A., Karki, Rajeshri G., Nicklaus, Marc C., Pathak, Vinay K., Pommier, Yves, Burke, Terrence R. Jr.

المصدر: ChemInform ; volume 34, issue 29 ; ISSN 0931-7597 1522-2667

الاتاحة: http://dx.doi.org/10.1002/chin.200329076
https://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1002%2Fchin.200329076
https://onlinelibrary.wiley.com/doi/pdf/10.1002/chin.200329076

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13

Academic Journal

Chicoric acid analogues as HIV-1 integrase inhibitors

المؤلفون: Lin, Zhaiwei, Neamati, Nouri, Zhao, He, Kiryu, Yoshimitsu, Turpin, Jim A, Aberham, Claudia, Strebel, Klaus, Kohn, Kurt, Witvrouw, Myriam, Pannecouque, Christophe, Debyser, Zeger, De Clercq, Erik, Rice, William G, Pommier, Yves, Burke, Terrence R Jr.

مصطلحات موضوعية: Animals, Anti-HIV Agents, Caffeic Acids, Cell Line, Drug Evaluation, Preclinical, HIV Integrase, HIV Integrase Inhibitors, HIV-1, HIV-2, Humans, Stereoisomerism, Structure-Activity Relationship, Succinates, Virus Replication

Relation: Journal of Medicinal Chemistry vol:42 issue:8 pages:1401-14; https://lirias.kuleuven.be/handle/123456789/12006; http://dx.doi.org/10.1021/jm980531m

الاتاحة: https://lirias.kuleuven.be/handle/123456789/12006
https://doi.org/10.1021/jm980531m

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14

Electronic Resource

An NMR strategy for fragment-based ligand screening utilizing a paramagnetic lanthanide probe

المؤلفون: Saio, Tomohide, Ogura, Kenji, Shimizu, Kazumi, Yokochi, Masashi, Burke, Terrence R., Jr., 1000070011757, Inagaki, Fuyuhiko

مصطلحات الفهرس: Ligand screening, Fragment-based drug design (FBDD), Protein-ligand structure, Lanthanide-binding peptide tag (LBT), Paramagnetic relaxation enhancement (PRE), Pseudo-contact shift (PCS), 464, Journal Article, VoR

URL: http://hdl.handle.net/2115/47385
https://eprints.lib.hokudai.ac.jp/dspace/bitstream/2115/47385/1/JBN51-3_395-408.pdf
https://doi.org/10.1007/s10858-011-9566-5
https://doi.org/10.1007/s10858-011-9566-5

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15

Academic Journal

Hydroxylated Aromatic Inhibitors of HIV-1 Integrase

المؤلفون: Burke, Terrence R. Jr., Fesen, Mark, Mazumder, Abhijit, Yung, Jessie, Wang, Jian, Carothers, Adelaide M., Grunberger, Dezider, Driscoll, John, Pommier, Yves, Kohn, Kurt

المصدر: Journal of Medicinal Chemistry ; volume 38, issue 21, page 4171-4178 ; ISSN 0022-2623 1520-4804

الاتاحة: http://dx.doi.org/10.1021/jm00021a006
https://pubs.acs.org/doi/pdf/10.1021/jm00021a006

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16

Academic Journal

An NMR strategy for fragment-based ligand screening utilizing a paramagnetic lanthanide probe

المؤلفون: Saio, Tomohide, Ogura, Kenji, Shimizu, Kazumi, Yokochi, Masashi, Burke, Terrence R., Jr., Inagaki, Fuyuhiko

مصطلحات موضوعية: Ligand screening, Fragment-based drug design (FBDD), Protein-ligand structure, Lanthanide-binding peptide tag (LBT), Paramagnetic relaxation enhancement (PRE), Pseudo-contact shift (PCS)

Time: 464

Relation: http://hdl.handle.net/2115/47385; Journal of Biomolecular NMR, 51(3): 395-408; http://dx.doi.org/10.1007/s10858-011-9566-5

الاتاحة: http://hdl.handle.net/2115/47385
https://doi.org/10.1007/s10858-011-9566-5

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17

Academic Journal

Enhancing precision in colorectal cancer surgery: development of an LGR5-targeting RSPO1 peptide mimetic as a contrast agent for intraoperative fluorescence molecular imaging.

المؤلفون: Parasido, Erika¹ (AUTHOR), Ribeiro, Patricia¹ (AUTHOR), Chingle, Ramesh M.² (AUTHOR), Rohwetter, Thomas¹ (AUTHOR), Gupta, Nikita¹ (AUTHOR), Avetian, George¹ (AUTHOR), Bladelli, Elisa³ (AUTHOR), Pierobon, Mariaelena³ (AUTHOR), Chen, Yu⁴ (AUTHOR), Tang, Qinggong⁵ (AUTHOR), Schnermann, Martin² (AUTHOR), Rodriguez, Olga¹ (AUTHOR), Robbins, David¹ (AUTHOR), Burke, Terrence R. Jr.² (AUTHOR), Albanese, Chris¹ (AUTHOR) albanese@georgetown.edu, Ihemelandu, Chukwuemeka¹ (AUTHOR)

المصدر: Cell Cycle. Jul2024, p1-12. 12p. 6 Illustrations.

مصطلحات موضوعية: *CONTRAST media, *COLORECTAL cancer, *PEPTIDES, *PROCTOLOGY, *CARCINOGENESIS, *LEUCINE

مصطلحات جغرافية: UNITED States

18

Academic Journal

Design and Synthesis of Phosphonodifluoromethyl Phenylalanine (F2Pmp): A Useful Phosphotyrosyl Mimetic.

المؤلفون: Burke, Terrence R. Jr.

المصدر: ChemInform; Mar2007, Vol. 38 Issue 10, pno-no, 1p

19

Academic Journal

A One-Step Synthesis of N^α-Fmoc-4-O- [O′,O′′-di-tert-butyl-2-(2-fluoromalonyl)]-L-tyrosine from Commercially Available Starting Material.

المؤلفون: Kang, Sang Uk, Burke, Terrence R. Jr.

المصدر: ChemInform; Feb2005, Vol. 36 Issue 7, pno-no, 1p

20

Academic Journal

Acylsulfonamide-Containing PTP1B Inhibitors Designed to Mimic an Enzyme-Bound Water of Hydration.

المؤلفون: Liu, Ding-Guo, Gao, Yang, Voigt, Johannes H., Lee, Kyeong, Nicklaus, Marc C., Wu, Li, Zhang, Zhong-Yin, Burke, Terrence R. Jr.

المصدر: ChemInform; Jan2004, Vol. 35 Issue 1, pno-no, 1p

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