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1
المؤلفون: Paul M. Slattum, J. Adam Willardsen, Weston R Judd, Brita Brown, Liwen Huang, Daniel Wettstein, Kirill Ostanin, Khanh C. Hoang, Glen L Alberts, Bruce D. Roth, Burt Richards, Liisa Valppu, Leena Bhoite
المصدر: Journal of Medicinal Chemistry. 54:5031-5047
مصطلحات موضوعية: Methyltransferase, Cell Survival, Stereochemistry, Antineoplastic Agents, Stereoisomerism, Gene Knockout Techniques, Structure-Activity Relationship, chemistry.chemical_compound, Cytosol, Cell Line, Tumor, Drug Discovery, Humans, Structure–activity relationship, Protein Methyltransferases, Viability assay, Cell Proliferation, Pyrans, Chemistry, Cell growth, Farnesyltransferase inhibitor, Recombinant Proteins, Biochemistry, Cell culture, ras Proteins, Molecular Medicine, Drug Screening Assays, Antitumor, Growth inhibition
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2
المؤلفون: Bruce D. Roth, Ann E. Weber, Ruth R. Wexler, Scott D. Edmondson, Jason Elliott
المصدر: Medicinal Chemistry Reviews ISBN: 9780996293211
Medicinal Chemistry Reviews -
3
المؤلفون: Randy Ramharack, Peggy Liao, Janak Khimchand Padia, Bruce D. Roth, Patt William Chester, Helen Tsenwhei Lee, Mark A Spahr, Jason K. Pontrello, Karen Elaine Sexton, Mark A. Massa
المصدر: Bioorganic & Medicinal Chemistry. 11:4827-4845
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Mice, Transgenic, Pharmacology, Biochemistry, Chemical synthesis, Cell Line, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, In vivo, Oral administration, Drug Discovery, Animals, Humans, Structure–activity relationship, Amino Acids, Molecular Biology, chemistry.chemical_classification, Sulfonamides, Dose-Response Relationship, Drug, biology, Chemistry, Organic Chemistry, Haplorhini, Lipoprotein(a), Amino acid, Dose–response relationship, biology.protein, Molecular Medicine, Lipoprotein
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4
المؤلفون: Jay R. Luly, Kenneth G. Carson, David J Heilig, Wen Song Yue, Shixin Qin, Jie Jack Li, David T. Connor, Joseph Edwin Low, Roberta A Glynn, Bharat K. Trivedi, Qing Ye, Stephen W. Hunt, Steven R. Miller, Bruce D. Roth, Weixing Yang
المصدر: Bioorganic & Medicinal Chemistry. 11:3777-3790
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Anti-Inflammatory Agents, Pharmaceutical Science, Antineoplastic Agents, Diamines, Biochemistry, Chemical synthesis, Receptors, Interleukin-8A, Structure-Activity Relationship, Quinoxalines, Drug Discovery, Humans, Structure–activity relationship, Interleukin 8, Receptor, Molecular Biology, Bicyclic molecule, Chemistry, Chemotaxis, Organic Chemistry, Interleukin-8 receptor, Small molecule, In vitro, Molecular Medicine, Calcium
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5
المؤلفون: Burt Richards, Mark A. Poritz, Bruce D. Roth, Bob Risley, David H.-F. Teng, Tanya Sandrock, Harry A. Austin, Mark Stump, Karen Repetny, Forrest Hsu, Alexander Kamb, Sanghee Yoo, Marianne K.-H. Kim
المصدر: Molecular Therapy. 4(5):398-406
مصطلحات موضوعية: Blotting, Western, Genetic Vectors, Green Fluorescent Proteins, Gene Expression, Peptide, Biology, Retinoblastoma Protein, Protein expression, Green fluorescent protein, Cell Line, Mice, Genes, Reporter, Transduction, Genetic, Drug Discovery, medicine, Genetics, Animals, Humans, Expressivity (genetics), Cloning, Molecular, Molecular Biology, Cyclin-Dependent Kinase Inhibitor p16, Gene Library, chemistry.chemical_classification, Pharmacology, Cell growth, Retinoblastoma, Proteins, Genetic Therapy, Oncogene Proteins, Viral, medicine.disease, Flow Cytometry, Phenotype, Molecular biology, Peptide Fragments, Leukemia Virus, Murine, Luminescent Proteins, Retroviridae, chemistry, Cell culture, Protein Biosynthesis, Molecular Medicine, Peptides
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6
المؤلفون: Giordano Caponigro, Mark A. Poritz, Michael John Feldhaus, Tanya Sandrock, Marianne Kim, Bruce D. Roth, Alexander Kamb
المصدر: Yeast. 19:1-7
