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المؤلفون: Maria Galvez-Llompart, Jorge Galvez, Riccardo Zanni
المصدر: RIUCV. Repositorio de la Universidad Católica de Valencia San Vicente Mártir
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RIUCV: Repositorio de la Universidad Católica de Valencia San Vicente Mártir
Universidad Católica de Valencia San Vicente Mártirمصطلحات موضوعية: medicine.drug_class, Antibiotics, 2415 Biología Molecular, Computational biology, medicine.disease_cause, Azithromycin, Virus, 2302.22 Farmacología Molecular, chemistry.chemical_compound, 32 Ciencias Médicas, Clarithromycin, medicine, Repurposing, Coronavirus, 2302.21 Biología Molecular, Molecular topology, 12 Matemáticas, business.industry, Topología molecular, COVID-19, Drugs, Lopinavir, chemistry, Fármacos, Brecanavir, business, Tipología molecular, medicine.drug
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المؤلفون: Emile J. Velthuisen, Todd M. Baughman, Brian A. Johns, David P. Temelkoff, Jason G. Weatherhead
المصدر: European Journal of Medicinal Chemistry. 63:202-212
مصطلحات موضوعية: Metabolic Clearance Rate, Stereochemistry, Bond breaking, chemistry.chemical_compound, Pharmacokinetics, Drug Discovery, Kinetic isotope effect, medicine, Animals, Humans, Benzodioxoles, Pharmacology, Molecular Structure, Organic Chemistry, HIV Protease Inhibitors, General Medicine, Metabolic stability, Deuterium, Rate-determining step, Combinatorial chemistry, Protease inhibitor (biology), Rats, Models, Chemical, chemistry, Area Under Curve, Hepatocytes, Brecanavir, Administration, Intravenous, Carbamates, medicine.drug
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المؤلفون: Lys A. Braga-Silva, André L.S. Santos
المصدر: Current Medicinal Chemistry. 18:2401-2419
مصطلحات موضوعية: Antifungal Agents, Aspartic Acid Proteases, medicine.medical_treatment, Virulence, HIV Infections, Biochemistry, Microbiology, Structure-Activity Relationship, chemistry.chemical_compound, Candida albicans, Drug Discovery, medicine, Animals, Humans, Protease Inhibitors, Protease inhibitor (pharmacology), Pathogen, Pharmacology, Protease, biology, Organic Chemistry, Candidiasis, biology.organism_classification, Corpus albicans, chemistry, Fungal behavior, Immunology, Brecanavir, Molecular Medicine
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المؤلفون: Jacob Lalezari, Douglas J. Ward, Harmony P. Garges, Susan A. Tomkins
المصدر: Journal of Antimicrobial Chemotherapy. 60:170-174
مصطلحات موضوعية: Adult, Male, Microbiology (medical), Anti-HIV Agents, medicine.medical_treatment, HIV Infections, Pharmacology, Virus, chemistry.chemical_compound, HIV Protease, Drug Resistance, Viral, Humans, Medicine, HIV Protease Inhibitor, Pharmacology (medical), Protease inhibitor (pharmacology), Benzodioxoles, Adverse effect, Darunavir, Chemotherapy, Ritonavir, business.industry, HIV Protease Inhibitors, Middle Aged, CD4 Lymphocyte Count, Treatment Outcome, Infectious Diseases, Amino Acid Substitution, chemistry, HIV-1, Brecanavir, RNA, Viral, Reverse Transcriptase Inhibitors, Drug Therapy, Combination, Female, Carbamates, business, medicine.drug
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المصدر: Expert Opinion on Therapeutic Patents. 16:1067-1091
مصطلحات موضوعية: Pharmacology, business.industry, virus diseases, Fosamprenavir, General Medicine, biochemical phenomena, metabolism, and nutrition, Virology, Amprenavir, chemistry.chemical_compound, Nelfinavir, chemistry, immune system diseases, Indinavir, Drug Discovery, medicine, Brecanavir, business, Tipranavir, Saquinavir, Darunavir, medicine.drug
