-
1Academic Journal
المؤلفون: Pippione, A.C., Kilic-Kurt, Z., Kovachka, S., Sainas, S., Rolando, B., Denasio, E., Pors, Klaus, Adinolfi, S., Zonari, D., Bagnati, R., Lolli, M.L., Spyrakis, F., Oliaro-Bosso, S., Boschi, D.
مصطلحات موضوعية: Aldo-keto reductase 1C3 (AKR1C3), Castration Resistant Prostate Cancer (CRPC), Bioisosteric modulation, Hydroxytriazole scaffold
الاتاحة: http://hdl.handle.net/10454/19070
-
2Academic Journal
المؤلفون: Santos, Ana R.N., Sheldrake, Helen M., Ibrahim, Ali I.M., Danta, Chhanda C., Bonanni, D., Daga, M., Oliaro-Bosso, s., Boschi, D., Lolli, M.L., Pors, Klaus
مصطلحات موضوعية: Tetrahydroisoquinoline, THIQ
الاتاحة: http://hdl.handle.net/10454/17252
-
3Academic Journal
المؤلفون: Pippione, A.C., Carnovale, I.M., Bonanni, D., Sini, Marcella, Goyal, P., Marini, E., Pors, Klaus, Adinolfi, S., Zonari, D., Festuccia, C., Wahlgren, W.Y., Friemann, R., Bagnati, R., Boschi, D., Oliaro-Bosso, S., Lolli, M.L.
مصطلحات موضوعية: Aldo-keto reductase 1C3, AKR1C3, 17β-HSD5, Prostate cancer (PCa), CRPC, Bioisosterism, Scaffold hopping, Inhibitors, X-ray crystallography
الاتاحة: http://hdl.handle.net/10454/16082
-
4Academic Journal
المؤلفون: Pippione, A.C., Giraudo, A., Bonanni, D., Carnovale, I.M., Marini, E., Cena, C., Costale, A., Zonari, D., Pors, Klaus, Sadiq, Maria, Boschi, D., Oliaro-Bosso, S., Lolli, M.L.
مصطلحات موضوعية: Aldo-keto reductase 1C3, AKR1C3, 17β-HSD5, Prostate cancer, CRPC, Bioisosterism, Scaffold hopping, Inhibitors
الاتاحة: http://hdl.handle.net/10454/13966
-
5Academic Journal
المؤلفون: Calistri, A, Luganini, A, Mognetti, B, Elder, E, Sibille, G, Conciatori, V, Del Vecchio, C, Sainas, S, Boschi, D, Montserrat, N, Mirazimi, A, Lolli, ML, Gribaudo, G, Parolin, C
المصدر: Microorganisms. 9(8)
مصطلحات موضوعية: Medicin och hälsovetenskap
-
6Academic Journal
المؤلفون: Pippione A. C., Kilic-Kurt Z., Kovachka S., Sainas S., Rolando B., Denasio E., Pors K., Adinolfi S., Zonari D., Bagnati R., Lolli M. L., Spyrakis F., Oliaro-Bosso S., Boschi D.
المساهمون: Pippione A.C., Kilic-Kurt Z., Kovachka S., Sainas S., Rolando B., Denasio E., Pors K., Adinolfi S., Zonari D., Bagnati R., Lolli M.L., Spyrakis F., Oliaro-Bosso S., Boschi D.
مصطلحات موضوعية: AKR1C3 inhibitors, prostate cancer, triazoles, aldo-keto reductase
Relation: info:eu-repo/semantics/altIdentifier/pmid/35447434; info:eu-repo/semantics/altIdentifier/wos/WOS:000793638500009; volume:237; firstpage:114366; lastpage:114384; numberofpages:19; journal:EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY; http://hdl.handle.net/2318/1859921; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85128267024; https://www-scopus-com.bibliopass.unito.it/record/display.uri?eid=2-s2.0-85128267024&origin=resultslist&sort=plf-f&src=s&st1=10.1016/j.ejmech.2022.114366&sid=07f6cd37fbeafef783a3f166320d8feb&sot=b&sdt=b&sl=33&s=DOI(10.1016/j.ejmech.2022.114366)&relpos=0&citeCnt=0&searchTerm=&featureToggles=FEATURE_NEW_DOC_DETAILS_EXPORT:1
الاتاحة: http://hdl.handle.net/2318/1859921
https://doi.org/10.1016/j.ejmech.2022.114366
https://www-scopus-com.bibliopass.unito.it/record/display.uri?eid=2-s2.0-85128267024&origin=resultslist&sort=plf-f&src=s&st1=10.1016/j.ejmech.2022.114366&sid=07f6cd37fbeafef783a3f166320d8feb&sot=b&sdt=b&sl=33&s=DOI(10.1016/j.ejmech.2022.114366)&relpos=0&citeCnt=0&searchTerm=&featureToggles=FEATURE_NEW_DOC_DETAILS_EXPORT:1 -
7Academic Journal
المؤلفون: Rubin E., Pippione A. C., Boyko M., Einaudi G., Sainas S., Collino M., Cifani C., Lolli M. L., Abu-Freha N., Kaplanski J., Boschi D., Azab A. N.