مصطلحات موضوعية: Saccharomyces cerevisiae Proteins, Green Fluorescent Proteins, Saccharomyces cerevisiae, Gene Expression, Bioengineering, Applied Microbiology and Biotechnology, Biochemistry, Pheromones, Green fluorescent protein, Fungal Proteins, Gene expression, Genetics, Zinc finger, Pheromone response, biology, Membrane Proteins, Signal transducing adaptor protein, Zinc Fingers, biology.organism_classification, Penetrance, Vesicular transport protein, Adaptor Proteins, Vesicular Transport, Luminescent Proteins, Peptides, Biotechnology
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7
المؤلفون: Anthony D. Sercel, Kuai-Lin Sun, Yuntao Song, Bruce D. Roth, Norman L. Colbry, D. R. Johnson
المصدر: Tetrahedron Letters. 41:8225-8230
مصطلحات موضوعية: chemistry.chemical_classification, Chemistry, Reductive methylation, Organic Chemistry, Drug Discovery, lipids (amino acids, peptides, and proteins), Alkylation, Biochemistry, Medicinal chemistry, Amino acid, Catalysis
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8Addition reactions of allyl stannanes to an indolo[2′,3′:3,4]pyrido[1,2-b]isoquinoline imminium salt
المؤلفون: David T. Connor, Bruce D. Roth, Paul C. Unangst, Larry D. Bratton, Bharat K. Trivedi, J. Ronald Rubin
المصدر: Journal of Heterocyclic Chemistry. 37:1081-1087
مصطلحات موضوعية: chemistry.chemical_classification, Addition reaction, Organic Chemistry, chemistry.chemical_element, Salt (chemistry), Medicinal chemistry, Adduct, chemistry.chemical_compound, chemistry, Reagent, Yield (chemistry), Proton NMR, Isoquinoline, Tin
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9
المؤلفون: Alexander Pavlovsky, Claude Forsey Purchase, V. Dhanaraj, Bruce D. Roth, Donald Hupe, Mark G. Williams, Ye Qi-Zhuang, Christine Humblet, Tom L. Blundell, Daniel F. Ortwine, Andrew D. White, Johnson Linda Lea
المصدر: Protein Science. 8:1455-1462
مصطلحات موضوعية: Models, Molecular, chemistry.chemical_classification, Metalloproteinase, Binding Sites, biology, Stereochemistry, Active site, Peptide, Matrix Metalloproteinase Inhibitors, Matrix metalloproteinase, Crystallography, X-Ray, Biochemistry, Enzyme, chemistry, Catalytic Domain, Hydrolase, biology.protein, Humans, Moiety, Matrix Metalloproteinase 3, Protease Inhibitors, Selectivity, Molecular Biology, Protein Binding, Research Article
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10
المؤلفون: Bruce D. Roth, Jie Jack Li, J. Ronald Rubin, Bharat K. Trivedi
المصدر: Tetrahedron Letters. 39:6111-6114
مصطلحات موضوعية: chemistry.chemical_classification, Organic Chemistry, Alkaloid synthesis, Iminium, Salt (chemistry), Biochemistry, Enamine, chemistry.chemical_compound, chemistry, Acetyl chloride, Reagent, Drug Discovery, Robinson annulation, Organic chemistry
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11
المؤلفون: Helen T. Lee, Brian R. Krause, Bruce D. Roth, R. L. Stanfield, W. H. Roark, Joseph Armand Picard, Drago Robert Sliskovic, R. F. Bousley, K. L. Hamelehle
المصدر: Bioorganic & Medicinal Chemistry Letters. 8:289-294
مصطلحات موضوعية: medicine.drug_class, Stereochemistry, Clinical Biochemistry, Sterol O-acyltransferase, Pharmaceutical Science, Carboxamide, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Organophosphorus Compounds, Microsomes, Drug Discovery, medicine, Animals, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, Sulfonamides, biology, Cholesterol, Anticholesteremic Agents, Organic Chemistry, Phosphoramidate, Enzyme, chemistry, Acyltransferases, Enzyme inhibitor, biology.protein, Molecular Medicine, Rabbits, Sterol O-Acyltransferase
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12
المؤلفون: Bruce D. Roth
المصدر: Drug Discovery Today. 3:19-25
مصطلحات موضوعية: Pharmacology, Biochemistry, Enzyme inhibitor, Drug Discovery, Sterol O-acyltransferase, Atherosclerotic disease, biology.protein, Biology, Clinical success, Cholesterol absorption
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13
المؤلفون: N. Suman-Chauhan, Louise Webdale, Bharat K. Trivedi, Terri S. Purchase, Bruce D. Roth, Bradley Dean Tait, Michael W. Wilson, C.E. Augelli-Szafran
المصدر: Bioorganic & Medicinal Chemistry Letters. 7:2009-2014
