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1
المؤلفون: Thomas F. Walsh, Nancy A. Nolan, Douglas J. Pettibone, William J. Greenlee, Stacey O'Malley, Raymond S.L. Chang, Kenneth J. Fitch, D. F. Veber, David L. Williams, Kathryn L. Murphy, Bradley V. Clineschmidt
المصدر: Bioorganic & Medicinal Chemistry Letters. 5:1155-1158
مصطلحات موضوعية: Angiotensin receptor, Chemistry, Ligand binding assay, Organic Chemistry, Clinical Biochemistry, Antagonist, Pharmaceutical Science, Biochemistry, Angiotensin II, Part iii, Drug Discovery, Molecular Medicine, Endothelin receptor, Molecular Biology
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2
المؤلفون: N. P. Gould, James B. Hoffman, D. F. Veber, Doug W. Hobbs, Doug J. Pettibone, Roger M. Freidinger, Bradley V. Clineschmidt
المصدر: Bioorganic & Medicinal Chemistry Letters. 5:119-122
مصطلحات موضوعية: Chemistry, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Combinatorial chemistry, Non peptide, Camphor, chemistry.chemical_compound, Oxytocin, Drug Discovery, Aspartic acid, medicine, Molecular Medicine, Molecular Biology, hormones, hormone substitutes, and hormone antagonists, medicine.drug
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3
المؤلفون: Bradley V. Clineschmidt, Richard G. Ball, Douglas J. Pettibone, Daniel F. Veber, Joseph M. Pawluczyk, J. Chris Culberson, Roger M. Freidinger, Jill M. Erb, Peter D. Williams, Debra S. Perlow
المصدر: Bioorganic & Medicinal Chemistry. 2:971-985
مصطلحات موضوعية: Male, Models, Molecular, Receptors, Vasopressin, Stereochemistry, Molecular Sequence Data, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Kidney, Oxytocin, Tritium, Biochemistry, Molecular mechanics, Piperazines, Structure-Activity Relationship, Uterine Contraction, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, Amino Acid Sequence, Receptor, Molecular Biology, Sulfonamides, Chemistry, Uterus, Organic Chemistry, Antagonist, Camphor, Rats, Kinetics, Liver, Receptors, Oxytocin, Molecular Medicine, Female, Selectivity, Acyl group, medicine.drug
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4
المؤلفون: Tsing-B. Chen, Kristie A. Faust, Elizabeth M. Naylor, Bradley V. Clineschmidt, Prasun K. Chakravarty, Victor J. Lotti, Robert J. Bendesky, Stacey A. O'Malley, Paul J. Kling, Raymond S.L. Chang, Arthur A. Patchett, William J. Greenlee
المصدر: Drug Development Research. 32:161-171
مصطلحات موضوعية: Agonist, medicine.medical_specialty, Angiotensin II receptor type 1, Aldosterone, medicine.drug_class, Antagonist, Molecular biology, Angiotensin II, chemistry.chemical_compound, Endocrinology, chemistry, Internal medicine, Drug Discovery, Renin–angiotensin system, medicine, Receptor, IC50
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5
المؤلفون: C. J. Woyden, M. J. Novy, Mark G. Bock, Bradley V. Clineschmidt, B. E. Evans, E V Lis, Terry W. Schorn, K. L. Thompson, Peter K. S. Siegl, Douglas J. Pettibone, Duane R. Reiss, Peter D. Williams, Doug W. Hobbs, M. A. Cukierski, Maribeth T. Guidotti, Roger M. Freidinger, D. F. Veber, G. J. Haluska, M. J. Cook, M. J. Kaufman, S.-H. L. Chiu
المصدر: Drug Development Research. 30:129-142
مصطلحات موضوعية: Tocolytic agent, medicine.medical_specialty, Antagonist, Pharmacology, Biology, Oxytocin Antagonist, Endocrinology, Oxytocin, In vivo, Internal medicine, Tocolytic, Drug Discovery, medicine, Receptor, L-368,899, medicine.drug
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6
المؤلفون: Mark G. Bock, B. E. Evans, Peter D. Williams, Roger M. Freidinger, Douglas J. Pettibone, D. F. Veber, Bradley V. Clineschmidt
المصدر: Regulatory Peptides. 45:289-293
مصطلحات موضوعية: medicine.medical_specialty, Vasopressin, Preterm labor, Physiology, Clinical Biochemistry, Neuropeptide, Peptide, Pharmacology, Oxytocin, Peptides, Cyclic, Biochemistry, Cellular and Molecular Neuroscience, Endocrinology, Pregnancy, Internal medicine, medicine, Animals, chemistry.chemical_classification, business.industry, Antagonist, Tocolytic Agents, chemistry, Female, business, medicine.drug
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7
المؤلفون: Bradley V. Clineschmidt, Gino Salituro, Deborah L. Zink, Joanne M. Williamson, Douglas J. Pettibone