المساهمون: Rubin E., Pippione A.C., Boyko M., Einaudi G., Sainas S., Collino M., Cifani C., Lolli M.L., Abu-Freha N., Kaplanski J., Boschi D., Azab A.N.
مصطلحات موضوعية: Depression, Inflammation, Ischemic stroke, Mortality, NF-κB, Stroke
Relation: info:eu-repo/semantics/altIdentifier/pmid/35053779; info:eu-repo/semantics/altIdentifier/wos/WOS:000757682800001; volume:12; issue:1; firstpage:35; lastpage:51; numberofpages:17; journal:BRAIN SCIENCES; http://hdl.handle.net/2318/1851978; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85122150981
-
8Academic Journal
المؤلفون: Houshmand M., Vitale N., Orso F., Cignetti A., Molineris I., Gaidano V., Sainas S., Giorgis M., Boschi D., Fava C., Passoni A., Gai M., Geuna M., Sora F., Iurlo A., Abruzzese E., Breccia M., Mulas O., Caocci G., Castagnetti F., Taverna D., Oliviero S., Pane F., Lolli M. L., Circosta P., Saglio G.
المساهمون: Houshmand M., Vitale N., Orso F., Cignetti A., Molineris I., Gaidano V., Sainas S., Giorgis M., Boschi D., Fava C., Passoni A., Gai M., Geuna M., Sora F., Iurlo A., Abruzzese E., Breccia M., Mulas O., Caocci G., Castagnetti F., Taverna D., Oliviero S., Pane F., Lolli M.L., Circosta P., Saglio G.
مصطلحات موضوعية: Drug Resistance, Neoplasm, Fusion Proteins, bcr-abl, Human, Protein Kinase Inhibitor, Dihydroorotate Dehydrogenase, Leukemia, Myelogenous, Chronic, BCR-ABL Positive
وصف الملف: ELETTRONICO
Relation: info:eu-repo/semantics/altIdentifier/pmid/35773274; info:eu-repo/semantics/altIdentifier/wos/WOS:000819455900003; volume:13; issue:6; firstpage:1; lastpage:13; numberofpages:13; journal:CELL DEATH & DISEASE; https://hdl.handle.net/11585/905782; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85133235930; https://www.nature.com/articles/s41419-022-05028-9#Ack1
-
9Academic Journal
المؤلفون: Sainas S., Giorgis M., Circosta P., Gaidano V., Bonanni D., Pippione A. C., Bagnati R., Passoni A., Qiu Y., Cojocaru C. F., Canepa B., Bona A., Rolando B., Mishina M., Ramondetti C., Buccinna B., Piccinini M., Houshmand M., Cignetti A., Giraudo E., Al-Karadaghi S., Boschi D., Saglio G., Lolli M. L.
المساهمون: Sainas S., Giorgis M., Circosta P., Gaidano V., Bonanni D., Pippione A.C., Bagnati R., Passoni A., Qiu Y., Cojocaru C.F., Canepa B., Bona A., Rolando B., Mishina M., Ramondetti C., Buccinna B., Piccinini M., Houshmand M., Cignetti A., Giraudo E., Al-Karadaghi S., Boschi D., Saglio G., Lolli M.L.
مصطلحات موضوعية: Animal, Apoptosi, Binding Site, Biphenyl Compound, Cell Differentiation, Cell Line, Tumor, Drug Design, Enzyme Inhibitor, Female, Half-Life, Human, Leukemia, Myeloid, Acute, Male, Mice, Inbred BALB C, Microsomes, Liver, Molecular Docking Simulation, Oxidoreductases Acting on CH-CH Group Donor, Pyrazole, Pyridine, Rat, Rats, Sprague-Dawley, Structure-Activity Relationship
Relation: info:eu-repo/semantics/altIdentifier/pmid/33844533; info:eu-repo/semantics/altIdentifier/wos/WOS:000651785800011; volume:64; issue:9; firstpage:5404; lastpage:5428; numberofpages:25; journal:JOURNAL OF MEDICINAL CHEMISTRY; https://hdl.handle.net/2318/1795212; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85102878882
-
10Academic Journal
المؤلفون: Gaidano V., Houshmand M., Vitale N., Carra G., Morotti A., Tenace V., Rapelli S., Sainas S., Pippione A. C., Giorgis M., Boschi D., Lolli M. L., Cilloni D., Cignetti A., Saglio G., Circosta P.