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المؤلفون: Bruno D. Chapsal, Arun K. Ghosh
المصدر: Aspartic Acid Proteases as Therapeutic Targets
مصطلحات موضوعية: business.industry, Fosamprenavir, Drug resistance, medicine.disease, Virology, Atazanavir, chemistry.chemical_compound, Acquired immunodeficiency syndrome (AIDS), chemistry, Brecanavir, Medicine, HIV Protease Inhibitor, Ritonavir, business, Darunavir, medicine.drug
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المؤلفون: Mark Johnson, Maggie T. Anderson, Y. Sunila Reddy, Susan L. Ford, Judith Ng-Cashin, Sharon C. Murray
المصدر: Antimicrobial agents and chemotherapy. 51(4)
مصطلحات موضوعية: Adult, Male, HIV Infections, Pharmacology, Antiviral Agents, Drug Administration Schedule, chemistry.chemical_compound, Pharmacokinetics, Medicine, Humans, Pharmacology (medical), Benzodioxoles, Adverse effect, IC50, Ritonavir, Dose-Response Relationship, Drug, business.industry, HIV Protease Inhibitors, Middle Aged, Dose–response relationship, Drug Combinations, Infectious Diseases, Tolerability, chemistry, Area Under Curve, Toxicity, Brecanavir, HIV-1, Female, Carbamates, Safety, business, medicine.drug
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المؤلفون: Andrea De Luca
مصطلحات موضوعية: medicine.medical_treatment, Immunology, resistance, HIV protease inhibitors, Salvage therapy, Pharmacology, Settore MED/17 - MALATTIE INFETTIVE, chemistry.chemical_compound, Virology, medicine, HIV Protease Inhibitor, Darunavir, Protease, Oncology (nursing), INVESTIGATIONAL AGENTS, business.industry, Hematology, Infectious Diseases, Oncology, chemistry, Brecanavir, business, Tipranavir, HIV drug resistance, medicine.drug
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المؤلفون: Pedro Fernandez, Maggie T. Anderson, Mark Johnson, Daniel S. Stein, Y. Sunila Reddy, Susan L. Ford, Sharon C. Murray
مصطلحات موضوعية: Adult, Diarrhea, Male, Administration, Oral, Capsules, Pharmacology, Clinical Therapeutics, Drug Administration Schedule, chemistry.chemical_compound, Pharmacokinetics, Double-Blind Method, Oral administration, HIV Protease Inhibitor, Medicine, Flatulence, Humans, Pharmacology (medical), Benzodioxoles, Ritonavir, Dose-Response Relationship, Drug, business.industry, Headache, Nausea, HIV Protease Inhibitors, Middle Aged, Virology, Dose–response relationship, Drug Combinations, Infectious Diseases, Tolerability, chemistry, Area Under Curve, Toxicity, Brecanavir, Carbamates, business, Gels, medicine.drug, Half-Life
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المؤلفون: David J. Reynolds, Ed W. McLean, Istvan Kaldor, Robert X. Xu, Elizabeth M. Turner, Douglas M. Sammond, C. Webster Andrews, Furfine Eric Steven, Michael R. Hale, Andrew Spaltenstein, Michael Stephen Brieger, Ronald George Sherrill, Mary H. Hanlon, Richard J. Hazen, Roger D. Tung, John F. Miller
المصدر: Bioorganicmedicinal chemistry letters. 16(7)
مصطلحات موضوعية: medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Virus, chemistry.chemical_compound, Amprenavir, Drug Discovery, medicine, HIV Protease Inhibitor, Protease inhibitor (pharmacology), Molecular Biology, chemistry.chemical_classification, Sulfonamides, Protease, biology, Molecular Structure, Organic Chemistry, HIV Protease Inhibitors, Virology, Enzyme, chemistry, Enzyme inhibitor, Brecanavir, biology.protein, Molecular Medicine, medicine.drug