المصدر: Bioorganic & Medicinal Chemistry Letters. 3:337-340
مصطلحات موضوعية: Natural product, Chemistry, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Peptide hormone, Pharmacology, Biochemistry, Oxytocin receptor, chemistry.chemical_compound, Oxytocin, Drug Discovery, medicine, Natural source, Molecular Medicine, Molecular Biology, medicine.drug
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8
المؤلفون: Erb Jm, Douglas J. Pettibone, D. S. Perlow, S.-H. L. Chiu, Peter D. Williams, Roger M. Freidinger, Mark G. Bock, L. A. Carroll, Steven M. Pitzenberger, Michael J. Kaufman, J. C. Culberson, B. E. Evans, J. S. Murphy, G. F. Lundell, S. L. Fitzpatrick, Bradley V. Clineschmidt, Joseph M. Pawluczyk, Richard G. Ball, P. S. Anderson
المصدر: ChemInform. 25
مصطلحات موضوعية: chemistry.chemical_classification, Sulfonyl, Piperazine, chemistry.chemical_compound, chemistry, Preterm labor, Bicyclic molecule, Stereochemistry, General Medicine, Bridged compounds, L-368,899, Oxytocin Antagonist, Bioavailability
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9
المؤلفون: Douglas J. Pettibone, Peter D. Williams, C. J. Woyden, Roger M. Freidinger, Erb Jm, E V Lis, Duane R. Reiss, Bradley V. Clineschmidt, D. F. Veber, Maribeth T. Guidotti, Joseph M. Pawluczyk
المصدر: ChemInform. 27
مصطلحات موضوعية: chemistry.chemical_compound, L-371,257, Chemistry, Stereochemistry, General Medicine, Non peptide, Oxytocin Antagonist, Bioavailability
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10
المؤلفون: J. A. Totaro, Roger M. Freidinger, Mark G. Bock, Gretchen S. Young, Bradley V. Clineschmidt, Douglas J. Pettibone, Peter D. Williams, Richard W. Ransom, D. F. Veber, E V Lis
المصدر: European Journal of Pharmacology. 196:233-237
مصطلحات موضوعية: Agonist, Vasopressin, medicine.medical_specialty, medicine.drug_class, Inositol Phosphates, Bradykinin, Biology, Oxytocin, Tritium, Peptides, Cyclic, Oxytocin Antagonist, Uterine Contraction, chemistry.chemical_compound, Internal medicine, medicine, Animals, IC50, Pharmacology, Uterus, Antagonist, Rats, Inbred Strains, Biological activity, Rats, Endocrinology, chemistry, Female, medicine.drug
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11Academic Journal
المؤلفون: Robert G. Pendleton, Robert J. Bendesky, Bradley V. Clineschmidt, Schaffer Thomas E. Nolan
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.1025.9331; http://jpet.aspetjournals.org/content/241/1/110.full.pdf
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12
المؤلفون: Chen A, Dhanoa Dm, E V Lis, T. F. Walsh, Nancy A. Nolan, Stephen Krause, Kathy L. Murphy, Kenneth J. Fitch, Prasun K. Chakravarty, Douglas J. Pettibone, Julie A. O'Brien, Elizabeth M. Naylor, W.J. Greenlee, Scott W. Bagley, David L. Williams, Bradley V. Clineschmidt, Daniel F. Veber
المصدر: Life sciences. 58(14)
مصطلحات موضوعية: Agonist, medicine.hormone, Endothelin Receptor Antagonists, Male, medicine.medical_specialty, medicine.drug_class, Biological Availability, Blood Pressure, CHO Cells, Dioxoles, Pharmacology, Biology, In Vitro Techniques, Phosphatidylinositols, General Biochemistry, Genetics and Molecular Biology, Endothelins, Iodine Radioisotopes, Rats, Sprague-Dawley, Mice, Structure-Activity Relationship, Dogs, Internal medicine, Cricetinae, medicine, Animals, Humans, General Pharmacology, Toxicology and Pharmaceutics, Receptor, IC50, Receptors, Endothelin, Chinese hamster ovary cell, Hydrolysis, Antagonist, Ferrets, Imidazoles, General Medicine, Receptor antagonist, Rats, Kinetics, Endocrinology, Female, Endothelin receptor, Muscle Contraction
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13
المؤلفون: Douglas J. Pettibone, J. C. Culberson, Doug W. Hobbs, R. M. Freidinger, Peter D. Williams, N. P. Gould, Bradley V. Clineschmidt, James B. Hoffman, D. F. Veber
المصدر: Peptides 1994 ISBN: 9789072199218
Peptides 1994مصطلحات موضوعية: Oxytocin, Chemistry, medicine, Pharmacology, medicine.drug, Bioavailability
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14