المساهمون: Gaidano V., Houshmand M., Vitale N., Carra G., Morotti A., Tenace V., Rapelli S., Sainas S., Pippione A.C., Giorgis M., Boschi D., Lolli M.L., Cilloni D., Cignetti A., Saglio G., Circosta P.
مصطلحات موضوعية: Acute myeloid leukemia, Apoptosi, Cancer metabolism, DHODH, Differentiation, Dipyridamole, Pyrimidine depletion
Relation: volume:13; issue:5; firstpage:1; lastpage:22; numberofpages:22; journal:CANCERS; http://hdl.handle.net/2318/1784382; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85101684784
-
11Report
-
12Report
المؤلفون: Boschi, D., Branca, S., De Martini, F., Hardy, L., Popescu, S.
المصدر: Phys.Rev.Lett. 80 (1998) 1121-1125
مصطلحات موضوعية: Quantum Physics
URL الوصول: http://arxiv.org/abs/quant-ph/9710013
-
13Conference
المؤلفون: Sainas S., Pippione A. C., Bonanni D., Giorgis Marta, Lupino E., Circosta P., Gaidano V., Cignetti A., Piccinini M., Saglio G., Al-Karadaghi S., Boschi D., Lolli M. L.
المساهمون: Sainas S., Pippione A. C., Bonanni D., Giorgis Marta, Lupino E. , Circosta P. , Gaidano V. , Cignetti A. , Piccinini M. , Saglio G. , Al-Karadaghi S. , Boschi D., Lolli M.L.
Relation: ispartofbook:Book of Abstract Postgraduate symposium XII: biological and medicinal chemistry symposium for postgraduates; Postgraduate symposium XII: biological and medicinal chemistry symposium for postgraduates; firstpage:1; lastpage:1; numberofpages:1; http://hdl.handle.net/2318/1689220
الاتاحة: http://hdl.handle.net/2318/1689220
-
14Book
المؤلفون: Sainas S., Dosio F., Boschi D., Lolli M. L.
المساهمون: Botta, Maurizio, Sainas, S., Dosio, F., Boschi, D., Lolli, M.L.
مصطلحات موضوعية: Chitinase, Ivermectin, Neglected tropical disease, Onchocerca volvulu, Onchocerciasi, Scaffold hopping, Biochemistry, Organic Chemistry
Relation: info:eu-repo/semantics/altIdentifier/isbn/9780128151433; info:eu-repo/semantics/altIdentifier/wos/WOS:000452396400002; ispartofbook:Annual Reports in Medicinal Chemistry; volume:51; firstpage:1; lastpage:38; numberofpages:38; http://hdl.handle.net/2318/1678654; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85054152543; http://www.elsevier.com/wps/find/bookdescription.cws_home/BS_ARMC/description#description
-
15Academic Journal
المؤلفون: Giraudo A., Krall J., Bavo F., Nielsen B., Kongstad K. T., Rolando B., De Blasio R., Gloriam D. E., Loffler R., Thiesen L., Harpsoe K., Frydenvang K., Boschi D., Wellendorph P., Lolli M. L., Jensen A. A., Frolund B.
المساهمون: Giraudo A., Krall J., Bavo F., Nielsen B., Kongstad K.T., Rolando B., De Blasio R., Gloriam D.E., Loffler R., Thiesen L., Harpsoe K., Frydenvang K., Boschi D., Wellendorph P., Lolli M.L., Jensen A.A., Frolund B.
مصطلحات موضوعية: PHARMACOLOGICAL CHARACTERIZATION, BINDING, ANALOGS, GLUTAMATE, GLYCINE, SELECTIVITY, ANTAGONISTS, MODULATION, SUBTYPES, AGONISTS
Relation: info:eu-repo/semantics/altIdentifier/pmid/31117514; info:eu-repo/semantics/altIdentifier/wos/WOS:000473251200005; volume:62; issue:12; firstpage:5797; lastpage:5809; numberofpages:13; journal:JOURNAL OF MEDICINAL CHEMISTRY; http://hdl.handle.net/2318/1719861; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85068187580; http://pubs.acs.org/jmc
-
16Academic Journal
المؤلفون: Santos A. R. N., Sheldrake H. M., Ibrahim A. I. M., Danta C. C., Bonanni D., Daga M., Oliaro-Bosso S., Boschi D., Lolli M. L., Pors K.
