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1Academic Journal
المؤلفون: María Ángeles Márquez-Moñino, Raquel Ortega-García, Hayley Whitfield, Andrew M. Riley, Lourdes Infantes, Shane W. Garrett, Megan L. Shipton, Charles A. Brearley, Barry V. L. Potter, Beatriz González
المصدر: Nature Communications, Vol 15, Iss 1, Pp 1-16 (2024)
مصطلحات موضوعية: Science
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2041-1723
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2Academic Journal
المؤلفون: Huanchen Wang, Lalith Perera, Nikolaus Jork, Guangning Zong, Andrew M. Riley, Barry V. L. Potter, Henning J. Jessen, Stephen B. Shears
المصدر: Nature Communications, Vol 13, Iss 1, Pp 1-13 (2022)
مصطلحات موضوعية: Science
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2041-1723
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3Academic Journal
المؤلفون: Xiangdong Su, Wolfgang Dohle, Stephen J. Mills, Joanna M. Watt, Ana M. Rossi, Colin W. Taylor, Barry V. L. Potter
المصدر: ACS Omega, Vol 5, Iss 44, Pp 28793-28811 (2020)
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2470-1343
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4Academic Journal
المؤلفون: Ruqaiyyah Siddiqui, Mutasem Rawas-Qalaji, Mohammed I. El-Gamal, Sreedevi Sajeev, Jayalakshmi Jagal, Seyed-Omar Zaraei, Rawan M. Sbenati, Hanan S. Anbar, Wolfgang Dohle, Barry V. L. Potter, Naveed Ahmed Khan
المصدر: Antibiotics, Vol 12, Iss 3, p 561 (2023)
مصطلحات موضوعية: Acanthamoeba castellanii, CNS infections, free-living amoebae, irosustat, PLGA nanoparticles, STX140, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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5Academic Journal
المؤلفون: Wolfgang Dohle, Xiangdong Su, Yamni Nigam, Edward Dudley, Barry V. L. Potter
المصدر: Molecules, Vol 28, Iss 1, p 5 (2022)
مصطلحات موضوعية: benzyl guanidine, benzyl aminoguanidine hydrazone, guanylation, antimicrobial activity, methicillin-resistant Staphylococcus aureus (MRSA), Organic chemistry, QD241-441
وصف الملف: electronic resource
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6Academic Journal
المؤلفون: Yu-chi Shen, Caroline Arellano-Garcia, Rosa E. Menjivar, Ethan M. Jewett, Wolfgang Dohle, Sofiia Karchugina, Jonathan Chernoff, Barry V. L. Potter, Kate F. Barald
المصدر: BMC Pharmacology and Toxicology, Vol 20, Iss 1, Pp 1-13 (2019)
مصطلحات موضوعية: Neurofibromatosis 2, Nonsteroidal sulfamate derivatives, Tumour treatment, Cytoskeleton, Therapeutics. Pharmacology, RM1-950, Toxicology. Poisons, RA1190-1270
وصف الملف: electronic resource
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7Academic Journal
المؤلفون: Scott D. Hargrave, Anna M. Joubert, Barry V. L. Potter, Wolfgang Dohle, Sumari Marais, Anne E. Mercier
المصدر: Molecules, Vol 27, Iss 12, p 3819 (2022)
مصطلحات موضوعية: cancer, 2-methoxyestradiol, tetrahydroisoquinoline analog (STX3451), radiosensitization, reactive oxygen species, apoptosis, Organic chemistry, QD241-441
وصف الملف: electronic resource
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8Academic Journal
المؤلفون: Wolfgang Dohle, Andrea E. Prota, Grégory Menchon, Ernest Hamel, Michel O. Steinmetz, Barry V. L. Potter
المصدر: ACS Omega, Vol 4, Iss 1, Pp 755-764 (2019)
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2470-1343
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9Academic Journal
المؤلفون: Dharshini Ganeshapillai, L. W. Lawrence Woo, Mark P. Thomas, Atul Purohit, Barry V. L. Potter
المصدر: ACS Omega, Vol 3, Iss 9, Pp 10748-10772 (2018)
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2470-1343
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10Academic Journal
المؤلفون: Joanna M. Watt, Richard Graeff, Barry V. L. Potter
المصدر: Molecules, Vol 26, Iss 23, p 7165 (2021)
مصطلحات موضوعية: synthesis, cADPR, cyclase, nucleotide, fragment, Organic chemistry, QD241-441
وصف الملف: electronic resource
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11Academic Journal
المؤلفون: Nigel Vicker, Helen V. Bailey, Joanna M. Day, Mary F. Mahon, Andrew Smith, Helena J. Tutill, Atul Purohit, Barry V. L. Potter
المصدر: Molecules, Vol 26, Iss 23, p 7166 (2021)
مصطلحات موضوعية: prostate cancer, synthesis, dehydrogenase, homology modelling, chiral chromatography, X-ray crystallography, Organic chemistry, QD241-441
وصف الملف: electronic resource