المؤلفون: James B. Hoffman, Jill M. Erb, Kevin F. Gilbert, Daniel F. Veber, Roger M. Freidinger, Mark G. Bock, Robert M. DiPardo, Ben E. Evans, James L. Leighton, George F. Lundell, Douglas J. Pettibone, Bradley V. Clineschmidt, Willie L. Whitter, Roger D. Tung, Peter D. Williams, N. P. Gould, Debra S. Perlow
المصدر: Peptides ISBN: 9789401090681
Peptides 1992
Peptides 1992 ISBN: 9789401046466مصطلحات موضوعية: Oxytocin, Chemistry, medicine, Pharmacology, medicine.drug
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15
المؤلفون: Ben E. Evans, James L. Leighton, Kenneth E. Rittle, Kevin F. Gilbert, George F. Lundell, Norman P. Gould, Doug W. Hobbs, Robert M. DiPardo, Daniel F. Veber, Douglas J. Pettibone, Bradley V. Clineschmidt, Paul S. Anderson, Roger M. Freidinger
المصدر: Journal of medicinal chemistry. 35(21)
مصطلحات موضوعية: Receptors, Vasopressin, Magnetic Resonance Spectroscopy, Administration, Oral, Biological Availability, Peptide, Pharmacology, Oxytocin, Structure-Activity Relationship, Obstetric Labor, Premature, Piperidines, In vivo, Pregnancy, Drug Discovery, medicine, Structure–activity relationship, Animals, Spiro Compounds, Receptor, chemistry.chemical_classification, Receptors, Angiotensin, Antagonist, Biological activity, Rats, chemistry, Biochemistry, Receptors, Oxytocin, Molecular Medicine, Female, Hormone, medicine.drug
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16
المؤلفون: Bradley V. Clineschmidt, Peter D. Williams, Jill M. Erb, Douglas J. Pettibone, George F. Lundell, R. M. Freidinger, D. S. Perlow, Mark G. Bock, D. F. Veber, R. D. Tung, Robert M. DiPardo
المصدر: Peptides 1990 ISBN: 9789072199089
Peptides 1990مصطلحات موضوعية: Oxytocin, Chemistry, medicine, Pharmacology, medicine.drug
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17
المصدر: European Journal of Pharmacology. 44:65-74
مصطلحات موضوعية: Male, Serotonin, Crossed extensor reflex, Time Factors, Central nervous system, Motor Activity, Pharmacology, Piperazines, chemistry.chemical_compound, Reflex, polycyclic compounds, medicine, Animals, Xylamidine, 5-HT receptor, MK-212, Behavior, Animal, musculoskeletal, neural, and ocular physiology, Antagonist, Pargyline, Electric Stimulation, Rats, medicine.anatomical_structure, chemistry, Pyrazines, Anesthesia, Female, Serotonin Antagonists, psychological phenomena and processes, Muscle Contraction, medicine.drug
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18
المؤلفون: Michael Williams, Bradley V. Clineschmidt, J. A. Totaro, Patricia R. Bunting, John J. Witoslawski, Edwin A. Risley
المصدر: Drug Development Research. 2:147-163
مصطلحات موضوعية: medicine.drug_class, medicine.medical_treatment, Pharmacology, Anxiolytic, Chlordiazepoxide, Apomorphine, chemistry.chemical_compound, Anticonvulsant, Muscimol, chemistry, Dihydroalprenolol, Drug Discovery, medicine, Licking, Diazepam, medicine.drug
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19A Structurally Unique, Potent, and Selective Oxytocin Antagonist Derived from Streptomyces silvensis
المؤلفون: Roger M. Freidinger, Jerrold M. Liesch, Lawrence R. Koupal, Paul S. Anderson, Michael A. Goetz, Joanne M. Williamson, Otto D. Hensens, Douglas J. Pettibone, Bradley V. Clineschmidt, George F. Lundell, James P. Springer, Cheryl D. Schwartz
المصدر: Endocrinology. 125:217-222
مصطلحات موضوعية: Receptors, Vasopressin, medicine.medical_specialty, Vasopressin, Arginine, In Vitro Techniques, Peptide hormone, Biology, Oxytocin, Peptides, Cyclic, Cyclase, Oxytocin Antagonist, Endocrinology, Internal medicine, medicine, Animals, Receptor, Receptors, Angiotensin, urogenital system, Uterus, Antagonist, Rats, Inbred Strains, Streptomyces, Rats, Arginine Vasopressin, Liver, Receptors, Oxytocin, Female, Peptides, hormones, hormone substitutes, and hormone antagonists, medicine.drug
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20
المصدر: European Journal of Pharmacology. 35:211-214
مصطلحات موضوعية: Serotonin, medicine.medical_specialty, Time Factors, Fenfluramine, Dopamine, Pharmacology, Dose level, Single oral dose, Norepinephrine, Internal medicine, medicine, Animals, Diminution, business.industry, Brain, Rats, Inbred Strains, Rat brain, Rats, Endocrinology, Depression, Chemical, business, medicine.drug