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1Academic Journal
المؤلفون: Cipriano, Alessandra, Milite, Ciro, Feoli, Alessandra, Viviano, Monica, Pepe, Giacomo, Campiglia, Pietro, Sarno, Giuliana, Picaud, Sarah, Imaide, Satomi, Makukhin, Nikolai, Filippakopoulos, Panagis, Ciulli, Alessio, Castellano, Sabrina, Sbardella, Gianluca
المصدر: Cipriano , A , Milite , C , Feoli , A , Viviano , M , Pepe , G , Campiglia , P , Sarno , G , Picaud , S , Imaide , S , Makukhin , N , Filippakopoulos , P , Ciulli , A , Castellano , S & Sbardella , G 2022 , ' Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain ' , ChemMedChem , vol. 17 , no. 20 , e202200343 . https://doi.org/10.1002/cmdc.202200343
مصطلحات موضوعية: Benzimidazole-6-sulfonamide, Bromodomain, Bioisosteres, Selectivity, Structure-activity relationships
وصف الملف: application/pdf
الاتاحة: https://discovery.dundee.ac.uk/en/publications/9262919b-076d-4f3a-b6e8-482a936747cd
https://doi.org/10.1002/cmdc.202200343
https://discovery.dundee.ac.uk/ws/files/86582869/ChemMedChem_2022_Cipriano_Discovery_of_Benzo_d_imidazole_6_sulfonamides_as_Bromodomain_and_Extra_Terminal_Domain_BET.pdf
http://www.scopus.com/inward/record.url?scp=85138079605&partnerID=8YFLogxK -
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المؤلفون: Alessandra Cipriano, Ciro Milite, Alessandra Feoli, Monica Viviano, Giacomo Pepe, Pietro Campiglia, Giuliana Sarno, Sarah Picaud, Satomi Imaide, Nikolai Makukhin, Panagis Filippakopoulos, Alessio Ciulli, Sabrina Castellano, Gianluca Sbardella
مصطلحات موضوعية: Male, Pharmacology, Sulfonamides, Bioisosteres, Organic Chemistry, Imidazoles, Nuclear Proteins, Bromodomain, Cell Cycle Proteins, Structure-activity relationships, Biochemistry, Benzimidazole-6-sulfonamide, Selectivity, Drug Discovery, Benzo(a)pyrene, Humans, Molecular Medicine, Benzimidazoles, General Pharmacology, Toxicology and Pharmaceutics, Transcription Factors