المساهمون: Santos A.R.N., Sheldrake H.M., Ibrahim A.I.M., Danta C.C., Bonanni D., Daga M., Oliaro-Bosso S., Boschi D., Lolli M.L., Pors K.
مصطلحات موضوعية: AKR1C3, INHIBITORS, Tetrahydroisoquinoline
Relation: info:eu-repo/semantics/altIdentifier/pmid/31673310; info:eu-repo/semantics/altIdentifier/wos/WOS:000481437100020; volume:10; issue:8; firstpage:1476; lastpage:1480; numberofpages:5; journal:MEDCHEMCOMM; http://hdl.handle.net/2318/1719859; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85070714488; http://pubs.rsc.org/en/journals/journal/md
-
17Conference
المؤلفون: Pippione Agnese Chiara, Iakovleva M., Vottero, C., Sainas, S, Kilic-Kurt, Z., Rolando, B, Kovachka, S, Spyrakis, F, Buschini, A., Montalbano, S., Oliaro Bosso, S., Lolli M. L, Boschi D.
المساهمون: Pippione Agnese Chiara , Iakovleva, M., Vottero, C., Sainas, S, Kilic-Kurt, Z., Rolando, B, Kovachka, S, Spyrakis, F, Buschini, A., Montalbano, S., Oliaro Bosso, S., Lolli, M.L, Boschi, D.
Relation: ispartofbook:"-"; 27th National Meeting in Medicinal Chemistry (NMMC27); firstpage:157; lastpage:157; numberofpages:1; https://hdl.handle.net/2318/1909291
الاتاحة: https://hdl.handle.net/2318/1909291
-
18Academic Journal
المؤلفون: Houshmand M., Vitale N., Orso F., Cignetti A., Molineris I., Gaidano V., Sainas S., Giorgis M., Boschi D., Fava C., Iurlo A., Abruzzese E., Breccia M., Mulas O., Caocci G., Castagnetti F., Taverna D., Pane F., Lolli M., Circosta P., Saglio G.
المساهمون: Houshmand M., Vitale N., Orso F., Cignetti A., Molineris I., Gaidano V., Sainas S., Giorgis M., Boschi D., Fava C., Iurlo A., Abruzzese E., Breccia M., Mulas O., Caocci G., Castagnetti F., Taverna D., Pane F., Lolli M., Circosta P., Saglio G.
مصطلحات موضوعية: chronic myeloid leukemia (CML), CML, dihydroorotate dehydrogenase, Meds433
وصف الملف: ELETTRONICO
Relation: volume:22; firstpage:288; lastpage:289; numberofpages:2; journal:CLINICAL LYMPHOMA MYELOMA & LEUKEMIA; https://hdl.handle.net/11585/905767; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85138589925
الاتاحة: https://hdl.handle.net/11585/905767
https://doi.org/10.1016/S2152-2650(22)01366-0 -
19Book
المؤلفون: Pippione A. C., Sainas S., Boschi D., Lolli M. L.
المساهمون: Pippione A.C., Sainas S., Boschi D., Lolli M.L.
مصطلحات موضوعية: Bioisostere, Bioisosterism, Carboxylic group, Drug design, Fused system, Hydroxyazole, Isosterism, Phenol, Scaffold hopping
Relation: info:eu-repo/semantics/altIdentifier/isbn/9780128201817; ispartofbook:Advances in Heterocyclic Chemistry; volume:134; firstpage:273; lastpage:311; numberofpages:39; http://hdl.handle.net/2318/1795165; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85100084670
-
20Book
المؤلفون: Sainas S., Pippione A. C., Boschi D., Lolli M. L.
المساهمون: Sainas S., Pippione A.C., Boschi D., Lolli M.L.
مصطلحات موضوعية: Bioisosterism, Carboxylic group, Drug design, Hydroxyazole, Isosterism, Phenol, Scaffold hopping
Relation: info:eu-repo/semantics/altIdentifier/isbn/9780128201817; ispartofbook:Advances in Heterocyclic Chemistry; volume:134; firstpage:185; lastpage:272; numberofpages:88; http://hdl.handle.net/2318/1795166; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85102462386