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1
المؤلفون: Bradley Dean Tait, H. William Tedford, Chad A. Finkenbinder, Gary L. Benzon, Bruce A. Steinbaugh, Whitney Smith, Anna Tempczyk-Russell, Lin Bao, Robert M. Kennedy
المصدر: Pesticide Biochemistry and Physiology. 106:124-140
مصطلحات موضوعية: chemistry.chemical_classification, biology, Chemistry, Stereochemistry, Health, Toxicology and Mutagenesis, In silico, fungi, Mutagenesis (molecular biology technique), Peptide, General Medicine, Aedes aegypti, Computational biology, Spodoptera, biology.organism_classification, Beet armyworm, Exigua, Pharmacophore, Agronomy and Crop Science
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2
المؤلفون: Larry J. Markoski, Stephen J. Gracheck, Carolyn Nouhan, Peter J. Tummino, Steven VanderRoest, James Saunders, J. V. N. Vara Prasad, Krishna R. Iyer, Christopher Gajda, Fred E. Boyer, Donna Ferguson, Elizabeth A. Lunney, John M. Domagala, Bradley Dean Tait, Michael Sinz, Donald Hupe, Tod P. Holler, Susan Elizabeth Hagen, Edmund L. Ellsworth
المصدر: Bioorganic & Medicinal Chemistry Letters. 9:2217-2222
مصطلحات موضوعية: Models, Molecular, Dihydropyran, Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Chemical synthesis, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Moiety, HIV Protease Inhibitor, Disulfides, Molecular Biology, chemistry.chemical_classification, Protease, Protease binding, Organic Chemistry, HIV, HIV Protease Inhibitors, Enol, chemistry, Pyrones, Molecular Medicine, Sulfonic Acids, Lactone
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3
المؤلفون: Peter J. Tummino, James Saunders, Stephen J. Gracheck, Bradley Dean Tait, J. V. N. Vara Prasad, Joanne I. Brodfuehrer, Christopher Andrew Gajda, Krishna R. Iyer, Tod P. Holler, Susan Elizabeth Hagen, Steven VanderRoest, Edmund L. Ellsworth, Fred E. Boyer, Carolyn Nouhan, Donna Ferguson, Larry James Markoski, Michael Sinz, Donald Hupe, Elizabeth A. Lunney, John M. Domagala
المصدر: Bioorganic & Medicinal Chemistry Letters. 9:1481-1486
مصطلحات موضوعية: Models, Molecular, Anti-HIV Agents, Dihydropyran, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Thio, Carboxamide, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Drug Discovery, medicine, Animals, Moiety, HIV Protease Inhibitor, Molecular Biology, Pyrans, chemistry.chemical_classification, biology, Chemistry, Organic Chemistry, HIV Protease Inhibitors, Kinetics, Enzyme inhibitor, biology.protein, Molecular Medicine, Lactone
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4
المؤلفون: Bradley Dean Tait, Francis Y. Chung, Barbra H. Stewart, O. Helen Chan, C. John
المصدر: Pharmaceutical Research. 15:1401-1406
مصطلحات موضوعية: Pharmacology, chemistry.chemical_classification, Intestinal permeability, Chromatography, Organic Chemistry, Human immunodeficiency virus (HIV), Synthetic membrane, Pharmaceutical Science, Biology, medicine.disease_cause, medicine.disease, digestive system, Enzyme, chemistry, Biochemistry, Enzyme inhibitor, biology.protein, medicine, Molecular Medicine, HIV Protease Inhibitor, Pharmacology (medical), Intracellular, Biotechnology, Drug transport
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5
المؤلفون: Elizabeth A. Lunney, Frederick E. Boyer, J. V. N. Vara Prasad, Stephen J. Gracheck, Carolyn Nouhan, Edmund L. Ellsworth, Bradley Dean Tait, Donna Ferguson, Susan Elizabeth Hagen, Steven VanderRoest, Larry J. Markoski, James Saunders, Harriet W. Hamilton, B. A. Steinbaugh, Peter J. Tummino, John M. Domagala, Donald Hupe, Christopher Gajda
المصدر: Journal of Medicinal Chemistry. 40:3707-3711
مصطلحات موضوعية: Chemical Phenomena, Anti-HIV Agents, Stereochemistry, Chemical synthesis, Virus, Mice, Structure-Activity Relationship, HIV-1 protease, In vivo, Drug Discovery, medicine, Animals, Structure–activity relationship, chemistry.chemical_classification, biology, Chemistry, Physical, Chemistry, HIV Protease Inhibitors, In vitro, Kinetics, Biochemistry, Pyrones, HIV-1, biology.protein, Molecular Medicine, Ritonavir, Lactone, medicine.drug
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6