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12Academic Journal
المؤلفون: Marco Mottinelli, Mathew P. Leese, Barry V. L. Potter
المصدر: Beilstein Journal of Organic Chemistry, Vol 13, Iss 1, Pp 1871-1878 (2017)
مصطلحات موضوعية: cyclization, Pomeranz–Fritsch, steroidomimetic, synthesis, tetrahydroisoquinoline, Science, Organic chemistry, QD241-441
وصف الملف: electronic resource
Relation: https://doaj.org/toc/1860-5397
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13Academic Journal
المؤلفون: Peter J. Watson, Christopher J. Millard, Andrew M. Riley, Naomi S. Robertson, Lyndsey C. Wright, Himali Y. Godage, Shaun M. Cowley, Andrew G. Jamieson, Barry V. L. Potter, John W. R. Schwabe
المصدر: Nature Communications, Vol 7, Iss 1, Pp 1-13 (2016)
مصطلحات موضوعية: Science
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2041-1723
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14Academic Journal
المؤلفون: Ylana Adami Franco, Manoel Oliveira de Moraes, Larissa A. C. Carvalho, Wolfgang Dohle, Renaira Oliveira da Silva, Isabella Harumi Yonehara Noma, Keli Lima, Barry V. L. Potter, João A. Machado-Neto, Silvya Stuchi Maria-Engler
المصدر: International Journal of Molecular Sciences, Vol 24, Iss 14, p 11314 (2023)
مصطلحات موضوعية: STX140, estradiol analogue, melanoma, senescence, B-raf-inhibitor resistance, Biology (General), QH301-705.5, Chemistry, QD1-999
Relation: https://www.mdpi.com/1422-0067/24/14/11314; https://doaj.org/toc/1661-6596; https://doaj.org/toc/1422-0067; https://doaj.org/article/b68f60ce70a9417ab3d6190a93e3a97e
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15Academic Journal
المصدر: ChemistryOpen, Vol 9, Iss 11, Pp 1113-1122 (2020)
مصطلحات موضوعية: Microwave, optimisation, quinoline, synthesis, X-ray crystallography, Chemistry, QD1-999
Relation: https://doi.org/10.1002/open.202000247; https://doaj.org/toc/2191-1363; https://doaj.org/article/6dd4e0b176994deb903ddea9352755b1
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16
المؤلفون: Megan L. Shipton, Fathima A. Jamion, Simon Wheeler, Andrew M. Riley, Felix Plasser, Barry V. L. Potter, Stephen J. Butler
مصطلحات موضوعية: General Chemistry
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17Academic Journal
المؤلفون: Barry V L Potter
المصدر: Proceedings, Vol 22, Iss 1, p 25 (2019)
مصطلحات موضوعية: Estrogens, Cancer, Sulfatase, Inhibition, Synthesis, General Works
Relation: https://www.mdpi.com/2504-3900/22/1/25; https://doaj.org/toc/2504-3900; https://doaj.org/article/4bd2399d3bec4f05adaa52c88bf3a4c9
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18
المؤلفون: Wolfgang Dohle, Hannah Asiki, Wojciech Gruchot, Paul A. Foster, Havreen K. Sahota, Ruoli Bai, Kirsten E. Christensen, Ernest Hamel, Barry V. L. Potter
المصدر: ChemMedChem. 17
مصطلحات موضوعية: Pharmacology, Organic Chemistry, Drug Discovery, Molecular Medicine, General Pharmacology, Toxicology and Pharmaceutics, Biochemistry
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19
المؤلفون: Wolfgang Dohle, Hannah Asiki, Wojciech Gruchot, Paul A. Foster, Havreen K. Sahota, Ruoli Bai, Kirsten E. Christensen, Ernest Hamel, Barry V. L. Potter
مصطلحات موضوعية: Pharmacology, Organic Chemistry, Drug Discovery, Molecular Medicine, General Pharmacology, Toxicology and Pharmaceutics, Biochemistry
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20
المصدر: Potter, B, Mottinelli, M & Leese, M P 2021, ' N-Phenyl-1,2,3,4-tetrahydroisoquinoline: an alternative scaffold for design of 17-hydroxysteroid dehydrogenase 1 inhibitors ', ChemMedChem, vol. 16, no. 1, pp. 259-291 . https://doi.org/10.1002/cmdc.202000762
مصطلحات موضوعية: 17-Hydroxysteroid Dehydrogenases, Stereochemistry, medicine.medical_treatment, Molecular Conformation, Estrone, 01 natural sciences, Biochemistry, Steroid, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, SDG 3 - Good Health and Well-being, Tetrahydroisoquinolines, Drug Discovery, medicine, Humans, Enzyme Inhibitors, General Pharmacology, Toxicology and Pharmaceutics, Hydroxysteroid dehydrogenase, Pharmacology, chemistry.chemical_classification, 010405 organic chemistry, Tetrahydroisoquinoline, Organic Chemistry, Estrogen Receptor alpha, In vitro, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Enzyme, chemistry, Nuclear receptor, Drug Design, THIQ, Molecular Medicine, medicine.drug
وصف الملف: application/pdf