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1
المؤلفون: Mark L. Lewis, Charlotte Alice Louise Lane, Blanda Luzia Christa Stammen, David James Rawson, Peter J. Bungay, William A. Million, Stephen Martin Denton, Sharan K. Bagal, Tanya L. Hay, C. Elizabeth Payne, Lisa R. Thompson, Maw Graham Nigel, Cedric Poinsard, Karl Richard Gibson, Kemp Mark Ian, Edward B. Stevens, Melanie S. Glossop
المصدر: ACS Medicinal Chemistry Letters. 6:650-654
مصطلحات موضوعية: business.industry, Sodium channel, Organic Chemistry, Drug Discovery, NAV1, Medicine, Pharmacology, Subtype selective, business, Inflammatory pain, Biochemistry
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2
المؤلفون: Steven M. Gaulier, Dafydd R. Owen, Margarita Rodriguez-Lens, Huw Rees, Valerie A. Horne, Blanda Luzia Christa Stammen, Martin Corless, Maw Graham Nigel, Thomas Ryckmans, David W. Pearce, Ross A. Kinloch, Tracy J. Ringer
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:1702-1706
مصطلحات موضوعية: Agonist, ERG1 Potassium Channel, medicine.drug_class, Chemistry, Pharmaceutical, Clinical Biochemistry, hERG, Pharmaceutical Science, Carboxamide, Pharmacology, Biochemistry, Cell Line, δ-opioid receptor, Structure-Activity Relationship, Opioid receptor, Receptors, Opioid, delta, Drug Discovery, medicine, Animals, Combinatorial Chemistry Techniques, Humans, 4-Aminopyridine, Receptor, Molecular Biology, Ion channel, biology, Electromyography, Chemistry, Organic Chemistry, Ether-A-Go-Go Potassium Channels, Rats, Analgesics, Opioid, Models, Chemical, Drug Design, Neuropathic pain, biology.protein, Molecular Medicine
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3
المؤلفون: Gemma C. Parsons, Peter T. Stephenson, Michelle Y. Platts, Barber Christopher Gordon, Blanda Luzia Christa Stammen, David C. Pryde, David Ellis, David W. Gordon, Helen J. Mason, Rachel L. Eastwood, Catherine Burt, Donald Stuart Middleton, David Bachelor, Martin Corless, Keith Statham, Anthony Wood, Wolfgang Klute, Kerry A. Paradowski, David C. Blakemore, David R. Fenwick
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:1084-1088
مصطلحات موضوعية: ERG1 Potassium Channel, Anti-HIV Agents, Stereochemistry, Clinical Biochemistry, Human immunodeficiency virus (HIV), Pharmaceutical Science, CCR5 receptor antagonist, medicine.disease_cause, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Piperidines, Amide, Drug Discovery, medicine, Combinatorial Chemistry Techniques, Humans, Structure–activity relationship, Molecular Biology, Primary (chemistry), Molecular Structure, Drug discovery, Organic Chemistry, Amides, Combinatorial chemistry, Ether-A-Go-Go Potassium Channels, chemistry, Drug Design, CCR5 Receptor Antagonists, HIV-1, Microsomes, Liver, Molecular Medicine, Piperidine
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4
المؤلفون: Marcel J. de Groot, David Price, Blanda Luzia Christa Stammen, Manos Perros, Anthony Wood, Armour Duncan Robert, Derek J. Leishman, Carolyn Napier
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:4633-4637
مصطلحات موضوعية: Models, Molecular, congenital, hereditary, and neonatal diseases and abnormalities, Receptors, CCR5, medicine.drug_class, Clinical Biochemistry, hERG, Pharmaceutical Science, Carboxamide, CCR5 receptor antagonist, Antiviral Agents, Biochemistry, Cell Line, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Humans, Structure–activity relationship, cardiovascular diseases, Chemokine CCL4, Molecular Biology, Ion channel, Maraviroc, Molecular Structure, biology, Ligand binding assay, Organic Chemistry, HIV, Macrophage Inflammatory Proteins, Ether-A-Go-Go Potassium Channels, Potassium channel, chemistry, CCR5 Receptor Antagonists, biology.protein, Biophysics, Molecular Medicine
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5
المؤلفون: Anthony Wood, Armour Duncan Robert, David Price, Marcel J. de Groot, Martin Paul Edwards, Manos Perros, Blanda Luzia Christa Stammen
المصدر: ChemMedChem. 1:706-709
مصطلحات موضوعية: Benzimidazole, Anti-HIV Agents, Human immunodeficiency virus (HIV), HIV Infections, CCR5 receptor antagonist, medicine.disease_cause, Biochemistry, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Text mining, Drug Discovery, medicine, Humans, General Pharmacology, Toxicology and Pharmaceutics, Receptor, Maraviroc, Pharmacology, business.industry, Organic Chemistry, Hit to lead, Virology, chemistry, CCR5 Receptor Antagonists, Molecular Medicine, Benzimidazoles, business, Cyclobutanes
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6
المصدر: Synthetic Communications. 28:623-632
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Propane, Thermometer, Organic Chemistry, Molecule, Excimer, Medicinal chemistry, Fluorescence
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7
المصدر: Helvetica Chimica Acta, Vol. 80, No 3 (1997) pp. 623-639