المؤلفون: John W. Erickson, Donald Hupe, Eric T. Baldwin, J. R. Rubin, and Sergei V. Gulnik, Christine Humblet, Susan Elizabeth Hagen, Christopher Gajda, Harriet W. Hamilton, Carolyn Nouhan, Beishan Liu, J. V. N. Vara Prasad, Neil Graham, Edmund L. Ellsworth, Peter J. Tummino, John M. Domagala, Alexander Pavlovsky, Donna Ferguson, Elizabeth A. Lunney, T. N. Bhat, Bradley Dean Tait, Stephen J. Gracheck
المصدر: Journal of Medicinal Chemistry. 40:3781-3792
مصطلحات موضوعية: Anti-HIV Agents, Stereochemistry, medicine.medical_treatment, Thio, Crystallography, X-Ray, Chemical synthesis, Structure-Activity Relationship, HIV Protease, Coumarins, Drug Discovery, medicine, Structure–activity relationship, chemistry.chemical_classification, Binding Sites, Protease, biology, Active site, Stereoisomerism, HIV Protease Inhibitors, Amino acid, Enzyme, chemistry, Pyrones, Enzyme inhibitor, Drug Design, HIV-1, biology.protein, Molecular Medicine
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7
المؤلفون: N. Suman-Chauhan, Louise Webdale, Bharat K. Trivedi, Terri S. Purchase, Bruce D. Roth, Bradley Dean Tait, Michael W. Wilson, C.E. Augelli-Szafran
المصدر: Bioorganic & Medicinal Chemistry Letters. 7:2009-2014
مصطلحات موضوعية: chemistry.chemical_classification, Indole test, Stereochemistry, medicine.drug_class, Organic Chemistry, Clinical Biochemistry, Antagonist, Pharmaceutical Science, Biological activity, Receptor antagonist, Biochemistry, Chemical synthesis, CI-988, chemistry, Heterocyclic compound, Drug Discovery, medicine, Molecular Medicine, Moiety, Molecular Biology
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8
المؤلفون: Alan Daugherty, Kathryn Welch, Richard D. Dyer, Joseph A. Cornicelli, Thomas M.A. Bocan, Sandra M. Sendobry, Bharat K. Trivedi, Steven J. Feinmark, Norman L. Colbry, Bradley Dean Tait
المصدر: British Journal of Pharmacology. 120:1199-1206
مصطلحات موضوعية: Pharmacology, medicine.medical_specialty, Antioxidant, biology, Cholesterol, medicine.medical_treatment, Arteriosclerosis, medicine.disease, chemistry.chemical_compound, Endocrinology, ABAP, chemistry, Enzyme inhibitor, In vivo, Internal medicine, medicine, biology.protein, computer, Ex vivo, Lipoprotein, computer.programming_language
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9
المؤلفون: Christopher Gajda, Bradley Dean Tait, Peter J. Tummino, Harriet W. Hamilton, Susan Elizabeth Hagen, Alexander Pavlovsky, Donna Ferguson, Elizabeth A. Lunney
المصدر: Bioorganic & Medicinal Chemistry Letters. 6:719-724
مصطلحات موضوعية: chemistry.chemical_classification, Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, chemistry.chemical_compound, Enzyme, Pyran, Drug Discovery, Molecular Medicine, HIV Protease Inhibitor, Molecular Biology, Alkyl
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10
المؤلفون: Elizabeth A. Lunney, Donna Ferguson, Edmund L. Ellsworth, Bradley Dean Tait, Donald Hupe, Christopher Gajda, John M. Domagala, Peter J. Tummino
المصدر: Journal of Molecular Recognition. 9:139-142
مصطلحات موضوعية: Protease, biology, Chemistry, Stereochemistry, medicine.medical_treatment, Human immunodeficiency virus (HIV), Active site, medicine.disease_cause, Non peptide, Template, Structural Biology, biology.protein, medicine, Molecular Biology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::d281638c28cd1eb87b9535e9b0eda4c5
https://doi.org/10.1002/(sici)1099-1352(199603)9:2<139::aid-jmr249>3.0.co;2-h -
11
المؤلفون: Linda Guilds-Zamarka, Dirk A. Bornemeier, Maritza Oxender, Bruce J. Auerbach, Bharat K. Trivedi, Bradley Dean Tait, Bruce D. Roth, Richard D. Dyer, Joseph A. Cornicelli
المصدر: Bioorganic & Medicinal Chemistry Letters. 6:93-96
مصطلحات موضوعية: Catechol, biology, Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Lipoxygenase, chemistry.chemical_compound, Drug Discovery, biology.protein, Molecular Medicine, Moiety, Molecular Biology, Mass screening
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12
المؤلفون: Peter J. Tummino, C.M. Jacobs, Elizabeth A. Lunney, Bradley Dean Tait, D. Ferguson, L. Hupe, D. Hupe
المصدر: Archives of Biochemistry and Biophysics. 316:523-528