مصطلحات موضوعية: chemistry.chemical_classification, Indole test, Stereochemistry, medicine.drug_class, Organic Chemistry, Clinical Biochemistry, Antagonist, Pharmaceutical Science, Biological activity, Receptor antagonist, Biochemistry, Chemical synthesis, CI-988, chemistry, Heterocyclic compound, Drug Discovery, medicine, Molecular Medicine, Moiety, Molecular Biology
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14
المؤلفون: Bruce D. Roth, Karen Lackey
المصدر: Methods and Principles in Medicinal Chemistry ISBN: 9783527677252
Medicinal Chemistry Approaches to Personalized Medicineمصطلحات موضوعية: business.industry, Medicine, Personalized medicine, business, Medicinal chemistry
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15
المؤلفون: Bruce D. Roth, Karen Lackey
المصدر: Medicinal Chemistry Approaches to Personalized Medicine
مصطلحات موضوعية: Engineering, business.industry, Drug discovery, Personalized medicine, business, Medicinal chemistry
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16
المؤلفون: Martyn Clive Pritchard, Bruce D. Roth, N. Suman-Chauhan, Daniel F. Ortwine, C.E. Augelli-Szafran, David R. Hill, David Christopher Horwell, Clare O. Kneen, Bharat K. Trivedi, Louise Webdale, Terri S. Purchase
المصدر: Bioorganic & Medicinal Chemistry. 4:1733-1745
مصطلحات موضوعية: Steric effects, Indoles, Stereochemistry, Carboxylic acid, Clinical Biochemistry, Substituent, Pharmaceutical Science, Ring (chemistry), Biochemistry, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Hormone Antagonists, Meglumine, Drug Discovery, Animals, Moiety, Molecular Biology, chemistry.chemical_classification, digestive, oral, and skin physiology, Organic Chemistry, Receptor, Cholecystokinin B, Rats, Receptor, Cholecystokinin A, chemistry, Lipophilicity, Polar effect, Molecular Medicine, Receptors, Cholecystokinin, Selectivity
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17
المؤلفون: Bruce D. Roth
المصدر: Current Pharmaceutical Design. 2:139-154
مصطلحات موضوعية: Pharmacology, Drug Discovery
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18
المؤلفون: Linda Guilds-Zamarka, Dirk A. Bornemeier, Maritza Oxender, Bruce J. Auerbach, Bharat K. Trivedi, Bradley Dean Tait, Bruce D. Roth, Richard D. Dyer, Joseph A. Cornicelli
المصدر: Bioorganic & Medicinal Chemistry Letters. 6:93-96
مصطلحات موضوعية: Catechol, biology, Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Lipoxygenase, chemistry.chemical_compound, Drug Discovery, biology.protein, Molecular Medicine, Moiety, Molecular Biology, Mass screening
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19
المؤلفون: Maureen K. Anderson, Patrice Lee, J. F. Reindel, K. L. Hamelehle, R. L. Stanfield, Drago Sliskovic, J. A. Picard, Bruce D. Roth, B.R. Krause, D. Turluck, Andrew D. White, Sandra Bak Mueller, Reynold Homan, Thomas M.A. Bocan, Patrick Michael O'brien, Helen Tsenwhei Lee, Claude Forsey Purchase, R. F. Bousley
المصدر: Journal of Medicinal Chemistry. 39:2354-2366
مصطلحات موضوعية: Male, Arteriosclerosis, Stereochemistry, Guinea Pigs, Hypercholesterolemia, Drug Evaluation, Preclinical, Tetrazoles, Cholesterol, Dietary, Structure-Activity Relationship, chemistry.chemical_compound, Amide, Drug Discovery, Animals, Moiety, Tetrazole, Enzyme Inhibitors, Fatty acid amide, Molecular Structure, Cholesterol, Anticholesteremic Agents, Macrophages, Biological activity, Rats, chemistry, Drug Design, Microsomes, Liver, Microsome, Molecular Medicine, Rabbits, Acetamide, Sterol O-Acyltransferase
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20
المؤلفون: Maureen K. Anderson, Reynold Homan, Joseph Armand Picard, R. L. Stanfield, Bruce D. Roth, Brian R. Krause, K. L. Hamelehle, W. Howard Roark, R. F. Bousley
المصدر: Bioorganic & Medicinal Chemistry Letters. 5:2367-2370
مصطلحات موضوعية: chemistry.chemical_classification, medicine.drug_class, Organic Chemistry, Clinical Biochemistry, Sterol O-acyltransferase, Pharmaceutical Science, Biochemistry, Sulfonylurea, In vitro, Enzyme, Plasma cholesterol, chemistry, In vivo, Drug Discovery, medicine, Molecular Medicine, lipids (amino acids, peptides, and proteins), Molecular Biology