مصطلحات موضوعية: Bicyclic molecule, Stereochemistry, Monoterpene, Organic Chemistry, chemistry.chemical_element, Biochemistry, Catalysis, Inorganic Chemistry, chemistry.chemical_compound, chemistry, Dibenzylideneacetone, Intramolecular force, ddc:540, Drug Discovery, Thujone, Physical and Theoretical Chemistry, Palladium
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8
المؤلفون: Simon Gayton, Andrew N. Warren, Blanda Luzia Christa Stammen, Matthew D. Selby, Jens Ahman, Sarah Haycock-Lewandowski, David Price
المصدر: Tetrahedron Letters. 46:5005-5007
مصطلحات موضوعية: Coupling (electronics), chemistry.chemical_compound, chemistry, Amide, Reagent, Organic Chemistry, Drug Discovery, Organic chemistry, Tropane, Biochemistry, Combinatorial chemistry, Polymer supported, Maraviroc
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9
المصدر: Case Studies in Modern Drug Discovery and Development
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, business.industry, Human immunodeficiency virus (HIV), Medicine, CCR5 receptor antagonist, business, medicine.disease_cause, Virology, Maraviroc
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10
المؤلفون: David C. Pryde, Chris Pickford, Paul Targett-Adams, Helen Lavender, Mike Westby, Amy Palmer, Stephen M. Shaw, Tram T. Tran, Florian Wakenhut, Blanda Luzia Christa Stammen, Jenny Middleton, Emily J. S. Graham, Philip Brain, Lyn H. Jones
المصدر: Journal of virology. 85(13)
مصطلحات موضوعية: Models, Molecular, Pyrrolidines, Hepatitis C virus, viruses, Immunology, Hepacivirus, Biology, Viral Nonstructural Proteins, medicine.disease_cause, Endoplasmic Reticulum, Virus Replication, Microbiology, Antiviral Agents, Small Molecule Libraries, Inhibitory Concentration 50, Interferon, Virology, Lipid droplet, Cell Line, Tumor, Vaccines and Antiviral Agents, medicine, Humans, NS5A, Microscopy, Confocal, Endoplasmic reticulum, Imidazoles, virus diseases, Valine, biochemical phenomena, metabolism, and nutrition, Small molecule, Lipids, In vitro, digestive system diseases, Biochemistry, Viral replication, Insect Science, Hepatocytes, Replicon, Carbamates, medicine.drug
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11
المصدر: ChemInform. 29
مصطلحات موضوعية: chemistry.chemical_compound, Chemistry, Propane, Thermometer, Organic chemistry, Molecule, General Medicine, Excimer, Medicinal chemistry, Fluorescence
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12
المؤلفون: David Price, Armour Duncan Robert, Carolyn Napier, Manos Perros, Derek J. Leishman, Anthony Wood, Marcel J. de Groot, Blanda Luzia Christa Stammen
المصدر: Current topics in medicinal chemistry. 8(13)
مصطلحات موضوعية: congenital, hereditary, and neonatal diseases and abnormalities, Receptors, CCR5, Anti-HIV Agents, hERG, Drug Evaluation, Preclinical, CCR5 receptor antagonist, Pharmacology, Maraviroc, chemistry.chemical_compound, Cyclohexanes, Drug Discovery, Humans, cardiovascular diseases, Ion channel, biology, Drug discovery, Ligand binding assay, General Medicine, Triazoles, Ether-A-Go-Go Potassium Channels, chemistry, Lipophilicity, CCR5 Receptor Antagonists, biology.protein, Pharmacophore
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13
المؤلفون: Manos Perros, Marcel J. de Groot, Armour Duncan Robert, David Price, Anthony Wood, Blanda Luzia Christa Stammen, Catherine Burt
المصدر: Chemical biologydrug design. 67(4)
مصطلحات موضوعية: Models, Molecular, Benzimidazole, Receptors, CCR5, Stereochemistry, Chemokine receptor CCR5, Anti-HIV Agents, CCR5 receptor antagonist, Pharmacology, Biochemistry, chemistry.chemical_compound, Structure-Activity Relationship, Piperidines, Cytochrome P-450 CYP2D6 Inhibitors, Drug Discovery, Structure–activity relationship, Moiety, Humans, skin and connective tissue diseases, biology, Organic Chemistry, Tropane, Ligand (biochemistry), chemistry, CCR5 Receptor Antagonists, biology.protein, HIV-1, Molecular Medicine, Piperidine, Tropanes
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14
المؤلفون: Julie Mori, Blanda Luzia Christa Stammen, Manos Perros, Armour Duncan Robert, Anthony Wood, Carolyn Napier, Becky Irvine, David Price, Susan Dobbs, Paul Griffin, Patrick Dorr, Caroline Smith-Burchnell, Mike Westby, Malcolm Macartney, Graham Rickett, Rob Webster
المصدر: Antimicrobial agents and chemotherapy. 49(11)
مصطلحات موضوعية: Male, Receptors, CCR5, Chemokine receptor CCR5, Anti-HIV Agents, Aplaviroc, viruses, Biological Availability, CCR5 receptor antagonist, Pharmacology, Membrane Fusion, Antiviral Agents, Maraviroc, Rats, Sprague-Dawley, chemistry.chemical_compound, Dogs, Viral envelope, In vivo, Viral entry, Cyclohexanes, Drug Resistance, Viral, medicine, Animals, Humans, Pharmacology (medical), Acquired Immunodeficiency Syndrome, biology, Triazoles, Virology, Rats, Infectious Diseases, chemistry, CCR5 Receptor Antagonists, biology.protein, HIV-1, Vicriviroc, Drug Therapy, Combination, medicine.drug, HeLa Cells