مصطلحات موضوعية: Models, Molecular, Stereochemistry, medicine.medical_treatment, Carboxylic acid, Molecular Sequence Data, Carboxylic Acids, Biophysics, Biochemistry, Sulfone, chemistry.chemical_compound, Non-competitive inhibition, HIV-1 protease, medicine, Phenyl group, Computer Simulation, Amino Acid Sequence, Molecular Biology, chemistry.chemical_classification, Biphenyl, Binding Sites, Protease, biology, Biphenyl Compounds, HIV Protease Inhibitors, Recombinant Proteins, Kinetics, Solubility, chemistry, Drug Design, HIV-1, biology.protein, Lineweaver–Burk plot
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13
المؤلفون: Bradley Dean Tait, William A. Pryor, Joseph A. Cornicelli, Mingdan Wu, D. T. Witiak, L. J. Devall, B. K. Trivedi
المصدر: The Journal of Organic Chemistry. 58:3521-3532
مصطلحات موضوعية: Absorption (pharmacology), Antioxidant, Chromatography, Autoxidation, medicine.medical_treatment, Linoleic acid, Organic Chemistry, Micelle, chemistry.chemical_compound, ABAP, Reaction rate constant, chemistry, medicine, Sodium dodecyl sulfate, computer, computer.programming_language
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14
المؤلفون: D. T. Witiak, B. K. Trivedi, Joseph A. Cornicelli, Mingdan Wu, Bradley Dean Tait, L. J. Devall, William A. Pryor
المصدر: ChemInform. 24
مصطلحات موضوعية: Absorption (pharmacology), Chromatography, Antioxidant, Autoxidation, Linoleic acid, medicine.medical_treatment, General Medicine, Combinatorial chemistry, Micelle, chemistry.chemical_compound, ABAP, Reaction rate constant, chemistry, medicine, Sodium dodecyl sulfate, computer, computer.programming_language
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15
المؤلفون: Susan Elizabeth Hagen, Bradley Dean Tait, Elizabeth A. Lunney, Christopher Gajda, Alexander Pavlovsky, Donna Ferguson, Harriet W. Hamilton, Peter J. Tummino
المصدر: ChemInform. 27
مصطلحات موضوعية: chemistry.chemical_classification, chemistry.chemical_compound, Enzyme, Chemistry, Pyran, Stereochemistry, HIV Protease Inhibitor, General Medicine, Alkyl
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16
المؤلفون: N. Suman-Chauhan, Bradley Dean Tait, Bharat K. Trivedi, Bruce D. Roth, Terri S. Purchase, Michael W. Wilson, C.E. Augelli-Szafran, Louise Webdale
المصدر: ChemInform. 28
مصطلحات موضوعية: Indole test, Stereochemistry, Chemistry, medicine.drug_class, medicine, Antagonist, Moiety, Biological activity, General Medicine, Receptor antagonist, Combinatorial chemistry, CI-988
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17
مصطلحات موضوعية: chemistry.chemical_classification, Enzyme, Protease, chemistry, Pharmacokinetics, medicine.medical_treatment, medicine, Potency, Pharmacology, Blood proteins, Virus, Mass screening, Bioavailability
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18
المؤلفون: Donald Hupe, Alexander Pavlovsky, Donna Ferguson, John M. Domagala, Peter J. Tummino, Susan Elizabeth Hagen, Thomas J. McQuade, Neil Graham, John W. Erickson, Edmund L. Ellsworth, Stephen J. Gracheck, Christopher Gajda, Carolyn Nouhan, J. V. N. Vara Prasad, Kimberly Suzanne Para, Bradley Dean Tait, Elizabeth A. Lunney
المصدر: Bioorganicmedicinal chemistry. 4(9)
مصطلحات موضوعية: Models, Molecular, Molecular model, Chemical Phenomena, Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Crystallography, X-Ray, Biochemistry, HIV-1 protease, Drug Discovery, medicine, Potency, Humans, Benzopyrans, Molecular Biology, IC50, Mass screening, Protease, biology, Chemistry, Organic Chemistry, Active site, HIV Protease Inhibitors, Hydrogen-Ion Concentration, Combinatorial chemistry, In vitro, biology.protein, Molecular Medicine
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19
المؤلفون: J. V. N. Vara Prasad, Elizabeth A. Lunney, Donald Hupe, Peter J. Tummino, Donna Ferguson, Bradley Dean Tait, James B. Dunbar, Kimberly Suzanne Para, Daniel F. Ortwine
المصدر: Journal of the American Chemical Society. 116:6989-6990
مصطلحات موضوعية: Colloid and Surface Chemistry, HIV-1 protease, biology, Chemistry, Stereochemistry, biology.protein, General Chemistry, Biochemistry, Catalysis